cisapride and gr 113808

cisapride has been researched along with gr 113808 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (33.33)18.2507
2000's6 (50.00)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bockaert, J; Claeysen, S; Dumuis, A; Journot, L; Sebben, M1
Bender, E; Gommeren, W; Jurzak, M; Leysen, J; Luyten, W; Van den Wyngaert, I; Verhasselt, P1
Bender, E; Gommeren, W; Jurzak, M; Leysen, J; Luyten, W; Pindon, A; van Oers, I; Verhasselt, P; Zhang, YB1
Berque-Bestel, I; Fischmeister, R; Langlois, M; Lezoualc'h, F; Mialet, J; Sicsic, S1
Bach, T; Brattelid, T; Kaumann, AJ; Krobert, KA; Kvingedal, AM; Levy, FO; Syversveen, T1
Alisi, MA; Apicella, C; Capezzone de Joannon, A; Cazzolla, N; Costi, R; Cuzzucoli Crucitti, G; Di Santo, R; Furlotti, G; Garrone, B; Iacovo, A; Magarò, G; Mangano, G; Miele, G; Ombrato, R; Pescatori, L; Polenzani, L; Rosi, F; Vitiello, M1
Mizutani, Y; Suzuki, T; Takeda, M; Taniyama, K; Tsukamoto, K1
Akkermans, LM; Briejer, MR; Lefebvre, RA; Prins, NH; Schuurkes, JA; Van Haselen, JF1
Cartier, D; Contesse, V; Delarue, C; Duparc, C; Fischmeister, R; Godin, M; Kuhn, JM; Lefebvre, H; Lihrmann, I; Vaudry, H1
Debonnel, G; Lucas, G1
Fujii, H; Kadowaki, M; Kojima, Y; Nakagawa, T; Nakajima, Y; Shimatani, H; Takaki, M1
Chai, W; Chan, KY; Danser, AH; de Maeyer, JH; de Vries, R; MaassenVanDenBrink, A; Saxena, PR; Schuurkes, JA; van den Bogeardt, AJ; Villalón, CM1

Trials

1 trial(s) available for cisapride and gr 113808

ArticleYear
Characterization of serotonin(4) receptors in adrenocortical aldosterone-producing adenomas: in vivo and in vitro studies.
    The Journal of clinical endocrinology and metabolism, 2002, Volume: 87, Issue:3

    Topics: Adenoma; Adrenal Cortex Neoplasms; Adult; Aldosterone; Cisapride; Female; Humans; In Vitro Techniques; Indoles; Male; Middle Aged; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2002

Other Studies

11 other study(ies) available for cisapride and gr 113808

ArticleYear
Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor.
    FEBS letters, 1996, Nov-25, Volume: 398, Issue:1

    Topics: Age Factors; Amino Acid Sequence; Animals; Animals, Newborn; Base Sequence; Binding Sites; Brain; Brain Chemistry; Cloning, Molecular; Inferior Colliculi; Mice; Molecular Sequence Data; Rats; Rats, Inbred Strains; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Transfection

1996
Cloning and expression of a human serotonin 5-HT4 receptor cDNA.
    Journal of neurochemistry, 1997, Volume: 69, Issue:5

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Brain; Cell Membrane; Cloning, Molecular; COS Cells; Cytosine; DNA Primers; Frameshift Mutation; Guinea Pigs; Humans; Indoles; Kinetics; Molecular Sequence Data; Open Reading Frames; Polymerase Chain Reaction; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Sulfonamides; Swine; Transfection

1997
Structure of the human serotonin 5-HT4 receptor gene and cloning of a novel 5-HT4 splice variant.
    Journal of neurochemistry, 2000, Volume: 74, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; COS Cells; DNA, Recombinant; Genetic Variation; Humans; Molecular Sequence Data; Protein Isoforms; Receptors, Serotonin; RNA, Messenger; Tissue Distribution

2000
Pharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cells.
    British journal of pharmacology, 2000, Volume: 131, Issue:4

    Topics: Animals; CHO Cells; Cricetinae; Cyclic AMP; Humans; Indoles; Protein Isoforms; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Structure-Activity Relationship; Sulfonamides

2000
5HT4(a) and 5-HT4(b) receptors have nearly identical pharmacology and are both expressed in human atrium and ventricle.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:2

    Topics: Adenylyl Cyclases; Adult; Animals; Base Sequence; Cell Line; Cloning, Molecular; Cyclic AMP; DNA, Recombinant; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Mice; Middle Aged; Molecular Sequence Data; Myocardium; Protein Isoforms; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2001
Discovery and pharmacological profile of new 1H-indazole-3-carboxamide and 2H-pyrrolo[3,4-c]quinoline derivatives as selective serotonin 4 receptor ligands.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Animals; Computational Biology; Dogs; Drug Design; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Ligands; Macaca fascicularis; Mice; Microsomes, Liver; Molecular Structure; Nociception; Protein Binding; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin, 5-HT4; Structure-Activity Relationship; Swine

2012
Identification of SK-951, a novel benzofuran derivative, as an agonist to 5-HT4 receptors.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:2

    Topics: Acetylcholine; Animals; Benzofurans; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Cisapride; Electric Stimulation; Esophagus; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Muscarinic; Serotonin Receptor Agonists; Sulfonamides

1999
Pharmacological characterization of 5-HT4 receptors mediating relaxation of canine isolated rectum circular smooth muscle.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: 5-Methoxytryptamine; Animals; Cisapride; Colon; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Indoles; Male; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Rectum; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

1999
5-HT4 receptors exert a frequency-related facilitatory control on dorsal raphé nucleus 5-HT neuronal activity.
    The European journal of neuroscience, 2002, Volume: 16, Issue:5

    Topics: 4-Aminobenzoic Acid; Action Potentials; Animals; Benzofurans; Cisapride; Electrophysiology; Indoles; Male; Neurons; para-Aminobenzoates; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2002
A 5-HT4 agonist mosapride enhances rectorectal and rectoanal reflexes in guinea pigs.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:2

    Topics: Anal Canal; Animals; Benzamides; Cisapride; Guinea Pigs; Indoles; Injections, Intravenous; Male; Morpholines; Muscle Contraction; Muscle Relaxation; Receptors, Serotonin; Rectum; Reflex; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Transducers, Pressure

2003
Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.
    Life sciences, 2012, Apr-09, Volume: 90, Issue:13-14

    Topics: 5-Methoxytryptamine; Adolescent; Adult; Aged; Benzofurans; Calcium Channels; Child; Cisapride; Female; Gastrointestinal Agents; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Middle Aged; Muscle Contraction; Myocardium; Pyridines; Quinuclidines; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Sulfonamides; Young Adult

2012