cisapride and td-5108

cisapride has been researched along with td-5108 in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (50.00)29.6817
2010's7 (43.75)24.3611
2020's1 (6.25)2.80

Authors

AuthorsStudies
Cange, L; Finizia, C; Lundell, L; Ruth, M1
Olden, KW1
Kamm, MA1
Kawatsu, R; Kohmura, Y; Toga, T1
Armstrong, SR; Beattie, DT; Humphrey, PP; Marquess, D; Sandlund, C; Shaw, JP; Smith, JA; Taylor, JA1
Beattie, DT; Humphrey, PP; Marquess, D; Shaw, JP; Smith, JA; Vickery, RG1
Vakil, N1
Barberich, TJ; Hewitt, MC; Shao, L; Wang, F1
Ajdary, S; Ataee, R; Rezayat, M; Shahriari, S; Shokrgozar, MA; Zarrindast, MR1
Heras, J; Mas, M; Mearín, F; Plazas, MJ1
Chai, W; Chan, KY; Danser, AH; de Maeyer, JH; de Vries, R; MaassenVanDenBrink, A; Saxena, PR; Schuurkes, JA; van den Bogeardt, AJ; Villalón, CM1
Camilleri, M; Chang, L; Chey, WD; De Maeyer, JH; Galligan, JJ; Lacy, BE; Müller-Lissner, S; Quigley, EM; Schuurkes, J; Stanghellini, V; Tack, J1
Amagasu, SM; Beattie, DT; Ero, MP; Higgins, DL; Hopkins, A; Kersey, K; Smith, JA; Vickery, RG1
Burgard, EC; Kullmann, FA; Kurihara, R; McKenna, DG; Thor, KB; Wells, GI; Ye, L1
Camilleri, M; Chedid, V; Erwin, PJ; Mandawat, A; Murad, MH; Vijayvargiya, P1
Fujio, Y; Hamatani, T; Kaji, Y; Kakuyama, H; Kawai, H; Noda, N; Takagaki, T; Yodo, Y1

Reviews

4 review(s) available for cisapride and td-5108

ArticleYear
Pharmacological treatment of irritable bowel syndrome--from concept to sales.
    The European journal of surgery. Supplement. : = Acta chirurgica. Supplement, 2002, Issue:587

    Topics: Antidepressive Agents; Benzofurans; Carbolines; Cisapride; Constipation; Drug Industry; Gastrointestinal Agents; Humans; Indoles; Irritable Bowel Syndrome; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2002
New pharmacological agents for the treatment of gastroesophageal reflux disease.
    Reviews in gastroenterological disorders, 2008,Spring, Volume: 8, Issue:2

    Topics: Anti-Ulcer Agents; Benzamides; Cisapride; Esophageal Sphincter, Lower; Gastroesophageal Reflux; Humans; Imidazoles; Proton Pump Inhibitors; Pyridines; Quinuclidines; Serotonin 5-HT4 Receptor Agonists

2008
Systematic review: cardiovascular safety profile of 5-HT(4) agonists developed for gastrointestinal disorders.
    Alimentary pharmacology & therapeutics, 2012, Volume: 35, Issue:7

    Topics: Cardiovascular Diseases; Cisapride; Gastrointestinal Agents; Gastrointestinal Diseases; Humans; Indoles; Randomized Controlled Trials as Topic; Serotonin 5-HT4 Receptor Agonists

2012
Effects of Promotility Agents on Gastric Emptying and Symptoms: A Systematic Review and Meta-analysis.
    Gastroenterology, 2019, Volume: 156, Issue:6

    Topics: Breath Tests; Cisapride; Domperidone; Dopamine D2 Receptor Antagonists; Dyspepsia; Gastric Emptying; Gastroparesis; Ghrelin; Humans; Macrocyclic Compounds; Oligopeptides; Radionuclide Imaging; Randomized Controlled Trials as Topic; Serotonin 5-HT4 Receptor Agonists; Symptom Assessment

2019

Trials

2 trial(s) available for cisapride and td-5108

ArticleYear
The effect of mosapride on oesophageal motor function and acid reflux in patients with gastro-oesophageal reflux disease.
    European journal of gastroenterology & hepatology, 2003, Volume: 15, Issue:10

    Topics: Adult; Aged; Benzamides; Cisapride; Cross-Over Studies; Double-Blind Method; Drug Administration Schedule; Esophagus; Female; Gastroesophageal Reflux; Gastrointestinal Agents; Humans; Hydrogen-Ion Concentration; Male; Manometry; Middle Aged; Morpholines; Peristalsis; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists

2003
Thorough QT/QTc Study Shows That a Novel 5-HT
    Clinical pharmacology in drug development, 2020, Volume: 9, Issue:8

