cimetidine has been researched along with thiazoles in 165 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 128 (77.58) | 18.7374 |
1990's | 27 (16.36) | 18.2507 |
2000's | 5 (3.03) | 29.6817 |
2010's | 5 (3.03) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Buck, SH; Gilman, DJ; Jones, DF; Wardleworth, JM; Yellin, TO | 1 |
Bertaccini, G; Coruzzi, G; Musso, E | 1 |
Bertaccini, G; Impicciatore, M; Morini, G | 1 |
Hough, LB; Nalwalk, JW | 1 |
Ianelli, S; Pelizzi, G | 1 |
Chia, SC; Chong, YY; Fock, KM; Yap, CK | 1 |
Nowak, JZ; Sek, B | 1 |
Hoshino, R; Kagoshima, M; Shimada, H | 1 |
Goddard, CJ; Hakkinen, JP; Holt, WF; Maciejko, JJ; Murphy, WR; Oates, PJ; Reiter, LA | 1 |
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P | 1 |
Bruno, M; Grassi, A; Ippen, J; Thomas, G | 1 |
Best, KL; Goode, RL; Hirsch, KS; Lin, TM; Neubauer, BL; Pioch, RP; Probst, KS; Shaar, CJ; Tinsley, FC | 1 |
Fagan, TC; Fennerty, B; Lipsy, RJ | 1 |
Madrid, JA; Pariente, JA; Salido, GM | 2 |
Frank, N; Frei, E; Kato, T; Ohgaki, H; Sato, S; Tsuda, M | 1 |
Arrang, JM; Garbarg, M; Schwartz, JC | 1 |
Edvinsson, L; Jansen, I; Ottosson, A | 1 |
Eberle, NB; Glick, SD; Gogas, KR; Hough, LB; Lyon, RA; Parsons, ME; Ward, SJ; Young, RC | 1 |
Hirsch, E | 1 |
Amoruso, A; Barone, M; Di Leo, A; Francavilla, A; Ingrosso, M; Makowka, L; Panella, C; Polimeno, L; Starzl, TE | 1 |
Fujimoto, K; Fukagawa, K; Ookuma, K; Sakata, T; Shiraishi, T; Wada, H; Yoshimatsu, H | 1 |
Chremos, AN; Lin, ET; Sambol, NC; Upton, RA; Williams, RL | 1 |
Levine, JB | 1 |
De Natale, F; De Natale, G; Marino, A | 1 |
Cherner, JA; Cloud, ML; Latz, JE; Offen, WW | 1 |
Bast, A; Smid, K; Timmerman, H | 1 |
Rovers, JP; Souney, PF | 1 |
Dammann, HG; Dreyer, M; Gottlieb, WR; Müller, P; Simon, B; Wolf, N | 1 |
Alvarez, A; Barrio, E; Conchillo, F; Dieguez, P; Forné, M; Muñoz, M; Panés, J; Rodrigo, L; Viver, J; Zozaya, JM | 1 |
Bode, JC; Klotz, U; Krishna, DR; Walker, S | 1 |
Calogero, A; Cramarossa, L; Famularo, G; Filingeri, V; Giacomelli, R; Iacona, A; Nardi, S; Rosati, R; Sacchetti, S; Stortoni, F | 1 |
Chapman, JM; Kosh, JW; Sowell, JW | 1 |
Gardner, JD; Jensen, RT; Maton, PN | 1 |
Galbraith, RA; Jellinck, PH | 1 |
Hajos, ZG; Press, JB; Sanfilippo, PJ; Scott, CK; Shriver, DA; Urbanski, M | 1 |
Cherner, JA; Chremos, AN; Ciarleglio, CA; Collen, MJ; Cornelius, MJ; Gardner, JD; Howard, JM; Jensen, RT; Maton, PN; McArthur, KE | 1 |
Chremos, AN; Gamal, MA; Graham, DY; Smith, JL | 1 |
Cook, PG; Mangel, AW; Pendleton, RG; Shepherd-Rose, A | 1 |
Chremos, AN; Huber, PB; Kuljian, B; McCallum, RW; Tupy-Visich, MA | 1 |
Arvela, P; Klotz, U; Rosenkranz, B | 1 |
Smith, JL | 1 |
Bianchi Porro, G | 1 |
Kuroiwa, Y; Misawa, S; Tanaka, E | 1 |
Greenblatt, DJ; Harmatz, JS; Locniskar, A; Shader, RI; Zinny, MA | 1 |
Aono, M; Mizuta, K; Moriga, M; Narusawa, H | 1 |
Imai, Y; Inada, M; Kawata, S; Minami, Y; Noda, S; Tamura, S; Tarui, S | 1 |
Nielsen, ST | 2 |
Evans, DC; Lin, TM; Pioch, RP; Warrick, MW | 1 |
Gardner, JD; Howard, JM; Jensen, RT; Maton, PN; Slaff, JI; Vinayek, R; Wank, SA | 1 |
Knigge, U; Matzen, S; Warberg, J | 1 |
Arvela, P; Klotz, U; Pasanen, M; Pelkonen, O; Sotaniemi, E | 1 |
Dammann, HG; Dreyer, M; Gottlieb, WR; Keohane, P; Müller, P; Simon, B; Walter, TA | 1 |
Hashimoto, Y; Iwatsuki, N; Koga, Y | 1 |
Mahachai, V; Thomson, AB | 1 |
Gardner, JD; Howard, JM; Jensen, RT; Maton, PN; Vinayek, R; Wank, SA | 1 |
Hagiwara, T; Namiki, A; Omote, K; Sumita, S; Takahashi, T; Ujike, Y | 1 |
Humphries, TJ | 1 |
Baba, S; Daikuhara, Y; Gohda, E; Hirono, S; Miyazaki, H; Nakayama, H; Sakiyama, O; Takahashi, K; Tamada, F; Tsubouchi, H | 1 |
Freston, JW | 1 |
Bertaccini, G; Coruzzi, G; Poli, E | 1 |
Gavaler, JS; Heyl, A; Susen, B; Van Thiel, DH | 1 |
Hammond, JB; Offen, WW | 1 |
Chiou, R; Chremos, AN; Lin, JH; Williams, R; Yeh, KC | 1 |
Heim, J; Kaufmann, D; Krammisch, H; Mappes, A; Merki, HS; Neumann, J; Roehmel, J; Scheurle, E; Walt, RP; Witzel, L | 1 |
Akamatsu, K; Hirabayashi, Y; Kanaoka, M; Masumoto, S; Nakanishi, K; Nishinobu, M; Ohta, Y; Okada, S; Sakaue, H; Sasaki, T | 1 |
Calcutt, CR; Ganellin, CR; Griffiths, R; Leigh, BK; Maguire, JP; Mitchell, RC; Mylek, ME; Parsons, ME; Smith, IR; Young, RC | 1 |
Matsumoto, C; McMahon, FG; Offen, WW; Regel, G; Ryan, J; Vargas, R | 1 |
Dicke, JM; Henderson, GI; Johnson, RF; Kuehl, TJ; Schenker, S | 1 |
Amplatz, S; Comberlato, M; de Pretis, G; Dobrilla, G | 1 |
Brambilla, A; De Paoli, AM; Ghiorzi, A; Giachetti, A | 1 |
Berardi, RR; Nostrant, TT; Tankanow, RM | 1 |
Kuroiwa, Y; Misawa, S; Nakamura, K; Tanaka, E | 1 |
Argenbright, LS; Lu, AY; Miwa, GT; Wang, RW | 1 |
Gillam, EM; Mason, SR; Reilly, PE | 1 |
Luskin, AT; Tomasko, MA | 1 |
Klotz, U; Kuhlmann, U; Machleidt, C; Mettang, T; Weber, J | 1 |
Berta, L; Crua, MR; Dusio, P; Fazzari, A; Fortunati, N; Frairia, R; Gaidano, G | 1 |
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I | 1 |
Nakamura, K; Tanaka, E | 1 |
Astengo, M; Basso, C; Bennicelli, C; Camoirano, A; De Flora, S; Zanacchi, P | 1 |
Forsyth, DR; Jayasinghe, KS; Roberts, CJ | 1 |
Brockmeier, D; Lameire, N; Rosenkranz, B | 1 |
Ciarleglio, CA; Collen, MJ; Stanczak, VJ | 1 |
Al-Gadi, M; Hill, SJ | 1 |
Fölsch, UR; Hartmann, H | 1 |
Ahmed, W; Qureshi, H; Zuberi, SJ | 1 |
Baronti, A; Di Carlo, S; Verdiani, P | 1 |
Bellini, M; Cipparrone, G; Costa, F; Greco, A; Maltinti, G; Marchi, S; Polloni, A | 1 |
Imai, Y; Inada, M; Kawata, S; Minami, Y; Tamura, S; Tarui, S | 1 |
Lewis, JH | 1 |
Dammann, HG; Mueller, P; Simon, B; Walter, TA | 1 |
Jantos, H; Monti, JM; Pellejero, T | 1 |
Burget, DW; Howden, CW; Hunt, RH; Jones, DB | 1 |
Hazama, H; Murase, T; Okuno, H; Sameshima, Y; Shiozaki, Y | 1 |
