ciglitazone and thiazoles

ciglitazone has been researched along with thiazoles in 135 studies

Research

Studies (135)

TimeframeStudies, this research(%)All Research%
pre-199027 (20.00)18.7374
1990's22 (16.30)18.2507
2000's83 (61.48)29.6817
2010's3 (2.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gill, AM; Powell, JG; Sampson, BM; Yen, TT1
Dietrich, A; Harrison, MC; Hohman, TC; McCaleb, M; Millen, J; Sredy, J; Sullivan, D; Woolson, SA; Wrobel, J1
Cheeseman, RS; Christos, TE; Kees, KL; McCaleb, ML; Patt, WC; Prozialeck, DH; Smith, TM; Steiner, KE1
Alessi, TR; Bagli, JF; Dolak, TM; Ellinboe, JW; Guzzo, F; McCaleb, ML; Nguyen, TT; Tomer, JD1
Gill, AM; Yen, TT1
Jirkovsky, I; McCaleb, ML; Nowicki, JW; Zask, A1
Ikeda, H; Kawamatsu, Y; Meguro, K; Momose, Y; Sohda, T; Sugiyama, Y1
Belin, D; Bruzzone, R; Trimble, ER1
Caro, JF; Ittoop, O; Sinha, MK1
Chisholm, DJ; James, DE; Jenkins, AB; Kraegen, EW; Storlien, LH1
Lien, EL; Steiner, KE1
Chang, AY; Wyse, BM1
Diani, AR; Sawada, GA; Wyse, BM1
Colca, JR; Connell, CL; Diani, AR; Fletcher-McGruder, BL; Jodelis, KS; Palazuk, BJ; Sawada, G; Wyse, BM1
Kern, HF; Rausch, U; Trimble, ER1
Fujita, T; Taketomi, S; Yokono, K1
Antwi, D; Bray, GA; Chan, TM; Fukushima, M; Shargill, NS; Tatoyan, A1
Mercer, SW; Trayhurn, P1
Rothwell, NJ; Stock, MJ; Tedstone, AE1
Arch, JR; Thurlby, PL; Wilson, S1
Chang, AY; Diani, AR; Gilchrist, BJ; Hearron, AE; Jodelis, K; Peterson, T; Sawada, G; Wyse, BM1
Bachmann, W; Häring, HU; Kirsch, DM1
Iwasaki, M; Kobayashi, M; Maegawa, H; Ohgaku, S; Shigeta, Y; Watanabe, N1
Fujita, T; Iwatsuka, H; Kawamatsu, Y; Sohda, T; Sugiyama, Y; Suzuoki, Z; Taketomi, S1
Chang, AY; Diani, AR; Gilchrist, BJ; Peterson, T; Wyse, BM1
Chang, AY; Gilchrist, BJ; Wyse, BM2
Chang, AY; Diani, AR; Gilchrist, BJ; Hearron, AE; Peterson, T; Sawada, GA; Wyse, BM1
Kawamatsu, Y; Meguro, K; Sohda, T1
Kawamatsu, Y; Mizuno, K; Sohda, T1
Fujita, T; Sugiyama, Y; Tanayama, S; Torii, H; Yoshida, K1
Tanayama, S; Torii, H; Tsukamoto, T; Yoshida, K1
Cox, JW; Pullen, RH1
Fujita, T; Imamiya, E; Kawamatsu, Y; Mizuno, K; Sohda, T; Sugiyama, Y1
Benson, S; Feuerstein, BG; Hyun, WC; Kurtz, TW; Pershadsingh, HA; Szollosi, J1
Kliewer, SA; Lehmann, JM; Lenhard, JM; Morris, DC; Patel, I; Willson, TM1
Umeda, F1
Lambe, KG; Tugwood, JD1
Clark, DA; Genereux, PE; Gibbs, EM; Hulin, B; Lewis, DM; Newton, LS1
Connell, J; Petrie, J; Small, M1
Benson, SC; Kurtz, TW; Morikang, E; Pershadsingh, HA1
Bucher, NL; Farmer, SR; Morrison, RF; Wu, Z; Xie, Y1
Akatsuka, H; Arakawa, K; Homma, K; Iijima, I; Inamasu, M; Kawanami, S; Matsumoto, M; Okumura, K; Ozeki, M; Saiga, Y; Watanabe, A; Yasuda, K1
Goldammer, T; Kanitz, W; Löhrke, B; Pöhland, R; Shahi, SK; Viergutz, T; Walzel, H; Wollenhaupt, K1
Dandine, M; Dauzats, M; Daviaud, D; Langin, D; Saulnier-Blache, JS; Viguerie-Bascands, N1
Gerritsen, ME; Kowalski, J; Xin, X; Yang, S1
Gebicke-Haerter, PJ; Kakimura, J; Kitamura, Y; Matsuoka, Y; Nomura, Y; Taniguchi, T1
Combs, CK; Doller, C; Fitch, MT; Landreth, GE; Silver, J1
Kniss, DA; Li, HM; Liu, L; Sabourin, CL; Seewaldt, V; Smith, PJ; Yee, LD1
Casini, A; Ceni, E; Crabb, D; Galli, A; Price, D; Salzano, R; Surrenti, C1
Bishop-Bailey, D; Clark, RB; Estrada-Hernandez, T; Hla, T; Padula, SJ; Puddington, L1
Dietl, G; Krüger, B; Löhrke, B; Renne, U; Schmidt, P; Shahi, SK1
Kuzuya, T1
Ikeda, H; Murase, K; Sugiyama, Y1
Demer, LL; Jackson, SM1
Loitsch, SM; Stein, J; Wächtershäuser, A1
Black, PM; Brown, EM; Chattopadhyay, N; Godbole, MM; Heese, O; Singh, DP; Sinohara, T1
Chiang, HT; Ho, LL; Li, HF; Wu, SN1
Cho, D; Chung, SW; Kang, BY; Kim, SH; Kim, TS; Pak, YK; Trinchieri, G1
Adzet, T; Alegret, M; Cabrero, A; Laguna, JC; Sánchez, RM; Vázquez, M1
Aleo, MD; Avery, MJ; Beierschmitt, WP; Drupa, CA; Fortner, JH; Kaplan, AH; Navetta, KA; Shepard, RM; Walsh, CM1
Cao, HJ; Kaur, K; Padilla, J; Phipps, RP; Smith, TJ1
Brüne, B; Von Knethen A, A1
Kagechika, H; Kawashima, S; Sato, M; Tanaka, K; Yajima, Y1
Dixon, C; Hilbelink, T; Lu, L; Rovin, BH; Wilmer, WA1
Gunawan, I; Malamas, MS; McCaleb, M; Mihan, B; Sredy, J; Sullivan, D1
Harris, SG; Phipps, RP1
Conrad, DJ; Dai, X; Luu, B; Wang, AC1
Albajar, M; Galetto, R; Polanco, JI; Rodríguez-Rey, JC; Zakin, MM1
Hupfeld, CJ; Weiss, RH1
Bláha, L; Hofmanová, J; Kozubík, A; Minksová, K; Soucek, K; Stika, J; Vondrácek, J1
Frucht, H; Yang, WL1
Kang, K; Pariza, MW1
Dulak, J; Huk, I; Jozkowicz, A; Nanobashvili, J; Nigisch, A; Prager, M; Weigel, G; Winter, B1
Levine, L1
Berry, E; Gilmour, R; Helliwell, R; Keelan, J; Marvin, K; Mitchell, M; Nijmeijer, B; Sato, T1
Coffey, MJ; Hayes, MM; King, SR; Lane, BR; Markovitz, DM1
Marra, F; Pastacaldi, S1
Archer, DC; Cunard, R; DiCampli, D; Glass, CK; Kahn, DA; Kelly, CJ; Ricote, M1
Brüne, B; Fischer, B; von Knethen, A1
Dixon, C; Doseff, AI; Hilbelink, T; Kotur, M; Lu, L; Rovin, BH; Wilmer, WA1
Chang, TH; Szabo, E1
Bright, JJ; Natarajan, C1
Dembinska-Kiec, A; Dulak, J; Jozkowicz, A; Piatkowska, E; Placha, W1
Breyer, B; Cheng, H; Feng, T; Haydon, RC; He, TC; Ishikawa, A; Jiang, W; Montag, A; Peabody, T; Simon, MA; Zhou, L1
Baik, EJ; Kim, EJ; Kwon, KJ; Lee, SH; Moon, CH; Park, JY1
Dessouroux, A; Lennon, AM; Pierre, M; Ramaugé, M1
Blaschke, F; Bungenstock, A; Eilers, F; Fleck, E; Goetze, S; Graf, K; Gräfe, M; Kintscher, U; Law, RE; Stawowy, P1
Feinstein, D; Grommes, C; Heneka, MT; Klockgether, T; Koenigsknecht, J; Kraus, JA; Landreth, G; Schlegel, U; Zander, T1
Frauwirth, KA; Lazar, MA; Rangwala, SM; Thompson, CB; Wang, YL1
Chi, KH; Chio, CC; Huang, WC; Lin, WW; Wu, HM1
Chatterjee, PK; Cuzzocrea, S; Hattori, Y; McDonald, MC; Mota-Filipe, H; Pisano, B; Thiemermann, C; Wayman, NS1
Miyazaki, Y; Tachibana, H; Yamada, K1
Büchele, B; Jendrach, M; Schüle, A; Simmet, T; Syrovets, T1
Battarbee, H; Coates, G; Nissim, I; Welbourne, T1
Cho, H; Tai, HH2
Fujimura, Y; Tachibana, H; Yamada, K1
Chan, UP; Chen, GG; Ip, PC; Lau, WY; Lee, JF; Wang, SH1
Greenberg, AS; Mathys, JM; Rabbi, MF; Skolnik, PR1
Cammarota, S; Chiariotti, L; Fusco, A; Iuliano, R; Kroll, T; Le Pera, I; Martelli, ML; Monaco, C; Sama', I; Santoro, M1
Hansen, M; Maisch, B; Rupp, H; Wahl, R1
Bungenstock, A; Czupalla, C; Eilers, F; Fleck, E; Goetze, S; Graf, K; Gräfe, M; Kintscher, U; Law, RE; Nürnberg, B; Spencer-Hänsch, C; Stawowy, P1
Fujita, T; Ikeda, H; Kawamatsu, Y; Meguro, K; Sohda, T1
Jensen, BA; Mann, KK; Ryu, HY; Schlezinger, JJ; Sherr, DH1
Corbett, L; Knox, AJ; Nie, M; Pang, L1
Calnek, DS; Hart, CM; Mazzella, L; Roman, J; Roser, S1
Aruna, B; Ehtesham, NZ; Ghosh, S; Mukhopadhyay, S; Singh, AK1
Belvisi, MG; Bishop-Bailey, D; Mitchell, JA; Patel, HJ; Yacoub, MH1
Brune, K; Hinz, B; Pahl, A1
Chen, YE; Fu, M; Lin, Y; Mao, Z; Zhang, J; Zhu, X1
Kehrer, JP; Tong, Z; Wu, X1
Burghardt, R; Qin, C; Safe, S; Smith, R; Stewart, J; Wormke, M1
Han, S; Huang, RP; Sidell, N; Wanichkul, T1
Chao, VA; Hornung, D; Taylor, RN; Vigne, JL; Wallwiener, D1
Slomiany, A; Slomiany, BL1
Ethridge, RT; Evers, BM; Hashimoto, K1
Broaddus, RR; Copland, JA; Fischer, SM; Gottardis, MM; Houston, KD; Walker, CL1
Brüne, B; Tautenhahn, A; von Knethen, A1
Bradbury, J; Clinton, SK; Guo, Y; Seewaldt, VL; Suster, S; Yee, LD1
Holman, NA; May, FJ; Monteith, GR; Roberts-Thomson, SJ; Robinson, JA; Smith, SA1
Burgermeister, E; Liscovitch, M; Tencer, L1
Dawson, MI; James, SY; Kolluri, SK; Lin, F; Zhang, XK1
Dai, J; Remick, DG; Wang, X; Zeng, X1
Auwerx, J; Capron, M; Dombrowicz, D; Honda, K; Loyens, M; Papin, JP; Staels, B; Woerly, G1
Fu, J; Gaetani, S; Lin, E; Oveisi, F; Piomelli, D1
Knight, B; Olynyk, JK; Yeap, BB; Yeoh, GC1
Cabot, PJ; Davis, B; Monteith, GR; Roberts-Thomson, SJ; Robinson, JA; Venkata, NG1
Brunskill, NJ; Chana, RS1
Futagami, M; Mizunuma, H; Shigeto, T; Xin, B; Yokoyama, Y1
Elias, PM; Feingold, KR; Jiang, YJ; Kim, P; Lu, B; Paragh, G; Schmitz, G1
Guo, SW; Wu, Y1
Baron, DM; Hudec, X; Kaindl, U; Koneczny, I; König, JS; Marian, B; Röhrl, C1
Buono, C; Busch, S; Chibout, SD; Cruz, E; Gurnani, M; McLean, LA; Moulin, P; Patel, P; Pognan, F; Reising, A; Sampath, S; Shangari, N; Wolf, A1
Caballero, J; Fuentes, E; Muñoz-Gutiérrez, C; Palomo, I; Sepúlveda, C1

