cimetidine has been researched along with antipyrine in 74 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 47 (63.51) | 18.7374 |
1990's | 5 (6.76) | 18.2507 |
2000's | 12 (16.22) | 29.6817 |
2010's | 10 (13.51) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Blake, JF; Curatolo, WJ; Lombardo, F | 1 |
Artursson, P; Luthman, K; Norinder, U; Stenberg, P | 1 |
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA | 1 |
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL | 1 |
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY | 2 |
Artursson, P; Bergström, CA; Matsson, P; Nagahara, N; Norinder, U; Tavelin, S | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S | 1 |
Campillo, NE; Guerra, A; Páez, JA | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Avdeef, A; Tam, KY | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K | 1 |
Barber, S; Dew, TP; Farrell, TL; Poquet, L; Williamson, G | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Atwood, JL; Breckenridge, AM; Mossman, S; Serlin, MJ; Sibeon, RG; Williams, JR; Willoughby, JM | 1 |
Bianchetti, G; Desager, JP; Harvengt, C; Hulhoven, R | 1 |
Rieth, H; Sauerbrey, N | 1 |
Nakamura, K; Tanaka, E | 1 |
Desager, JP; Harvengt, C; Horsmans, Y; Leclercq, V; Van Nieuwenhuyze, Y | 1 |
Fribourg, HA; Heitmann, RN; McLaren, JB; Zanzalari, KP | 1 |
Breimer, DD; Brugman, M; Schellens, JH; van der Wart, JH | 1 |
Akamatsu, K; Hirabayashi, Y; Kanaoka, M; Masumoto, S; Nakanishi, K; Nishinobu, M; Ohta, Y; Okada, S; Sakaue, H; Sasaki, T | 1 |
Dicke, JM; Henderson, GI; Johnson, RF; Kuehl, TJ; Schenker, S | 1 |
Kuroiwa, Y; Misawa, S; Nakamura, K; Tanaka, E | 1 |
Crewe, HK; Lennard, MS; Tucker, GT; Woods, HF | 1 |
Larsson, H; Lorentzon, P; Wallmark, B | 1 |
Back, DJ; Mönig, H; Ohnhaus, EE; Park, BK; Tjia, J | 1 |
Eksymä, S; Gachalyi, B; Hämäläinen, A; Lahtela, JT; Sotaniemi, EA | 1 |
Csillag, K; Gachályi, B; Káldor, A; Kocsis, F; Nagy, B; Vas, A | 2 |
Døssing, M; Jørgensen, BG; Loft, S; Petersen, KT; Poulsen, HE; Sonne, J | 1 |
Døssing, M; Loft, S; Pilsgaard, H; Poulsen, HE; Rasmussen, B; Sonne, J | 1 |
Ching, MS; Date, NM; Hardy, KJ; Mihaly, GW; Morgan, DJ; Smallwood, RA | 1 |
Desager, JP; Dumont, E; Harvengt, C | 1 |
Adamska-Dyniewska, I; Chojnacki, J; Jabłkowski, M; Tkaczewski, W | 1 |
Døssing, M; Loft, S; Pilsgaard, H; Poulsen, E; Sonne, J | 1 |
Breckenridge, AM; Edwards, G; Mihaly, GW; Nicholl, DD; Ward, SA | 1 |
Banditt, P; Kettner, W; Schröter, U; Walther, H | 1 |
Breimer, DD; de Leede, LG; Kleinbloesem, CH; Teunissen, MW | 1 |
Aarons, L; Adedoyin, A; Houston, JB | 1 |
Bell, GD; Henry, DA; Kitchingman, G; Langman, MJ; Macdonald, IA | 1 |
Henry, DA; Langman, MJ | 1 |
Breen, KJ; Bury, R; Desmond, PV; Mashford, ML; Morphett, B; Shaw, RG; Westwood, B | 1 |
Jones, DB; Smallwood, RA; Webster, LK | 1 |
Dammann, HG; DeVries, JX; Koroknay, B; Müller, P; Simon, B; Staiger, C; Weber, E | 1 |
Agnew, E; Brodie, MJ; Macphee, GJ; McColl, KE; Murray, T; Park, BK; Scobie, G; Thompson, GG | 1 |