    Topics: Administration, Oral; Adult; Anti-Bacterial Agents; Arrhythmias, Cardiac; Asian People; Benzamides; Case-Control Studies; Cisapride; Cross-Over Studies; Double-Blind Method; Electrocardiography; Female; Humans; Indoles; Irritable Bowel Syndrome; Long QT Syndrome; Male; Morpholines; Moxifloxacin; Piperidines; Placebos; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists

2020

Other Studies

10 other study(ies) available for cisapride and td-5108

ArticleYear
Therapy for irritable bowel syndrome.
    The New England journal of medicine, 2004, Mar-18, Volume: 350, Issue:12

    Topics: Antidepressive Agents; Cisapride; Female; Humans; Indoles; Irritable Bowel Syndrome; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
The 5-HT(4) agonists cisapride, mosapride, and CJ-033466, a Novel potent compound, exhibit different human ether-a-go-go-related gene (hERG)-blocking activities.
    Journal of pharmacological sciences, 2007, Volume: 105, Issue:2

    Topics: Aminopyridines; Arrhythmias, Cardiac; Benzamides; Cell Line; Cisapride; Electrophysiology; Ether-A-Go-Go Potassium Channels; Humans; Imidazoles; Inhibitory Concentration 50; Morpholines; Patch-Clamp Techniques; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists

2007
The in vivo gastrointestinal activity of TD-5108, a selective 5-HT(4) receptor agonist with high intrinsic activity.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:1

    Topics: Administration, Oral; Animals; Azabicyclo Compounds; Benzamides; Cisapride; Colon; Dogs; Dose-Response Relationship, Drug; Esophagus; Female; Gastrointestinal Transit; Guinea Pigs; Indoles; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Rats; Rats, Sprague-Dawley; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists

2008
The in vitro pharmacological profile of TD-5108, a selective 5-HT(4) receptor agonist with high intrinsic activity.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:1

    Topics: Animals; Azabicyclo Compounds; Benzamides; Cell Line; Cisapride; Colon; Cyclic AMP; Esophagus; Ether-A-Go-Go Potassium Channels; Guinea Pigs; Humans; Indoles; Kidney; Morpholines; Protein Binding; Rats; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists

2008
mu-Opioid/5-HT4 dual pharmacologically active agents-efforts towards an effective opioid analgesic with less GI and respiratory side effects (Part I).
    Bioorganic & medicinal chemistry letters, 2009, Oct-01, Volume: 19, Issue:19

    Topics: Analgesics, Opioid; Cisapride; Gastrointestinal Transit; Humans; Metoclopramide; Receptors, Opioid, mu; Receptors, Serotonin, 5-HT4; Respiratory System; Serotonin 5-HT4 Receptor Agonists; Stereoisomerism; Tramadol

2009
Study of 5HT3 and HT4 receptor expression in HT29 cell line and human colon adenocarcinoma tissues.
    Archives of Iranian medicine, 2010, Volume: 13, Issue:2

    Topics: Adenocarcinoma; Aminobenzoates; Biguanides; Blotting, Western; Bridged Bicyclo Compounds, Heterocyclic; Cell Proliferation; Cisapride; Colonic Neoplasms; HT29 Cells; Humans; Oxazines; para-Aminobenzoates; Piperidines; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2010
[Cardiac safety of cinitapride].
    Gastroenterologia y hepatologia, 2010, Volume: 33, Issue:8

    Topics: Arrhythmias, Cardiac; Aryl Hydrocarbon Hydroxylases; Benzamides; Cisapride; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Drug Interactions; Dyspepsia; Electrocardiography; Gastrointestinal Agents; Humans; Ketoconazole; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists

2010
Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.
    Life sciences, 2012, Apr-09, Volume: 90, Issue:13-14

    Topics: 5-Methoxytryptamine; Adolescent; Adult; Aged; Benzofurans; Calcium Channels; Child; Cisapride; Female; Gastrointestinal Agents; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Middle Aged; Muscle Contraction; Myocardium; Pyridines; Quinuclidines; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Sulfonamides; Young Adult

2012
An in vitro investigation of the cardiovascular effects of the 5-HT(4) receptor selective agonists, velusetrag and TD-8954.
    Vascular pharmacology, 2013, Volume: 58, Issue:1-2

    Topics: Adult; Animals; Azabicyclo Compounds; Benzimidazoles; CHO Cells; Cisapride; Coronary Vessels; Cricetinae; Cricetulus; Dogs; Ether-A-Go-Go Potassium Channels; Female; Humans; In Vitro Techniques; Indoles; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin 5-HT4 Receptor Agonists; Swine

2013
Effects of the 5-HT4 receptor agonist, cisapride, on neuronally evoked responses in human bladder, urethra, and ileum.
    Autonomic neuroscience : basic & clinical, 2013, Volume: 176, Issue:1-2

    Topics: Adult; Aged; Cisapride; Electric Stimulation; Evoked Potentials; Female; Humans; Ileum; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Neurons; Organ Culture Techniques; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Urethra; Urinary Bladder

2013