cimetidine and 4-methylhistamine

cimetidine has been researched along with 4-methylhistamine in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199014 (51.85)18.7374
1990's8 (29.63)18.2507
2000's3 (11.11)29.6817
2010's1 (3.70)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Nowak, JZ; Sek, B1
Bugajski, J; Gadek-Michalska, A1
Cortijo, J; Esplugues, J; Morcillo, EJ; Orón, JD; Ortiz, JL; Perpiñá, M; Sanz, C1
Adaikan, PG; Lau, LC; Ratnam, SS1
Knigge, U; Matzen, S; Warberg, J1
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I1
Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Tang, ZC; Xu, YH1
Kannisto, P; Owman, C; Schmidt, G; Sjöberg, NO1
Adachi, K; Aoyagi, T; Halprin, KM; Levine, V; Woodyard, CW1
Robichaud, L; Schwender, CF; Tecle, H1
Tomioka, K; Yamada, T1
Bugajski, J; Gadek, A1
Brink, C; Douglas, JS; Duncan, PG1
Kamei, C; Tasaka, K; Tsujimoto, S; Yoshida, T1
Banchelli, G; Buffoni, F; Conforti, L; Ignesti, G; Pirisino, R; Raimondi, L1
Fukuda, K; Matsumura, F; Tanaka, S1
Alemany, G; López-García, JA; Nicolau, MC; Planas, B; Ramis, C; Rial, R1
KAMEI, CH1
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E1
Abe, T; Kamei, C; Mio, M; Shimada, K; Zhao, Q1
Belon, P; Sainte-Laudy, J1
Dartt, DA; Hayashi, C; Hayashi, D; Hodges, RR; Li, D; Shatos, M1
Keuschler, J; Kržan, M; Mavri, J; Vianello, R1

Reviews

1 review(s) available for cimetidine and 4-methylhistamine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

26 other study(ies) available for cimetidine and 4-methylhistamine

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Responses to histamine and selective H2-receptor agonists in lung parenchymal strips from normal and sensitized guinea-pigs.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Animals; Benzimidazoles; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; Isoproterenol; Lung; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine H2; Thiourea

1989
Effect of histamine on human vas deferens in vitro.
    British journal of urology, 1989, Volume: 64, Issue:4

    Topics: Burimamide; Cimetidine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Humans; Male; Methylhistamines; Muscle Contraction; Pyrilamine; Vas Deferens

1989
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
    Acta endocrinologica, 1988, Volume: 119, Issue:4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea

1988
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
    International archives of allergy and applied immunology, 1986, Volume: 79, Issue:3

    Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Comparison of the effects of 4-methylhistamine on the cell-cycle response between CFU-s and its subpopulation.
    International journal of cell cloning, 1987, Volume: 5, Issue:6

    Topics: Animals; Bone Marrow; Bone Marrow Cells; Cell Cycle; Cell Survival; Cells, Cultured; Cimetidine; Colony-Forming Units Assay; Female; Hematopoietic Stem Cells; Hydroxyurea; Male; Methylhistamines; Mice; Mice, Inbred Strains; Spleen

1987
Alteration by histamine of the sympathetic nerve-mediated contractions in the bovine ovarian follicle wall in vitro.
    European journal of pharmacology, 1987, Mar-03, Volume: 135, Issue:1

    Topics: Animals; Cattle; Cimetidine; Electrolytes; Female; Glucose; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Norepinephrine; Ovary; Proteins; Pyrilamine; Sympathetic Nervous System

1987
The effect of histamine on epidermal outgrowth: its possible dual role as an inhibitor and stimulator.
    The Journal of investigative dermatology, 1981, Volume: 76, Issue:1

    Topics: Animals; Cells, Cultured; Cimetidine; Cyclic AMP; Cyclic GMP; Epidermis; Epinephrine; Histamine; Histamine H1 Antagonists; Methylhistamines; Swine

1981
Potential histamine H2-receptor blockers. 3- and 2-indole derivatives as immobile analogues of tautomeric forms of cimetidine.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:9

    Topics: Animals; Chemical Phenomena; Chemistry; Cimetidine; Guanidines; Guinea Pigs; Heart Rate; Histamine H2 Antagonists; Indoles; Male; Methylhistamines; Stereoisomerism

1981
Effects of histamine H2-receptor agonists and antagonists on isolated guinea-pig airway muscles.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 255, Issue:1

