Page last updated: 2024-09-04

cilomilast and warfarin

cilomilast has been researched along with warfarin in 4 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(warfarin)
Trials
(warfarin)
Recent Studies (post-2010) (warfarin)
162134236,5732,14314,728

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)warfarin (IC50)
Vitamin K epoxide reductase complex subunit 1 Homo sapiens (human)0.0088

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Clark, DJ; Fuder, H; Kelly, J; Murdoch, RD; Webber, DM1

Trials

1 trial(s) available for cilomilast and warfarin

ArticleYear
Warfarin pharmacodynamics unaffected by cilomilast.
    The Annals of pharmacotherapy, 2001, Volume: 35, Issue:12

    Topics: Adult; Anticoagulants; Bronchodilator Agents; Carboxylic Acids; Cyclohexanecarboxylic Acids; Double-Blind Method; Drug Interactions; Humans; International Normalized Ratio; Male; Middle Aged; Nitriles; Phosphodiesterase Inhibitors; Warfarin

2001

Other Studies

3 other study(ies) available for cilomilast and warfarin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010