Hall, ST; Houston, JB; Rhodes, JC | 1 |
de Vries, J; Staiger, C; Wang, NS; Weber, E | 1 |
Døssing, M; Pilsgaard, H; Poulsen, HE; Rasmussen, B | 1 |
Foote, SE; Paton, DM; Paxton, JW | 1 |
Feely, J; Guy, E; Hockings, N; Pereira, L | 1 |
Daneshmend, TK; Ene, MD; Parker, G; Roberts, CJ | 1 |
Slusher, LB; Vesell, ES | 1 |
Dammann, HG; Devries, JX; Korodnay, B; Müller, P; Simon, B; Staiger, C; Weber, E | 1 |
Klotz, U; Reimann, I | 1 |
Abernethy, DR; Divoll, M; Greenblatt, DJ; Shader, RI | 1 |
Abernethy, DR; Ameer, B; Divoll, M; Greenblatt, DJ; Shader, RI | 1 |
Bradbear, RA; Grice, J; O'Toole, J; Roberts, RK; Shepherd, RW | 1 |
Grice, J; McGuffie, C; Petroff, V; Roberts, RK; Wood, L | 1 |
Kaste, M; Neuvonen, PJ; Tokola, RA | 1 |
Pelkonen, O; Puurunen, J; Sotaniemi, E | 1 |
Bassily, M; Ghabrial, H; Morgan, DJ; Smallwood, RA | 1 |
Janus, K; Suszycka, J | 1 |
Berry, MN; Efthivoulou, MA | 1 |
Bauman, JH; Fuentes, RJ | 1 |
Ekblad, U; Heikkinen, T; Laine, K; Rahi, M; Rönnemaa, T; Tertti, K | 1 |
9 trial(s) available for cimetidine and antipyrine
Article | Year |
---|---|
Cimetidine: interaction with oral anticoagulants in man.
Topics: Acenocoumarol; Administration, Oral; Adult; Aged; Antipyrine; Biological Availability; Cimetidine; Clinical Trials as Topic; Drug Synergism; Female; Guanidines; Half-Life; Humans; Male; Middle Aged; Phenindione; Prothrombin Time; Warfarin | 1979 |
Effect of cimetidine on the pharmacodynamics, pharmacokinetics and biotransformation of a single oral dose of alpidem.
Topics: Administration, Oral; Adult; Anti-Anxiety Agents; Antipyrine; Biotransformation; Cimetidine; Drug Interactions; Female; Humans; Imidazoles; Liver; Male; Mixed Function Oxygenases; Psychometrics; Pyridines | 1990 |
[Interaction studies with fluconazole, a new triazole antifungal drug].
Topics: Adult; Antipyrine; Cimetidine; Clinical Trials as Topic; Contraceptives, Oral; Cyclosporins; Double-Blind Method; Drug Interactions; Female; Fluconazole; Humans; Male; Testosterone; Tolbutamide; Warfarin | 1989 |
The effect of roxatidine acetate and cimetidine on hepatic drug clearance assessed by simultaneous administration of three model substrates.
Topics: Adult; Antipyrine; Cimetidine; Half-Life; Histamine H2 Antagonists; Humans; Indocyanine Green; Liver; Male; Pharmaceutical Preparations; Piperidines; Trimethadione | 1989 |
The effect of liver microsomal enzyme inducing and inhibiting drugs on insulin mediated glucose metabolism in man.
Topics: Adult; Antipyrine; Benzhydryl Compounds; Cimetidine; Enzyme Induction; Enzyme Inhibitors; Female; Glucose; Humans; Insulin; Kinetics; Male; Microsomes, Liver; Phenobarbital | 1986 |
[The acetylator phenotype affects the antipyrine metabolism inhibiting action of cimetidine].
Topics: Acetylation; Antipyrine; Cimetidine; Clinical Trials as Topic; Drug Evaluation; Female; Humans; Male; Middle Aged; Peptic Ulcer; Phenotype | 1986 |
Cimetidine and ranitidine: comparison of effects on hepatic drug metabolism.
