cimetidine and thioperamide

cimetidine has been researched along with thioperamide in 52 studies

Research

Studies (52)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's32 (61.54)18.2507
2000's18 (34.62)29.6817
2010's2 (3.85)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Pratim Roy, P; Roy, K1
Arrang, JM; de Waele, C; Khateb, A; Mulhethaler, M; Serafin, M; Vibert, N; Vidal, PP; Yabe, T1
Bent, S; Braam, U; Fehling, U; Schmutzler, W; Schunack, W1
Barnes, PJ; Ichinose, M1
Bolser, DC; Chapman, RW; DeGennaro, FC; Hey, JA; O'Reilly, S1
Fujimoto, K; Gotoh, Y; Granger, DN; Kang, M; Sakai, T; Sakata, T; Tso, P; Tsunada, S1
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H1
Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M1
Kohno, S; Nabe, T; Ogawa, K; Ohata, K; Yamamura, H1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Hey, JA; Hutchison, RW1
Gertner, SB; Hey, JA; McLeod, RL1
Kamondi, A; Reiner, PB1
Koss, MC1
Kamei, C; Tasaka, K1
Arrang, JM; de Waele, C; Mühlethaler, M; Serafin, M; Vibert, N; Vidal, PP; Yabe, T1
Fort, P; Jones, BE; Khateb, A; Mühlethaler, M; Pegna, A1
Fujimoto, K; Gotoh, Y; Ogata, S; Ohyama, T; Okamoto, K; Ootani, A; Sakata, T; Tsunada, S1
Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Corbel, S; Dy, M1
KAMEI, CH1
Ea-Kim, L; Javellaud, J; Oudart, N1
Akiyama, K; Maeda, Y; Mita, H; Saito, H; Shimizu, H1
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Hough, LB; Li, BY; Nalwalk, JW1
Harada, N; Iwai, H; Nagata, M; Tomoda, K; Yamashita, T1
Bivalacqua, TJ; Champion, HC; Czapla, MA; Ilgenfritz, C; Kadowitz, PJ; Santiago, JA1
Laurikainen, E; Miller, JM; Nuttall, AL; Quirk, WS1
Acuña, Y; Campos, HA; Israel, A; Mathison, Y1
Flood, JF; Morley, JE; Uezu, K1
Bacciottini, L; Blandina, P; Chiappetta, M; Giovannini, MG; Mannaioni, PF1
Gao, C; Hu, Hz; Liu, S; Ren, J; Wood, JD; Xia, Y1
Bacciottini, L; Blandina, P; Cangioli, I; Mannaioni, PF; Passani, MB1
Anichtchik, OV; Panula, P; Peitsaro, N1
Ikarashi, Y; Ishige, A; Kuribara, H; Maruyama, Y; Sasaki, H; Yuzurihara, M1
Ghosh, AK; Hirasawa, N; Ohuchi, K1
Anai, M; Asano, T; Fukushima, Y; Ishikawa, M; Ishikawa, T; Kajiwara, T; Katsube, T; Mori, H; Ogawa, K; Ohkawa, S; Omata, M; Otsuka, H; Saitoh, T; Takahashi, H; Tamai, M1
Gründemann, D; Haag, C; Honold, C; Koschker, AC; Schömig, E; Zimmermann, T1
Desmecht, D; Jolly, S1
Bischoff, AM; Büsselberg, D; Dutschmann, M; Richter, DW1
Bacon, KB; Gantner, F; Sakai, K; Takeshita, K1
Gálfi, M; Juhász, A; László, F; László, FA; Molnár, A; Radács, M; Varga, C1
Anichtchik, OV; Kaslin, J; Panula, P; Peitsaro, N; Sundvik, M1
Alò, R; Canonaco, M; Crudo, M; Facciolo, RM; Giusi, G1
Brus, R; Jochem, J; Josko, J; Kostrzewa, RM; Noras, L; Nowak, P; Zwirska-Korczala, K1
Hirasawa, N; Hong, J; Ishihara, K; Katoh, G; Ohsawa, Y; Ohuchi, K; Seyama, T; Shibata, K; Tamura, S1
Drevensek, G; Ziberna, L; Zorman, T1
Giardini, JL; Heyland, A; Leguia, M; Nguyen, J; Sutherby, J; Wessel, G1
Barbaro, KC; Basílio, ABC; Boia-Ferreira, M; Chaim, OM; da Silva, LP; Donatti, L; Gremski, LH; Moreno, KG; Senff-Ribeiro, A; Soley, B; Veiga, SS; Vuitika, L; Wille, ACM1

