cilomilast has been researched along with 2-methyl-4(3h)-quinazolinone in 1 studies
Studies (cilomilast) | Trials (cilomilast) | Recent Studies (post-2010) (cilomilast) | Studies (2-methyl-4(3h)-quinazolinone) | Trials (2-methyl-4(3h)-quinazolinone) | Recent Studies (post-2010) (2-methyl-4(3h)-quinazolinone) |
---|---|---|---|---|---|
162 | 13 | 42 | 20 | 0 | 10 |
Protein | Taxonomy | cilomilast (IC50) | 2-methyl-4(3h)-quinazolinone (IC50) |
---|---|---|---|
Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | 3.405 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
de Esch, IJ; de Graaf, C; Jansen, C; Kanev, GK; Kooistra, AJ; Leurs, R | 1 |
1 other study(ies) available for cilomilast and 2-methyl-4(3h)-quinazolinone
Article | Year |
---|---|
PDEStrIAn: A Phosphodiesterase Structure and Ligand Interaction Annotated Database As a Tool for Structure-Based Drug Design.
Topics: Databases, Protein; Dose-Response Relationship, Drug; Drug Design; Humans; Ligands; Models, Molecular; Molecular Structure; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Structure-Activity Relationship | 2016 |