    Topics: Airway Resistance; Animals; Cimetidine; Dimaprit; Drug Interactions; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1982
Effect of intracerebroventricular impromidine on pituitary-adrenocortical response to stress in rats.
    Agents and actions, 1984, Volume: 14, Issue:5-6

    Topics: Adrenal Cortex; Animals; Atropine; Cimetidine; Corticosterone; Dimaprit; Imidazoles; Impromidine; Injections, Intraventricular; Male; Methylhistamines; Pituitary Gland; Propranolol; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Sympatholytics; Thiourea

1984
Changes in the response of guinea-pig airways in vivo and in vitro to cimetidine and propranolol during development.
    British journal of pharmacology, 1982, Volume: 75, Issue:3

    Topics: Aging; Airway Resistance; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Propranolol; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1982
Changes in plasma adrenocorticotropic hormone and cortisol levels induced by intracerebroventricular injection of histamine and its related compounds in dogs.
    Pharmacology, 1993, Volume: 47, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Dogs; Hexamethonium; Hexamethonium Compounds; Histamine; Hydrocortisone; Hypophysectomy; Injections, Intraventricular; Male; Methylhistamines; Pyrilamine

1993
Histamine lipolytic activity and semicarbazide-sensitive amine oxidase (SSAO) of rat white adipose tissue (WAT).
    Biochemical pharmacology, 1993, Oct-19, Volume: 46, Issue:8

    Topics: Adipose Tissue; Amine Oxidase (Copper-Containing); Animals; Benzylamines; Cimetidine; Histamine; Isoproterenol; Kinetics; Lipolysis; Male; Methylhistamines; Pyrilamine; Rats; Rats, Wistar; Semicarbazides

1993
Histamine H2 receptor mediates keratan sulfate secretion in rabbit chondrocytes: role of cAMP.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Animals; Bucladesine; Cartilage, Articular; Cells, Cultured; Cholera Toxin; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dinoprostone; Enzyme-Linked Immunosorbent Assay; Keratan Sulfate; Kinetics; Methylhistamines; Parathyroid Hormone; Proteoglycans; Rabbits; Receptors, Histamine H2; Sulfates; Sulfur Radioisotopes

1993
Histaminergic drugs in the rat caudate nucleus: effects on learned helplessness.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:2

    Topics: Animals; Astemizole; Caudate Nucleus; Cimetidine; Helplessness, Learned; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles

1993
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:4

    Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P

1996
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
    Endocrinology, 1999, Volume: 140, Issue:8

    Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea

1999
Effects of histamine and related compounds on the differentiation of HL-60-Eo cells into eosinophils.
    Methods and findings in experimental and clinical pharmacology, 2001, Volume: 23, Issue:7

    Topics: Cell Differentiation; Cell Division; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Eosinophils; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; HL-60 Cells; Humans; Impromidine; Methylhistamines; Ranitidine; Receptors, Histamine H2; Thymidine; Time Factors; Tritium

2001
Inhibition of basophil activation by histamine: a sensitive and reproducible model for the study of the biological activity of high dilutions.
    Homeopathy : the journal of the Faculty of Homeopathy, 2009, Volume: 98, Issue:4

    Topics: Alcian Blue; Animals; Antigens, CD; Basophils; Cimetidine; Coloring Agents; Enzyme Inhibitors; Flow Cytometry; Histamine; Histamine Agonists; Histamine H2 Antagonists; Histidine; Humans; Methylhistamines; Mice; Platelet Membrane Glycoproteins; Staining and Labeling; Tetraspanin 30

2009
Role of histamine and its receptor subtypes in stimulation of conjunctival goblet cell secretion.
    Investigative ophthalmology & visual science, 2012, May-17, Volume: 53, Issue:6

    Topics: Animals; Blotting, Western; Cells, Cultured; Cimetidine; Conjunctiva; Conjunctivitis, Allergic; Dose-Response Relationship, Drug; Fluorescent Antibody Technique; Goblet Cells; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Indoles; Male; Methylhistamines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles

2012
Relevance of Hydrogen Bonds for the Histamine H2 Receptor-Ligand Interactions: A Lesson from Deuteration.
    Biomolecules, 2020, 01-29, Volume: 10, Issue:2

    Topics: Binding Sites; Cimetidine; Density Functional Theory; Deuterium; Drug Design; Famotidine; Humans; Hydrogen Bonding; Ligands; Methylhistamines; Normal Distribution; Protein Binding; Protons; Receptors, Histamine H2; Water

2020