Fukuda, S; Hotta, T; Itoh, H; Kawasaki, T; Komatsu, K; Kuwayama, H; Matsuo, Y; Ohsaka, Y; Seki, A | 1 |
Coombes, JD; Norris, DB; Rising, TJ; Ross, BC; Steward, A | 2 |
Dammann, HG; Müller, P; Simon, B; Walter, TA | 1 |
Levi, R; Trzeciakowski, JP | 1 |
Brater, C; Feldman, M; Richardson, CT; Welborn, J | 1 |
Brater, DC; Feldman, M; Kaojarern, S; Richardson, CT | 1 |
Domschke, S; Domschke, W | 1 |
Vohra, MM | 1 |
Douglas, AP; Strecker, RB; Valenzuela, JE | 1 |
Cheret, AM; Lewin, MJ; Pignal, F | 1 |
Avant, GR; Mitchell, MC; Patwardhan, RV; Schenker, S; Speeg, KV | 1 |
Bertaccini, G; Coruzzi, G | 1 |
Barker, LA | 1 |
Maeno, H; Takagi, T; Takeda, M | 2 |
Batzri, S; Dyer, J; Harmon, JW; Thompson, WF | 1 |
Maeno, H; Takagi, T; Takeda, M; Yashima, Y | 1 |
Buyniski, JP; Cavanagh, RL; Usakewicz, JJ | 1 |
Dinoso, VP | 1 |
Baldwin, JJ; Bolhofer, WA; Cragoe, EJ; Habecker, CN; Hoffman, JM; Lumma, WC; Phillips, BT; Pietruszkiewicz, AM; Torchiana, ML | 1 |
Radbil', OS; Sukherova, MI | 1 |
Flannery, MC; Johnston, BJ; McIsaac, RL | 1 |
Harada, M; Maeno, H; Terai, M | 1 |
Ishihara, Y; Okabe, S | 1 |
Dammann, HG; Müller, P; Simon, B | 1 |
Brittain, RT; Jack, D | 1 |
Chung, C; Clineschmidt, BV; Cook, P; Pendleton, RG; Torchiana, ML; Wiese, S | 1 |
Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
Hösli, E; Hösli, L; Schneider, U; Wiget, W | 1 |
Miwa, T; Tani, N; Watanabe, K; Watanabe, T; Watanabe, Y | 1 |
Dammann, HG; DeVries, JX; Koroknay, B; Müller, P; Simon, B; Staiger, C; Weber, E | 1 |
Yellin, TO; Zavecz, JH | 1 |
Lewis, S; Rising, TJ | 1 |
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G | 1 |
Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC | 1 |
Daly, MJ; Humphray, JM; Stables, R | 1 |
Miwa, M; Miwa, T; Tani, N | 1 |
Bartsch, H; Cassale, V; Crespi, M; Forichon, J; Lambert, R; Minaire, Y; Muñoz, N; Ohshima, H; Ramazotti, V; Walters, CL | 1 |
Fujiwara, T; Kohchi, M; Matsumoto, H; Miyoshi, A; Nakamura, M; Ohe, K | 1 |
Mori, H | 1 |
Dammann, HG; Devries, JX; Korodnay, B; Müller, P; Simon, B; Staiger, C; Weber, E | 1 |
Gómez, F; Ortíz, JA; Romero, A; Sacristán, A; Villamayor, F | 1 |
Wong, CL | 1 |
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
Akaike, N; Munakata, M | 1 |
Fujihara, A; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H | 1 |
Kweon, DS; Lee, MH; Shim, CK | 1 |
Alemany, G; López-García, JA; Nicolau, MC; Planas, B; Ramis, C; Rial, R | 1 |
Borda, ES; Goren, N; Leiros, CP; Sterin-Borda, L | 1 |
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J | 1 |
Busch, U; Heinzel, G; Narjes, H; Nehmiz, G | 1 |
Agut, J; Ortiz, JA; Sacristán, A; Sánchez, JC | 1 |
Conejo, L; Ortiz, JA; Palop, D; Romero, A; Sacristán, A; Villamayor, F | 1 |
Ballesta, A; Gómez, F; Ortiz, JA; Romero, A; Sacristán, A; Villamayor, F | 1 |
Agúndez, JA; Albet, C; Benítez, J; Carrillo, JA; Herrero, E; Márquez, M; Martínez, C; Ortiz, JA | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E | 1 |
Folger, CJ; Geoffroy, P; Hansen, RA; Wilner, KD | 1 |
Bateman, R; Eckers, C; Giles, K; Sage, AB; Wolff, JC | 1 |
Durán, N; Haun, M; Melo, PS | 1 |
Hough, LB; Lu, Q; Montero, MJ; Nalwalk, JW; Shan, Z; Svokos, K; Wentland, MP | 1 |
Schipper, HG; Simsek, S; van Agtmael, MA; van Lienden, KP | 1 |
Abe, T; Maruyama, S; Nonomura, K; Sato, S; Sazawa, A; Shindo, J; Shinohara, N; Suzuki, S | 1 |
Dartt, DA; Hayashi, C; Hayashi, D; Hodges, RR; Li, D; Shatos, M | 1 |
Kang, JH; Kim, HJ; Kim, HM; Kim, YL; Lee, AY; Lee, CH; Lee, EJ; Lee, HJ; Park, MK | 1 |
Bastide, C; Bruyere, F; Caremel, R; Castel-Lacanal, E; Cornu, JN; Guy, L; Karsenty, G; Kerdraon, J | 1 |
Bannister, R; Birkus, G; Cihlar, T; Hao, J; Huang, J; Huang, Y; Kosaka, A; Lepist, EI; Murray, BP; Ray, AS; Zhang, X | 1 |
13 review(s) available for cimetidine and thiazoles
Article | Year |
---|---|
Clinical review of histamine2 receptor antagonists.
Topics: Cimetidine; Drug Interactions; Duodenal Ulcer; Famotidine; Histamine H2 Antagonists; Humans; Nizatidine; Ranitidine; Stomach Ulcer; Thiazoles | 1990 |
[Drugs used in the therapy of peptic ulcer with special reference to H2 receptor blockaders].
Topics: Antacids; Anti-Ulcer Agents; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Omeprazole; Peptic Ulcer; Pirenzepine; Ranitidine; Thiazoles | 1989 |
A critical review of continuous infusion H2 receptor therapy.
Topics: Cimetidine; Famotidine; Gastric Juice; Histamine H2 Antagonists; Humans; Hydrogen-Ion Concentration; Infusion Pumps; Infusions, Parenteral; Intensive Care Units; Ranitidine; Thiazoles | 1989 |
Recent advances in the management of gastric acid hypersecretion in patients with Zollinger-Ellison syndrome.
Topics: Cimetidine; Famotidine; Gastric Acid; Histamine H2 Antagonists; Humans; Nizatidine; Omeprazole; Parasympatholytics; Ranitidine; Thiazoles; Zollinger-Ellison Syndrome | 1989 |
Pharmacological management of patients with peptic ulcer disease: prospects for the late 1980's.
Topics: Alprostadil; Antacids; Anti-Ulcer Agents; Cimetidine; Drug Resistance; Enprostil; Famotidine; Histamine H2 Antagonists; Humans; Misoprostol; Omeprazole; Peptic Ulcer; Pirenzepine; Prostaglandins; Prostaglandins E, Synthetic; Ranitidine; Sucralfate; Thiazoles | 1987 |
Famotidine: a notable lack of drug interactions.
Topics: Animals; Cimetidine; Cytochrome P-450 Enzyme System; Drug Interactions; Famotidine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Oxidation-Reduction; Ranitidine; Thiazoles | 1987 |
H2-antagonists and motility of the upper gastrointestinal tract in man.
Topics: Cimetidine; Clinical Trials as Topic; Esophagus; Famotidine; Gastrointestinal Motility; Histamine H2 Antagonists; Humans; Peristalsis; Ranitidine; Thiazoles | 1988 |
Comparison of famotidine with cimetidine and ranitidine.