Reviews

6 review(s) available for ciglitazone and thiazoles

ArticleYear
Hypoglycaemic agents which do not release insulin.
    Progress in medicinal chemistry, 1987, Volume: 24

    Topics: Animals; Fatty Acids; Humans; Hypoglycemic Agents; Insulin; Somatostatin; Thiazoles; Thiazolidinediones

1987
Potential role of thiazolidinediones in older diabetic patients.
    Drugs & aging, 1995, Volume: 7, Issue:5

    Topics: Aged; Aging; Animals; Benzopyrans; Chromans; Diabetes Mellitus, Type 2; Double-Blind Method; Glucose Tolerance Test; Humans; Hypoglycemic Agents; Insulin Resistance; Japan; Mice; Pioglitazone; Randomized Controlled Trials as Topic; Rats; Thiazoles; Thiazolidinediones; Troglitazone

1995
[The development of thiazolidinedione drugs as anti-diabetic agents].
    Nihon rinsho. Japanese journal of clinical medicine, 2000, Volume: 58, Issue:2

    Topics: Animals; Chemical and Drug Induced Liver Injury; Chromans; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Insulin Resistance; Mice; Rosiglitazone; Thiazoles; Thiazolidinediones; Troglitazone

2000
[Mechanisms of thiazolidinedione derivatives for hypoglycemic and insulin sensitizing effects].
    Nihon rinsho. Japanese journal of clinical medicine, 2000, Volume: 58, Issue:2

    Topics: Animals; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Insulin; Insulin Resistance; Lipid Metabolism; Pioglitazone; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Necrosis Factor-alpha

2000
[Thiazolidinediones and PPARgamma system in repair of liver damage].
    Recenti progressi in medicina, 2002, Volume: 93, Issue:1

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Antioxidants; Arteriosclerosis; Chromans; Diabetes Mellitus, Type 2; Eicosanoids; Fatty Acids; Forecasting; Humans; Hypoglycemic Agents; In Vitro Techniques; Inflammation; Liver Cirrhosis; Neoplasms; Obesity; Receptors, Cytoplasmic and Nuclear; Research; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2002
[Discovery and development of a new insulin sensitizing agent, pioglitazone].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2002, Volume: 122, Issue:11

    Topics: Animals; Clinical Trials as Topic; Clofibrate; Diabetes Mellitus; Diabetes Mellitus, Experimental; Drug Design; Humans; Hypoglycemic Agents; Insulin Resistance; Mice; Pioglitazone; Thiazoles; Thiazolidinediones

2002

Other Studies

129 other study(ies) available for ciglitazone and thiazoles

ArticleYear
Ciglitazone prevents and reverses dexamethasone-induced hyperglycemia in female viable yellow mice.
    International journal of obesity and related metabolic disorders : journal of the International Association for the Study of Obesity, 1992, Volume: 16, Issue:11

    Topics: Administration, Oral; Animals; Blood Glucose; Body Weight; Corticosterone; Dexamethasone; Dose-Response Relationship, Drug; Female; Hyperglycemia; Hypoglycemic Agents; Insulin; Male; Mice; Thiazoles; Thiazolidinediones

1992
Novel spirosuccinimides with incorporated isoindolone and benzisothiazole 1,1-dioxide moieties as aldose reductase inhibitors and antihyperglycemic agents.
    Journal of medicinal chemistry, 1992, Nov-27, Volume: 35, Issue:24

    Topics: Aldehyde Reductase; Animals; Blood Glucose; Cattle; Diabetes Mellitus, Experimental; Glyceraldehyde; Hypoglycemic Agents; Indoles; Male; Mice; Mice, Inbred C57BL; Molecular Structure; Rats; Structure-Activity Relationship; Succinimides; Thiazoles; Thiazolidinediones

1992
Perfluorocarbon-based antidiabetic agents.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Female; Fluorocarbons; Hypoglycemic Agents; Insulin; Mice; Mice, Obese; Molecular Structure; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

1992
Antihyperglycemic activity of novel substituted 3H-1,2,3,5-oxathiadiazole 2-oxides.
    Journal of medicinal chemistry, 1992, Apr-03, Volume: 35, Issue:7

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Male; Mice; Mice, Inbred C57BL; Molecular Structure; Rats; Rats, Zucker; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

1992
Effects of ciglitazone on endogenous plasma islet amyloid polypeptide and insulin sensitivity in obese-diabetic viable yellow mice.
    Life sciences, 1991, Volume: 48, Issue:7

    Topics: Amyloid; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Insulin; Islet Amyloid Polypeptide; Mice; Mice, Obese; Reference Values; Thiazoles; Thiazolidinediones; Triglycerides

1991
Synthesis and antihyperglycemic activity of novel 5-(naphthalenylsulfonyl)-2,4-thiazolidinediones.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:5

    Topics: Animals; Blood Glucose; Chemical Phenomena; Chemistry; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Lactates; Male; Mice; Naphthalenes; Rats; Rats, Zucker; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

1990
Studies on antidiabetic agents. Synthesis and hypoglycemic activity of 5-[4-(pyridylalkoxy)benzyl]-2,4-thiazolidinediones.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:1

    Topics: Animals; Chemical Phenomena; Chemistry; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Male; Mice; Mice, Inbred Strains; Mice, Obese; Pioglitazone; Pyridines; Thiazoles; Thiazolidinediones; Triglycerides

1990
Insulin resistance is accompanied by impairment of amylase-gene expression in the exocrine pancreas of the obese Zucker rat.
    The Biochemical journal, 1986, Aug-01, Volume: 237, Issue:3

    Topics: Amylases; Animals; Female; Gene Expression Regulation; Glucose; Insulin Resistance; Obesity; Pancreas; Protein Biosynthesis; Rats; Rats, Mutant Strains; Rats, Zucker; RNA, Messenger; Thiazoles; Thiazolidinediones

1986
Glyburide but not ciglitazone enhances insulin action in the liver independent of insulin receptor kinase activation.
    Metabolism: clinical and experimental, 1989, Volume: 38, Issue:7

