Page last updated: 2024-09-04

cilomilast and sitagliptin

cilomilast has been researched along with sitagliptin in 3 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(sitagliptin)
Trials
(sitagliptin)
Recent Studies (post-2010) (sitagliptin)
162134297070

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)sitagliptin (IC50)
Chain A, Dipeptidyl peptidase IVHomo sapiens (human)0.018
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)0.0255
Thromboxane-A synthase Homo sapiens (human)0.0194
Dipeptidyl peptidase 4Homo sapiens (human)0.0236
Dipeptidyl peptidase 4Mus musculus (house mouse)0.046
Prolyl endopeptidase FAPHomo sapiens (human)2.93
Dipeptidyl peptidase 8Homo sapiens (human)0.4715
Dipeptidyl peptidase 9Homo sapiens (human)1.539
Dipeptidyl peptidase 2Homo sapiens (human)0.022

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1

Other Studies

3 other study(ies) available for cilomilast and sitagliptin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010