Topics: Cimetidine; Famotidine; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles | 1988 |
Pharmacokinetics of histamine (H2)-receptor antagonists, including roxatidine, in chronic renal failure.
Topics: Anti-Ulcer Agents; Cimetidine; Famotidine; Histamine H2 Antagonists; Humans; Kidney Failure, Chronic; Piperidines; Ranitidine; Renal Dialysis; Thiazoles | 1988 |
New histamine H2-receptor antagonists.
Topics: Animals; Anticoagulants; Chemical Phenomena; Chemistry; Cimetidine; Confusion; Dogs; Drug Interactions; Duodenal Ulcer; Furans; Gastric Juice; Gastric Mucosa; Guanidines; Gynecomastia; Histamine H2 Antagonists; Humans; Imidazoles; Male; Molecular Conformation; Ranitidine; Spermatozoa; Thiazoles | 1980 |
[New generation of histamine H2 receptor blockaders].
Topics: Animals; Anti-Ulcer Agents; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Imidazoles; Ranitidine; Thiazoles | 1982 |
Histamine H2-antagonists--past, present and future.
Topics: Animals; Aspirin; Burimamide; Chemical Phenomena; Chemistry; Cimetidine; Dogs; Furans; Gastric Acid; Guanidines; Guinea Pigs; Half-Life; Histamine H2 Antagonists; Humans; Imidazoles; Methylamines; Ranitidine; Rats; Stomach; Thiazoles; Triazoles | 1983 |
[Drug therapy of bladder dysfunction].
Topics: Acetanilides; Anti-Inflammatory Agents; Botulinum Toxins, Type A; Cholinergic Antagonists; Cimetidine; Cyclosporine; Dimethyl Sulfoxide; Histamine H2 Antagonists; Humans; Immunosuppressive Agents; Muscarinic Antagonists; Neuromuscular Agents; Phosphodiesterase Inhibitors; Thiazoles; Urinary Bladder; Urinary Bladder Diseases; Urination; Urodynamics | 2013 |
32 trial(s) available for cimetidine and thiazoles
Article | Year |
---|---|
Nizatidine versus cimetidine in the treatment of duodenal ulcers.
Topics: Adult; Aged; Cimetidine; Duodenal Ulcer; Endoscopy, Gastrointestinal; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Nizatidine; Thiazoles; Wound Healing | 1991 |
A comparison of the influence of famotidine and cimetidine on phenytoin elimination and hepatic blood flow.
Topics: Cimetidine; Cytochrome P-450 Enzyme System; Drug Evaluation; Famotidine; Female; Histamine H2 Antagonists; Humans; Indocyanine Green; Liver Circulation; Male; Phenytoin; Random Allocation; Thiazoles | 1989 |
Comparison of nizatidine and cimetidine as once-nightly treatment of acute duodenal ulcer. Nizatidine Multicenter Duodenal Ulcer Study Group.
Topics: Acute Disease; Adult; Aged; Aged, 80 and over; Alcohol Drinking; Cimetidine; Creatinine; Double-Blind Method; Drug Administration Schedule; Duodenal Ulcer; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Multicenter Studies as Topic; Nizatidine; Patient Compliance; Random Allocation; Smoking; Thiazoles | 1989 |
[Inhibition of 24-hour acidity by nizatidine].
Topics: Cimetidine; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Famotidine; Gastric Acid; Gastric Acidity Determination; Histamine H2 Antagonists; Humans; Nizatidine; Random Allocation; Ranitidine; Thiazoles | 1989 |
A multicenter, randomized, double-blind study comparing famotidine with cimetidine in the treatment of active duodenal ulcer disease.
Topics: Adult; Cimetidine; Double-Blind Method; Drug Administration Schedule; Duodenal Ulcer; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Multicenter Studies as Topic; Random Allocation; Thiazoles | 1989 |
MK-208, a novel histamine H2-receptor inhibitor with prolonged antisecretory effect.
Topics: Adult; Cimetidine; Famotidine; Gastric Acid; Gastric Juice; Gastric Mucosa; Histamine H2 Antagonists; Humans; Hydrogen-Ion Concentration; Middle Aged; Pentagastrin; Thiazoles | 1985 |
Famotidine, a new H2-receptor antagonist, does not affect hepatic elimination of diazepam or tubular secretion of procainamide.
Topics: Adult; Cimetidine; Diazepam; Famotidine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Kidney Tubules; Kinetics; Liver; Male; Microsomes, Liver; Middle Aged; Procainamide; Random Allocation; Thiazoles | 1985 |
Famotidine in the treatment of gastric and duodenal ulceration: overview of clinical experience.
Topics: Acute Disease; Chronic Disease; Cimetidine; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Duodenal Ulcer; Endoscopy; Famotidine; Gefarnate; Histamine H2 Antagonists; Humans; Ranitidine; Stomach Ulcer; Thiazoles; Time Factors | 1985 |
Famotidine in the therapy of gastric hypersecretory states.
Topics: Adult; Aged; Cimetidine; Clinical Trials as Topic; Drug Therapy, Combination; Famotidine; Female; Gastric Acid; Histamine H2 Antagonists; Humans; Longitudinal Studies; Male; Middle Aged; Parasympatholytics; Ranitidine; Thiazoles; Zollinger-Ellison Syndrome | 1986 |
Nocturnal acid suppression with a new H2 receptor antagonist--nizatidine.
Topics: Adult; Cimetidine; Drug Evaluation; Gastric Acid; Gastric Acidity Determination; Histamine H2 Antagonists; Humans; Male; Nizatidine; Random Allocation; Ranitidine; Thiazoles; Time Factors | 1986 |
Famotidine: effective treatment of Zollinger-Ellison syndrome.
Topics: Adult; Aged; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Gastric Acid; Histamine H2 Antagonists; Humans; Male; Middle Aged; Ranitidine; Thiazoles; Zollinger-Ellison Syndrome | 1987 |
H2-receptor antagonists and duodenal ulcer recurrence: analysis of efficacy and commentary on safety, costs, and patient selection.
Topics: Cimetidine; Clinical Trials as Topic; Costs and Cost Analysis; Duodenal Ulcer; Famotidine; Histamine H2 Antagonists; Humans; Ranitidine; Recurrence; Risk Factors; Thiazoles; Time Factors | 1987 |
An evaluation of the anti-androgen effects associated with H2 antagonist therapy.
Topics: Adolescent; Adult; Cimetidine; Histamine H2 Antagonists; Humans; Hypothalamo-Hypophyseal System; Male; Nizatidine; Pituitary Hormones, Anterior; Sperm Count; Testis; Testosterone; Thiazoles; Thyroxine | 1987 |
Effect of nizatidine and cimetidine on betazole-stimulated gastric secretion of normal subjects: comparison of effects on acid, water, and pepsin.
Topics: Adult; Aged; Betazole; Body Water; Cimetidine; Dose-Response Relationship, Drug; Double-Blind Method; Gastric Acid; Gastric Juice; Histamine H2 Antagonists; Humans; Hydrogen-Ion Concentration; Male; Middle Aged; Nizatidine; Pepsin A; Pyrazoles; Random Allocation; Thiazoles | 1988 |
Comparative effect of famotidine and cimetidine on the pharmacokinetics of theophylline in normal volunteers.
Topics: Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Injections, Intravenous; Male; Theophylline; Thiazoles | 1987 |
Double blind comparison of the effects of cimetidine, ranitidine, famotidine, and placebo on intragastric acidity in 30 normal volunteers.
Topics: Cimetidine; Double-Blind Method; Drug Evaluation; Famotidine; Female; Gastric Acid; Gastric Acidity Determination; Histamine H2 Antagonists; Humans; Male; Ranitidine; Thiazoles; Time Factors | 1988 |
Pharmacokinetics and pharmacodynamics of oral nizatidine.
Topics: Administration, Oral; Adult; Cimetidine; Dietary Proteins; Gastric Acid; Gastrins; Histamine H2 Antagonists; Humans; Hydrogen-Ion Concentration; Male; Nizatidine; Thiazoles; Time Factors | 1988 |
H2-antagonists and motility of the upper gastrointestinal tract in man.
Topics: Cimetidine; Clinical Trials as Topic; Esophagus; Famotidine; Gastrointestinal Motility; Histamine H2 Antagonists; Humans; Peristalsis; Ranitidine; Thiazoles | 1988 |
Effects of H2-receptor antagonists on ethanol metabolism in Japanese volunteers.
Topics: Acetaldehyde; Adult; Cimetidine; Ethanol; Famotidine; Histamine H2 Antagonists; Humans; Japan; Male; Ranitidine; Thiazoles | 1988 |
Do nizatidine and cimetidine interact with ibuprofen?
