cimetidine and burimamide

cimetidine has been researched along with burimamide in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199024 (77.42)18.7374
1990's5 (16.13)18.2507
2000's2 (6.45)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Durant, GJ; Emmett, JC; Ganellin, CR; Miles, PD; Parsons, ME; Prain, HD; White, GR1
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Cross, SA1
Ryss, ES1
Maśliński, C; Nowak, JZ; Pilc, A1
Eschchar, I; Neuman, M; Pavlotzky, M1
Barth, H; Lorenz, W1
McCulloch, MW; Medgett, IC; Rand, MJ1
Festen, HP; Lamersen, CB; van Tongeren, JH1
Corbett, R; Greaves, MW1
Sajewicz, Z1
Drazen, JM; Soter, NA; Venugopalan, CS1
Chand, N; Eyre, P1
Brink, C; Gorenne, I; Labat, C; Norel, X; Ortiz, JL; Verley, J1
Arrang, JM; Garbarg, M; Schwartz, JC1
Adaikan, PG; Lau, LC; Ratnam, SS1
Dracott, BN; Fallowfield, C; Milliner, KJ; Vickers, MR1
Nowak, JZ1
Amos, RJ; Horton, MA; Jones, RJ1
Brittain, RT; Jack, D1
Bianucci, AM; Da Settimo, A; Martinelli, A1
Carella, G1
Pounder, RE1
Duncan, WA; Parsons, ME1
Bonasera, L; Pontieri, GM; Tolone, G1
Molinder, HK1
Alewijnse, AE; Blauw, J; Leurs, R; Roovers, E; Smit, MJ; Timmerman, H; Van De Vrede, Y; Van Nieuw Amerongen, GP1
Alewijnse, AE; Hoffmann, M; Leurs, R; Smit, MJ; Timmerman, H; Verzijl, D1
Hough, LB; Leurs, R; Menge, WM; Nalwalk, JW; Timmerman, H1

Reviews

7 review(s) available for cimetidine and burimamide

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990
[Current antihistaminic preparations in treatment of peptic ulcer (review of foreign literature)].
    Klinicheskaia meditsina, 1978, Volume: 56, Issue:6

    Topics: Animals; Burimamide; Cimetidine; Dogs; Drug Evaluation; Gastric Juice; Histamine; Histamine H2 Antagonists; Humans; Metiamide; Peptic Ulcer; Pyrrolidines; Thiophenes

1978
[Cimetidine and other H2 receptor blockers].
    Harefuah, 1978, Oct-01, Volume: 95, Issue:7

    Topics: Burimamide; Cimetidine; Esophagitis; Esophagitis, Peptic; Gastrointestinal Hemorrhage; Guanidines; Histamine H2 Antagonists; Humans; Metiamide

1978
[Cimetidine; new hope for ulcer patients?].
    Nederlands tijdschrift voor geneeskunde, 1978, Jun-17, Volume: 122, Issue:24

    Topics: Burimamide; Cimetidine; Creatinine; Duodenal Ulcer; Esophagitis, Peptic; Gastric Juice; Gastritis; Guanidines; Humans; Metiamide; Peptic Ulcer; Receptors, Histamine; Transaminases; Zollinger-Ellison Syndrome

1978
Histamine H2-antagonists--past, present and future.
    Journal of clinical gastroenterology, 1983, Volume: 5 Suppl 1

    Topics: Animals; Aspirin; Burimamide; Chemical Phenomena; Chemistry; Cimetidine; Dogs; Furans; Gastric Acid; Guanidines; Guinea Pigs; Half-Life; Histamine H2 Antagonists; Humans; Imidazoles; Methylamines; Ranitidine; Rats; Stomach; Thiazoles; Triazoles

1983
[Antagonists of histamine H1 and H2 receptors: pharmacologic aspects and clinical significance].
    La Clinica terapeutica, 1984, Aug-31, Volume: 110, Issue:4

    Topics: Burimamide; Cardiovascular System; Chlorpheniramine; Cimetidine; Duodenal Ulcer; Gastric Acid; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Neoplasms; Ranitidine; Urticaria

1984
Histamine H2-receptor antagonists and gastric acid secretion.
    Pharmacology & therapeutics, 1984, Volume: 26, Issue:2