Topics: Aminopyrine; Antipyrine; Cimetidine; Furans; Guanidines; Half-Life; Histamine H2 Antagonists; Humans; Microsomes, Liver; Ranitidine | 1980 |
[Comparative study of the effect of famotidine and cimetidine on antipyrine pharmacokinetics in the human].
Topics: Adult; Antipyrine; Cimetidine; Famotidine; Female; Histamine H1 Antagonists; Humans; Kinetics; Male; Thiazoles | 1984 |
[Effect of metronidazole on phenazone metabolism].
Topics: Adult; Antipyrine; Cimetidine; Drug Interactions; Female; Humans; Hydroxylation; Kinetics; Male; Metronidazole; Time Factors | 1984 |
65 other study(ies) available for cimetidine and antipyrine
Article | Year |
---|---|
Computation of brain-blood partitioning of organic solutes via free energy calculations.
Topics: Animals; Blood-Brain Barrier; Brain; Cattle; Cells, Cultured; Endothelium, Vascular; Membrane Lipids; Microcirculation; Molecular Conformation; Molecular Structure; Monte Carlo Method; Permeability; Pharmaceutical Preparations; Software; Solubility; Thermodynamics | 1996 |
Experimental and computational screening models for the prediction of intestinal drug absorption.
Topics: Biological Transport; Carbon Radioisotopes; Cell Line; Cell Membrane; Cell Membrane Permeability; Ciprofloxacin; Computational Biology; Drug Design; Foscarnet; Humans; Hydrogen Bonding; Intestinal Absorption; Intestinal Mucosa; Lactulose; Mannitol; Models, Biological; Raffinose; Surface Properties; Tritium; Verapamil | 2001 |
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water | 2001 |
Cheminformatic models to predict binding affinities to human serum albumin.
Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids | 2001 |
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding | 2002 |
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution | 2004 |
Exploring the role of different drug transport routes in permeability screening.
Topics: Administration, Oral; Biological Transport; Caco-2 Cells; Cell Line; Humans; Intestinal Absorption; Intestinal Mucosa; Intestine, Small; Membranes, Artificial; Models, Biological; Molecular Conformation; Monte Carlo Method; Permeability; Pharmaceutical Preparations; Pharmacokinetics | 2005 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship | 2008 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship | 2009 |
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
QSAR-based permeability model for drug-like compounds.
Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2011 |
Predicting phenolic acid absorption in Caco-2 cells: a theoretical permeability model and mechanistic study.
Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Cinnamates; Enterocytes; Humans; Hydrophobic and Hydrophilic Interactions; Intestinal Absorption; Kinetics; Models, Biological; Molecular Conformation; Osmolar Concentration; Phenols | 2012 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity | 2013 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Influence of rifampicin, phenobarbital and cimetidine on mixed function monooxygenase in extensive and poor metabolizers of debrisoquine.
Topics: Adult; Antipyrine; Biotransformation; Cimetidine; Debrisoquin; Half-Life; Humans; Hydroxylation; Isoquinolines; Male; Mixed Function Oxygenases; Phenobarbital; Phenotype; Rifampin | 1989 |
Effects of endophyte-infected fescue and cimetidine on respiration rates, rectal temperatures and hepatic mixed function oxidase activity as measured by hepatic antipyrine metabolism in sheep.
Topics: Alkaloids; Animal Feed; Animals; Antipyrine; Blood Flow Velocity; Body Temperature; Cimetidine; Female; Food Contamination; Liver; Mixed Function Oxygenases; Respiration; Sheep | 1989 |
Influence of enzyme induction and inhibition on the oxidation of nifedipine, sparteine, mephenytoin and antipyrine in humans as assessed by a "cocktail" study design.
Topics: Adult; Antipyrine; Cimetidine; Enzyme Induction; Female; Humans; Hydantoins; Male; Mephenytoin; Metabolic Clearance Rate; Nifedipine; Oxidation-Reduction; Phenobarbital; Smoking; Sparteine | 1989 |
Effects of prolonged oral cimetidine, ranitidine, and famotidine therapy on antipyrine elimination.