Topics: Adult; Cimetidine; Double-Blind Method; Drug Interactions; Half-Life; Histamine H2 Antagonists; Humans; Ibuprofen; Male; Nizatidine; Thiazoles | 1988 |
Famotidine versus cimetidine in the treatment of acute duodenal ulcer. Double-blind, randomized clinical trial comparing nocturnal administration of 40 mg famotidine to 800 mg cimetidine.
Topics: Acute Disease; Adult; Aged; Anti-Ulcer Agents; Cimetidine; Clinical Trials as Topic; Double-Blind Method; Duodenal Ulcer; Famotidine; Female; Humans; Male; Middle Aged; Pain; Random Allocation; Thiazoles | 1988 |
Famotidine effects on theophylline pharmacokinetics in subjects affected by COPD. Comparison with cimetidine and placebo.
Topics: Aged; Cimetidine; Famotidine; Female; Half-Life; Humans; Lung Diseases, Obstructive; Male; Metabolic Clearance Rate; Middle Aged; Theophylline; Thiazoles | 1988 |
Famotidine in the short-term treatment of duodenal ulcer and of concomitant peptic lesions: comparison with cimetidine.
Topics: Cimetidine; Duodenal Ulcer; Famotidine; Female; Humans; Male; Middle Aged; Peptic Ulcer; Thiazoles | 1988 |
Summary of the 30th meeting of the Food and Drug Administration Gastrointestinal Drugs Advisory Committee January 16-17, 1986.
Topics: Aluminum; Cimetidine; Clinical Trials as Topic; Duodenal Ulcer; Famotidine; Humans; Peptic Ulcer; Sucralfate; Thiazoles; United States; United States Food and Drug Administration | 1986 |
Effects of 800 mg cimetidine once daily on gastric acid secretion.
Topics: Administration, Oral; Cimetidine; Circadian Rhythm; Clinical Trials as Topic; Duodenal Ulcer; Famotidine; Gastric Acid; Humans; Ranitidine; Thiazoles | 1986 |
Tiotidine, a new long-acting histamine H2-receptor antagonist: comparison with cimetidine.
Topics: Adult; Cimetidine; Duodenal Ulcer; Gastric Acid; Gastric Emptying; Gastrins; Guanidines; Histamine H2 Antagonists; Humans; Middle Aged; Polyethylene Glycols; Thiazoles | 1981 |
Tiotidine, a new H2-receptor antagonist, is a potent inhibitor of nocturnal acid secretion in duodenal ulcer patients.
Topics: Adult; Cimetidine; Drug Evaluation; Duodenal Ulcer; Gastric Acid; Guanidines; Histamine H2 Antagonists; Humans; Middle Aged; Thiazoles | 1981 |
24 hour intragastric acidity and single night-time dose of three H-2-blockers.
Topics: Cimetidine; Clinical Trials as Topic; Double-Blind Method; Famotidine; Gastric Acidity Determination; Histamine H2 Antagonists; Humans; Random Allocation; Ranitidine; Thiazoles | 1983 |
[Comparative study of the effect of famotidine and cimetidine on antipyrine pharmacokinetics in the human].
Topics: Adult; Antipyrine; Cimetidine; Famotidine; Female; Histamine H1 Antagonists; Humans; Kinetics; Male; Thiazoles | 1984 |
Interaction of meloxicam with cimetidine, Maalox, or aspirin.
Topics: Administration, Oral; Adult; Aluminum Hydroxide; Antacids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Aspirin; Biological Availability; Chromatography, High Pressure Liquid; Cimetidine; Cross-Over Studies; Drug Combinations; Drug Interactions; Histamine H2 Antagonists; Humans; Magnesium Hydroxide; Male; Meloxicam; Middle Aged; Thiazines; Thiazoles | 1996 |
Comparative in vitro and in vivo inhibition of cytochrome P450 CYP1A2, CYP2D6, and CYP3A by H2-receptor antagonists.
Topics: Adult; Anti-Anxiety Agents; Antitussive Agents; Aryl Hydrocarbon Hydroxylases; Benzenesulfonates; Caffeine; Central Nervous System Stimulants; Cimetidine; Cytochrome P-450 CYP1A2 Inhibitors; Cytochrome P-450 CYP2D6 Inhibitors; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Dextromethorphan; Double-Blind Method; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Methylation; Microsomes, Liver; Midazolam; Oxidoreductases, N-Demethylating; Psychomotor Performance; Ranitidine; Thiazoles | 1999 |
The pharmacokinetics of ziprasidone in healthy volunteers treated with cimetidine or antacid.
Topics: Adult; Antacids; Anti-Ulcer Agents; Antipsychotic Agents; Area Under Curve; Cimetidine; Cross-Over Studies; Drug Interactions; Female; Half-Life; Humans; Male; Piperazines; Thiazoles | 2000 |
121 other study(ies) available for cimetidine and thiazoles
Article | Year |
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ICI 125,211: a new gastric antisecretory agent acting on histamine H2-receptors.
Topics: Animals; Cimetidine; Dogs; Female; Gastric Mucosa; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; Myocardial Contraction; Thiazoles; Thiourea; Time Factors | 1979 |
[Histamine receptors in the guinea pig papillary muscle].
Topics: Animals; Cimetidine; Epinephrine; Female; Guinea Pigs; Histamine; Male; Papillary Muscles; Pyrilamine; Receptors, Histamine; Thiazoles; Thiourea | 1977 |
The effects of stimulants and inhibitors of histamine receptors on acid secretion from guinea pig gastric fundus.
Topics: Animals; Cimetidine; Female; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Male; Methylhistamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Time Factors | 1978 |
Inhibition of morphine antinociception by centrally administered histamine H2 receptor antagonists.
Topics: Animals; Benzothiazoles; Brain; Cimetidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Morphine; Nociceptors; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles | 1992 |
Structural studies on H2-antagonists: crystal and molecular structure of N-cyano-N'-methyl-N"-(2-[(2-amino-5-thiazolyl)methylthio]ethyl) guanidine and N-cyano-3-[(2-guanidino-5-thiazolyl)methylthio]propionamidine.
Topics: Cimetidine; Crystallization; Famotidine; Guanidines; Histamine H2 Antagonists; Molecular Conformation; Thiazoles; X-Ray Diffraction | 1992 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
[Effects of NIK-228 on gastric acid secretion in rats using the congo red sprayed method].
Topics: Animals; Atropine; Benzothiazoles; Bethanechol; Bethanechol Compounds; Cimetidine; Congo Red; Deoxyglucose; Depression, Chemical; Gastric Acid; Imidazoles; Male; Rats; Rats, Inbred Strains; Staining and Labeling; Thiazoles; Vagus Nerve | 1991 |
CP-66,948: an antisecretory histamine H2-receptor antagonist with mucosal protective properties.
Topics: Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Ethanol; Gastric Acid; Gastric Mucosa; Gastrointestinal Hemorrhage; Guinea Pigs; Heart Rate; Histamine; Imidazoles; In Vitro Techniques; Indomethacin; Male; Pentagastrin; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Time Factors | 1991 |
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil | 1991 |
BAY P 1455, a thiazolylaminobenzimidazole derivative with gastroprotective properties in the rat.
Topics: Adrenalectomy; Animals; Anti-Ulcer Agents; Benzimidazoles; Cimetidine; Corticosterone; Cysteamine; Duodenal Ulcer; Ethanol; Female; Gastric Acid; Immersion; In Vitro Techniques; Indomethacin; Male; Pirenzepine; Prostaglandins E; Pylorus; Rats; Rats, Inbred Strains; Rioprostil; Stomach Ulcer; Stress, Psychological; Thiazoles | 1991 |
Endocrine effects of a new histamine H2-receptor antagonist, nizatidine (LY139037), in the male rat.
Topics: Androgens; Animals; Cimetidine; Gastric Acid; Histamine H2 Antagonists; Hypothalamus; Male; Metribolone; Molecular Structure; Nizatidine; Orchiectomy; Organ Size; Pituitary Gland; Preoptic Area; Prolactin; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen; Seminal Vesicles; Testis; Thiazoles | 1990 |
Role of histamine receptors in rabbit pancreatic exocrine secretion stimulated by cholecystokinin and secretin.
Topics: Animals; Chlorpheniramine; Cholecystokinin; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Secretin; Thiazoles; Thiourea | 1990 |
Detoxifying potential of thioproline against N-nitroso compounds, N-nitrosodimethylamine and N-nitrosocimetidine.
