Page last updated: 2024-09-04

cilomilast and labetalol

cilomilast has been researched along with labetalol in 2 studies

Compound Research Comparison

Studies
(cilomilast)
Trials
(cilomilast)
Recent Studies (post-2010)
(cilomilast)
Studies
(labetalol)
Trials
(labetalol)
Recent Studies (post-2010) (labetalol)
16213421,980450327

Protein Interaction Comparison

ProteinTaxonomycilomilast (IC50)labetalol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.016
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)3.354
Beta-1 adrenergic receptorHomo sapiens (human)0.01
Cytochrome P450 2D6Homo sapiens (human)0.8
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.393
Sodium-dependent noradrenaline transporter Homo sapiens (human)3.354
Alpha-1D adrenergic receptorHomo sapiens (human)0.521
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.393
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.037
Sodium-dependent dopamine transporter Homo sapiens (human)1.607
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.815

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1

Other Studies

2 other study(ies) available for cilomilast and labetalol

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009