Reviews

1 review(s) available for cimetidine and thioperamide

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

51 other study(ies) available for cimetidine and thioperamide

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Comparative chemometric modeling of cytochrome 3A4 inhibitory activity of structurally diverse compounds using stepwise MLR, FA-MLR, PLS, GFA, G/PLS and ANN techniques.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:7

    Topics: Algorithms; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Enzyme Inhibitors; Factor Analysis, Statistical; Least-Squares Analysis; Linear Models; Models, Molecular; Neural Networks, Computer; Quantitative Structure-Activity Relationship; Reproducibility of Results

2009
An in vivo and in vitro study of the vestibular nuclei histaminergic receptors in the guinea pig.
    Annals of the New York Academy of Sciences, 1992, May-22, Volume: 656

    Topics: Animals; Brain Stem; Cimetidine; Electric Stimulation; Eye Movements; Guanidines; Guinea Pigs; Head; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Piperidines; Receptors, Histamine; Receptors, Histamine H2; Reflex, Vestibulo-Ocular; Rotation; Vestibular Nuclei

1992
The influence of H1-, H2- and H3-receptors on the spontaneous and ConA induced histamine release from human adenoidal mast cells.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenoids; Cimetidine; Concanavalin A; Guanidines; Histamine Antagonists; Humans; Hydroxyzine; Imidazoles; Impromidine; Mast Cells; Meclizine; Methylhistamines; Piperidines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3

1991
Histamine H3 receptors modulate antigen-induced bronchoconstriction in guinea pigs.
    The Journal of allergy and clinical immunology, 1990, Volume: 86, Issue:4 Pt 1

    Topics: Animals; Antigens; Bronchoconstriction; Cimetidine; Dose-Response Relationship, Drug; Dose-Response Relationship, Immunologic; Guinea Pigs; Histamine; Immunization; Male; Ovalbumin; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Skin Tests

1990
Pharmacological studies of allergic cough in the guinea pig.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Administration, Oral; Aerosols; Albuterol; Analysis of Variance; Animals; Antitussive Agents; Capsaicin; Chlorpheniramine; Cimetidine; Codeine; Cough; Drug Hypersensitivity; Guinea Pigs; Hexamethonium; Histamine Antagonists; Indomethacin; Injections, Subcutaneous; Ipratropium; Loratadine; Male; Ovalbumin; Piperidines; Receptors, Histamine H1; Receptors, Histamine H2

1995
Role of histamine receptors in intestinal repair after ischemia-reperfusion in rats.
    Gastroenterology, 1994, Volume: 107, Issue:5

    Topics: Animals; Biological Transport; Chlorpheniramine; Cimetidine; Dietary Fats; Histamine Antagonists; Histamine Release; Intestinal Mucosa; Intestines; Lymph; Male; Ornithine Decarboxylase; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Reperfusion Injury

1994
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:2

    Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1994
R-alpha-methylhistamine-induced inhibition of gastric acid secretion in pylorus-ligated rats via central histamine H3 receptors.
    British journal of pharmacology, 1995, Volume: 115, Issue:7

    Topics: Animals; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; Injections, Intraventricular; Methylhistamines; Piperidines; Pylorus; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1995
Dimaprit, a histamine H2-agonist, inhibits anaphylactic histamine release from mast cells and the decreased release is restored by thioperamide (H3-antagonist), but not by cimetidine (H2-antagonist).
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:1

    Topics: Anaphylaxis; Animals; Anticonvulsants; Betahistine; Cimetidine; Dimaprit; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Indicators and Reagents; Male; Mast Cells; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Pharmacological characterization of the inhibitory effect of (R)-alpha-methylhistamine on sympathetic cardiopressor responses in the pithed guinea-pig.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:6