Topics: Animals; Cimetidine; Cytochrome P-450 CYP2E1; Dimethylnitrosamine; Formaldehyde; In Vitro Techniques; Inactivation, Metabolic; Male; Microsomes, Liver; Nitroso Compounds; Oxidoreductases, N-Demethylating; Rats; Rats, Inbred F344; Rats, Inbred Strains; Thiazoles; Thiazolidines | 1990 |
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
Topics: Animals; Burimamide; Cerebral Cortex; Cimetidine; Histamine; Histamine Release; Hypothalamus; Hypothalamus, Posterior; Imidazoles; Impromidine; Male; Potassium; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Synaptosomes; Thiazoles | 1987 |
Pharmacological characterization of histamine receptors in the human temporal artery.
Topics: Adult; Cimetidine; Dinoprost; Female; Histamine; Humans; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Pyridines; Pyrilamine; Receptors, Histamine; Temporal Arteries; Thiazoles; Vasoconstriction; Vasodilation | 1989 |
A role for histamine and H2-receptors in opioid antinociception.
Topics: Analgesia; Animals; Benzothiazoles; Cimetidine; Histamine; Male; Morphine; Phenoxypropanolamines; Piperidines; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Receptors, Opioid; Thiazoles | 1989 |
Famotidine and ranitidine, but not cimetidine, cause severe, disabling headache.
Topics: Adult; Cimetidine; Famotidine; Female; Headache; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles | 1989 |
Effect of cimetidine, ranitidine, famotidine and omeprazole on hepatocyte proliferation in vitro.
Topics: Animals; Cell Division; Cells, Cultured; Cimetidine; DNA; Famotidine; Hepatectomy; Histamine H2 Antagonists; Hormones; Liver; Omeprazole; Osmolar Concentration; Ranitidine; Rats; Rats, Inbred F344; Thiazoles | 1989 |
Neuronal histamine modulates feeding behavior through H1-receptor in rat hypothalamus.
Topics: Animals; Chlorpheniramine; Cimetidine; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Motor Activity; Neurons; Promethazine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Reference Values; Thiazoles | 1989 |
Safety profile of H2-receptor antagonists: current status of famotidine.
Topics: Anti-Ulcer Agents; Cimetidine; Drug Interactions; Famotidine; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles | 1989 |
The effects of cimetidine, ranitidine and famotidine on rat hepatic microsomal cytochrome P-450 activities.
Topics: Animals; Binding Sites; Cimetidine; Cytochrome P-450 Enzyme System; Famotidine; Histamine H2 Antagonists; In Vitro Techniques; Male; Microsomes, Liver; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles | 1989 |
Frequent non-response to histamine H2-receptor antagonists in cirrhotics.
Topics: Anti-Ulcer Agents; Cimetidine; Esophagitis, Peptic; Famotidine; Female; Gastric Acidity Determination; Gastritis; Histamine H2 Antagonists; Humans; Liver Cirrhosis; Male; Middle Aged; Peptic Ulcer; Ranitidine; Thiazoles | 1989 |
Evidence of drug interaction between cyclosporin A and H2-receptor antagonists (cimetidine, ranitidine and famotidine) in Sprague-Dawley rats.
Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Cimetidine; Creatinine; Cyclosporins; Drug Interactions; Famotidine; Histamine H2 Antagonists; Kidney; Liver; Male; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles | 1989 |
Histamine receptors in unstimulated pancreatic exocrine secretion of the rabbit.
Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Kinetics; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1989 |
A comparison of the cholinergic activity of selected H2-antagonists and sulfoxide metabolites.
Topics: Acetylcholine; Animals; Brain Chemistry; Cholinesterase Inhibitors; Cimetidine; Famotidine; Furans; Histamine H2 Antagonists; Ileum; Male; Mice; Nizatidine; Parasympathomimetics; Ranitidine; Structure-Activity Relationship; Sulfoxides; Thiazoles | 1989 |
Differential effects of cimetidine, ranitidine and famotidine on the hepatic metabolism of estrogen and testosterone in male rats.
Topics: Animals; Cimetidine; Estrogens; Famotidine; Liver; Male; Ranitidine; Rats; Rats, Inbred Strains; Testosterone; Thiazoles | 1989 |
Synthesis of (aryloxy)alkylamines. 1. Novel antisecretory agents with H+K+-ATPase inhibitory activity.
Topics: Adenosine Triphosphatases; Amines; Aminopyrine; Animals; Benzothiazoles; Benzoxazoles; Bucladesine; Chemical Phenomena; Chemistry; Cimetidine; Gastric Acid; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Histamine; Ligation; Male; Omeprazole; Parietal Cells, Gastric; Pyloric Antrum; Ranitidine; Rats; Structure-Activity Relationship; Thiazoles | 1988 |
Famotidine, a new, potent, long-acting histamine H2-receptor antagonist: comparison with cimetidine and ranitidine in the treatment of Zollinger-Ellison syndrome.
Topics: Aged; Cimetidine; Delayed-Action Preparations; Famotidine; Histamine H2 Antagonists; Humans; Middle Aged; Ranitidine; Thiazoles; Zollinger-Ellison Syndrome | 1985 |
Famotidine, a new H2-receptor antagonist. Effect on parietal, nonparietal, and pepsin secretion in man.
Topics: Adult; Cimetidine; Famotidine; Gastric Acidity Determination; Gastric Juice; Histamine H2 Antagonists; Humans; Male; Parietal Cells, Gastric; Pentagastrin; Pepsin A; Thiazoles; Time Factors | 1985 |
Effects of H2-receptor antagonists upon physiological acid secretory states in animals.
Topics: Animals; Benzimidazoles; Cimetidine; Famotidine; Gastric Emptying; Gastric Juice; Histamine H2 Antagonists; Male; Omeprazole; Rats; Secretory Rate; Thiadiazoles; Thiazoles | 1985 |
Clinical pharmacology of famotidine.
Topics: Animals; Cimetidine; Circadian Rhythm; Dogs; Dose-Response Relationship, Drug; Duodenal Ulcer; Famotidine; Food; Gastric Acid; Half-Life; Histamine; Histamine H2 Antagonists; Humans; Kinetics; Pentagastrin; Pepsin A; Prolactin; Rats; Tetragastrin; Thiazoles; Time Factors | 1985 |
Comparative effects of famotidine and cimetidine on trimethadione metabolism in the rat.
Topics: Animals; Cimetidine; Famotidine; Histamine H2 Antagonists; Kinetics; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxazoles; Rats; Thiazoles; Trimethadione | 1986 |
Interaction of diazepam with famotidine and cimetidine, two H2-receptor antagonists.
Topics: Adult; Biotransformation; Cimetidine; Diazepam; Drug Interactions; Famotidine; Half-Life; Histamine H2 Antagonists; Humans; Infusions, Parenteral; Kinetics; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam; Thiazoles | 1986 |
Cholinergic effects of histamine-H2 receptor antagonists partly through inhibition of acetylcholinesterase.
Topics: Animals; Butyrylcholinesterase; Cholinesterase Inhibitors; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Ranitidine; Thiazoles | 1986 |
Interaction of famotidine with rat liver microsomes, a study showing less inhibition of drug metabolism than with cimetidine.
Topics: Aminopyrine N-Demethylase; Animals; Cimetidine; Cytochrome P-450 Enzyme System; Famotidine; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylcholanthrene; Microsomes, Liver; Phenobarbital; Rats; Rats, Inbred Strains; Thiazoles | 1986 |
Inhibition of gastric acid secretion by H2-receptor antagonists.
Topics: Animals; Benzothiazoles; Cimetidine; Depression, Chemical; Gastric Acid; Guinea Pigs; Heart Rate; Histamine H2 Antagonists; In Vitro Techniques; Male; Pylorus; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles | 1986 |
Actions of nizatidine, a selective histamine H2-receptor antagonist, on gastric acid secretion in dogs, rats and frogs.
Topics: Administration, Oral; Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Gastric Acid; Histamine H2 Antagonists; Infusions, Parenteral; Molecular Weight; Nizatidine; Rana catesbeiana; Rats; Tetragastrin; Thiazoles | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
Effect of five structurally diverse H2-receptor antagonists on drug metabolism.
Topics: 7-Alkoxycoumarin O-Dealkylase; Animals; Aryl Hydrocarbon Hydroxylases; Biotransformation; Cimetidine; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Diazepam; Famotidine; Histamine H2 Antagonists; Humans; Imidazoles; Kinetics; Male; Microsomes, Liver; Nizatidine; Oxidoreductases; Oxygenases; Pharmaceutical Preparations; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles | 1986 |
Direct effects of H2-receptor antagonists on airway smooth muscle and on responses mediated by H1- and H2-receptors.
