cl 277082 has been researched along with pd 128042 in 3 studies
| Studies (cl 277082) | Trials (cl 277082) | Recent Studies (post-2010) (cl 277082) | Studies (pd 128042) | Trials (pd 128042) | Recent Studies (post-2010) (pd 128042) |
|---|---|---|---|---|---|
| 25 | 1 | 0 | 66 | 0 | 14 |
| Protein | Taxonomy | cl 277082 (IC50) | pd 128042 (IC50) |
|---|---|---|---|
| Sterol O-acyltransferase 1 | Rattus norvegicus (Norway rat) | 2.1277 | |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | 0.14 | |
| Sterol O-acyltransferase 1 | Homo sapiens (human) | 1.7444 | |
| Sterol O-acyltransferase 1 | Mus musculus (house mouse) | 0.31 | |
| Acyl-CoA:cholesterol acyltransferase | Oryctolagus cuniculus (rabbit) | 0.1487 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 3 (100.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Berger, JG; Burrier, RE; Clader, JW; Davis, HR; Domalski, M; Dugar, S; Kogan, TP; Salisbury, B; Vaccaro, W | 1 |
| Harte, RA; Jackson, B; Suckling, KE; Yeaman, SJ | 1 |
| Aragane, K; Kitamine, T; Kusunoki, J; Ohnishi, H; Yamaura, T | 1 |
3 other study(ies) available for cl 277082 and pd 128042
| Article | Year |
|---|---|
Substituted (1,2-diarylethyl)amide acyl-CoA:cholesterol acyltransferase inhibitors: effect of polar groups on in vitro and in vivo activity.
Topics: Amides; Animals; Anticholesteremic Agents; Cricetinae; Male; Mesocricetus; Microsomes, Liver; Sterol O-Acyltransferase; Structure-Activity Relationship | 1995 |
Effect of membrane environment on inhibition of acyl-CoA:cholesterol acyltransferase by a range of synthetic inhibitors.
Topics: Anilides; Animals; Cholesterol; Detergents; Enzyme Inhibitors; Esterification; Imidazoles; Liposomes; Male; Microsomes, Liver; Oleic Acid; Oleic Acids; Phenylurea Compounds; Phosphatidylcholines; Rats; Rats, Wistar; Solubility; Sterol O-Acyltransferase; Tumor Cells, Cultured; Urea | 1995 |
[Effect of F-1394, a potent and selective inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), on esterification of cholesterol and basolateral secretion of cholesteryl ester in Caco-2 cells].
Topics: Anilides; Anticholesteremic Agents; Caco-2 Cells; Cholesterol; Cholesterol Esters; Clofibrate; Cyclohexanes; Dioxanes; Esterification; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Intestinal Mucosa; Phenylurea Compounds; Pravastatin; Probucol; Simvastatin; Sterol O-Acyltransferase | 1997 |