    Topics: Adrenalectomy; Animals; Blood Pressure; Chlorpheniramine; Cimetidine; Drug Interactions; Electric Stimulation; Epinephrine; Guinea Pigs; Heart; Heart Rate; Histamine Agonists; Male; Methylhistamines; Piperidines; Prazosin; Spinal Cord; Sympathetic Nervous System; Vagotomy; Yohimbine

1994
Species differences in the cardiovascular responses to histamine H3 receptor activation.
    European journal of pharmacology, 1994, Jul-01, Volume: 259, Issue:2

    Topics: Animals; Blood Pressure; Cimetidine; Guinea Pigs; Heart Rate; Hemodynamics; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Piperidines; Rabbits; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Receptors, Histamine H3; Species Specificity

1994
Mechanisms of antihistamine-induced sedation in the human brain: H1 receptor activation reduces a background leakage potassium current.
    Neuroscience, 1994, Volume: 59, Issue:3

    Topics: Cerebral Cortex; Cimetidine; Evoked Potentials; Histamine; Histamine Antagonists; Humans; Hypnotics and Sedatives; Membrane Potentials; Neurons; Piperidines; Potassium Channels; Pyrilamine; Receptors, Histamine H1

1994
Histamine H3 receptor activation inhibits sympathetic-cholinergic responses in cats.
    European journal of pharmacology, 1994, May-12, Volume: 257, Issue:1-2

    Topics: Animals; Cats; Chlorpheniramine; Cimetidine; Electric Stimulation; Female; Histamine Agonists; Male; Methacholine Chloride; Methylhistamines; Parasympathetic Nervous System; Piperidines; Receptors, Histamine H3; Skin; Sympathetic Nervous System

1994
Effect of histamine on memory retrieval in old rats.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:2

    Topics: Acetylcholine; Aging; Animals; Anticonvulsants; Avoidance Learning; Cerebrovascular Circulation; Cimetidine; Dose-Response Relationship, Drug; Exploratory Behavior; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Motor Activity; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Medial vestibular nucleus in the guinea-pig: histaminergic receptors. II. An in vivo study.
    Experimental brain research, 1993, Volume: 93, Issue:2

    Topics: Animals; Anticonvulsants; Cimetidine; Electroencephalography; Guinea Pigs; Impromidine; Injections, Intraperitoneal; Perfusion; Piperidines; Posture; Receptors, Histamine; Reflex, Vestibulo-Ocular; Vestibular Nuclei

1993
Cholinergic nucleus basalis neurons are excited by histamine in vitro.
    Neuroscience, 1995, Volume: 69, Issue:2

    Topics: Action Potentials; Animals; Cholinergic Fibers; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Neurons; Piperidines; Substantia Innominata

1995
Histaminergic control of mucosal repair in the small intestine.
    Obesity research, 1995, Volume: 3 Suppl 5

    Topics: Animals; Biological Transport; Chlorpheniramine; Cimetidine; Enzyme Inhibitors; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; Intestinal Mucosa; Ischemia; Lipid Metabolism; Lymph; Male; Methylhistidines; Piperidines; Rats; Rats, Sprague-Dawley; Reperfusion

1995
Effect of oxitropium bromide on histamine-induced airway goblet cell secretion.
    American journal of respiratory and critical care medicine, 1996, Volume: 154, Issue:1

    Topics: Administration, Inhalation; Aerosols; Animals; Atropine; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; Histocytochemistry; Injections, Intravenous; Male; Mucus; Muscarinic Antagonists; Piperidines; Pyrilamine; Receptors, Histamine; Scopolamine Derivatives; Trachea; Vagus Nerve

1996
Evidence for bidirectional histamine transport by murine hematopoietic progenitor cells.
    FEBS letters, 1996, Aug-12, Volume: 391, Issue:3

    Topics: Animals; Biological Transport; Calcium; Cell Line; Cetirizine; Cimetidine; Female; Hematopoietic Stem Cells; Histamine; Histamine Antagonists; Interleukin-3; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrimidinones; Sodium

