clonidine and agmatine

clonidine has been researched along with agmatine in 49 studies

Research

Studies (49)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's22 (44.90)18.2507
2000's20 (40.82)29.6817
2010's7 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Botta, B; Botta, M; Carmignani, M; Corelli, F; De Bonnevaux, SC; De Luca, C; Delle Monache, F; Delle Monache, G; Espinal, R; Vitali, A; Volpe, AR1
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Andruszkiewicz, R; Ford, C; Hudson, AL; Treder, AP; Zgoda, W1
Andruszkiewicz, R; Ford, C; Hudson, AL; Treder, AP; Walkowiak, A; Zgoda, W1
Hussain, JF; Kendall, DA; Pinthong, D; Wilson, VG1
Limberger, N; Starke, K; Szabo, B; Urban, R1
Li, G; Regunathan, S; Reis, DJ1
Atlas, D2
Hanmer, C; Kendall, DA; Mason, R; Millns, P; Pinthong, D; Wilson, VG; Wright, IK1
Chikkala, DN; Ernsberger, P; Piletz, JE1
Barrow, CJ; Cooper, R; Eshraghi, J; Li, G; Regunathan, S; Reis, DJ1
Baker, GB; Holt, A1
Regunathan, S; Reis, DJ2
da Costa Santos, W; Garcez do Carmo, L; Hirata, H; Jurkiewicz, A; Jurkiewicz, NH1
Chan, CK; Godwin, SJ; Head, GA1
Bramwell, S; McGowan, D; Regunathan, S; Reis, DJ; Wang, H1
Angelini, R; Ascenzi, P; Ercolini, L; Federico, R; Mattevi, A; Venturini, G1
Dillon, MP; Eglen, RM; Hudson, AL; Kendall, DA; Morgan, NG; Nutt, DJ; Wilson, VG1
Chan, SL1
Chun, J; Dominiak, P; Qadri, F; Raasch, W; Schäfer, U1
Danbury, TC; Hudson, AL; Kestin, SC; Ruban, B; Waterman-Pearson, AE1
Li, J; Li, X; Pei, G; Qin, BY1
Göthert, M; Menzel, S; Molderings, GJ1
Dendorfer, A; Dominiak, P; Raasch, W1
Gandía, L; García, AG; Hernández-Guijo, JM; Jurkiewicz, A; Olivares, R; Ruiz-Nuño, A; Santos, WC1
Angelini, R; Ascenzi, P; Binda, C; Botta, M; Federico, R; Leone, L; Venturini, G1
Chun, J; Dominiak, P; Raasch, W; Schäfer, U1
Dominiak, P; Qadri, F; Raasch, W; Schäfer, U1
Ascenzi, P; Fasano, M; Federico, R; Marino, M; Venturini, G1
Ascenzi, P; Marino, M; Pallottini, V1
Garcez-do-Carmo, L; Jurkiewicz, A; Piçarro, I; Santos, WC; Smaili, SS1
Ren, LM; Zhao, D1
Roerig, SC1
Shen, FM; Su, DF; Wang, WZ; Yang, J1
Cheng, JT; Hwang, SL; Liu, IM; Tzeng, TF1
Briaud, S; Sannajust, F; Zhang, BL1
Garcez-do-Carmo, L; Santos, WC1
Coskun, I; Dogrul, A; Uzbay, T1
Gabilan, NH; Rodrigues, AL; Rosa, AO; Zeidan, MP; Zomkowski, AD1
Centurión, D; Cobos-Puc, LE; Márquez-Conde, JA; Monroy-Ordoñez, EB; Sánchez-López, A; Villalón, CM1
Chopde, CT; Kotagale, NR; Patel, MR; Shelkar, GP; Taksande, BG; Ugale, RR1
Chopde, CT; Gahane, AY; Kotagale, NR; Taksande, BG; Ugale, RR1
Cowan, A; Hirsch, DD; Kim, J; Lisek, R; Rawls, SM; Raymondi, N; Rosenthal, A1
Chopde, CT; Hirani, K; Kokare, DM; Kotagale, NR; Mali, PD; Nakhate, KT; Subhedar, NK; Taksande, BG; Ugale, RR1
He, HM; Lu, HG; Ren, LM; Tian, HL; Zhao, D1
Aglawe, MM; Chopde, CT; Kotagale, NR; Taksande, BG; Tripathi, SJ; Umekar, MJ1