    Topics: Burimamide; Chemical Phenomena; Chemistry; Cimetidine; Duodenal Ulcer; Esophagitis, Peptic; Gastric Acid; Gastrins; Gastrointestinal Hemorrhage; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Hypersensitivity; Intrinsic Factor; Kinetics; Malabsorption Syndromes; Metiamide; Pancreas; Pepsin A; Ranitidine; Receptors, Histamine H2; Stomach Ulcer; Stress, Psychological; Zollinger-Ellison Syndrome

1984

Trials

1 trial(s) available for cimetidine and burimamide

ArticleYear
Burimamide, metiamide, cimetidine...
    Lancet (London, England), 1975, Oct-25, Volume: 2, Issue:7939

    Topics: Bone Marrow; Burimamide; Cimetidine; Clinical Trials as Topic; Duodenal Ulcer; Guanidines; Humans; Metiamide; Thiourea

1975

Other Studies

23 other study(ies) available for cimetidine and burimamide

ArticleYear
Cyanoguanidine-thiourea equivalence in the development of the histamine H2-receptor antagonist, cimetidine.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:7

    Topics: Chemical Phenomena; Chemistry, Physical; Drug Stability; Guanidines; Histamine H2 Antagonists; Imidazoles; Molecular Conformation; Structure-Activity Relationship; Thiourea

1977
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Localization of histamine and histamine H2-receptor antagonists in the gastric mucosa.
    The Histochemical journal, 1977, Volume: 9, Issue:5

    Topics: Animals; Autoradiography; Burimamide; Carbonic Anhydrases; Cimetidine; Dogs; Female; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Male; Metiamide; Rats

1977
An interaction of histamine H2-receptor antagonists with the noradrenergic system in rat brain.
    European journal of pharmacology, 1978, Sep-01, Volume: 51, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Burimamide; Cimetidine; Dopamine; Female; Histamine H2 Antagonists; In Vitro Techniques; Metiamide; Motor Activity; Norepinephrine; Rats; Time Factors

1978
[Histamine and its role in peptic gastric diseases: the discovery of histamine-H2-receptor antagonists].
    Acta medica Austriaca, 1978, Volume: 5, Issue:2

    Topics: Animals; Burimamide; Cats; Cimetidine; Dogs; Duodenal Ulcer; Gastric Juice; Gastric Mucosa; Histamine H2 Antagonists; Histamine N-Methyltransferase; Humans; Male; Mast Cells; Pentagastrin; Peptic Ulcer; Rats; Receptors, Histamine H2; Vagotomy

1978
Effects of the histamine H2-receptor blocking drugs burimamide and cimetidine on noradrenergic transmission in the isolated aorta of the rabbit and atria of the guinea-pig.
    British journal of pharmacology, 1979, Volume: 67, Issue:4

    Topics: Animals; Aorta, Thoracic; Burimamide; Cimetidine; Cocaine; Female; Guanidines; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Rabbits; Synaptic Transmission; Thiourea

1979
Histamine H2-receptor antagonists inhibit enzymic histamine degradation in human skin.
    Clinical and experimental dermatology, 1979, Volume: 4, Issue:1

    Topics: Amodiaquine; Burimamide; Cimetidine; Guanidines; Histamine N-Methyltransferase; Humans; In Vitro Techniques; Methyltransferases; Skin; Thiourea

1979
[Current views on the role of histamine and histamine H2 receptors of parietal cells in the process of gastric secretion].
    Polski tygodnik lekarski (Warsaw, Poland : 1960), 1979, Jul-16, Volume: 34, Issue:29

    Topics: Burimamide; Chemical Phenomena; Chemistry; Cimetidine; Gastric Juice; Gastric Mucosa; Histamine; Humans; Metiamide; Models, Biological; Receptors, Histamine; Receptors, Histamine H2; Stimulation, Chemical

1979
H2 receptor mediated inhibition of immediate type hypersensitivity reactions in vivo.
    The American review of respiratory disease, 1978, Volume: 117, Issue:3

    Topics: Anaphylaxis; Animals; Burimamide; Cimetidine; Feedback; Guinea Pigs; Lung; Lung Volume Measurements; Male; Methylhistamines; Metiamide; Receptors, Histamine; Receptors, Histamine H2

1978
Spasmolytic action of histamine in airway smooth muscle of horse.
    Agents and actions, 1978, Volume: 8, Issue:3

    Topics: Animals; Atropine; Bronchi; Burimamide; Cimetidine; Histamine; Horses; In Vitro Techniques; Indomethacin; Metiamide; Muscle Contraction; Muscle, Smooth; Propranolol; Pyrilamine; Respiratory System; Trachea

