Page last updated: 2024-09-02

cl 218872 and kainic acid

cl 218872 has been researched along with kainic acid in 4 studies

Compound Research Comparison

Studies
(cl 218872)
Trials
(cl 218872)
Recent Studies (post-2010)
(cl 218872)
Studies
(kainic acid)
Trials
(kainic acid)
Recent Studies (post-2010) (kainic acid)
158039,54031,775

Protein Interaction Comparison

ProteinTaxonomycl 218872 (IC50)kainic acid (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 2Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 3Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 4Rattus norvegicus (Norway rat)4.2857
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 1Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 2Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 3Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 4Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.0126

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19903 (75.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Biggio, G; Corda, MG; Porceddu, ML; Sanna, E1
Bates, JF; Hall, TW; Peake, L; Standish, LJ; Swearengen, ES1
Pan, HS; Penney, JB; Young, AB1

Other Studies

4 other study(ies) available for cl 218872 and kainic acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Increase in nigral type II benzodiazepine recognition sites following striatonigral denervation.
    European journal of pharmacology, 1985, Jun-07, Volume: 112, Issue:2

    Topics: Animals; Carbolines; Corpus Striatum; Denervation; Flunitrazepam; Kainic Acid; Male; Neural Pathways; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1985
CL 218-872 pretreatment and intervention block kainate-induced convulsions and neuropathology.
    Behavioral neuroscience, 1988, Volume: 102, Issue:1

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Kainic Acid; Male; Organ Specificity; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1988
Characterization of benzodiazepine receptor changes in substantia nigra, globus pallidus and entopeduncular nucleus after striatal lesions.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:3

    Topics: Animals; Binding, Competitive; Corpus Striatum; Flunitrazepam; Globus Pallidus; Glutamates; Glutamic Acid; Kainic Acid; Male; Pyridazines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra; Time Factors

1984