    Topics: Animals; Cells, Cultured; Drug Synergism; Glyburide; Hypoglycemic Agents; Insulin; Kinetics; Liver; Macromolecular Substances; Phosphorylation; Protein-Tyrosine Kinases; Rats; Receptor, Insulin; Thiazoles; Thiazolidinediones

1989
A potent in vivo effect of ciglitazone on muscle insulin resistance induced by high fat feeding of rats.
    Metabolism: clinical and experimental, 1989, Volume: 38, Issue:11

    Topics: Animals; Blood Glucose; Deoxyglucose; Dietary Fats; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Muscles; Phosphorylation; Rats; Rats, Inbred Strains; Thiazoles; Thiazolidinediones

1989
The hypoglycemic effect of ciglitazone in obese, hyperglycemic animal models.
    Progress in clinical and biological research, 1988, Volume: 265

    Topics: Adipose Tissue; Adipose Tissue, Brown; Animals; Blood Glucose; Disease Models, Animal; Glycolysis; Hyperglycemia; Hypoglycemic Agents; Insulin; Male; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Mice, Obese; Mitochondria; Obesity; Oxygen Consumption; Receptor, Insulin; Thiazoles; Thiazolidinediones

1988
A review of the effects of ciglitazone on the pancreatic islets of obese, hyperglycemic mice.
    Progress in clinical and biological research, 1988, Volume: 265

    Topics: Animals; Hyperglycemia; Hypoglycemic Agents; Insulin; Islets of Langerhans; Male; Mice; Mice, Obese; Obesity; Thiazoles; Thiazolidinediones

1988
Ciglitazone, a hypoglycemic agent: early effects on the pancreatic islets of ob/ob mice.
    Metabolism: clinical and experimental, 1988, Volume: 37, Issue:3

    Topics: Animals; Blood Glucose; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Thiazoles; Thiazolidinediones

1988
Changes in individual rates of pancreatic enzyme and isoenzyme biosynthesis in the obese Zucker rat.
    The Biochemical journal, 1987, Dec-15, Volume: 248, Issue:3

    Topics: Amino Acids; Animals; Blood Glucose; Eating; Insulin; Isoelectric Focusing; Isoenzymes; Kinetics; Obesity; Pancreas; Proteins; Rats; Rats, Zucker; Thiazoles; Thiazolidinediones

1987
Insulin receptor and postbinding defects in KK mouse adipocytes and improvement by ciglitazone.
    Diabetes research and clinical practice, 1988, Jul-13, Volume: 5, Issue:2

    Topics: 3-O-Methylglucose; Adipose Tissue; Animals; Carbon Radioisotopes; Cells, Cultured; Diabetes Mellitus, Experimental; Glucose; Glycolysis; Hypoglycemic Agents; Insulin Resistance; Kinetics; Male; Methylglucosides; Methylglycosides; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Receptor, Insulin; Thiazoles; Thiazolidinediones; Tritium

1988
Effect of ciglitazone on glucose uptake and insulin sensitivity in skeletal muscle of the obese (ob/ob) mouse: distinct insulin and glucocorticoid effects.
    Metabolism: clinical and experimental, 1986, Volume: 35, Issue:1

    Topics: Adrenal Cortex; Animals; Deoxyglucose; Glucocorticoids; Gluconeogenesis; Glucose; Hypoglycemic Agents; Insulin; Liver; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Muscles; Thiazoles; Thiazolidinediones

1986
Effects of ciglitazone on insulin resistance and thermogenic responsiveness to acute cold in brown adipose tissue of genetically obese (ob/ob) mice.
    FEBS letters, 1986, Jan-20, Volume: 195, Issue:1-2

    Topics: Adipose Tissue, Brown; Animals; Cold Temperature; Guanosine Diphosphate; Insulin; Insulin Resistance; Lipids; Male; Mice; Mice, Obese; Mitochondria; Thiazoles; Thiazolidinediones

1986
Effects of ciglitazone on energy balance, thermogenesis and brown fat activity in the rat.
    Molecular and cellular endocrinology, 1987, Volume: 51, Issue:3

    Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Body Weight; Eating; Energy Metabolism; Male; Oxygen Consumption; Propranolol; Purine Nucleotides; Rats; Rats, Inbred Strains; Thiazoles; Thiazolidinediones

1987
Ciglitazone is not itself thermogenic but increases the potential for thermogenesis in lean mice.
    Bioscience reports, 1987, Volume: 7, Issue:7

    Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Calorimetry; Energy Metabolism; Female; Guanosine Diphosphate; Hypoglycemic Agents; Mice; Thiazoles; Thiazolidinediones

1987
Ciglitazone, a new hypoglycemic agent. 5. Effect on renal lesions in C57BL/KsJ-db/db mice.
    Nephron, 1986, Volume: 42, Issue:1

    Topics: Animals; Blood Glucose; Diabetic Nephropathies; Drug Evaluation, Preclinical; Glomerular Mesangium; Glycogen; Histocytochemistry; Hypoglycemic Agents; Immunoglobulin G; Immunoglobulin M; Kidney; Kidney Tubules; Male; Mice; Mice, Inbred C57BL; Thiazoles; Thiazolidinediones

1986
Ciglitazone reverses cAMP-induced post-insulin receptor resistance in rat adipocytes in vitro.
    FEBS letters, 1984, Oct-15, Volume: 176, Issue:1

    Topics: 3-O-Methylglucose; Adipose Tissue; Animals; Biological Transport; Cyclic AMP; Insulin; Insulin Resistance; Isoproterenol; Male; Methylglucosides; Rats; Receptor, Insulin; Thiazoles; Thiazolidinediones

1984
A new potentiator of insulin action. Post-receptor activation in vitro.
    FEBS letters, 1983, Oct-31, Volume: 163, Issue:1

    Topics: Adipose Tissue; Animals; Biological Transport, Active; Blood Glucose; Body Weight; Deoxyglucose; Diabetes Mellitus, Experimental; Drug Synergism; Glucose; Glycolysis; Insulin; Kinetics; Obesity; Rats; Rats, Inbred Strains; Receptor, Insulin; Thiazoles; Thiazolidinediones

1983
Reduction of insulin resistance in obese and/or diabetic animals by 5-[4-(1-methylcyclohexylmethoxy)benzyl]-thiazolidine-2,4-dione (ADD-3878, U-63,287, ciglitazone), a new antidiabetic agent.
    Diabetes, 1983, Volume: 32, Issue:9

    Topics: Animals; Blood Glucose; Cholesterol; Diabetes Mellitus; Diabetes Mellitus, Experimental; Dogs; Fatty Acids, Nonesterified; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Mice; Mice, Obese; Obesity; Phospholipids; Rats; Rats, Inbred Strains; Thiazoles; Thiazolidinediones; Triglycerides

1983
Ciglitazone, a new hypoglycemic agent. I. Studies in ob/ob and db/db mice, diabetic Chinese hamsters, and normal and streptozotocin-diabetic rats.
    Diabetes, 1983, Volume: 32, Issue:9

    Topics: Animals; Blood Glucose; Cricetinae; Cricetulus; Diabetes Mellitus, Experimental; Fatty Acids, Nonesterified; Glucagon; Hypoglycemic Agents; Insulin; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Rats; Thiazoles; Thiazolidinediones; Triglycerides

1983
Ciglitazone, a new hypoglycemic agent. II. Effect on glucose and lipid metabolisms and insulin binding in the adipose tissue of C57BL/6J-ob/ob and -+/? mice.
    Diabetes, 1983, Volume: 32, Issue:9

    Topics: Adipose Tissue; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Fatty Acids, Nonesterified; Hypoglycemic Agents; Insulin; Insulin Resistance; Lipids; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Thiazoles; Thiazolidinediones

1983
Ciglitazone, a new hypoglycaemic agent. 4. Effect on pancreatic islets of C57BL/6J-ob/ob and C57BL/KsJ-db/db mice.
    Diabetologia, 1984, Volume: 27, Issue:2

    Topics: Animals; Blood Glucose; Cytoplasmic Granules; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Insulin; Islets of Langerhans; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Microscopy, Electron; Thiazoles; Thiazolidinediones

1984
Studies on antidiabetic agents. IV. Synthesis and activity of the metabolites of 5-[4-(1-methylcyclohexylmethoxy)benzyl]-2,4-thiazolidinedione (ciglitazone).
    Chemical & pharmaceutical bulletin, 1984, Volume: 32, Issue:6

    Topics: Animals; Blood Glucose; Chemical Phenomena; Chemistry; Hypoglycemic Agents; Hypolipidemic Agents; Mice; Mice, Obese; Thiazoles; Thiazolidinediones; Triglycerides

1984
Studies on antidiabetic agents. VI. Asymmetric transformation of (+/-)-5-[4-(1-methylcyclohexylmethoxy)benzyl]-2,4- thiazolidinedione(ciglitazone) with optically active 1-phenylethylamines.
    Chemical & pharmaceutical bulletin, 1984, Volume: 32, Issue:11

    Topics: Animals; Chemical Phenomena; Chemistry, Physical; Hypoglycemic Agents; Mice; Mice, Obese; Phenethylamines; Stereoisomerism; Thiazoles; Thiazolidinediones

1984
Ciglitazone, a new hypoglycaemic agent. 3. Effect on glucose disposal and gluconeogenesis in vivo in C57BL/6J-ob/ob and -+/? mice.
    Diabetologia, 1983, Volume: 25, Issue:6

    Topics: Animals; Blood Glucose; Gluconeogenesis; Glucose; Glycogen; Hypoglycemic Agents; Kinetics; Lipid Metabolism; Liver; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Proteins; Thiazoles; Thiazolidinediones

1983
Rat-plasma metabolites of ciglitazone, a new antidiabetic agent.
    Xenobiotica; the fate of foreign compounds in biological systems, 1984, Volume: 14, Issue:3