1996
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:4

    Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P

1996
Reduction of the pressor response to nicotine in the guinea pigs by a histamine (H3) agonist is attenuated by an inhibitor of nitric oxide synthesis.
    Journal of cardiovascular pharmacology, 1996, Volume: 27, Issue:4

    Topics: Adrenalectomy; Animals; Arginine; Blood Pressure; Cimetidine; Guinea Pigs; Heart Rate; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; NG-Nitroarginine Methyl Ester; Nicotine; Nitric Oxide Synthase; Piperidines

1996
Histamine augments VCAM-1 expression on IL-4- and TNF-alpha-stimulated human umbilical vein endothelial cells.
    International archives of allergy and immunology, 1996, Volume: 111, Issue:2

    Topics: Amanitins; Antibodies, Blocking; Antigens, CD; Cell Adhesion; Cells, Cultured; Cimetidine; Eosinophils; Histamine; Histamine Antagonists; Humans; Immunohistochemistry; Integrin alpha4; Interleukin-4; Piperidines; Platelet Activating Factor; Pyrilamine; Tumor Necrosis Factor-alpha; Umbilical Veins; Vascular Cell Adhesion Molecule-1

1996
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
    Brain research bulletin, 1996, Volume: 41, Issue:4

    Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1996
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Effects of naltrexone and histamine antagonists on the antinociceptive activity of the cimetidine analog SKF92374 in rats.
    Brain research, 1997, Feb-14, Volume: 748, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Animals; Cimetidine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Naltrexone; Narcotic Antagonists; Nociceptors; Piperidines; Rats; Rats, Sprague-Dawley; Stereoisomerism

1997
Effect of histamine on intracellular Ca2+ concentration in guinea pig isolated vestibular hair cells.
    Acta oto-laryngologica. Supplementum, 1997, Volume: 528

    Topics: Afferent Pathways; Animals; Calcium; Cimetidine; Cytoplasm; Endolymphatic Sac; Extracellular Space; Fluorescent Dyes; Fura-2; Guinea Pigs; Hair Cells, Vestibular; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Mast Cells; Piperidines; Promethazine; Receptors, Cell Surface; Signal Transduction; Vestibular Nerve

1997
Comparison of responses to T-kinin and bradykinin in the mesenteric vascular bed of the cat.
    Peptides, 1997, Volume: 18, Issue:9

    Topics: Adamantane; Analysis of Variance; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cats; Cimetidine; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Female; Histamine Antagonists; Male; Meclofenamic Acid; Mesentery; Morpholines; NG-Nitroarginine Methyl Ester; Piperidines; Potassium Channels; Pyrilamine

1997
The vascular mechanism of action of betahistine in the inner ear of the guinea pig.
    European archives of oto-rhino-laryngology : official journal of the European Federation of Oto-Rhino-Laryngological Societies (EUFOS) : affiliated with the German Society for Oto-Rhino-Laryngology - Head and Neck Surgery, 1998, Volume: 255, Issue:3

    Topics: Animals; Betahistine; Cimetidine; Cochlea; Ear, Inner; Female; Guinea Pigs; Histamine Antagonists; Idazoxan; Male; Methylhistamines; Piperidines; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Vasodilator Agents

1998
Thioperamide, a histamine H3-receptor blocker, facilitates vasopressor response to footshocks.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cimetidine; Electric Stimulation; Enzyme Inhibitors; Heart Rate; Hindlimb; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistidines; Norepinephrine; Phentolamine; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Vasoconstrictor Agents

1998
Effect of histamine H2 and H3 receptor modulation in the septum on post-training memory processing.
    Psychopharmacology, 1998, Volume: 140, Issue:3

    Topics: Animals; Cimetidine; Dimaprit; Histamine Agonists; Histamine Antagonists; Imidazoles; Limbic System; Male; Memory; Mice; Piperidines; Thiourea

1998
Acetylcholine release from hippocampus of freely moving rats is modulated by thioperamide and cimetidine.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1999, Volume: 48 Suppl 1

