Page last updated: 2024-09-04

cilomilast and tamsulosin

cilomilast has been researched along with tamsulosin in 3 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(tamsulosin)
Trials
(tamsulosin)
Recent Studies (post-2010) (tamsulosin)
16213421,460468693

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)tamsulosin (IC50)
Alpha-1D adrenergic receptorHomo sapiens (human)0.0008
Alpha-1A adrenergic receptorHomo sapiens (human)0.0013
Alpha-1B adrenergic receptorHomo sapiens (human)0.0045
Alpha-1D adrenergic receptorMus musculus (house mouse)0.0018
Alpha-1B adrenergic receptorMus musculus (house mouse)0.0018
Alpha-1A adrenergic receptorMus musculus (house mouse)0.0018

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1

Other Studies

3 other study(ies) available for cilomilast and tamsulosin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010