Page last updated: 2024-09-04

cilomilast and prednisolone

cilomilast has been researched along with prednisolone in 5 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(prednisolone)
Trials
(prednisolone)
Recent Studies (post-2010) (prednisolone)
162134234,4143,3027,141

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)prednisolone (IC50)
Glucocorticoid receptorHomo sapiens (human)0.0278
Progesterone receptorHomo sapiens (human)2.08
Glucocorticoid receptorRattus norvegicus (Norway rat)0.0565
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.016
Mineralocorticoid receptor Homo sapiens (human)0.0322
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.016
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.016
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.016

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Cantinieaux, B; Cataldo, D; Delvaux, C; Dentener, M; Michel, O; Murdoch, RD; Vertongen, F1
Iwata, M; Kobayashi, M; Kubo, S; Miyata, K; Shimizu, Y; Takahashi, K1

Trials

1 trial(s) available for cilomilast and prednisolone

ArticleYear
Evaluation of oral corticosteroids and phosphodiesterase-4 inhibitor on the acute inflammation induced by inhaled lipopolysaccharide in human.
    Pulmonary pharmacology & therapeutics, 2007, Volume: 20, Issue:6

    Topics: Acute Disease; Administration, Oral; Adolescent; Adult; Anti-Inflammatory Agents; C-Reactive Protein; Carboxylic Acids; Cross-Over Studies; Cyclohexanecarboxylic Acids; Double-Blind Method; E-Selectin; Female; Glucocorticoids; Humans; Inflammation; Lipopolysaccharides; Male; Matrix Metalloproteinase 9; Middle Aged; Neutrophils; Nitriles; Phosphodiesterase Inhibitors; Prednisolone; Sputum; Tissue Inhibitor of Metalloproteinase-1; Tumor Necrosis Factor-alpha

2007

Other Studies

4 other study(ies) available for cilomilast and prednisolone

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Anti-neutrophilic inflammatory activity of ASP3258, a novel phosphodiesterase type 4 inhibitor.
    International immunopharmacology, 2012, Volume: 12, Issue:1

    Topics: Adult; Aminopyridines; Animals; Anti-Inflammatory Agents; Benzamides; Bronchoalveolar Lavage Fluid; Cells, Cultured; Chemokine CXCL1; Cyclohexanecarboxylic Acids; Cyclopropanes; Glucocorticoids; Humans; Lipopolysaccharides; Male; Naphthyridines; Neutrophils; Nitriles; Phosphodiesterase 4 Inhibitors; Pneumonia; Prednisolone; Rats; Rats, Wistar; Superoxides; Tumor Necrosis Factor-alpha

2012