Reviews

7 review(s) available for clonidine and agmatine

ArticleYear
Endogenous ligands of imidazoline receptors: classic and immunoreactive clonidine-displacing substance and agmatine.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Agmatine; Animals; Clonidine; Humans; Imidazoles; Imidazoline Receptors; Immunohistochemistry; Ligands; Receptors, Drug

1995
Molecular and physiological properties of clonidine-displacing substance.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Agmatine; Animals; Binding Sites; Clonidine; Humans; Imidazoline Receptors; Liver; Molecular Weight; Placenta; Receptors, Drug

1995
Imidazoline receptors and their endogenous ligands.
    Annual review of pharmacology and toxicology, 1996, Volume: 36

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Antihypertensive Agents; Binding, Competitive; Clonidine; GTP-Binding Proteins; Humans; Imidazoline Receptors; Ligands; Receptors, Adrenergic, alpha-2; Receptors, Drug; Signal Transduction; Structure-Activity Relationship; Synaptic Transmission; Tissue Distribution

1996
'Seeing through a glass darkly': casting light on imidazoline 'I' sites.
    Trends in pharmacological sciences, 1998, Volume: 19, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Allosteric Site; Animals; Binding, Competitive; Brain; Clonidine; Down-Regulation; Imidazoles; Kidney; Monoamine Oxidase; Neuroprotective Agents; Structure-Activity Relationship

1998
Clonidine-displacing substance and its putative role in control of insulin secretion: a minireview.
    General pharmacology, 1998, Volume: 31, Issue:4

    Topics: Agmatine; Animals; Binding Sites; Cells, Cultured; Clonidine; Humans; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans

1998
Agmatine: an endogenous ligand at imidazoline receptors is a novel neurotransmitter.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Animals; Arginine; Binding, Competitive; Brain; Clonidine; Humans; Imidazoline Receptors; Kinetics; Ligands; Receptors, Adrenergic, alpha-2; Receptors, Drug

1999
Biological significance of agmatine, an endogenous ligand at imidazoline binding sites.
    British journal of pharmacology, 2001, Volume: 133, Issue:6

    Topics: Agmatine; Animals; Binding Sites; Binding, Competitive; Blood Pressure; Clonidine; Heart Rate; Humans; Imidazoles; Ligands

2001

Other Studies

42 other study(ies) available for clonidine and agmatine

ArticleYear
Further hypotensive metabolites from Verbesina caracasana.
    Bioorganic & medicinal chemistry letters, 1999, Nov-15, Volume: 9, Issue:22

    Topics: Animals; Antihypertensive Agents; Asteraceae; Mass Spectrometry; Rats

1999
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

2003
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
New analogues of agmatine with higher affinity to imidazoline receptors.
    Bioorganic & medicinal chemistry letters, 2009, Feb-01, Volume: 19, Issue:3

    Topics: Agmatine; Chemistry, Pharmaceutical; Clonidine; Drug Design; Drug Evaluation, Preclinical; Guanidine; Humans; Imidazoles; Imidazoline Receptors; Inhibitory Concentration 50; Kinetics; Models, Chemical; Protein Binding; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins

2009
New imidazoline/α(2)-adrenoceptors affecting compounds-4(5)-(2-aminoethyl)imidazoline (dihydrohistamine) derivatives. Synthesis and receptor affinity studies.
    Bioorganic & medicinal chemistry, 2011, Jan-01, Volume: 19, Issue:1

    Topics: Imidazoles; Magnetic Resonance Spectroscopy; Receptors, Adrenergic, alpha-2

2011
Comparison of the interaction of agmatine and crude methanolic extracts of bovine lung and brain with alpha 2-adrenoceptor binding sites.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Binding, Competitive; Brimonidine Tartrate; Cattle; Cerebral Cortex; Clonidine; Dioxanes; Idazoxan; Imidazoles; Lung; Methanol; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Yohimbine

1995
Cardiovascular effects of agmatine, a "clonidine-displacing substance", in conscious rabbits.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 351, Issue:3

    Topics: Action Potentials; Agmatine; Animals; Binding, Competitive; Blood Pressure; Cerebral Cortex; Cisterna Magna; Clonidine; Electric Stimulation; Female; Heart Rate; Hemodynamics; In Vitro Techniques; Injections; Kidney; Male; Rabbits; Receptors, Adrenergic, alpha-2; Sympathetic Nervous System; Yohimbine

1995
Agmatine recognizes alpha 2-adrenoceptor binding sites but neither activates nor inhibits alpha 2-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 351, Issue:1

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Clonidine; Cyclic AMP; In Vitro Techniques; Male; Quinoxalines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2