    Topics: Animals; Body Weight; Dose-Response Relationship, Drug; Feeding Behavior; Female; Gas Chromatography-Mass Spectrometry; Hydroxylation; Hypoglycemic Agents; Male; Mice; Mice, Obese; Rats; Rats, Inbred Strains; Stereoisomerism; Thiazoles; Thiazolidinediones

1984
Disposition in rats and dogs of ciglitazone, a new antidiabetic agent.
    Xenobiotica; the fate of foreign compounds in biological systems, 1984, Volume: 14, Issue:3

    Topics: Administration, Oral; Animals; Bile; Blood Proteins; Dogs; Erythrocytes; Feces; Female; Hypoglycemic Agents; Male; Maternal-Fetal Exchange; Pregnancy; Protein Binding; Rats; Rats, Inbred Strains; Thiazoles; Thiazolidinediones; Tissue Distribution

1984
Isomodal column switching high-performance liquid chromatographic technique for the analysis of ciglitazone and its metabolites in human serum.
    Journal of chromatography, 1984, Apr-13, Volume: 307, Issue:1

    Topics: Adult; Chromatography, High Pressure Liquid; Humans; Hypoglycemic Agents; Isomerism; Male; Reference Standards; Thiazoles; Thiazolidinediones

1984
Studies on antidiabetic agents. II. Synthesis of 5-[4-(1-methylcyclohexylmethoxy)-benzyl]thiazolidine-2,4-dione (ADD-3878) and its derivatives.
    Chemical & pharmaceutical bulletin, 1982, Volume: 30, Issue:10

    Topics: Animals; Hypoglycemic Agents; Male; Mice; Mice, Obese; Thiazoles; Thiazolidinediones

1982
Effects of ciglitazone on blood pressure and intracellular calcium metabolism.
    Hypertension (Dallas, Tex. : 1979), 1993, Volume: 21, Issue:6 Pt 2

    Topics: Animals; Blood Pressure; Calcium; Female; Insulin; Intracellular Membranes; Obesity; Platelet-Derived Growth Factor; Rats; Rats, Zucker; Signal Transduction; Thiazoles; Thiazolidinediones; Tumor Cells, Cultured

1993
A prostaglandin J2 metabolite binds peroxisome proliferator-activated receptor gamma and promotes adipocyte differentiation.
    Cell, 1995, Dec-01, Volume: 83, Issue:5

    Topics: Adipocytes; Animals; Binding, Competitive; Cell Differentiation; Cells, Cultured; Fibroblasts; Hypoglycemic Agents; Ligands; Mice; Microbodies; Prostaglandin D2; Prostaglandins; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; Rosiglitazone; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation

1995
A human peroxisome-proliferator-activated receptor-gamma is activated by inducers of adipogenesis, including thiazolidinedione drugs.
    European journal of biochemistry, 1996, Jul-01, Volume: 239, Issue:1

    Topics: Adipose Tissue; Amino Acid Sequence; Animals; Base Sequence; Benzopyrans; Chromans; DNA, Complementary; Fatty Acids; Humans; Mice; Molecular Sequence Data; Pioglitazone; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation; Troglitazone

1996
Hypoglycemic activity of a series of alpha-alkylthio and alpha-alkoxy carboxylic acids related to ciglitazone.
    Journal of medicinal chemistry, 1996, Sep-27, Volume: 39, Issue:20

    Topics: 3T3 Cells; Adipocytes; Animals; Benzofurans; Carboxylic Acids; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Mice; Mice, Mutant Strains; Mice, Obese; Molecular Structure; Oxazoles; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

1996
"Glitazones", a prospect for non-insulin-dependent diabetes.
    Lancet (London, England), 1997, Jan-11, Volume: 349, Issue:9045

    Topics: Chromans; Diabetes Mellitus, Type 2; Humans; Hyperinsulinism; Hypoglycemic Agents; Insulin Resistance; Pioglitazone; Thiazoles; Thiazolidinediones; Troglitazone

1997
Effects of thiazolidinediones on growth and differentiation of human aorta and coronary myocytes.
    American journal of hypertension, 1997, Volume: 10, Issue:4 Pt 1

    Topics: Aorta; Cell Division; Cells, Cultured; Chromans; Coronary Vessels; Humans; Hypoglycemic Agents; Muscle, Smooth, Vascular; Thiazoles; Thiazolidinediones; Troglitazone

1997
PPARgamma induces the insulin-dependent glucose transporter GLUT4 in the absence of C/EBPalpha during the conversion of 3T3 fibroblasts into adipocytes.
    The Journal of clinical investigation, 1998, Jan-01, Volume: 101, Issue:1

    Topics: 3T3 Cells; Adaptor Protein Complex 2; Adaptor Protein Complex alpha Subunits; Adaptor Proteins, Vesicular Transport; Adipocytes; Animals; CCAAT-Enhancer-Binding Proteins; Cell Differentiation; Complement Factor D; Dexamethasone; DNA-Binding Proteins; Gene Expression; Glucose Transporter Type 4; Hypoglycemic Agents; Insulin; Ligands; Membrane Proteins; Mice; Monosaccharide Transport Proteins; Muscle Proteins; Nuclear Proteins; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; RNA, Messenger; Serine Endopeptidases; Thiazoles; Thiazolidinediones; Transcription Factors

1998
Novel benzoxazole 2,4-thiazolidinediones as potent hypoglycemic agents. Synthesis and structure-activity relationships.
    Chemical & pharmaceutical bulletin, 1997, Volume: 45, Issue:12

    Topics: Animals; Benzopyrans; Benzoxazoles; Chromans; Diabetes Mellitus; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Male; Mice; Obesity; Pioglitazone; Rosiglitazone; Structure-Activity Relationship; Thiazoles; Thiazolidinediones; Troglitazone

1997
Detection and functional characterisation of the transcription factor peroxisome proliferator-activated receptor gamma in lutein cells.
    The Journal of endocrinology, 1998, Volume: 159, Issue:3

    Topics: Analysis of Variance; Animals; Aurintricarboxylic Acid; Cattle; Cell Cycle; Dose-Response Relationship, Drug; Female; Flow Cytometry; Granulosa Cells; Hypoglycemic Agents; Luteal Cells; Luteinizing Hormone; Microscopy, Fluorescence; Progesterone; Prostaglandin D2; Protein Isoforms; Receptors, Cytoplasmic and Nuclear; Receptors, LH; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors

1998
Increase in uncoupling protein-2 mRNA expression by BRL49653 and bromopalmitate in human adipocytes.
    Biochemical and biophysical research communications, 1999, Mar-05, Volume: 256, Issue:1

    Topics: Adipocytes; Adipose Tissue; Adult; Cells, Cultured; Culture Techniques; Dose-Response Relationship, Drug; Female; Gene Expression Regulation; Humans; Ion Channels; Leptin; Membrane Transport Proteins; Middle Aged; Mitochondrial Proteins; Palmitates; Proteins; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors; Transcriptional Activation; Tumor Necrosis Factor-alpha; Uncoupling Protein 2

1999
Peroxisome proliferator-activated receptor gamma ligands are potent inhibitors of angiogenesis in vitro and in vivo.
    The Journal of biological chemistry, 1999, Mar-26, Volume: 274, Issue:13

    Topics: Animals; Cell Differentiation; Cell Division; Cells, Cultured; Cornea; Eicosanoids; Endothelium, Vascular; Gene Expression Regulation; Humans; Ligands; Neovascularization, Physiologic; Prostaglandin D2; Rats; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors

1999
Activators of peroxisome proliferator-activated receptor-gamma (PPARgamma) inhibit inducible nitric oxide synthase expression but increase heme oxygenase-1 expression in rat glial cells.
    Neuroscience letters, 1999, Mar-05, Volume: 262, Issue:2

    Topics: Alitretinoin; Animals; Anti-Inflammatory Agents, Non-Steroidal; Brain; Cells, Cultured; Dinoprostone; Enzyme Induction; Gene Expression Regulation, Enzymologic; Heme Oxygenase (Decyclizing); Heme Oxygenase-1; Interferon-gamma; Lipopolysaccharides; Neuroglia; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitrites; Prostaglandin D2; Pyrimidines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin

1999
Cellular and molecular mechanisms of glial scarring and progressive cavitation: in vivo and in vitro analysis of inflammation-induced secondary injury after CNS trauma.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Oct-01, Volume: 19, Issue:19

    Topics: Animals; Animals, Newborn; Astrocytes; Axons; Brain Injuries; Cell Movement; Cells, Cultured; Cerebral Cortex; Ganglia, Spinal; Gene Expression Regulation; Glial Fibrillary Acidic Protein; Indomethacin; Inflammation; Lipopolysaccharides; Macrophage Activation; Macrophages, Peritoneal; Microscopy, Video; Neurites; Neuroglia; Neurons; Proteoglycans; Rats; Rats, Sprague-Dawley; Thiazoles; Thiazolidinediones; Zymosan

1999
Peroxisome proliferator-activated receptor gamma activation in human breast cancer.
    International journal of oncology, 1999, Volume: 15, Issue:5

    Topics: Breast Neoplasms; Cell Division; DNA-Binding Proteins; Female; Genes, Reporter; Humans; Hypoglycemic Agents; Prostaglandins; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Recombinant Proteins; Retinoid X Receptors; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured

1999
Peroxisome proliferator-activated receptor gamma transcriptional regulation is involved in platelet-derived growth factor-induced proliferation of human hepatic stellate cells.
    Hepatology (Baltimore, Md.), 2000, Volume: 31, Issue:1

    Topics: Cell Differentiation; Cell Division; Cells, Cultured; Gene Expression; Gene Expression Regulation; Humans; Liver; Platelet-Derived Growth Factor; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Transfection