Topics: Administration, Oral; Adolescent; Adult; Aged; Antipyrine; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Liver; Male; Metabolic Clearance Rate; Middle Aged; Ranitidine; Thiazoles | 1987 |
A comparative evaluation of the transport of H2-receptor antagonists by the human and baboon placenta.
Topics: Adolescent; Adult; Animals; Antipyrine; Biological Transport; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; In Vitro Techniques; Maternal-Fetal Exchange; Nizatidine; Papio; Perfusion; Placenta; Pregnancy; Ranitidine; Thiazoles | 1988 |
The effect of H2-receptor antagonists on antipyrine and pentobarbital metabolism in male and female rats.
Topics: Animals; Antipyrine; Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Male; Microsomes, Liver; Mixed Function Oxygenases; Pentobarbital; Ranitidine; Rats; Rats, Inbred Strains; Sex Factors; Thiazoles | 1988 |
Metoprolol oxidation by rat liver microsomes. Inhibition by debrisoquine and other drugs.
Topics: Animals; Antipyrine; Cimetidine; Debrisoquin; Guanidines; Isoquinolines; Metoprolol; Microsomes, Liver; Ranitidine; Rats; Rats, Inbred Strains | 1986 |
The mechanism of action of omeprazole--a survey of its inhibitory actions in vitro.
Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Antipyrine; Benzimidazoles; Bucladesine; Cimetidine; Gastric Acid; Gastric Mucosa; Guinea Pigs; Histamine; Male; Omeprazole; Parietal Cells, Gastric; Sodium-Potassium-Exchanging ATPase; Stomach; Swine | 1985 |
Selective inhibition of drug oxidation after simultaneous administration of two probe drugs, antipyrine and tolbutamide.
Topics: Adult; Antipyrine; Cimetidine; Female; Half-Life; Humans; Male; Oxidation-Reduction; Pharmaceutical Preparations; Primaquine; Sulfaphenazole; Tolbutamide | 1988 |
Inhibition and induction of metronidazole and antipyrine metabolism.
Topics: Adult; Antipyrine; Cimetidine; Drug Interactions; Female; Humans; Hydroxylation; Kinetics; Male; Metronidazole; Phenobarbital | 1987 |
Effect of concomitant administration of cimetidine and phenobarbital on antipyrine elimination and metabolite formation.
Topics: Adult; Antipyrine; Biotransformation; Cimetidine; Female; Humans; Male; Phenobarbital | 1987 |
Low clearance of cimetidine across the human placenta.
Topics: Antipyrine; Cimetidine; Female; Humans; Leucine; Maternal-Fetal Exchange; Mathematics; Metabolic Clearance Rate; Placenta; Pregnancy | 1987 |
The urinary 6 beta-hydroxycortisol excretion in man on inducers and inhibitors of the hepatic mixed function oxidase.
Topics: Antipyrine; Cimetidine; Enzyme Induction; Humans; Hydrocortisone; Liver; Mixed Function Oxygenases | 1987 |
[Effect of combined therapy with cimetidine and (+)-cyanidanol-3 on the hepatic clearance of antipyrine].
Topics: Adolescent; Adult; Antipyrine; Catechin; Cimetidine; Drug Therapy, Combination; Female; Humans; Liver; Male; Metabolic Clearance Rate; Middle Aged; Peptic Ulcer | 1986 |
Pharmacogenetic differences in the inhibitory effect of cimetidine on the metabolism of antipyrine.
Topics: Acetylation; Adult; Antipyrine; Cimetidine; Edaravone; Female; Glucaric Acid; Humans; Male; Metabolic Clearance Rate; Microsomes, Liver; Middle Aged; Pharmacogenetics; Phenotype | 1987 |
Inhibition of antipyrine elimination by disulfiram and cimetidine: the effect of concomitant administration.
Topics: Adult; Antipyrine; Cimetidine; Depression, Chemical; Disulfiram; Drug Interactions; Female; Humans; Liver; Male; Time Factors | 1986 |
The effects of primaquine stereoisomers and metabolites on drug metabolism in the isolated perfused rat liver and in vitro rat liver microsomes.
