Page last updated: 2024-09-03
cki 7 and pf 4800567
cki 7 has been researched along with pf 4800567 in 2 studies
Compound Research Comparison
Studies (cki 7) | Trials (cki 7) | Recent Studies (post-2010) (cki 7) | Studies (pf 4800567) | Trials (pf 4800567) | Recent Studies (post-2010) (pf 4800567) |
---|---|---|---|---|---|
35 | 0 | 7 | 10 | 0 | 9 |
Protein Interaction Comparison
Protein | Taxonomy | cki 7 (IC50) | pf 4800567 (IC50) |
---|---|---|---|
Chain A, Casein kinase I isoform delta | Homo sapiens (human) | 0.3715 | |
Chain A, Casein kinase I isoform epsilon | Homo sapiens (human) | 0.3715 | |
Gonadotropin-releasing hormone receptor | Homo sapiens (human) | 0.032 | |
Casein kinase I isoform delta | Homo sapiens (human) | 0.5413 | |
Casein kinase I isoform epsilon | Homo sapiens (human) | 0.032 |
Research
Studies (2)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Feng, S; Ji, P; Li, GB; Ma, S; Sun, QZ; Wang, ZR; Yan, HX; Yang, LL; Yang, SY; Zou, J | 1 |
Chen, T; Chen, Y; Feng, F; Guo, Q; Lin, H; Liu, W; Liu, Z; Qiao, Y; Qu, W; Sun, H; Yang, H | 1 |
Reviews
1 review(s) available for cki 7 and pf 4800567
Article | Year |
---|---|
Small molecule modulators targeting protein kinase CK1 and CK2.
Topics: Animals; Casein Kinase I; Casein Kinase II; Drug Discovery; Humans; Molecular Docking Simulation; Protein Kinase Inhibitors; Small Molecule Libraries | 2019 |
Other Studies
1 other study(ies) available for cki 7 and pf 4800567
Article | Year |
---|---|
Discovery of N6-phenyl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine derivatives as novel CK1 inhibitors using common-feature pharmacophore model based virtual screening and hit-to-lead optimization.
Topics: Casein Kinase I; Diamines; Dose-Response Relationship, Drug; Drug Discovery; High-Throughput Screening Assays; Models, Molecular; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship | 2012 |