Page last updated: 2024-09-04

cilomilast and trazodone

cilomilast has been researched along with trazodone in 2 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(trazodone)
Trials
(trazodone)
Recent Studies (post-2010) (trazodone)
16213421,466295312

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)trazodone (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.091
Alpha-2A adrenergic receptorHomo sapiens (human)0.909
D(2) dopamine receptorHomo sapiens (human)4.485
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.017
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.281
Alpha-2B adrenergic receptorHomo sapiens (human)0.389
Alpha-2C adrenergic receptorHomo sapiens (human)1.942
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.311
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.281
Alpha-1D adrenergic receptorHomo sapiens (human)0.265
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.1315
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.091
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.311
Sodium-dependent serotonin transporterHomo sapiens (human)0.192
Histamine H1 receptorHomo sapiens (human)0.361
D(3) dopamine receptorHomo sapiens (human)3.743
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.107
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.281
Sigma non-opioid intracellular receptor 1Homo sapiens (human)2.203

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1

Other Studies

2 other study(ies) available for cilomilast and trazodone

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010