Topics: Animals; Antipyrine; Cimetidine; Depression, Chemical; Drug Interactions; Kinetics; Liver; Male; Microsomes, Liver; Mixed Function Oxygenases; Perfusion; Primaquine; Rats; Rats, Inbred Strains; Stereoisomerism | 1985 |
[Effect of histamine H2 receptor blockers on hepatic elimination of drugs].
Topics: Adult; Antipyrine; Cimetidine; Half-Life; Humans; Liver; Male; Metabolic Clearance Rate; Peptic Ulcer | 1985 |
Influence of cimetidine on steady state concentration and metabolite formation from antipyrine infused with a rectal osmotic mini pump.
Topics: Adult; Antipyrine; Biotransformation; Cimetidine; Drug Interactions; Humans; Intestinal Absorption; Male; Metabolic Clearance Rate; Perfusion; Rectum; Saliva | 1985 |
High-performance liquid chromatographic method for the simultaneous determination of cimetidine and antipyrine in plasma.
Topics: Animals; Antipyrine; Chromatography, High Pressure Liquid; Cimetidine; Indicators and Reagents; Kinetics; Rats | 1985 |
The effects of H2 receptor antagonists on hepatic drug metabolism.
Topics: Adult; Aminopyrine; Antipyrine; Breath Tests; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Liver; Middle Aged; Ranitidine; Structure-Activity Relationship | 1981 |
Effects of cimetidine and ranitidine on hepatic drug metabolism.
Topics: Adult; Antipyrine; Cimetidine; Drug Interactions; Female; Furans; Guanidines; Half-Life; Histamine H2 Antagonists; Humans; Liver; Male; Mixed Function Oxygenases; Ranitidine; Theophylline | 1982 |
How potent is the inhibition of drug metabolism by omeprazole?
Topics: Animals; Antipyrine; Benzimidazoles; Cimetidine; Drug Interactions; Half-Life; Humans; Liver; Omeprazole; Pharmaceutical Preparations; Rats | 1984 |
Effects of cimetidine on carbamazepine auto- and hetero-induction in man.
Topics: 5-Aminolevulinate Synthetase; Adult; Antipyrine; Carbamazepine; Cimetidine; Half-Life; Humans; Leukocytes; Male; Time Factors | 1984 |
Inhibition of antipyrine metabolite formation in rats in vivo.
Topics: Animals; Antipyrine; Benzoflavones; Cimetidine; Cytochrome P-450 Enzyme System; Male; Metyrapone; Proadifen; Rats; Rats, Inbred Strains | 1984 |
Time course of phenobarbital and cimetidine mediated changes in hepatic drug metabolism.
Topics: Adult; Aminopyrine; Antipyrine; Biotransformation; Breath Tests; Cimetidine; Female; Half-Life; Humans; Liver; Male; Phenobarbital | 1983 |
No impairment of antipyrine elimination by the selective anticholinergic drug pirenzepine.
Topics: Adult; Anti-Ulcer Agents; Antipyrine; Benzodiazepinones; Cimetidine; Drug Interactions; Half-Life; Humans; Liver; Male; Mixed Function Oxygenases; Parasympatholytics; Pirenzepine | 1983 |
Factors affecting the response to inhibition of drug metabolism by cimetidine--dose response and sensitivity of elderly and induced subjects.
Topics: Adult; Aged; Aging; Antipyrine; Cimetidine; Dose-Response Relationship, Drug; Female; Humans; Male; Random Allocation; Rifampin; Saliva | 1984 |
Effects of chronic oral cimetidine on apparent liver blood flow and hepatic microsomal enzyme activity in man.
Topics: Adult; Antipyrine; Cimetidine; Female; Humans; Indocyanine Green; Kinetics; Liver Circulation; Male; Metabolic Clearance Rate; Microsomes, Liver; Middle Aged | 1984 |
Cimetidine-induced reduction in gastrointestinal absorption of antipyrine and rate constants for formation of its metabolites.