Topics: Animals; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ranitidine; Thiazoles; Trachea | 1987 |
Tiotidine and ICIA 5165 inhibit central and peripheral H2 receptors with equal potency.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cimetidine; Guanidines; Guinea Pigs; Heart Rate; Hippocampus; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Thiazoles | 1987 |
[Comparative studies on hemodynamic effects of intravenous cimetidine, ranitidine and famotidine in intensive care unit patients].
Topics: Adult; Aged; Aged, 80 and over; Cimetidine; Famotidine; Female; Hemodynamics; Histamine H2 Antagonists; Humans; Injections, Intravenous; Intensive Care Units; Male; Middle Aged; Ranitidine; Thiazoles | 1987 |
Effect of histamine H2-receptor antagonists on DNA synthesis in adult rat hepatocytes in primary culture. Cimetidine enhanced hepatocytes proliferation stimulated with insulin and epidermal growth factor.
Topics: Animals; Cell Division; Cimetidine; DNA; Epidermal Growth Factor; Famotidine; Histamine H2 Antagonists; Humans; Insulin; Liver; Protein Biosynthesis; Ranitidine; Rats; Thiazoles | 1987 |
[Action of famotidine, a new H2-receptor antagonist, on the papillary muscle and atrium of the guinea pig, in vitro].
Topics: Animals; Cimetidine; Famotidine; Guinea Pigs; Heart Rate; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Myocardial Contraction; Ranitidine; Thiazoles | 1987 |
Effects of prolonged oral cimetidine, ranitidine, and famotidine therapy on antipyrine elimination.
Topics: Administration, Oral; Adolescent; Adult; Aged; Antipyrine; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Liver; Male; Metabolic Clearance Rate; Middle Aged; Ranitidine; Thiazoles | 1987 |
Zolantidine (SK&F 95282) is a potent selective brain-penetrating histamine H2-receptor antagonist.
Topics: Animals; Benzothiazoles; Binding, Competitive; Brain Chemistry; Cimetidine; Cyclic AMP; Female; Guinea Pigs; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Male; Phenoxypropanolamines; Piperidines; Rats; Thiazoles; Uterus | 1988 |
A comparative evaluation of the transport of H2-receptor antagonists by the human and baboon placenta.
Topics: Adolescent; Adult; Animals; Antipyrine; Biological Transport; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; In Vitro Techniques; Maternal-Fetal Exchange; Nizatidine; Papio; Perfusion; Placenta; Pregnancy; Ranitidine; Thiazoles | 1988 |
Effect of mifentidine on mepirizole-induced duodenal ulcer in the rat.
Topics: Animals; Anti-Ulcer Agents; Cimetidine; Dose-Response Relationship, Drug; Duodenal Ulcer; Duodenum; Epirizole; Famotidine; Female; Histamine H2 Antagonists; Imidazoles; Intestinal Mucosa; Pyrazoles; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles | 1987 |
The effect of H2-receptor antagonists on antipyrine and pentobarbital metabolism in male and female rats.
Topics: Animals; Antipyrine; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Male; Microsomes, Liver; Mixed Function Oxygenases; Pentobarbital; Ranitidine; Rats; Rats, Inbred Strains; Sex Factors; Thiazoles | 1988 |
In vitro studies on the interaction of famotidine with liver microsomal cytochrome P-450.
Topics: Animals; Cimetidine; Cytochrome P-450 Enzyme System; Famotidine; Histamine H2 Antagonists; Humans; Male; Methylcholanthrene; Microsomes, Liver; Oxidation-Reduction; Phenobarbital; Rats; Rats, Inbred Strains; Spectrum Analysis; Thiadiazoles; Thiazoles | 1988 |
Differential inhibition of human liver phenacetin O-deethylation by histamine and four histamine H2-receptor antagonists.
Topics: Binding Sites; Binding, Competitive; Catalysis; Chromatography, Thin Layer; Cimetidine; Cytochrome P-450 CYP1A2; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Imidazoles; Microsomes, Liver; Oxidation-Reduction; Oxidoreductases; Ranitidine; Thiazoles | 1988 |
Recurrent parotitis with H2 receptor antagonists in a patient with Sjogren's syndrome.
Topics: Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Middle Aged; Parotitis; Ranitidine; Recurrence; Sjogren's Syndrome; Stomach Ulcer; Thiazoles | 1988 |
Cimetidine (but not ranitidine or famotidine) affects histamine determination.
Topics: Cimetidine; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles | 1988 |
Plasma sex steroid transport and histamine H2-receptor antagonists. Clinical implications.
Topics: Adult; Cimetidine; Famotidine; Gonadal Steroid Hormones; Histamine H2 Antagonists; Hormones; Humans; Male; Middle Aged; Peptic Ulcer; Ranitidine; Sex Hormone-Binding Globulin; Thiazoles; Thyroid Hormones | 1988 |
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea | 1988 |
Bacterial genotoxicity of nitrosated famotidine.
Topics: Animals; Biotransformation; Cimetidine; Escherichia coli; Famotidine; Histamine H1 Antagonists; Microsomes, Liver; Mutagenicity Tests; Mutation; Nitrites; Ranitidine; Rats; Rats, Inbred Strains; Salmonella typhimurium; Thiazoles | 1986 |
Refractory duodenal ulcers (nonhealing duodenal ulcers with standard doses of antisecretory medication).
Topics: Adult; Aged; Anti-Ulcer Agents; Cimetidine; Duodenal Ulcer; Famotidine; Female; Gastric Acid; Humans; Male; Middle Aged; Ranitidine; Smoking; Thiazoles | 1989 |
Characterization of histamine receptors mediating the stimulation of cyclic AMP accumulation in rabbit cerebral cortical slices.
Topics: Adenosine; Animals; Cerebral Cortex; Chlorpheniramine; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Imidazoles; Impromidine; Kinetics; Mathematics; Metiamide; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles | 1985 |
New H2-blockers: does more choice help?
Topics: Anti-Ulcer Agents; Cimetidine; Famotidine; Humans; Nizatidine; Peptic Ulcer; Ranitidine; Thiazoles | 1988 |
Healing and relapse rates of duodenal ulcer with various H2 receptor antagonists.
Topics: Adolescent; Adult; Anti-Ulcer Agents; Cimetidine; Duodenal Ulcer; Famotidine; Female; Humans; Male; Ranitidine; Retrospective Studies; Thiazoles | 1988 |
Comparative effects of famotidine and cimetidine on 7-ethoxycoumarin O-deethylase activity in human livers.
Topics: 7-Alkoxycoumarin O-Dealkylase; Cimetidine; Famotidine; Humans; Liver; Oxygenases; Thiazoles | 1986 |
Effects of H1- and H2-histamine receptor agonists and antagonists on sleep and wakefulness in the rat.
Topics: Animals; Cimetidine; Diphenhydramine; Electroencephalography; Injections, Intraperitoneal; Injections, Intraventricular; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sleep, REM; Thiazoles; Wakefulness | 1986 |
Comparison of the effects of gastric antisecretory agents in healthy volunteers and patients with duodenal ulcer.
Topics: Anti-Ulcer Agents; Cimetidine; Drug Administration Schedule; Duodenal Ulcer; Famotidine; Gastric Acidity Determination; Humans; Imidazoles; Omeprazole; Ranitidine; Thiazoles | 1986 |
Effect of H2-receptor antagonists on acetaminophen-induced hepatic injury.
Topics: Acetaminophen; Animals; Chemical and Drug Induced Liver Injury; Cimetidine; Famotidine; Glutathione; Liver; Liver Diseases; Male; Methylcholanthrene; Microsomes, Liver; Ranitidine; Rats; Thiazoles | 1986 |
Gastric anti-ulcer and cytoprotective properties of 2-(3,4-dimethoxyphenyl)-5-methyl-thiazolidine-4-one in rat experimental ulcers.
Topics: Acetates; Animals; Anti-Ulcer Agents; Cell Survival; Cimetidine; Ethanol; Gastric Mucosa; Indomethacin; Male; Rats; Rats, Inbred Strains; Regional Blood Flow; Stomach Ulcer; Thiazoles | 1986 |
In vitro histamine H2-antagonist activity of the novel compound HUK 978.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Cimetidine; Dose-Response Relationship, Drug; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Ileum; Receptors, Histamine; Receptors, Histamine H2; Thiazoles | 1985 |
Anti-secretory activity of the novel H2-antagonist, HUK 978, in rat, guinea-pig and dog.
Topics: Administration, Oral; Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Gastric Acid; Gastric Mucosa; Guanidines; Guinea Pigs; Injections, Intravenous; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Time Factors | 1985 |
[H2 receptor antagonists and intragastric acidity].