2000
The nuclear receptor PPAR gamma and immunoregulation: PPAR gamma mediates inhibition of helper T cell responses.
    Journal of immunology (Baltimore, Md. : 1950), 2000, Feb-01, Volume: 164, Issue:3

    Topics: Adjuvants, Immunologic; Animals; Binding Sites, Antibody; CD3 Complex; Clone Cells; Female; Immune Sera; Immunosuppressive Agents; Interleukin-2; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Microbodies; Nuclear Proteins; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Spleen; T-Lymphocytes, Helper-Inducer; Thiazoles; Thiazolidinediones; Transcription Factors

2000
Thiazolidinedione-induced activation of the transcription factor peroxisome proliferator-activated receptor gamma in cells adjacent to the murine skeletal muscle: implications for fibroblast functions.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 439, Issue:3

    Topics: Adipocytes; Animals; Blotting, Western; Cell Separation; DNA, Complementary; Down-Regulation; Fatty Acids; Fibroblasts; Flow Cytometry; Glucose; Homeostasis; Hypoglycemic Agents; Immunohistochemistry; Macrophages; Male; Mice; Mice, Obese; Muscle, Skeletal; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Necrosis Factor-alpha

2000
Peroxisome proliferator-activated receptor activators modulate the osteoblastic maturation of MC3T3-E1 preosteoblasts.
    FEBS letters, 2000, Apr-07, Volume: 471, Issue:1

    Topics: Animals; Bone Density; Cell Differentiation; Cells, Cultured; Humans; Mice; Osteoblasts; Protein Isoforms; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection

2000
PPAR-gamma is selectively upregulated in Caco-2 cells by butyrate.
    Biochemical and biophysical research communications, 2000, Jun-07, Volume: 272, Issue:2

    Topics: Alkaline Phosphatase; Blotting, Western; Butyrates; Caco-2 Cells; Cell Differentiation; Dose-Response Relationship, Drug; Enzyme Activation; Humans; Pentanoic Acids; Propionates; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Substrate Specificity; Thiazoles; Thiazolidinediones; Transcription Factors; Up-Regulation

2000
Expression of peroxisome proliferator-activated receptors (PPARS) in human astrocytic cells: PPARgamma agonists as inducers of apoptosis.
    Journal of neuroscience research, 2000, Jul-01, Volume: 61, Issue:1

    Topics: Apoptosis; Astrocytes; Caspase 3; Caspases; Cell Survival; DNA Fragmentation; Gene Expression; Humans; Hypoglycemic Agents; Peroxisomes; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors

2000
Regulation of Ca(2+)-activated K+ currents by ciglitazone in rat pituitary GH3 cells.
    Journal of investigative medicine : the official publication of the American Federation for Clinical Research, 2000, Volume: 48, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium; Hypoglycemic Agents; Membrane Potentials; Pituitary Gland; Potassium Channels; Rats; Thiazoles; Thiazolidinediones; Tumor Cells, Cultured

2000
Oxidized low density lipoprotein inhibits interleukin-12 production in lipopolysaccharide-activated mouse macrophages via direct interactions between peroxisome proliferator-activated receptor-gamma and nuclear factor-kappa B.
    The Journal of biological chemistry, 2000, Oct-20, Volume: 275, Issue:42

    Topics: Animals; Cells, Cultured; DNA-Binding Proteins; Female; Gene Expression Regulation; HeLa Cells; Humans; Hypoglycemic Agents; Interleukin-12; Lipopolysaccharides; Lipoproteins, LDL; Macrophages; Mice; Mice, Inbred DBA; NF-kappa B; Receptors, Cytoplasmic and Nuclear; Spleen; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Transfection

2000
Down-regulation of uncoupling protein-3 and -2 by thiazolidinediones in C2C12 myotubes.
    FEBS letters, 2000, Oct-27, Volume: 484, Issue:1

    Topics: Acyl-CoA Dehydrogenase; Animals; Atorvastatin; Bezafibrate; Carnitine O-Palmitoyltransferase; Carrier Proteins; Cell Line; Cholesterol; Chromans; Down-Regulation; Fatty Acid Desaturases; Heptanoic Acids; Hypoglycemic Agents; Ion Channels; Ligands; Membrane Transport Proteins; Mice; Mitochondrial Proteins; Muscles; Oleic Acid; Peroxisome Proliferators; Proteins; Pyrimidines; Pyrroles; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Triazenes; Troglitazone; Uncoupling Protein 2; Uncoupling Protein 3

2000
The use of explant lens culture to assess cataractogenic potential.
    Annals of the New York Academy of Sciences, 2000, Volume: 919

    Topics: Adenosine Triphosphate; Aminooxyacetic Acid; Animals; Benzopyrans; Biotransformation; Cataract; Drug-Related Side Effects and Adverse Reactions; Glutathione; Lens, Crystalline; Lipoxygenase Inhibitors; Male; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Thiazoles; Thiazolidinediones; Toxicity Tests; Xenobiotics

2000
Peroxisome proliferator activator receptor-gamma agonists and 15-deoxy-Delta(12,14)(12,14)-PGJ(2) induce apoptosis in normal and malignant B-lineage cells.
    Journal of immunology (Baltimore, Md. : 1950), 2000, Dec-15, Volume: 165, Issue:12

    Topics: Animals; Apoptosis; B-Lymphocytes; Cell Lineage; Cells, Cultured; Chromans; Dinoprost; Hypoglycemic Agents; Lymphoma, B-Cell; Male; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred DBA; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone; Tumor Cells, Cultured

2000
Delayed activation of PPARgamma by LPS and IFN-gamma attenuates the oxidative burst in macrophages.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2001, Volume: 15, Issue:2

    Topics: Animals; Cell Line; Cell Survival; Cells, Cultured; Escherichia coli; Genes, Reporter; Humans; Hypoglycemic Agents; Interferon-gamma; Lipopolysaccharides; Luciferases; Macrophages; Mice; Microbodies; Monocytes; NG-Nitroarginine Methyl Ester; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Recombinant Proteins; Respiratory Burst; Rosiglitazone; Tetradecanoylphorbol Acetate; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection

2001
Synergistic potentiation of thiazolidinedione-induced ST 13 preadipocyte differentiation by RAR synergists.
    Biochemical and biophysical research communications, 2001, Jan-26, Volume: 280, Issue:3

    Topics: Adipocytes; Aminobenzoates; Animals; Benzazepines; Benzoates; Bexarotene; Cell Differentiation; Cell Line; Dibenzazepines; Ligands; Mice; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection

2001
A cyclopentenone prostaglandin activates mesangial MAP kinase independently of PPARgamma.
    Biochemical and biophysical research communications, 2001, Feb-16, Volume: 281, Issue:1

    Topics: Cells, Cultured; Cyclopentanes; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glomerular Mesangium; Humans; Hypoglycemic Agents; Immunologic Factors; JNK Mitogen-Activated Protein Kinases; Ligands; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Prostaglandin D2; Prostaglandins; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors

2001
Antihyperglycemic activity of new 1,2,4-oxadiazolidine-3,5-diones.
    European journal of medicinal chemistry, 2001, Volume: 36, Issue:1

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Type 2; Disease Models, Animal; Female; Hypoglycemic Agents; Insulin; Male; Mice; Mice, Obese; Oxadiazoles; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

2001
The nuclear receptor PPAR gamma is expressed by mouse T lymphocytes and PPAR gamma agonists induce apoptosis.
    European journal of immunology, 2001, Volume: 31, Issue:4

    Topics: Animals; Antigen Presentation; Apoptosis; Cell Division; Cell Survival; Cells, Cultured; Chromans; Flow Cytometry; Immunohistochemistry; In Situ Nick-End Labeling; Ionomycin; Ligands; Lymphocyte Activation; Mice; Mice, Inbred BALB C; Mice, Transgenic; Prostaglandin D2; Pyrimidines; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Specific Pathogen-Free Organisms; T-Lymphocytes; Tetradecanoylphorbol Acetate; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2001
Peroxisome proliferator-activated receptor-gamma regulates airway epithelial cell activation.
    American journal of respiratory cell and molecular biology, 2001, Volume: 24, Issue:6

    Topics: Adjuvants, Immunologic; Cytokines; Down-Regulation; Humans; Inflammation Mediators; Interleukin-4; Interleukin-8; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Respiratory Mucosa; RNA, Messenger; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors

2001
Identification of a peroxisome-proliferator-activated-receptor response element in the apolipoprotein E gene control region.
    The Biochemical journal, 2001, Jul-15, Volume: 357, Issue:Pt 2

    Topics: Animals; Apolipoproteins E; Astrocytoma; Base Sequence; Binding Sites; CCAAT-Enhancer-Binding Protein-beta; CCAAT-Enhancer-Binding Protein-delta; CCAAT-Enhancer-Binding Proteins; Cell Line; Consensus Sequence; DNA-Binding Proteins; Gene Expression Regulation; Glioblastoma; Introns; Luciferases; Macrophages; Microbodies; Molecular Sequence Data; Protein Biosynthesis; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Transfection; Tumor Cells, Cultured

2001
TZDs inhibit vascular smooth muscle cell growth independently of the cyclin kinase inhibitors p21 and p27.
    American journal of physiology. Endocrinology and metabolism, 2001, Volume: 281, Issue:2

    Topics: Animals; Becaplermin; CDC2-CDC28 Kinases; Cell Cycle Proteins; Cell Division; Cells, Cultured; Culture Media, Serum-Free; Cyclin D1; Cyclin E; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinase 4; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cyclin-Dependent Kinases; Cyclins; DNA; Enzyme Inhibitors; Muscle, Smooth, Vascular; Oligonucleotides, Antisense; Platelet-Derived Growth Factor; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-sis; Rats; Receptors, Cytoplasmic and Nuclear; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Suppressor Proteins

