cimetidine and alpha-methylhistamine

cimetidine has been researched along with alpha-methylhistamine in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's16 (64.00)18.2507
2000's8 (32.00)29.6817
2010's1 (4.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arrang, JM; de Waele, C; Khateb, A; Mulhethaler, M; Serafin, M; Vibert, N; Vidal, PP; Yabe, T1
Anjelkovic, IZ; Collis, CS; Djuric, D; Rosic, M; Segal, MB; Zlokovic, BV1
Bent, S; Braam, U; Fehling, U; Schmutzler, W; Schunack, W1
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H1
Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Hey, JA; Hutchison, RW1
Gertner, SB; Hey, JA; McLeod, RL1
Garbarg, M; Kjaer, A; Knigge, U; Rouleau, A; Warberg, J1
Koss, MC1
Kamei, C; Tasaka, K1
Bach, FW; Kjaer, A; Knigge, U; Madsen, EL; Søe-Jensen, P; Warberg, J1
Assenmacher, I; Barbanel, G; Givalois, L; Ixart, G; Malaval, F; Mekaouche, M; Siaud, P1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Hough, LB; Li, BY; Nalwalk, JW1
Gao, C; Hu, Hz; Liu, S; Ren, J; Wood, JD; Xia, Y1
Anichtchik, OV; Panula, P; Peitsaro, N1
Hidaka, Y; Itadani, H; Nakamura, T; Ohta, M; Tanaka, K1
Kawarai, M; Koss, MC; Yu, Y1
Anai, M; Asano, T; Fukushima, Y; Ishikawa, M; Ishikawa, T; Kajiwara, T; Katsube, T; Mori, H; Ogawa, K; Ohkawa, S; Omata, M; Otsuka, H; Saitoh, T; Takahashi, H; Tamai, M1
Fogel, WA; Stasiak, A; Wagner, W1
Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW1
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1

Reviews

1 review(s) available for cimetidine and alpha-methylhistamine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

24 other study(ies) available for cimetidine and alpha-methylhistamine

ArticleYear
An in vivo and in vitro study of the vestibular nuclei histaminergic receptors in the guinea pig.
    Annals of the New York Academy of Sciences, 1992, May-22, Volume: 656

    Topics: Animals; Brain Stem; Cimetidine; Electric Stimulation; Eye Movements; Guanidines; Guinea Pigs; Head; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Piperidines; Receptors, Histamine; Receptors, Histamine H2; Reflex, Vestibulo-Ocular; Rotation; Vestibular Nuclei

1992
The effects of (R) alpha-methyl histamine on the isolated guinea pig aorta.
    Agents and actions. Supplements, 1991, Volume: 33

    Topics: Animals; Aorta; Cimetidine; Female; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; Imidazoles; Impromidine; Male; Methylhistamines; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H3; Vasoconstriction; Vasodilation

1991
The influence of H1-, H2- and H3-receptors on the spontaneous and ConA induced histamine release from human adenoidal mast cells.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenoids; Cimetidine; Concanavalin A; Guanidines; Histamine Antagonists; Humans; Hydroxyzine; Imidazoles; Impromidine; Mast Cells; Meclizine; Methylhistamines; Piperidines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3

1991
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:2

    Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1994
R-alpha-methylhistamine-induced inhibition of gastric acid secretion in pylorus-ligated rats via central histamine H3 receptors.
    British journal of pharmacology, 1995, Volume: 115, Issue:7

    Topics: Animals; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; Injections, Intraventricular; Methylhistamines; Piperidines; Pylorus; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1995
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Pharmacological characterization of the inhibitory effect of (R)-alpha-methylhistamine on sympathetic cardiopressor responses in the pithed guinea-pig.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:6

    Topics: Adrenalectomy; Animals; Blood Pressure; Chlorpheniramine; Cimetidine; Drug Interactions; Electric Stimulation; Epinephrine; Guinea Pigs; Heart; Heart Rate; Histamine Agonists; Male; Methylhistamines; Piperidines; Prazosin; Spinal Cord; Sympathetic Nervous System; Vagotomy; Yohimbine

1994
Species differences in the cardiovascular responses to histamine H3 receptor activation.
    European journal of pharmacology, 1994, Jul-01, Volume: 259, Issue:2

