cilengitide has been researched along with cyclic(arg-gly-asp-d-phe-val) in 5 studies
| Studies (cilengitide) | Trials (cilengitide) | Recent Studies (post-2010) (cilengitide) | Studies (cyclic(arg-gly-asp-d-phe-val)) | Trials (cyclic(arg-gly-asp-d-phe-val)) | Recent Studies (post-2010) (cyclic(arg-gly-asp-d-phe-val)) |
|---|---|---|---|---|---|
| 194 | 29 | 133 | 20 | 0 | 9 |
| Protein | Taxonomy | cilengitide (IC50) | cyclic(arg-gly-asp-d-phe-val) (IC50) |
|---|---|---|---|
| Integrin beta-3 | Homo sapiens (human) | 1.239 | |
| Integrin alpha-V | Homo sapiens (human) | 1.0243 | |
| Integrin beta-5 | Homo sapiens (human) | 0.0063 | |
| Integrin beta-6 | Homo sapiens (human) | 3.696 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 3 (60.00) | 29.6817 |
| 2010's | 2 (40.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Auzzas, L; Battistini, L; Belvisi, L; Burreddu, P; Casiraghi, G; Castorina, M; Curti, C; Gaetani, E; Giannini, G; Motto, I; Nicastro, G; Pisano, C; Rassu, G; Zanardi, F | 1 |
| Castorina, M; Dal Pozzo, A; de Castiglione, R; Giannini, G; Mazzini, S; Mondelli, R; Muzi, L; Ni, M; Penco, S; Pisano, C | 1 |
| Bottoncetti, A; Brandi, A; Cini, N; Cordero, FM; Gratteri, P; Melani, F; Pisaneschi, F; Salvati, M | 1 |
| Corti, A; Curnis, F; Ghitti, M; Gori, A; Musco, G; Nardelli, F; Paissoni, C; Quilici, G; Sacchi, A; Traversari, C; Valentinis, B | 1 |
| Kemker, I; Marion, A; Schnepel, C; Schröder, DC; Sewald, N | 1 |
5 other study(ies) available for cilengitide and cyclic(arg-gly-asp-d-phe-val)
| Article | Year |
|---|---|
Grafting aminocyclopentane carboxylic acids onto the RGD tripeptide sequence generates low nanomolar alphaVbeta3/alphaVbeta5 integrin dual binders.
Topics: Binding, Competitive; Crystallography, X-Ray; Cycloleucine; Integrin alphaVbeta3; Integrins; Models, Molecular; Molecular Structure; Oligopeptides; Peptides, Cyclic; Protein Binding; Radioligand Assay; Receptors, Vitronectin; Snake Venoms; Solutions; Structure-Activity Relationship | 2005 |
Incorporation of the unusual C(alpha)-fluoroalkylamino acids into cyclopeptides: synthesis of arginine-glycine-aspartate (RGD) analogues and study of their conformational and biological behavior.
Topics: Amino Acids; Dimethyl Sulfoxide; Fluorine; Integrin alphaVbeta3; Integrins; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Oligopeptides; Peptides, Cyclic; Receptors, Vitronectin; Stereoisomerism; Structure-Activity Relationship; Water | 2006 |
Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin alphavbeta3 and alphavbeta5 ligands.
Topics: Computer Simulation; Integrin alphaVbeta3; Integrins; Ligands; Models, Molecular; Molecular Structure; Oligopeptides; Peptides, Cyclic; Receptors, Vitronectin; Structure-Activity Relationship | 2008 |
Succinimide-Based Conjugates Improve IsoDGR Cyclopeptide Affinity to α
Topics: Allosteric Regulation; Binding, Competitive; Cell Line, Tumor; Cell Membrane; HEK293 Cells; Humans; Integrin alphaVbeta3; Magnetic Resonance Spectroscopy; Melanoma; Molecular Docking Simulation; Peptides, Cyclic; Protein Conformation; Snake Venoms; Structure-Activity Relationship; Succinimides; Tyrosine | 2018 |
Cyclization of RGD Peptides by Suzuki-Miyaura Cross-Coupling.
Topics: Boronic Acids; Cell Line, Tumor; Cyclization; Humans; Hydrocarbons, Halogenated; Models, Chemical; Molecular Dynamics Simulation; Molecular Structure; Oligopeptides; Solvents; Structure-Activity Relationship | 2019 |