Page last updated: 2024-09-04

cinacalcet and tacrolimus

cinacalcet has been researched along with tacrolimus in 5 studies

Compound Research Comparison

Studies
(cinacalcet)
Trials
(cinacalcet)
Recent Studies (post-2010)
(cinacalcet)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
1,07015562717,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomycinacalcet (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Asberg, A; Bergan, S; Falck, P; Holdaas, H; Midtvedt, K; Reubsaet, JL; Vethe, NT1
Heller, T; Koziolek, MJ; Maass, E; Mueller, GA1
Cointault, O; Durand, D; Esposito, L; Gandia, P; Gennero, I; Guitard, J; Kamar, N; Lavayssière, L; Rostaing, L; Spataru, L1
Edminister, JR; Huang, WW; Jorizzo, JL; Patel, HA; Pixley, JN1

Reviews

1 review(s) available for cinacalcet and tacrolimus

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for cinacalcet and tacrolimus

ArticleYear
Cinacalcet's effect on the pharmacokinetics of tacrolimus, cyclosporine and mycophenolate in renal transplant recipients.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 2008, Volume: 23, Issue:3

    Topics: Adult; Aged; Cinacalcet; Cyclosporine; Dose-Response Relationship, Drug; Female; Humans; Immunosuppressive Agents; Kidney; Kidney Transplantation; Male; Middle Aged; Mycophenolic Acid; Naphthalenes; Tacrolimus

2008

Other Studies

3 other study(ies) available for cinacalcet and tacrolimus

ArticleYear
Decrease in serum tacrolimus level and rise in serum creatinine under late addition of cinacalcet in a renal transplant recipient with hyperparathyroidism: a case report.
    Transplantation proceedings, 2007, Volume: 39, Issue:10

    Topics: Cinacalcet; Creatinine; Drug Interactions; Drug Therapy, Combination; Female; Humans; Hyperparathyroidism, Secondary; Immunosuppressive Agents; Kidney Transplantation; Middle Aged; Naphthalenes; Tacrolimus

2007
Pharmacodynamic effects of cinacalcet after kidney transplantation: once- versus twice-daily dose.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 2008, Volume: 23, Issue:11

    Topics: Adult; Aged; Calcium; Cinacalcet; Cyclosporine; Dose-Response Relationship, Drug; Female; Humans; Hypercalcemia; Hyperparathyroidism, Secondary; Kidney Failure, Chronic; Kidney Transplantation; Longitudinal Studies; Male; Middle Aged; Naphthalenes; Parathyroid Hormone; Phosphorus; Prospective Studies; Tacrolimus

2008
Improvement of Hailey-Hailey Disease With Topical Cinacalcet, 3%, Ointment.
    JAMA dermatology, 2023, 06-01, Volume: 159, Issue:6

    Topics: Cinacalcet; Humans; Ointments; Pemphigus, Benign Familial; Tacrolimus

2023