    Topics: Animals; Blood Pressure; Cimetidine; Guinea Pigs; Heart Rate; Hemodynamics; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Piperidines; Rabbits; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Receptors, Histamine H3; Species Specificity

1994
Dehydration-induced release of vasopressin involves activation of hypothalamic histaminergic neurons.
    Endocrinology, 1994, Volume: 135, Issue:2

    Topics: Animals; Arginine Vasopressin; Blood; Cimetidine; Dehydration; Histamine; Hypothalamus; Male; Methylhistamines; Methylhistidines; Neurons; Osmolar Concentration; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2

1994
Histamine H3 receptor activation inhibits sympathetic-cholinergic responses in cats.
    European journal of pharmacology, 1994, May-12, Volume: 257, Issue:1-2

    Topics: Animals; Cats; Chlorpheniramine; Cimetidine; Electric Stimulation; Female; Histamine Agonists; Male; Methacholine Chloride; Methylhistamines; Parasympathetic Nervous System; Piperidines; Receptors, Histamine H3; Skin; Sympathetic Nervous System

1994
Effect of histamine on memory retrieval in old rats.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:2

    Topics: Acetylcholine; Aging; Animals; Anticonvulsants; Avoidance Learning; Cerebrovascular Circulation; Cimetidine; Dose-Response Relationship, Drug; Exploratory Behavior; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Motor Activity; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Insulin/hypoglycemia-induced adrenocorticotropin and beta-endorphin release: involvement of hypothalamic histaminergic neurons.
    Endocrinology, 1993, Volume: 132, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Cetirizine; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Hypoglycemia; Hypothalamus; Insulin; Male; Methylhistamines; Neurons; Pyrilamine; Pyrimidinones; Rats; Rats, Wistar

1993
Involvement of central histamine in the early phase of ACTH and corticosterone responses to endotoxin in rats.
    Neuroendocrinology, 1996, Volume: 63, Issue:3

    Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Corticosterone; Escherichia coli; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Kinetics; Lipopolysaccharides; Male; Median Eminence; Methylhistamines; Pyrilamine; Rats; Rats, Sprague-Dawley

1996
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Effects of naltrexone and histamine antagonists on the antinociceptive activity of the cimetidine analog SKF92374 in rats.
    Brain research, 1997, Feb-14, Volume: 748, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Animals; Cimetidine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Naltrexone; Narcotic Antagonists; Nociceptors; Piperidines; Rats; Rats, Sprague-Dawley; Stereoisomerism

1997
Histamine H3 receptor-mediated suppression of inhibitory synaptic transmission in the submucous plexus of guinea-pig small intestine.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Male; Methylhistamines; Norepinephrine; Phentolamine; Piperidines; Receptors, Histamine H3; Submucous Plexus; Synaptic Transmission

2000
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish

2000
Molecular cloning and characterization of a new human histamine receptor, HH4R.
    Biochemical and biophysical research communications, 2000, Dec-20, Volume: 279, Issue:2

    Topics: Amino Acid Sequence; Binding, Competitive; Cell Line; Cimetidine; Cloning, Molecular; Colforsin; Cyclic AMP; Histamine Agonists; Histamine Antagonists; Humans; Leukocytes; Methylhistamines; Molecular Sequence Data; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Stereoisomerism; Transfection

2000
Histamine H3 receptor-mediated inhibition of sympathetically evoked mydriasis in rats.
    European journal of pharmacology, 2001, May-04, Volume: 419, Issue:1

    Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Methylhistamines; Mydriasis; Pupil; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Thiourea

2001
Effects of N-alpha-methyl-histamine on human H(2) receptors expressed in CHO cells.
    Gut, 2002, Volume: 50, Issue:6

    Topics: Animals; CHO Cells; Cimetidine; Cricetinae; Cyclic AMP; Famotidine; Female; Histamine Agonists; Histamine Antagonists; Histamine H2 Antagonists; Methylhistamines; Ovary; Piperidines; Receptors, Histamine H2; Receptors, Histamine H3

2002
Mouse mammary epithelial cells bear histamine receptors.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2002, Volume: 51 Suppl 1

    Topics: Animals; Binding Sites; Cimetidine; Epithelial Cells; Female; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Mammary Glands, Animal; Methylhistamines; Mice; Mice, Inbred BALB C; Pyrilamine; Radiopharmaceuticals; Receptors, Histamine

2002
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4

2002
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010