Compounds > cki 7
Page last updated: 2024-09-03

cki 7 and (R)-DRF053

cki 7 has been researched along with (R)-DRF053 in 1 studies

Compound Research Comparison

Studies
(cki 7)		Trials
(cki 7)		Recent Studies (post-2010)
(cki 7)		Studies
((R)-DRF053)		Trials
((R)-DRF053)		Recent Studies (post-2010) ((R)-DRF053)
3507706

Protein Interaction Comparison

ProteinTaxonomycki 7 (IC50)(R)-DRF053 (IC50)
Glycogen synthase kinase-3 beta Sus scrofa (pig)4.1
[Tau protein] kinase Sus scrofa (pig)4.1
Cyclin-T1Homo sapiens (human)8
Cyclin-dependent kinase 1Homo sapiens (human)1.96
G2/mitotic-specific cyclin-B1Homo sapiens (human)1.96
Cyclin-A2Homo sapiens (human)0.29
G1/S-specific cyclin-E1Homo sapiens (human)0.093
Cyclin-dependent kinase 2Homo sapiens (human)0.1915
Casein kinase I isoform alphaHomo sapiens (human)0.014
Cyclin-dependent kinase 7Homo sapiens (human)0.822
Cyclin-dependent kinase 9Homo sapiens (human)8
Cyclin-HHomo sapiens (human)0.822
CDK-activating kinase assembly factor MAT1Homo sapiens (human)0.822
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.1475
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.1475

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Feng, S; Ji, P; Li, GB; Ma, S; Sun, QZ; Wang, ZR; Yan, HX; Yang, LL; Yang, SY; Zou, J1

Other Studies

1 other study(ies) available for cki 7 and (R)-DRF053

ArticleYear
Discovery of N6-phenyl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine derivatives as novel CK1 inhibitors using common-feature pharmacophore model based virtual screening and hit-to-lead optimization.
    European journal of medicinal chemistry, 2012, Volume: 56

    Topics: Casein Kinase I; Diamines; Dose-Response Relationship, Drug; Drug Discovery; High-Throughput Screening Assays; Models, Molecular; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship

2012
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