2001
Inhibitors of arachidonic acid metabolism potentiate tumour necrosis factor-alpha-induced apoptosis in HL-60 cells.
    European journal of pharmacology, 2001, Jul-13, Volume: 424, Issue:1

    Topics: Apoptosis; Arachidonic Acid; Caspase 3; Caspases; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Cytochrome c Group; Cytosol; Dose-Response Relationship, Drug; Drug Synergism; HL-60 Cells; Humans; Indomethacin; Isoenzymes; Masoprocol; Membrane Proteins; Peroxisome Proliferators; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin; Tumor Necrosis Factor-alpha

2001
Activation of the PPAR pathway induces apoptosis and COX-2 inhibition in HT-29 human colon cancer cells.
    Carcinogenesis, 2001, Volume: 22, Issue:9

    Topics: Alitretinoin; Antineoplastic Agents; Apoptosis; Cell Division; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; DNA Fragmentation; Down-Regulation; Drug Synergism; Enzyme-Linked Immunosorbent Assay; Genes, cdc; HT29 Cells; Humans; Isoenzymes; Membrane Proteins; Prostaglandin-Endoperoxide Synthases; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin

2001
trans-10,cis-12-Conjugated linoleic acid reduces leptin secretion from 3T3-L1 adipocytes.
    Biochemical and biophysical research communications, 2001, Sep-21, Volume: 287, Issue:2

    Topics: 3T3 Cells; Adipocytes; Animals; Antioxidants; Hypoglycemic Agents; Leptin; Linoleic Acid; Male; Masoprocol; Mice; Mice, Inbred ICR; Thiazoles; Thiazolidinediones

2001
Prostaglandin-J2 induces synthesis of interleukin-8 by endothelial cells in a PPAR-gamma-independent manner.
    Prostaglandins & other lipid mediators, 2001, Volume: 66, Issue:3

    Topics: Cell Line; Cell Survival; Electrophoretic Mobility Shift Assay; Endothelium, Vascular; Humans; Interleukin-8; Ligands; NF-kappa B; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection; Up-Regulation

2001
Stimulated release of arachidonic acid by agonists of the peroxisome proliferator-activated receptor and retinoic acid receptors.
    Prostaglandins, leukotrienes, and essential fatty acids, 2001, Volume: 65, Issue:4

    Topics: Alitretinoin; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Celecoxib; Cell Line; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Drug Synergism; Indomethacin; Kinetics; Liver; Prostaglandin D2; Prostaglandins A; Pyrazoles; Rats; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Sulfonamides; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin

2001
15-deoxy-delta12,14-prostaglandin J2-induced apoptosis in amnion-like WISH cells.
    Prostaglandins & other lipid mediators, 2001, Volume: 66, Issue:4

    Topics: Amino Acid Chloromethyl Ketones; Amnion; Apoptosis; Caspase Inhibitors; Caspases; Cell Survival; Cells, Cultured; Cysteine Proteinase Inhibitors; Enzyme Activation; Humans; Hypoglycemic Agents; Immunologic Factors; Ligands; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Rosiglitazone; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors

2001
Peroxisome proliferator-activated receptor gamma agonists inhibit HIV-1 replication in macrophages by transcriptional and post-transcriptional effects.
    The Journal of biological chemistry, 2002, May-10, Volume: 277, Issue:19

    Topics: Cell Line; Cells, Cultured; Dactinomycin; Dose-Response Relationship, Drug; HeLa Cells; HIV-1; Humans; Hypoglycemic Agents; Macrophages; Plasmids; Promoter Regions, Genetic; Prostaglandins A; Protein Synthesis Inhibitors; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA Processing, Post-Transcriptional; RNA-Directed DNA Polymerase; RNA, Messenger; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors; Transcription, Genetic; Transfection; U937 Cells

2002
Regulation of cytokine expression by ligands of peroxisome proliferator activated receptors.
    Journal of immunology (Baltimore, Md. : 1950), 2002, Mar-15, Volume: 168, Issue:6

    Topics: Adjuvants, Immunologic; Animals; Concanavalin A; Cytokines; Female; Interleukin-4; Ligands; Lymphocyte Activation; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Microbodies; Promoter Regions, Genetic; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Receptors, IgE; RNA, Messenger; Spleen; T-Lymphocytes; Thiazoles; Thiazolidinediones; Transcription Factors; Up-Regulation

2002
Dualism of oxidized lipoproteins in provoking and attenuating the oxidative burst in macrophages: role of peroxisome proliferator-activated receptor-gamma.
    Journal of immunology (Baltimore, Md. : 1950), 2002, Mar-15, Volume: 168, Issue:6

    Topics: Animals; Cell Line; Cells, Cultured; Humans; Linoleic Acids; Linoleic Acids, Conjugated; Lipoproteins, LDL; Macrophage Activation; Macrophages; Mice; Monocytes; Reactive Oxygen Species; Receptors, Cytoplasmic and Nuclear; Respiratory Burst; Thiazoles; Thiazolidinediones; Transcription Factors; U937 Cells

2002
15-Deoxy-Delta12,14-prostaglandin J2 regulates mesangial cell proliferation and death.
    Kidney international, 2002, Volume: 61, Issue:4

    Topics: 1-Phosphatidylinositol 4-Kinase; Cell Death; Cell Division; Cells, Cultured; Chromans; Chromones; Enzyme Inhibitors; Glomerular Mesangium; Humans; Morpholines; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2002
Enhanced growth inhibition by combination differentiation therapy with ligands of peroxisome proliferator-activated receptor-gamma and inhibitors of histone deacetylase in adenocarcinoma of the lung.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2002, Volume: 8, Issue:4

    Topics: Adenocarcinoma; Basic Helix-Loop-Helix Leucine Zipper Transcription Factors; Blotting, Western; Carcinoma, Non-Small-Cell Lung; Cell Differentiation; Cell Division; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; DNA-Binding Proteins; Dose-Response Relationship, Drug; Drug Synergism; Gelsolin; Gene Expression Regulation, Neoplastic; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Hydroxamic Acids; Ligands; Lung Neoplasms; Phenylbutyrates; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; RNA; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Cells, Cultured

2002
Peroxisome proliferator-activated receptor-gamma agonists inhibit experimental allergic encephalomyelitis by blocking IL-12 production, IL-12 signaling and Th1 differentiation.
    Genes and immunity, 2002, Volume: 3, Issue:2

    Topics: Animals; Cell Differentiation; Cells, Cultured; DNA-Binding Proteins; Dose-Response Relationship, Drug; Encephalomyelitis, Autoimmune, Experimental; Immunologic Factors; Interleukin-12; Janus Kinase 2; Kinetics; Lymphocyte Activation; Macrophages; Mice; Microglia; Myelin Basic Protein; Prostaglandin D2; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Spinal Cord; Th1 Cells; Thiazoles; Thiazolidinediones; Transcription Factors

2002
Ligands of peroxisome proliferator-activated receptor-gamma increase the generation of vascular endothelial growth factor in vascular smooth muscle cells and in macrophages.
    Acta biochimica Polonica, 2000, Volume: 47, Issue:4

    Topics: Animals; Antineoplastic Agents; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Endothelial Growth Factors; Endothelium, Vascular; Hypoglycemic Agents; Interleukin-1; Ligands; Lipopolysaccharides; Lymphokines; Macrophages; Mice; Muscle, Smooth; Promoter Regions, Genetic; Prostaglandin D2; Rats; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation; Transfection; Up-Regulation; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Nuclear receptor agonists as potential differentiation therapy agents for human osteosarcoma.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2002, Volume: 8, Issue:5

    Topics: Alitretinoin; Antineoplastic Agents; Apoptosis; Cell Differentiation; Cell Division; Chromans; Dose-Response Relationship, Drug; Drug Synergism; Gene Expression Regulation, Neoplastic; HT29 Cells; Humans; Osteosarcoma; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Neoplasm; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors; Tretinoin; Troglitazone; Tumor Cells, Cultured

2002
Effects of peroxisome proliferator-activated receptor agonists on LPS-induced neuronal death in mixed cortical neurons: associated with iNOS and COX-2.
    Brain research, 2002, Jun-21, Volume: 941, Issue:1-2

    Topics: Animals; Cell Culture Techniques; Cell Death; Chromans; Clofibrate; Cyclooxygenase 2; Dinoprostone; Electrophoretic Mobility Shift Assay; Escherichia coli; Immunohistochemistry; In Situ Nick-End Labeling; Isoenzymes; Lipopolysaccharides; Mice; Mice, Inbred ICR; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Peroxisome Proliferators; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2002
MAP kinase cascades are activated in astrocytes and preadipocytes by 15-deoxy-Delta(12-14)-prostaglandin J(2) and the thiazolidinedione ciglitazone through peroxisome proliferator activator receptor gamma-independent mechanisms involving reactive oxygenat
    The Journal of biological chemistry, 2002, Aug-16, Volume: 277, Issue:33

    Topics: Adipocytes; Animals; Astrocytes; Cells, Cultured; Enzyme Activation; MAP Kinase Signaling System; Prostaglandin D2; Rats; Reactive Oxygen Species; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors

2002
PPAR activators inhibit endothelial cell migration by targeting Akt.
    Biochemical and biophysical research communications, 2002, May-24, Volume: 293, Issue:5

    Topics: Apoptosis; Blotting, Western; Cell Movement; Cells, Cultured; Chromans; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Fenofibrate; Flavonoids; Humans; Hypoglycemic Agents; Hypolipidemic Agents; In Situ Nick-End Labeling; Lipid Metabolism; Lymphokines; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Peroxisome Proliferators; Phosphatidylinositol 3-Kinases; Phosphorylation; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors; Troglitazone; Umbilical Veins; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Vasodilator Agents