1995
Comparison of the properties of agmatine and endogenous clonidine-displacing substance at imidazoline and alpha-2 adrenergic receptors.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:2

    Topics: Agmatine; Animals; Binding Sites; Cattle; Cells, Cultured; Clonidine; Imidazoline Receptors; Receptors, Adrenergic, alpha-2; Receptors, Drug

1995
Agmatine: an endogenous clonidine-displacing substance in the brain.
    Science (New York, N.Y.), 1994, Feb-18, Volume: 263, Issue:5149

    Topics: Adrenal Medulla; Agmatine; Animals; Binding Sites; Brain; Brain Chemistry; Carboxy-Lyases; Cattle; Cerebral Cortex; Clonidine; Epinephrine; Imidazoline Receptors; Neurotransmitter Agents; Norepinephrine; Rats; Receptors, Adrenergic, alpha; Receptors, Drug

1994
Identifying clonidine-displacing substance.
    Science (New York, N.Y.), 1994, Oct-21, Volume: 266, Issue:5184

    Topics: Agmatine; Animals; Brain Chemistry; Cattle; Clonidine; Humans

1994
Metabolism of agmatine (clonidine-displacing substance) by diamine oxidase and the possible implications for studies of imidazoline receptors.
    Progress in brain research, 1995, Volume: 106

    Topics: Agmatine; Amine Oxidase (Copper-Containing); Animals; Clonidine; Dose-Response Relationship, Drug; Imidazoline Receptors; Kidney; Kinetics; Rats; Receptors, Drug; Swine

1995
Functional properties of agmatine in rat vas deferens.
    European journal of pharmacology, 1996, Jul-04, Volume: 307, Issue:3

    Topics: Agmatine; Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Synaptic Transmission; Vas Deferens

1996
Central cardiovascular actions of agmatine, a putative clonidine-displacing substance, in conscious rabbits.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug

1997
An antiserum to idazoxan recognizes an immunoreactive substance in human serum and cerebral spinal fluid which is not agmatine.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Agmatine; Animals; Antibody Specificity; Antigens; Cattle; Clonidine; Humans; Idazoxan; Imidazoline Receptors; Immune Sera; Radioimmunoassay; Rats; Receptors, Drug; Serum Albumin, Bovine

1997
Competitive inhibition of swine kidney copper amine oxidase by drugs: amiloride, clonidine, and gabexate mesylate.
    Biochemical and biophysical research communications, 1997, Nov-07, Volume: 240, Issue:1

    Topics: Agmatine; Amiloride; Amine Oxidase (Copper-Containing); Animals; Binding, Competitive; Catalysis; Clonidine; Gabexate; Kidney; Kinetics; Oxidation-Reduction; Putrescine; Swine

1997
Effects of agmatine on the cardiovascular system of spontaneously hypertensive rats.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Animals; Blood Pressure; Clonidine; Diastole; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Injections, Intravenous; Male; Rats; Rats, Inbred SHR; Systole

1999
Imidazoline (I2) binding sites in chicken brain.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Amiloride; Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Chickens; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug; Tritium

1999
Analgesic effect of agmatine and its enhancement on morphine analgesia in mice and rats.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:1

    Topics: Agmatine; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Clonidine; Drug Synergism; Female; Imidazoles; Imidazoline Receptors; Male; Mice; Morphine; Rats; Rats, Wistar; Receptors, Drug

1999
Imidazoline derivatives and agmatine induce histamine release from the rat stomach.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Chromatography, High Pressure Liquid; Clonidine; Gastric Mucosa; Histamine Release; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoindoles; Rats; Rats, Wistar; Receptors, Drug; Tolazoline

1999
Positive inotropic effects of imidazoline derivatives are not mediated via imidazoline binding sites but alpha1-adrenergic receptors.
    Japanese journal of pharmacology, 2000, Volume: 84, Issue:1

    Topics: Agmatine; Animals; Binding, Competitive; Cardiotonic Agents; Clonidine; Heart; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Myocardial Contraction; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Drug

2000
Blockade by agmatine of catecholamine release from chromaffin cells is unrelated to imidazoline receptors.
    European journal of pharmacology, 2001, Apr-06, Volume: 417, Issue:1-2

    Topics: Acetylcholine; Agmatine; Animals; Benzofurans; Binding Sites; Binding, Competitive; Calcium Channels; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Imidazoles; Imidazoline Receptors; Membrane Potentials; Potassium; Potassium Channels; Receptors, Drug; Receptors, Nicotinic; Sodium Channels