Topics: Cimetidine; Drug Administration Schedule; Famotidine; Histamine Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Peptic Ulcer; Ranitidine; Thiazoles | 1984 |
The cardiac pharmacology of tiotidine (LCL 125, 211): a new histamine H2-receptor antagonist.
Topics: Animals; Arrhythmias, Cardiac; Atrioventricular Node; Cimetidine; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Thiazoles | 1980 |
New drugs for peptic ulcer.
Topics: Benzamides; Benzodiazepinones; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Morpholines; Parasympatholytics; Pepsin A; Peptic Ulcer; Piperazines; Pirenzepine; Prostaglandins E, Synthetic; Ranitidine; Thiazoles; Trimipramine | 1980 |
Tiotidine and cimetidine--kinetics and dynamics.
Topics: Adult; Cimetidine; Dose-Response Relationship, Drug; Female; Guanidines; Histamine H2 Antagonists; Humans; Intestinal Absorption; Male; Metabolic Clearance Rate; Middle Aged; Thiazoles; Time Factors | 1981 |
Species differences in the contractile response to two specific histamine H1-receptor agonists: 2-(2-pyridyl)-ethylamine and 2-(2-aminoethyl)-thiazole.
Topics: Animals; Cimetidine; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Species Specificity; Thiazoles; Vas Deferens | 1981 |
Effects of H2-receptor antagonists cimetidine, ranitidine, and ICI 125,211 on histamine-stimulated adenylate cyclase activity in guinea pig gastric mucosa.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Ranitidine; Structure-Activity Relationship; Thiazoles | 1981 |
Inhibition of microsomal drug metabolism by histamine H2-receptor antagonists studied in vivo and in vitro in rodents.
Topics: Aminopyrine; Aminopyrine N-Demethylase; Animals; Breath Tests; Cimetidine; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Furans; Guanidines; Histamine H2 Antagonists; Male; Mice; Mice, Inbred ICR; Microsomes, Liver; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Time Factors | 1982 |
Effect of some new Histamine H2-receptor antagonists on the guinea-pig papillary muscle.
Topics: Animals; Cimetidine; Furans; Guanidines; Guinea Pigs; Histamine Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Ranitidine; Thiazoles | 1981 |
Histamine H1- and muscarinic receptor antagonist activity of cimetidine and tiotidine in the guinea pig isolated ileum.
Topics: Animals; Carbachol; Cimetidine; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Thiazoles | 1981 |
Effect of a new potent H2-blocker, 3-]]]2-[(diaminomethylene)amino]-4-thiazolyl]methyl]-thio]-N2-sulfamoylpropionamidine (YM-11170) on gastric secretion induced by histamine and food in conscious dogs.
Topics: Animals; Cimetidine; Dogs; Famotidine; Food; Gastric Acid; Histamine; Histamine H2 Antagonists; Thiazoles | 1982 |
Interaction of histamine with gastric mucosal cells. Effect of histamine H2 antagonists on binding and biological response.
Topics: Animals; Cimetidine; Cyclic AMP; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Ranitidine; Receptors, Histamine; Thiazoles | 1982 |
Effect of a new potent H2-blocker, 3-[[[2-(diaminomethylene)amino]-4-thiazolyl]methyl]thio]-N2-sulfamoyl propionamidine (YM-11170), on gastric secretion, ulcer formation and weight of male accessory sex organs in rats.
Topics: Androgen Antagonists; Animals; Aspirin; Castration; Cimetidine; Famotidine; Gastric Juice; Gastric Mucosa; Genitalia, Male; Histamine H2 Antagonists; Male; Organ Size; Rats; Rats, Inbred Strains; Stomach Ulcer; Testosterone; Thiazoles | 1982 |
A comparison of some of the pharmacological properties of etintidine, a new histamine H2-receptor antagonist, with those of cimetidine, ranitidine and tiotidine.
Topics: Adrenergic beta-Antagonists; Animals; Cimetidine; Dogs; Female; Furans; Gastric Juice; Guanidines; Guinea Pigs; Heart Rate; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Parasympatholytics; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Uterine Contraction | 1983 |
The role of antagonists to acid secretion.
Topics: 16,16-Dimethylprostaglandin E2; Benzodiazepinones; Cimetidine; Furans; Gastric Acid; Gastrointestinal Diseases; Guanidines; Histamine H2 Antagonists; Humans; Pirenzepine; Proglumide; Ranitidine; Somatostatin; Thiazoles | 1982 |
Conformational requirements for histamine H2-receptor inhibitors: a structure-activity study of phenylene analogues related to cimetidine and tiotidine.
Topics: Animals; Benzene Derivatives; Biological Assay; Cimetidine; Dogs; Folic Acid; Gastric Juice; Guanidines; Guinea Pigs; Heart Atria; Histamine H2 Antagonists; Indicators and Reagents; Myocardial Contraction; Receptors, Histamine; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles | 1983 |
Dose-response curve analysis of gastric secretory responses in the dog and man to impromidine: a new histamine-H2-receptor agonist.
Topics: Adult; Animals; Binding, Competitive; Cimetidine; Dogs; Dose-Response Relationship, Drug; Female; Gastric Acid; Guanidines; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles | 1983 |
Effect of a new potent H2-receptor antagonist 3[[[2-[(diaminomethylene)amino]-4-thiazolyl]methyl]thio]-N2- sulfamoylpropionamidine (YM-11170) on gastric mucosal histamine-sensitive adenylate cyclase from guinea pig.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Dinoprostone; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Guinea Pigs; Hippocampus; Histamine; Histamine H2 Antagonists; Male; Prostaglandins E; Thiazoles | 1983 |
Effects of antiulcer agents on healing of mepirizole-induced duodenal ulcers in rats.
Topics: Aluminum Hydroxide; Animals; Anti-Ulcer Agents; Cimetidine; Drug Combinations; Duodenal Ulcer; Epirizole; Famotidine; Histamine H2 Antagonists; Magnesium Hydroxide; Male; Propantheline; Prostaglandins E, Synthetic; Pyrazoles; Rats; Rats, Inbred Strains; Thiazoles; Time Factors; Wound Healing | 1983 |
Kinetics of antisecretory action of a new H2-antagonist, YM-11170, in conscious dogs.
Topics: Animals; Atropine; Cimetidine; Dimaprit; Dogs; Famotidine; Gastric Acid; Gastric Mucosa; Histamine H2 Antagonists; Kinetics; Male; Methacholine Chloride; Methacholine Compounds; Pentagastrin; Thiazoles; Thiourea | 1983 |
Studies on MK-208 (YM-11170) a new, slowly dissociable H2-receptor antagonist.
Topics: Animals; Cimetidine; Famotidine; Female; Gastric Acid; Gastric Fistula; Guinea Pigs; Heart Atria; Heart Rate; Histamine H2 Antagonists; In Vitro Techniques; Male; Ranitidine; Rats; Thiazoles | 1983 |
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea | 1983 |
Evidence for the existence of histamine H1- and H2-receptors on astrocytes of cultured rat central nervous system.
Topics: Aminopyridines; Animals; Astrocytes; Brain Stem; Cells, Cultured; Cimetidine; Histamine; Histamine H1 Antagonists; Membrane Potentials; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Spinal Cord; Thiazoles | 1984 |
Method for detection of antibody against low molecular weight antigen (hapten)--production and detection of antibody against histamine H2 receptor of antibody against histamine H2 receptor antagonist "Famotidine".
Topics: Animals; Antibodies; Antibody Formation; Antibody Specificity; Cimetidine; Famotidine; Fluorescent Antibody Technique; Haptens; Histamine H2 Antagonists; Molecular Weight; Rabbits; Ranitidine; Thiazoles | 1983 |
Interaction of alpha-adrenergic imidazolines with cardiac histamine H2-receptors.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Drug Interactions; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine Release; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Receptors, Histamine; Receptors, Histamine H2; Stereoisomerism; Sympathomimetics; Tetrahydronaphthalenes; Thiazoles; Tolazoline | 1981 |
A species comparison of the histamine H2-receptor on mast cells and basophils.
Topics: Animals; Basophils; Cimetidine; Female; Furans; Guanidines; Guinea Pigs; Histamine H2 Antagonists; Histamine Release; Humans; In Vitro Techniques; Lung; Male; Mast Cells; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Thiazoles | 1982 |
A possible physiological role of histamine H2-receptors in rat mesenteric circulation.
Topics: Animals; Cimetidine; Dimaprit; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Splanchnic Circulation; Thiazoles; Thiourea; Vasodilation | 1983 |
Effects of histamine receptor stimulation on regional myocardial blood flow.
Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1983 |
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1982 |
Inhibition of gastric secretion by a new H2-antagonist, YM-11170 in healthy subjects.
Topics: Administration, Oral; Adult; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Juice; Humans; Male; Pepsin A; Ranitidine; Thiazoles; Time Factors | 1984 |
In-vivo nitrosation, precancerous lesions and cancers of the gastrointestinal tract. On-going studies and preliminary results.
Topics: Anemia, Pernicious; Cimetidine; Gastrectomy; Gastritis, Atrophic; Humans; Nitrosamines; Nitroso Compounds; Precancerous Conditions; Stomach Neoplasms; Thiazoles; Thiazolidines | 1984 |
Effect of H2-receptor antagonists, cimetidine and YM-11170, on serum gastrin levels in lumen-perfused rats.
Topics: Animals; Cimetidine; Famotidine; Gastric Acid; Gastric Acidity Determination; Gastric Mucosa; Gastrins; Histamine; Infusions, Parenteral; Male; Perfusion; Rats; Rats, Inbred Strains; Thiazoles | 1983 |
[Effects of protective agents on ulcer formation].
Topics: Adult; Animals; Cimetidine; Dogs; Duodenal Ulcer; Famotidine; Gastric Juice; Gastric Mucosa; Humans; Male; Peptic Ulcer; Stomach Ulcer; Thiazoles | 1984 |
Comparative effects of famotidine and cimetidine on antipyrine kinetics in healthy volunteers.
Topics: Adult; Antipyrine; Cimetidine; Famotidine; Female; Humans; Kinetics; Male; Thiazoles | 1984 |
Effect of ebrotidine on the density of antral G-cells in the gastric mucosa in the rat.
Topics: Animals; Benzenesulfonates; Cell Count; Cell Division; Cimetidine; Gastric Mucosa; Histamine H2 Antagonists; Immunohistochemistry; Male; Pyloric Antrum; Rats; Rats, Sprague-Dawley; Thiazoles | 1995 |
Effects of a histamine H2 receptor agonist and antagonist on restraint-induced antinociception in female mice.
Topics: Animals; Benzothiazoles; Cimetidine; Dimaprit; Female; Histamine Agonists; Histamine H2 Antagonists; Mice; Mice, Inbred Strains; Pain Measurement; Phenoxypropanolamines; Piperidines; Reaction Time; Restraint, Physical; Stress, Psychological; Thiazoles | 1995 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine | 1994 |
Antisecretory effects of a novel and long-lasting histamine H2-receptor antagonist, YM-14471, in rats and dogs.
Topics: Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H2 Antagonists; Infusions, Intravenous; Male; Omeprazole; Pyrimidinones; Rats; Rats, Wistar; Thiazoles | 1993 |
Effect of cimetidine on the pharmacokinetics of fentiazac in rats.
Topics: Acetates; Animals; Anti-Inflammatory Agents, Non-Steroidal; Biological Availability; Blood Proteins; Chromatography, High Pressure Liquid; Cimetidine; Half-Life; Injections, Intravenous; Male; Protein Binding; Rats; Rats, Wistar; Thiazoles | 1993 |
Histaminergic drugs in the rat caudate nucleus: effects on learned helplessness.
Topics: Animals; Astemizole; Caudate Nucleus; Cimetidine; Helplessness, Learned; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles | 1993 |
Increases in cyclic AMP levels couple to H1 receptors in atria from autoimmune myocarditis mice.
Topics: Animals; Autoimmune Diseases; Cimetidine; Cyclic AMP; Heart Atria; Histamine; Histamine Agonists; Histamine Antagonists; Male; Mice; Myocarditis; Phosphatidylinositols; Pyrilamine; Receptors, Histamine H1; Signal Transduction; Thiazoles | 1995 |
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles | 1996 |
Action of ebrotidine, ranitidine and cimetidine on the specific binding to histamine H1- and H2-receptors.
Topics: Animals; Benzenesulfonates; Cell Membrane; Cerebellum; Cerebral Cortex; Cimetidine; Depression, Chemical; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Isotope Labeling; Male; Protein Binding; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium | 1997 |
Effect of ebrotidine on ethanol-induced gastric mucosal damage in the rat. Comparative study with other H2-receptor antagonists.
Topics: Animals; Benzenesulfonates; Cimetidine; Dose-Response Relationship, Drug; Ethanol; Famotidine; Female; Gastric Mucosa; Histamine H2 Antagonists; Indomethacin; Peptic Ulcer; Ranitidine; Rats; Rats, Sprague-Dawley; Thiazoles | 1997 |
Comparative study of plasma gastrin levels in rats after two months of ebrotidine administration.
Topics: Animals; Benzenesulfonates; Cimetidine; Gastrins; Histamine H2 Antagonists; Male; Omeprazole; Ranitidine; Rats; Rats, Sprague-Dawley; Specific Pathogen-Free Organisms; Thiazoles | 1997 |
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea | 1999 |
Accurate mass liquid chromatography/mass spectrometry on quadrupole orthogonal acceleration time-of-flight mass analyzers using switching between separate sample and reference sprays. 2. Applications using the dual-electrospray ion source.
Topics: Calibration; Cimetidine; Indicators and Reagents; Rosiglitazone; Spectrometry, Mass, Electrospray Ionization; Thiazoles; Thiazolidinediones | 2001 |
Derivatives of dehydrocrotonin, a diterpene lactone isolated from Croton cajucara: cytotoxicity in rat cultured hepatocytes and in V79 cells.
Topics: Animals; Cell Line; Cell Survival; Cellular Senescence; Cimetidine; Cricetinae; Cricetulus; Croton; Culture Media, Conditioned; Diterpenes; Diterpenes, Clerodane; DNA; Dose-Response Relationship, Drug; Fibroblasts; Hepatocytes; Male; Neutral Red; Plants, Medicinal; Rats; Rats, Wistar; Succinate Dehydrogenase; Tetrazolium Salts; Thiazoles | 2002 |
Antinociceptive, brain-penetrating derivatives related to improgan, a non-opioid analgesic.
Topics: Algorithms; Analgesics; Animals; Behavior, Animal; Benzothiazoles; Brain; Cimetidine; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Molecular Structure; Pain; Pain Measurement; Phenoxypropanolamines; Piperidines; Quinazolines; Quinazolinones; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors; Triazoles | 2005 |
Bone hydatid disease refractory to nitazoxanide treatment.
Topics: Adult; Albendazole; Anthelmintics; Bone Diseases; Cimetidine; Drug Resistance; Echinococcosis; Histamine H2 Antagonists; Humans; Lumbar Vertebrae; Male; Nitro Compounds; Thiazoles | 2009 |
Interferon-α-based immunotherapy in metastatic renal cell carcinoma patients with the primary tumor in situ.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Carcinoma in Situ; Carcinoma, Renal Cell; Chemotherapy, Adjuvant; Cimetidine; Dexamethasone; Female; Humans; Immunotherapy; Interferon-alpha; Kaplan-Meier Estimate; Kidney Neoplasms; Male; Meloxicam; Middle Aged; Neoadjuvant Therapy; Nephrectomy; Thiazines; Thiazoles; Treatment Outcome | 2012 |
Role of histamine and its receptor subtypes in stimulation of conjunctival goblet cell secretion.
Topics: Animals; Blotting, Western; Cells, Cultured; Cimetidine; Conjunctiva; Conjunctivitis, Allergic; Dose-Response Relationship, Drug; Fluorescent Antibody Technique; Goblet Cells; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Indoles; Male; Methylhistamines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles | 2012 |
Histamine receptor 2-mediated growth-differentiation factor-15 expression is involved in histamine-induced melanogenesis.
Topics: Cell Line, Tumor; Cell Proliferation; Chemotaxis; Cimetidine; Gene Expression; Gene Expression Regulation; Growth Differentiation Factor 15; Histamine; Histamine Agonists; Humans; Intramolecular Oxidoreductases; Melanins; Membrane Glycoproteins; Monophenol Monooxygenase; Oxidoreductases; Receptors, Histamine H2; Thiazoles | 2012 |
Contribution of the organic anion transporter OAT2 to the renal active tubular secretion of creatinine and mechanism for serum creatinine elevations caused by cobicistat.
Topics: Animals; Biological Transport, Active; Carbamates; Cell Line; Cells, Cultured; CHO Cells; Cimetidine; Cobicistat; Creatinine; Cricetulus; Dogs; HEK293 Cells; Humans; Kidney Tubules; Kinetics; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Organic Cation Transporter 2; Recombinant Proteins; Thiazoles | 2014 |