1978
Histamine receptors on human isolated pulmonary arterial muscle preparations: effects of endothelial cell removal and nitric oxide inhibitors.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Arginine; Burimamide; Chlorpheniramine; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Pulmonary Artery; Receptors, Histamine; Serotonin; Tetraethylammonium; Tetraethylammonium Compounds; Thiourea

1992
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
    Neuroscience, 1987, Volume: 23, Issue:1

    Topics: Animals; Burimamide; Cerebral Cortex; Cimetidine; Histamine; Histamine Release; Hypothalamus; Hypothalamus, Posterior; Imidazoles; Impromidine; Male; Potassium; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Synaptosomes; Thiazoles

1987
Effect of histamine on human vas deferens in vitro.
    British journal of urology, 1989, Volume: 64, Issue:4

    Topics: Burimamide; Cimetidine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Humans; Male; Methylhistamines; Muscle Contraction; Pyrilamine; Vas Deferens

1989
The effects of histamine H2-receptor antagonists on PHA induced lymphocyte proliferation.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Burimamide; Cimetidine; Histamine H2 Antagonists; Histamine Release; Humans; In Vitro Techniques; Lymphocyte Activation; Phytohemagglutinins; Pyrimidinones; Ranitidine

1984
Interaction of histamine H2-receptor blocking drugs with the noradrenergic system in rat brain and heart.
    European journal of pharmacology, 1980, Nov-07, Volume: 68, Issue:1

    Topics: Animals; Brain; Burimamide; Cimetidine; Histamine H2 Antagonists; Male; Metiamide; Myocardium; Norepinephrine; Rats

1980
The effect of histamine H2 receptor antagonists on platelet aggregation in man.
    Scandinavian journal of haematology, 1983, Volume: 31, Issue:1

    Topics: Burimamide; Cimetidine; Dose-Response Relationship, Drug; Furans; Histamine H2 Antagonists; Humans; Imidazoles; Male; Metiamide; Platelet Aggregation; Ranitidine

1983
A conformational approach to histamine H2-receptor antagonists.
    Il Farmaco; edizione scientifica, 1984, Volume: 39, Issue:8

    Topics: Animals; Burimamide; Cimetidine; Dimaprit; Guinea Pigs; Histamine H2 Antagonists; Hydrogen-Ion Concentration; Metiamide; Molecular Conformation; Structure-Activity Relationship; Thiourea

1984
Reminiscences of the development of cimetidine.
    Gastroenterology, 1980, Volume: 78, Issue:3

    Topics: Burimamide; Cimetidine; Drug Industry; England; Guanidines; Histamine Antagonists; History, 20th Century

1980
Histamine binding to H2 receptors stimulates phospholipid methylation in mast cells.
    Experientia, 1982, Aug-15, Volume: 38, Issue:8

    Topics: Animals; Burimamide; Cimetidine; Histamine; Male; Mast Cells; Methylation; Phospholipids; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2

1982
The development of cimetidine: 1964-1976. A human story.
    Journal of clinical gastroenterology, 1994, Volume: 19, Issue:3

    Topics: Adult; Animals; Burimamide; Cimetidine; Dogs; Drug Industry; England; Histamine H2 Antagonists; History, 20th Century; Humans; Male; Metiamide; Peptic Ulcer; Research; United States

1994
Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Jun-25, Volume: 93, Issue:13

    Topics: Animals; Burimamide; CHO Cells; Cimetidine; Colforsin; Cricetinae; Cyclic AMP; Histamine Agonists; Histamine H2 Antagonists; Ranitidine; Receptors, Histamine H2; Transfection; Up-Regulation

1996
Constitutive activity and structural instability of the wild-type human H2 receptor.
    Journal of neurochemistry, 1998, Volume: 71, Issue:2

    Topics: Animals; Binding, Competitive; Burimamide; CHO Cells; Cimetidine; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Famotidine; Gene Expression; Histamine H2 Antagonists; Humans; Ranitidine; Receptors, Histamine H2; Up-Regulation

1998
Antinociceptive activity of derivatives of improgran and burimamide.
    Pharmacology, biochemistry, and behavior, 2000, Jan-01, Volume: 65, Issue:1

    Topics: Analgesics, Non-Narcotic; Animals; Burimamide; Cimetidine; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Structure-Activity Relationship

2000