cl 218872 has been researched along with beta-carboline-3-carboxylic acid ethyl ester in 17 studies
| Studies (cl 218872) | Trials (cl 218872) | Recent Studies (post-2010) (cl 218872) | Studies (beta-carboline-3-carboxylic acid ethyl ester) | Trials (beta-carboline-3-carboxylic acid ethyl ester) | Recent Studies (post-2010) (beta-carboline-3-carboxylic acid ethyl ester) |
|---|---|---|---|---|---|
| 158 | 0 | 3 | 240 | 0 | 9 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 14 (82.35) | 18.7374 |
| 1990's | 1 (5.88) | 18.2507 |
| 2000's | 1 (5.88) | 29.6817 |
| 2010's | 1 (5.88) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P | 1 |
| Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
| Clayton, T; Cook, JM; Cromer, BA; Ma, C; Majumder, S; Namjoshi, OA; Petrou, S; Platt, DM; Roth, BL; VanLinn, ML; Yin, W | 1 |
| Faull, RL; Villiger, JW | 1 |
| Arbilla, S; Langer, SZ; Lista, A | 1 |
| Biggio, G; Corda, MG; Porceddu, ML; Sanna, E | 1 |
| Gardner, CR; James, V | 1 |
| Cole, R; De Vellis, J; Noble, EP; Syapin, PJ | 1 |
| Sieghart, W | 2 |
| Herblin, WF | 1 |
| Eichinger, A; Möhler, H; Richards, JG; Sieghart, W | 1 |
| Faull, RL; Holford, NH; Villiger, JW | 1 |
| Eichinger, A; Sieghart, W | 1 |
| Gardner, CR | 1 |
| Drexler, G; Mayer, A; Sieghart, W | 1 |
| Beer, B; Lippa, AS; Meyerson, LR | 1 |
1 review(s) available for cl 218872 and beta-carboline-3-carboxylic acid ethyl ester
| Article | Year |
|---|---|
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles | 1982 |
16 other study(ies) available for cl 218872 and beta-carboline-3-carboxylic acid ethyl ester
| Article | Year |
|---|---|
Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship | 1998 |
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Design, synthesis, and subtype selectivity of 3,6-disubstituted β-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse.
Topics: Alcoholism; Animals; Benzodiazepines; Binding Sites; Carbolines; Cell Line; Computer Simulation; GABA-A Receptor Antagonists; Humans; Protein Subunits; Rats; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 2010 |
Multiple benzodiazepine receptors in the human basal ganglia: a detailed pharmacological and anatomical study.
Topics: Adolescent; Adult; Aged; Autoradiography; Basal Ganglia; Binding, Competitive; Carbolines; Caudate Nucleus; Child; Child, Preschool; Female; Flunitrazepam; Globus Pallidus; Humans; Male; Middle Aged; Putamen; Pyridazines; Receptors, GABA-A | 1988 |
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1988 |
Increase in nigral type II benzodiazepine recognition sites following striatonigral denervation.
Topics: Animals; Carbolines; Corpus Striatum; Denervation; Flunitrazepam; Kainic Acid; Male; Neural Pathways; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1985 |
Actions and interactions of benzodiazepine agonists, antagonists and inverse agonists on suprahyoid muscle twitching.
Topics: Amphetamine; Animals; Benzodiazepines; Carbolines; In Vitro Techniques; Male; Muscle Contraction; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A | 1985 |
Benzodiazepine receptors: multiple receptors or multiple conformations?
Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A | 1985 |
Characterization of benzodiazepine binding sites after short-wave photo-affinity labeling with flunitrazepam.
Topics: Affinity Labels; Animals; Binding Sites; Carbolines; Cell Membrane; Cerebral Cortex; Flunitrazepam; Male; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays | 1986 |
Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.
Topics: Aging; Animals; Animals, Newborn; Carbolines; Cell Membrane; Cerebellum; Clonazepam; Diazepam; Flunitrazepam; Inferior Colliculi; Pyridazines; Rats; Receptors, GABA-A | 1986 |
Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.
Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Molecular Weight; Photochemistry; Pyridazines; Rats; Receptors, GABA-A | 1987 |
Benzodiazepine receptors in the human cerebellar cortex: a quantitative autoradiographic and pharmacological study demonstrating the predominance of type I receptors.
Topics: Adult; Autoradiography; Binding, Competitive; Carbolines; Cerebellar Cortex; Female; Flunitrazepam; Humans; Male; Pyridazines; Receptors, GABA-A | 1987 |
Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Photochemistry; Pyridazines; Rats; Receptors, GABA-A; Temperature | 1984 |
Agonist and inverse agonist effects of CL 218872 on benzodiazepine receptors.
Topics: Action Potentials; Animals; Benzodiazepines; Carbolines; Male; Neural Inhibition; Purkinje Cells; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins.
Topics: Animals; Anti-Anxiety Agents; Carbolines; Cerebellum; Flunitrazepam; Hippocampus; In Vitro Techniques; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Tritium | 1983 |