2001
Inhibition of pig liver and Zea mays L. polyamine oxidase: a comparative study.
    Journal of enzyme inhibition, 2001, Volume: 16, Issue:2

    Topics: Agmatine; Amiloride; Amine Oxidase (Copper-Containing); Animals; Benzamidines; Cattle; Clonidine; Enzyme Inhibitors; Gabexate; Guanidines; Indoles; Kidney; Kinetics; Liver; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxidoreductases Acting on CH-NH Group Donors; Pisum sativum; Polyamine Oxidase; Structure-Activity Relationship; Swine; Trypsin; Trypsin Inhibitors; Zea mays

2001
Agmatine, an endogenous ligand at imidazoline binding sites, does not antagonize the clonidine-mediated blood pressure reaction.
    British journal of pharmacology, 2002, Volume: 135, Issue:3

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Aorta, Thoracic; Binding Sites; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Imidazoline Receptors; Ligands; Male; Muscle Contraction; Rats; Rats, Inbred SHR; Receptors, Drug; Vasoconstriction

2002
Agmatine oxidation by copper amine oxidase.
    European journal of biochemistry, 2002, Volume: 269, Issue:3

    Topics: Agmatine; Amine Oxidase (Copper-Containing); Animals; Binding, Competitive; Clonidine; Humans; Imidazoline Receptors; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Male; Membranes; Models, Molecular; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Oxidation-Reduction; Pisum sativum; Pyrrolidines; Rats; Rats, Wistar; Receptors, Drug; Trypsin

2002
Clonidine displacement from type 1 imidazoline receptor by p-aminobenzamidine, the prototype of trypsin-like serine protease inhibitors.
    IUBMB life, 2002, Volume: 54, Issue:5

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Benzamidines; Catalytic Domain; Clonidine; Dose-Response Relationship, Drug; Imidazoline Receptors; Kinetics; Ligands; Male; Models, Chemical; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Drug; Serine Proteinase Inhibitors; Trypsin

2002
Dual effect of agmatine in the bisected rat vas deferens.
    The Journal of pharmacy and pharmacology, 2003, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Epididymis; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Phenoxybenzamine; Potassium Chloride; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine

2003
Electrophysiological responses to imidazoline/alpha2-receptor agonists in rabbit sinoatrial node pacemaker cells.
    Acta pharmacologica Sinica, 2003, Volume: 24, Issue:12

    Topics: Action Potentials; Adrenergic alpha-2 Receptor Agonists; Agmatine; Animals; Antihypertensive Agents; Aorta, Thoracic; Clonidine; Imidazoles; Male; Rabbits; Sinoatrial Node; Vasoconstriction; Xylazine

2003
Spinal and supraspinal agmatine activate different receptors to enhance spinal morphine antinociception.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Analgesics, Opioid; Animals; Clonidine; Dose-Response Relationship, Drug; Injections, Spinal; Male; Mice; Morphine; Norepinephrine; Pain Measurement; Receptors, Adrenergic, alpha-2; Spinal Cord

2003
Cardiovascular effects of agmatine within the rostral ventrolateral medulla are similar to those of clonidine in anesthetized rats.
    Experimental brain research, 2005, Volume: 160, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Anesthesia; Animals; Baroreflex; Blood Pressure; Cardiovascular Physiological Phenomena; Clonidine; Efferent Pathways; Glutamic Acid; Heart Rate; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sympathetic Nervous System

2005
Activation of imidazoline receptors in adrenal gland to lower plasma glucose in streptozotocin-induced diabetic rats.
    Diabetologia, 2005, Volume: 48, Issue:4

    Topics: Adrenal Glands; Adrenal Medulla; Adrenalectomy; Agmatine; Animals; beta-Endorphin; Blood Glucose; Blood Pressure; Clonidine; Diabetes Mellitus, Experimental; Gene Expression; Glucose Transporter Type 4; Imidazoles; Imidazoline Receptors; Male; Monosaccharide Transport Proteins; Muscle Proteins; Phosphoenolpyruvate Carboxykinase (GTP); Rats; Rats, Wistar; Receptors, Drug; Receptors, Opioid, mu

2005
Central actions of agmatine in conscious spontaneously hypertensive rats.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2005, Volume: 27, Issue:8

    Topics: Agmatine; Animals; Antihypertensive Agents; Blood Pressure; Brain; Cardiovascular System; Clonidine; Consciousness; Dose-Response Relationship, Drug; Drug Interactions; Heart Rate; Hypertension; Injections, Intraventricular; Male; Movement; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