    Topics: Acetylcholine; Animals; Cimetidine; Hippocampus; Histamine Antagonists; Histamine H2 Antagonists; Male; Piperidines; Rats; Rats, Wistar

1999
Histamine H3 receptor-mediated suppression of inhibitory synaptic transmission in the submucous plexus of guinea-pig small intestine.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Male; Methylhistamines; Norepinephrine; Phentolamine; Piperidines; Receptors, Histamine H3; Submucous Plexus; Synaptic Transmission

2000
Thioperamide and cimetidine modulate acetylcholine release from the amygdala of freely moving rats.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2000, Volume: 49 Suppl 1

    Topics: Acetylcholine; Amygdala; Animals; Cimetidine; Histamine Antagonists; Histamine H2 Antagonists; Male; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3

2000
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish

2000
Effects of drugs acting as histamine releasers or histamine receptor blockers on an experimental anxiety model in mice.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:1

    Topics: Animals; Anxiety; Cimetidine; Disease Models, Animal; Histamine Antagonists; Histamine Release; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; p-Methoxy-N-methylphenethylamine; Piperidines; Pyrilamine

2000
Enhancement by histamine of vascular endothelial growth factor production in granulation tissue via H(2) receptors.
    British journal of pharmacology, 2001, Volume: 134, Issue:7

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cells, Cultured; Cimetidine; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Endothelial Growth Factors; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Granulation Tissue; Histamine; Histamine Antagonists; Immunohistochemistry; Indoles; Indomethacin; Inflammation; Isoquinolines; Lymphokines; Macrophages, Peritoneal; Male; Maleimides; Naphthalenes; Neovascularization, Pathologic; Piperidines; Protein Kinase C; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; RNA, Messenger; Specific Pathogen-Free Organisms; Sulfonamides; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2001
Effects of N-alpha-methyl-histamine on human H(2) receptors expressed in CHO cells.
    Gut, 2002, Volume: 50, Issue:6

    Topics: Animals; CHO Cells; Cimetidine; Cricetinae; Cyclic AMP; Famotidine; Female; Histamine Agonists; Histamine Antagonists; Histamine H2 Antagonists; Methylhistamines; Ovary; Piperidines; Receptors, Histamine H2; Receptors, Histamine H3

2002
Activation of the extraneuronal monoamine transporter (EMT) from rat expressed in 293 cells.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Biological Transport; Cell Line; Cimetidine; Cloning, Molecular; Corticosterone; Dose-Response Relationship, Drug; Gene Expression; Genetic Vectors; Humans; Imidazoles; Kinetics; Mice; Norepinephrine; Organic Cation Transport Proteins; Papaverine; Piperidines; Quinolines; Rats; Thiourea; Transfection; Tritium

2002
Functional identification of epithelial and smooth muscle histamine-dependent relaxing mechanisms in the bovine trachea, but not in bronchi.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2003, Volume: 134, Issue:1

    Topics: Animals; Bronchi; Cattle; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine H2 Antagonists; Muscle Relaxation; Muscle, Smooth; Piperidines; Receptors, Histamine H2; Receptors, Histamine H3; Respiratory Mucosa; Trachea

2003
Histaminergic modulation of the intact respiratory network of adult mice.
    Pflugers Archiv : European journal of physiology, 2003, Volume: 445, Issue:5

    Topics: Animals; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypoxia; Medulla Oblongata; Mice; Mice, Inbred C57BL; Nerve Net; Neurons; Phrenic Nerve; Piperidines; Pons; Pyrilamine; Receptors, Histamine H3; Respiratory System

2003
Critical role of histamine H4 receptor in leukotriene B4 production and mast cell-dependent neutrophil recruitment induced by zymosan in vivo.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:3

    Topics: Animals; Bone Marrow Cells; Carrageenan; Cimetidine; Cytokines; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Leukotriene B4; Mast Cells; Mice; Mice, Inbred BALB C; Neutrophil Infiltration; Piperidines; Pleurisy; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Zymosan

2003
Histamine-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue cultures.
    Regulatory peptides, 2006, May-15, Volume: 134, Issue:2-3

    Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Kinetics; Male; Oxytocin; Piperidines; Pituitary Gland, Posterior; Pyrilamine; Rats; Tissue Culture Techniques; Vasopressins

2006
Identification of zebrafish histamine H1, H2 and H3 receptors and effects of histaminergic ligands on behavior.
    Biochemical pharmacology, 2007, Apr-15, Volume: 73, Issue:8

    Topics: Animals; Behavior, Animal; Cimetidine; Histamine Agonists; Histamine Antagonists; Imidazoles; Piperidines; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Zebrafish

2007
Specific cerebral heat shock proteins and histamine receptor cross-talking mechanisms promote distinct lead-dependent neurotoxic responses in teleosts.
    Toxicology and applied pharmacology, 2008, Mar-01, Volume: 227, Issue:2

    Topics: Amino Acid Sequence; Animals; Behavior, Animal; Brain; Brain Chemistry; Cimetidine; Fishes; Fluoresceins; Fluorescent Dyes; Heat-Shock Proteins; Histamine H2 Antagonists; Histamine H3 Antagonists; HSP70 Heat-Shock Proteins; HSP90 Heat-Shock Proteins; In Situ Hybridization; Injections, Intraperitoneal; Lead Poisoning, Nervous System; Molecular Sequence Data; Organic Chemicals; Piperidines; Receptor Cross-Talk; Receptors, Histamine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2008
Ontogenetic noradrenergic lesion alters histaminergic activity in adult rats.
    Neurotoxicity research, 2008, Volume: 13, Issue:2

    Topics: Age Factors; Animals; Animals, Newborn; Benzylamines; Brain; Chlorpheniramine; Cimetidine; Exploratory Behavior; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine H3 Antagonists; Male; Motor Activity; Norepinephrine; Piperidines; Rats; Rats, Wistar; Sympathomimetics

2008
Modification of the picryl chloride-induced allergic dermatitis model in mouse ear lobes by 12-O-tetradecanoylphorbol 13-acetate, and analysis of the role of histamine in the modified model.
    International archives of allergy and immunology, 2009, Volume: 148, Issue:4

    Topics: Animals; Cell Count; Cimetidine; Cyclophosphamide; Cyclosporine; Cytokines; Dermatitis, Allergic Contact; Disease Models, Animal; Ear Auricle; Eosinophil Peroxidase; Eosinophils; Gene Expression; Histamine; Histamine Antagonists; Immunoglobulin E; Interferon-gamma; Interleukin-4; Male; Mast Cells; Mice; Mice, Inbred BALB C; Picryl Chloride; Piperidines; Pyrilamine; Tetradecanoylphorbol Acetate; Thymic Stromal Lymphopoietin

2009
Characterization of histamine-induced relaxation in pre-contracted rat aorta.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2009, Volume: 58 Suppl 1

    Topics: Animals; Aorta; Cimetidine; Ethylenediamines; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine H3 Antagonists; Male; Muscle Relaxation; Piperidines; Protein Isoforms; Rats; Rats, Wistar; Receptors, Histamine

2009
Histamine is a modulator of metamorphic competence in Strongylocentrotus purpuratus (Echinodermata: Echinoidea).
    BMC developmental biology, 2012, Apr-27, Volume: 12

    Topics: Animals; Apoptosis; Chlorpheniramine; Cimetidine; Ectoderm; Gene Expression Regulation, Developmental; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine H3 Antagonists; Histidine Decarboxylase; Larva; Metamorphosis, Biological; Methylhistidines; Organ Specificity; Piperidines; Receptors, Histamine H1; Strongylocentrotus purpuratus

2012
TCTP from
    Cells, 2019, 11-22, Volume: 8, Issue:12

    Topics: Animals; Biomarkers, Tumor; Cimetidine; Cromolyn Sodium; Dose-Response Relationship, Drug; Hypersensitivity; Inflammation; Injections, Intraperitoneal; Injections, Intravenous; Mast Cells; Mice; Phosphoric Diester Hydrolases; Piperidines; Promethazine; Rabbits; Rats; Skin Diseases; Spider Venoms; Tumor Cells, Cultured; Tumor Protein, Translationally-Controlled 1

2019