Topics: Adult; Antipyrine; Cimetidine; Drug Interactions; Humans; Intestinal Absorption; Kinetics; Male | 1984 |
Comparative effects of famotidine and cimetidine on antipyrine kinetics in healthy volunteers.
Topics: Adult; Antipyrine; Cimetidine; Famotidine; Female; Humans; Kinetics; Male; Thiazoles | 1984 |
Delayed clearance of diazepam due to cimetidine.
Topics: Adult; Antipyrine; Cimetidine; Diazepam; Drug Interactions; Drug Synergism; Female; Guanidines; Half-Life; Humans; Kinetics; Male; Nordazepam | 1980 |
Cimetidine impairs clearance of antipyrine and desmethyldiazepam in the elderly.
Topics: Adult; Aged; Antipyrine; Cimetidine; Clorazepate Dipotassium; Guanidines; Humans; Metabolic Clearance Rate; Middle Aged; Nordazepam | 1982 |
Differential effect of cimetidine on drug oxidation (antipyrine and diazepam) vs. conjugation (acetaminophen and lorazepam): prevention of acetaminophen toxicity by cimetidine.
Topics: Acetaminophen; Adult; Animals; Antipyrine; Biotransformation; Cimetidine; Diazepam; Guanidines; Humans; Kinetics; Lethal Dose 50; Lorazepam; Male; Mice; Oxidation-Reduction | 1983 |
Cimetidine use in children with cystic fibrosis: inhibition of hepatic drug metabolism.
Topics: Adolescent; Antipyrine; Child; Chromatography, High Pressure Liquid; Cimetidine; Guanidines; Humans; Liver; Saliva | 1982 |
Cimetidine impairs the elimination of theophylline and antipyrine.
Topics: Adult; Antipyrine; Cimetidine; Drug Synergism; Female; Guanidines; Humans; Kinetics; Male; Middle Aged; Theophylline | 1981 |
Cimetidine-phenytoin interaction: effect on serum phenytoin concentration and antipyrine test.
Topics: Adult; Aged; Antipyrine; Cimetidine; Drug Interactions; Female; Guanidines; Humans; Kinetics; Male; Middle Aged; Phenytoin; Prospective Studies | 1981 |
Effect of cimetidine on microsomal drug metabolism in man.
Topics: Adult; Antipyrine; Benzopyrene Hydroxylase; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Drug Interactions; Guanidines; Humans; In Vitro Techniques; Metabolic Clearance Rate; Microsomes; Microsomes, Liver; Pharmaceutical Preparations | 1980 |
Determinants of placental drug transfer: studies in the isolated perfused human placenta.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Antipyrine; Cimetidine; Diclofenac; Female; Histamine H2 Antagonists; Humans; In Vitro Techniques; Maternal-Fetal Exchange; Models, Biological; Perfusion; Placenta; Pregnancy | 1995 |
The effect of cimetidine on antipyrine metabolism in calves.
Topics: Administration, Oral; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Antipyrine; Cattle; Chromatography, High Pressure Liquid; Cimetidine; Drug Interactions; Edaravone; Female; Free Radical Scavengers; Histamine H2 Antagonists; Software | 1997 |
Antipyrine and aminopyrine induce acetaldehyde accumulation from ethanol in isolated hepatocytes.
Topics: Acetaldehyde; Aldehyde Dehydrogenase; Aminopyrine; Animals; Antipyrine; Cells, Cultured; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Ethanol; Liver; Male; Mitochondria, Liver; Oxidation-Reduction; Rats; Rats, Wistar | 1997 |
Cimetidine impairs the elimination of theophylline and antipyrine.
Topics: Antipyrine; Biotransformation; Bronchodilator Agents; Cimetidine; Drug Interactions; Enzyme Inhibitors; Humans; Theophylline | 1982 |
The role of organic cation transporters (OCTs) in the transfer of metformin in the dually perfused human placenta.
Topics: Antipyrine; Biological Transport, Active; Cimetidine; Female; Humans; Maternal-Fetal Exchange; Metformin; Organic Cation Transport Proteins; Perfusion; Placenta; Pregnancy | 2010 |