2005
L-NAME pre-treatment partially inhibits the agmatine-evoked depression of the electrically induced twitch contraction of isolated rat vas deferens.
    Life sciences, 2006, Jul-24, Volume: 79, Issue:9

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Agmatine; Animals; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Epididymis; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Rats; Rats, Wistar; S-Nitroso-N-Acetylpenicillamine; Synaptic Transmission; Vas Deferens

2006
The contribution of alpha-1 and alpha-2 adrenoceptors in peripheral imidazoline and adrenoceptor agonist-induced nociception.
    Anesthesia and analgesia, 2006, Volume: 103, Issue:2

    Topics: Adrenergic alpha-Agonists; Agmatine; Analgesics; Animals; Clonidine; Dose-Response Relationship, Drug; Hyperalgesia; Imidazoline Receptors; Male; Mice; Mice, Inbred BALB C; Norepinephrine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Yohimbine

2006
Evidence for imidazoline receptors involvement in the agmatine antidepressant-like effect in the forced swimming test.
    European journal of pharmacology, 2007, Jun-22, Volume: 565, Issue:1-3

    Topics: Agmatine; Animals; Antazoline; Antidepressive Agents; Benzofurans; Clonidine; Female; Imidazoles; Imidazoline Receptors; Male; Mice; Receptors, Adrenergic, alpha-2; Receptors, Drug; Receptors, N-Methyl-D-Aspartate; Swimming

2007
Evidence that some imidazoline derivatives inhibit peripherally the vasopressor sympathetic outflow in pithed rats.
    Autonomic neuroscience : basic & clinical, 2008, Dec-05, Volume: 143, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Blood Vessels; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Imidazoles; Imidazoline Receptors; Imidazolines; Injections, Intravenous; Male; Methoxamine; Rats; Rats, Wistar; Sympathetic Nervous System; Vasomotor System

2008
Agmatine, an endogenous imidazoline receptor ligand modulates ethanol anxiolysis and withdrawal anxiety in rats.
    European journal of pharmacology, 2010, Jul-10, Volume: 637, Issue:1-3

    Topics: Agmatine; Animals; Anti-Anxiety Agents; Anxiety; Arginine; Biguanides; Brain; Clonidine; Dose-Response Relationship, Drug; Eflornithine; Ethanol; Guanidines; Imidazoles; Imidazoline Receptors; Ligands; Maze Learning; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome

2010
Repeated agmatine treatment attenuates nicotine sensitization in mice: modulation by alpha2-adrenoceptors.
    Behavioural brain research, 2010, Dec-01, Volume: 213, Issue:2

    Topics: Agmatine; Animals; Arginine; Biguanides; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Eflornithine; Enzyme Inhibitors; Guanidines; Idazoxan; Male; Mice; Motor Activity; Nicotine; Receptors, Adrenergic, alpha-2; Yohimbine

2010
Icilin-evoked behavioral stimulation is attenuated by alpha₂-adrenoceptor activation.
    Brain research, 2011, Apr-12, Volume: 1384

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Agmatine; Analysis of Variance; Animals; Behavior, Animal; Clonidine; Disease Models, Animal; Dose-Response Relationship, Drug; Head Movements; Male; Movement Disorders; Pyrimidinones; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Time Factors; Yohimbine

2011
Agmatine in the hypothalamic paraventricular nucleus stimulates feeding in rats: involvement of neuropeptide Y.
    British journal of pharmacology, 2011, Volume: 164, Issue:2b

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Agmatine; Animals; Arcuate Nucleus of Hypothalamus; Arginine; Clonidine; Drug Synergism; Eating; Feeding Behavior; Hyperphagia; Male; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Neuropeptide Y; Yohimbine

2011
Effects of imidazolines on neurogenic contraction in isolated urinary bladder detrusor strips from rabbit.
    Canadian journal of physiology and pharmacology, 2012, Volume: 90, Issue:2

    Topics: Adenosine Triphosphate; Agmatine; Animals; Carbachol; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Imidazoles; Imidazolines; In Vitro Techniques; Male; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Purinergic Agonists; Rabbits; Synaptic Transmission; Urinary Bladder; Urinary Bladder, Neurogenic

2012
Evidences for the agmatine involvement in antidepressant like effect of bupropion in mouse forced swim test.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 107

    Topics: Agmatine; Animals; Antidepressive Agents; Arginine; Benzofurans; Biguanides; Bupropion; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Eflornithine; Guanidines; Idazoxan; Imidazoles; Immobility Response, Tonic; Injections, Intraventricular; Male; Mice; Motor Activity

2013