2002
Induction of apoptosis in human and rat glioma by agonists of the nuclear receptor PPARgamma.
    Journal of neurochemistry, 2002, Volume: 81, Issue:5

    Topics: Animals; Apoptosis; bcl-2-Associated X Protein; bcl-Associated Death Protein; Cadherins; Carrier Proteins; Cell Division; Cell Survival; DNA Fragmentation; Drug Evaluation, Preclinical; Glioma; Humans; Nuclear Proteins; Oligonucleotides, Antisense; Prostaglandin D2; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Pyrimidines; Rats; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Cells, Cultured

2002
Thiazolidinedione activation of peroxisome proliferator-activated receptor gamma can enhance mitochondrial potential and promote cell survival.
    The Journal of biological chemistry, 2002, Aug-30, Volume: 277, Issue:35

    Topics: Animals; Cell Death; Cell Survival; Cells, Cultured; Humans; Hypoglycemic Agents; Interleukin-3; Lymphocyte Activation; Membrane Potentials; Mice; Mice, Inbred C57BL; Mitochondria; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Recombinant Proteins; Rosiglitazone; T-Lymphocytes; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection; Up-Regulation

2002
Superoxide anion-dependent Raf/MEK/ERK activation by peroxisome proliferator activated receptor gamma agonists 15-deoxy-delta(12,14)-prostaglandin J(2), ciglitazone, and GW1929.
    Experimental cell research, 2002, Jul-15, Volume: 277, Issue:2

    Topics: Animals; Benzophenones; Cell Line; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Peroxisomes; Phosphatidylinositol 3-Kinases; Phosphorylation; Prostaglandin D2; Protein Kinase C; Proto-Oncogene Proteins c-raf; ras Proteins; Reactive Oxygen Species; Receptors, Cytoplasmic and Nuclear; Superoxides; Thiazoles; Thiazolidinediones; Transcription Factors; Tyrosine

2002
Ligands of the peroxisome proliferator-activated receptors (PPAR-gamma and PPAR-alpha) reduce myocardial infarct size.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2002, Volume: 16, Issue:9

    Topics: Adult; Animals; Cardiotonic Agents; Cell Adhesion Molecules; Cell Line; Cells, Cultured; Chemokine CCL2; Clofibrate; Heme Oxygenase (Decyclizing); Heme Oxygenase-1; Humans; Ligands; Male; Membrane Proteins; Myocardial Infarction; Myocardial Reperfusion Injury; Pioglitazone; Prostaglandin D2; Prostaglandins A; Protein Isoforms; Pyrimidines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors

2002
Inhibitory effect of peroxisome proliferator-activated receptor-gamma ligands on the expression of IgE heavy chain germline transcripts in the human B cell line DND39.
    Biochemical and biophysical research communications, 2002, Jul-12, Volume: 295, Issue:2

    Topics: B-Lymphocytes; Cell Line; Germ Cells; Humans; Immunoglobulin E; Immunoglobulin Heavy Chains; Interleukin-4; Ligands; Phosphorylation; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; STAT6 Transcription Factor; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors

2002
Ciglitazone inhibits plasmin-induced proinflammatory monocyte activation via modulation of p38 MAP kinase activity.
    Thrombosis and haemostasis, 2002, Volume: 88, Issue:2

    Topics: Chemotaxis, Leukocyte; Fibrinolysin; Humans; Inflammation; Interleukin-1; Mitogen-Activated Protein Kinases; Monocytes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Necrosis Factor-alpha

2002
Glitazones regulate glutamine metabolism by inducing a cellular acidosis in MDCK cells.
    American journal of physiology. Endocrinology and metabolism, 2002, Volume: 283, Issue:4

    Topics: Acidosis; Alanine Transaminase; Animals; Cell Line; Chromans; Epithelial Cells; Glutamine; Hydrogen-Ion Concentration; Hypoglycemic Agents; Kidney; L-Lactate Dehydrogenase; Nitrogen; Nitrogen Isotopes; Rosiglitazone; Thiazoles; Thiazolidinediones; Troglitazone

2002
Thiazolidinediones as a novel class of NAD(+)-dependent 15-hydroxyprostaglandin dehydrogenase inhibitors.
    Archives of biochemistry and biophysics, 2002, Sep-15, Volume: 405, Issue:2

    Topics: Drug Evaluation, Preclinical; Enzyme Inhibitors; Hydroxyprostaglandin Dehydrogenases; Imipramine; Kinetics; NAD; Structure-Activity Relationship; Thiazoles; Thiazolidinediones

2002
Peroxisome proliferator-activated receptor ligands negatively regulate the expression of the high-affinity IgE receptor Fc epsilon RI in human basophilic KU812 cells.
    Biochemical and biophysical research communications, 2002, Sep-20, Volume: 297, Issue:2

    Topics: Basophils; Flow Cytometry; Histamine Release; Humans; Ligands; Mast Cells; Peroxisome Proliferators; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Receptors, IgE; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Cells, Cultured

2002
Apoptosis induced by activation of peroxisome-proliferator activated receptor-gamma is associated with Bcl-2 and NF-kappaB in human colon cancer.
    Life sciences, 2002, Apr-19, Volume: 70, Issue:22

    Topics: Apoptosis; Cell Division; Cell Survival; Colon; Colonic Neoplasms; DNA-Binding Proteins; Electrophoretic Mobility Shift Assay; HT29 Cells; Humans; Hypoglycemic Agents; Immunoenzyme Techniques; Immunologic Factors; Ligands; NF-kappa B; Promoter Regions, Genetic; Prostaglandin D2; Proto-Oncogene Proteins c-bcl-2; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic

2002
Stimulation of peroxisome proliferator-activated receptors alpha and gamma blocks HIV-1 replication and TNFalpha production in acutely infected primary blood cells, chronically infected U1 cells, and alveolar macrophages from HIV-infected subjects.
    Journal of acquired immune deficiency syndromes (1999), 2002, Sep-01, Volume: 31, Issue:1

    Topics: Acquired Immunodeficiency Syndrome; Anti-HIV Agents; Cell Line; Chromans; Fenofibrate; HIV-1; Humans; Leukocytes, Mononuclear; Macrophages, Alveolar; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone; Tumor Necrosis Factor-alpha; Virus Replication

2002
Inhibitory effects of peroxisome poliferator-activated receptor gamma on thyroid carcinoma cell growth.
    The Journal of clinical endocrinology and metabolism, 2002, Volume: 87, Issue:10

    Topics: Apoptosis; Cell Cycle Proteins; Cell Division; Cyclin-Dependent Kinase Inhibitor p27; Cyclin-Dependent Kinases; DNA Mutational Analysis; Gene Expression; Humans; Mutation; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; Sequence Analysis, DNA; Thiazoles; Thiazolidinediones; Thyroid Gland; Thyroid Neoplasms; Transcription Factors; Transfection; Tumor Cells, Cultured; Tumor Suppressor Proteins

2002
Characterization of sucrose-induced changes in cardiac phenotype.
    Pflugers Archiv : European journal of physiology, 2002, Volume: 445, Issue:1

    Topics: Animals; Calcium; Dietary Sucrose; Heart; Hypoglycemic Agents; Imidazoles; Insulin; Myosin Heavy Chains; Phenotype; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Sympatholytics; Thiazoles; Thiazolidinediones; Ventricular Myosins

2002
Leptin induces endothelial cell migration through Akt, which is inhibited by PPARgamma-ligands.
    Hypertension (Dallas, Tex. : 1979), 2002, Volume: 40, Issue:5

    Topics: Androstadienes; Cell Line; Cell Movement; Chemotaxis; Chromans; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Leptin; Ligands; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphoric Monoester Hydrolases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; PTEN Phosphohydrolase; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone; Tumor Suppressor Proteins; Wortmannin

2002
Inhibition of NAD+-dependent 15-hydroxyprostaglandin dehydrogenase (15-PGDH) by cyclooxygenase inhibitors and chemopreventive agents.
    Prostaglandins, leukotrienes, and essential fatty acids, 2002, Volume: 67, Issue:6

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Hydroxyprostaglandin Dehydrogenases; Inhibitory Concentration 50; Isoenzymes; Kinetics; Membrane Proteins; NAD; Placenta; Prostaglandin-Endoperoxide Synthases; Thiazoles; Thiazolidinediones

2002
Peroxisome proliferator-activated receptor gamma-mediated NF-kappa B activation and apoptosis in pre-B cells.
    Journal of immunology (Baltimore, Md. : 1950), 2002, Dec-15, Volume: 169, Issue:12

    Topics: Animals; Apoptosis; B-Lymphocytes; Bone Marrow Cells; Cell Line; Cell Line, Transformed; Male; Mice; Mice, Inbred C57BL; NF-kappa B; Oxazoles; Peroxisome Proliferators; Peroxisomes; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Signal Transduction; Stem Cells; Thiazoles; Thiazolidinediones; Transcription Factors; Tyrosine

2002
Cyclooxygenase-2 expression by nonsteroidal anti-inflammatory drugs in human airway smooth muscle cells: role of peroxisome proliferator-activated receptors.
    Journal of immunology (Baltimore, Md. : 1950), 2003, Jan-15, Volume: 170, Issue:2

    Topics: Adjuvants, Immunologic; Anti-Inflammatory Agents, Non-Steroidal; Cell Line; Cell Survival; Cyclooxygenase 2; Dexamethasone; Dinoprostone; Flurbiprofen; Humans; Indomethacin; Isoenzymes; Lung; Membrane Proteins; Muscle, Smooth; NF-kappa B; Nitrobenzenes; Promoter Regions, Genetic; Prostaglandin Antagonists; Prostaglandin D2; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Protein Transport; Receptors, Cytoplasmic and Nuclear; Response Elements; Sulfonamides; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation

2003
Peroxisome proliferator-activated receptor gamma ligands increase release of nitric oxide from endothelial cells.
    Arteriosclerosis, thrombosis, and vascular biology, 2003, Jan-01, Volume: 23, Issue:1

    Topics: Animals; Aorta; Cells, Cultured; Endothelium, Vascular; Enzyme Induction; Humans; Immunologic Factors; Ligands; Nitric Oxide; Nitric Oxide Synthase; Prostaglandin D2; Pulmonary Artery; Receptors, Cytoplasmic and Nuclear; Swine; Thiazoles; Thiazolidinediones; Transcription Factors; Umbilical Veins

2003
The genomic organization of mouse resistin reveals major differences from the human resistin: functional implications.
    Gene, 2003, Feb-13, Volume: 305, Issue:1

    Topics: 3T3 Cells; Animals; Base Sequence; Binding Sites; DNA; Exons; Genes; Hormones, Ectopic; Humans; Intercellular Signaling Peptides and Proteins; Introns; Luciferases; Mice; Molecular Sequence Data; Nerve Growth Factor; Protein Binding; Proteins; Recombinant Fusion Proteins; Resistin; Sequence Analysis, DNA; Thiazoles; Thiazolidinediones; Transfection

2003
Activation of peroxisome proliferator-activated receptors in human airway smooth muscle cells has a superior anti-inflammatory profile to corticosteroids: relevance for chronic obstructive pulmonary disease therapy.
    Journal of immunology (Baltimore, Md. : 1950), 2003, Mar-01, Volume: 170, Issue:5

    Topics: Adolescent; Adult; Anti-Inflammatory Agents; Apoptosis; Blotting, Western; Cell Division; Cells, Cultured; Dexamethasone; DNA Fragmentation; Female; Granulocyte Colony-Stimulating Factor; Granulocyte-Macrophage Colony-Stimulating Factor; Growth Inhibitors; Humans; Interleukin-1; Ligands; Male; Middle Aged; Muscle, Smooth; Peroxisomes; Prostaglandin D2; Protein Isoforms; Pulmonary Disease, Chronic Obstructive; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Trachea; Transcription Factors

2003
15-Deoxy-Delta(12,14)-prostaglandin J2 inhibits the expression of proinflammatory genes in human blood monocytes via a PPAR-gamma-independent mechanism.
    Biochemical and biophysical research communications, 2003, Mar-07, Volume: 302, Issue:2

    Topics: Cyclooxygenase 2; Gene Expression; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Immunologic Factors; In Vitro Techniques; Inflammation; Interleukin-1; Interleukin-6; Isoenzymes; Lipopolysaccharides; Membrane Proteins; Monocytes; Prostaglandin D2; Prostaglandin-Endoperoxide Synthases; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Necrosis Factor-alpha

2003
Thiazolidinediones, a class of anti-diabetic drugs, inhibit Id2 expression through a PPARgamma-independent pathway in human aortic smooth muscle cells.
    Cellular and molecular life sciences : CMLS, 2003, Volume: 60, Issue:1

    Topics: Anilides; Aorta; Chromans; DNA-Binding Proteins; Dose-Response Relationship, Drug; Down-Regulation; Gene Expression Regulation; Humans; Hypoglycemic Agents; Inhibitor of Differentiation Protein 2; Muscle, Smooth, Vascular; Oxazoles; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; RNA, Messenger; Thiazoles; Thiazolidinediones; Time Factors; Transcription Factors; Troglitazone; Tyrosine

2003
Increased expression of the lipocalin 24p3 as an apoptotic mechanism for MK886.
    The Biochemical journal, 2003, May-15, Volume: 372, Issue:Pt 1

    Topics: Acute-Phase Proteins; Animals; Apoptosis; Carcinogens; Caspase 3; Caspases; Gene Expression Regulation; Indoles; Lipocalin-2; Lipocalins; Lipoxygenase Inhibitors; Mice; Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Pyrimidines; Thiazoles; Thiazolidinediones

2003
Peroxisome proliferator-activated receptor gamma agonists induce proteasome-dependent degradation of cyclin D1 and estrogen receptor alpha in MCF-7 breast cancer cells.
    Cancer research, 2003, Mar-01, Volume: 63, Issue:5

    Topics: Breast Neoplasms; Cell Division; Cyclin D1; Cysteine Endopeptidases; Down-Regulation; Estrogen Receptor alpha; G1 Phase; Humans; Multienzyme Complexes; Prostaglandin D2; Proteasome Endopeptidase Complex; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; RNA, Messenger; S Phase; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured; Ubiquitin

2003
Cytokine regulation by peroxisome proliferator-activated receptor gamma in human endometrial cells.
    Fertility and sterility, 2003, Volume: 79 Suppl 1

    Topics: Benzophenones; Colony-Stimulating Factors; Cytokines; Endometrium; Epithelial Cells; Female; Humans; Interleukin-6; Ligands; Phenylacetates; Prostaglandin D2; Protein Array Analysis; Protein Isoforms; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Tyrosine

2003
Thiazolidinedione inhibition of peritoneal inflammation.
    Gynecologic and obstetric investigation, 2003, Volume: 55, Issue:1

    Topics: Animals; Chemokine CCL5; Disease Models, Animal; Endometriosis; Female; Interleukin-1; Leukocyte Count; Macrophages, Peritoneal; Mice; Mice, Inbred C57BL; Peritonitis; Peroxisome Proliferators; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Thioglycolates; Tumor Necrosis Factor-alpha

2003
Suppression of gastric mucosal inflammatory responses to Helicobacter pylori lipopolysaccharide by peroxisome proliferator-activated receptor gamma activation.
    IUBMB life, 2002, Volume: 53, Issue:6

    Topics: Animals; Apoptosis; Cyclooxygenase 2; Gastric Mucosa; Gastritis; Helicobacter pylori; Inflammation; Isoenzymes; Ligands; Lipopolysaccharides; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors

2002
Peroxisome proliferator-activated receptor gamma ligand inhibits cell growth and invasion of human pancreatic cancer cells.
    International journal of gastrointestinal cancer, 2002, Volume: 32, Issue:1

    Topics: 3T3 Cells; Adenocarcinoma; alpha Catenin; Animals; Antineoplastic Agents; Apoptosis; beta Catenin; Cadherins; Caspase 3; Caspase 8; Caspase 9; Caspases; Cell Cycle; Cell Cycle Proteins; Cell Division; Collagen; Cyclin D1; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cyclins; Cyclooxygenase 2; Cytoskeletal Proteins; Drug Combinations; Enzyme Induction; Gene Expression Regulation, Neoplastic; Humans; Isoenzymes; Laminin; Ligands; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Membrane Proteins; Mice; Neoplasm Invasiveness; Neoplasm Proteins; Pancreatic Neoplasms; Prostaglandin D2; Prostaglandin-Endoperoxide Synthases; Proteoglycans; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors; Tumor Cells, Cultured; Tumor Suppressor Proteins

2002
Inhibition of proliferation and estrogen receptor signaling by peroxisome proliferator-activated receptor gamma ligands in uterine leiomyoma.
    Cancer research, 2003, Mar-15, Volume: 63, Issue:6

    Topics: Animals; Cell Division; Chromans; Docosahexaenoic Acids; Estradiol; Female; Humans; Leiomyoma; Ligands; Prostaglandin D2; Protein Isoforms; Rats; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; Signal Transduction; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone; Tumor Cells, Cultured; Uterine Neoplasms

2003
Activation-induced PPARgamma expression sensitizes primary human T cells toward apoptosis.
    Journal of leukocyte biology, 2003, Volume: 73, Issue:5

    Topics: Apoptosis; Cysteine Proteinase Inhibitors; Gene Expression Regulation; Humans; Hydrazines; Jurkat Cells; Lymphocyte Activation; Lymphopenia; Nitrogen Oxides; Phytohemagglutinins; Promoter Regions, Genetic; Prostaglandin D2; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; T-Lymphocytes; Thiazoles; Thiazolidinediones; Transcription Factors

2003
The antiproliferative effects of PPARgamma ligands in normal human mammary epithelial cells.
    Breast cancer research and treatment, 2003, Volume: 78, Issue:2

    Topics: Apoptosis; Breast; Cell Cycle; Cell Division; Cells, Cultured; Epithelial Cells; Female; Gene Expression; Humans; Hypoglycemic Agents; Ligands; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; Thiazoles; Thiazolidinediones; Transcription Factors

2003
Effects of peroxisome proliferator-activated receptor gamma ligands ciglitazone and 15-deoxy-delta 12,14-prostaglandin J2 on rat cultured cerebellar granule neuronal viability.
    Journal of neuroscience research, 2003, Jun-15, Volume: 72, Issue:6

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Dose-Response Relationship, Drug; Gene Expression Regulation; Ligands; Neurons; Prostaglandin D2; Proto-Oncogene Proteins c-jun; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors

2003
Peroxisome proliferator-activated receptor-gamma upregulates caveolin-1 and caveolin-2 expression in human carcinoma cells.
    Oncogene, 2003, Jun-19, Volume: 22, Issue:25

    Topics: Adenocarcinoma; Antigens, Differentiation; Antigens, Neoplasm; Breast Neoplasms; Caveolin 1; Caveolin 2; Caveolins; Cell Differentiation; Cell Line; Chromans; Colonic Neoplasms; Dimerization; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Gene Expression Regulation, Neoplastic; Genes, Dominant; Humans; Kidney; Ligands; Macromolecular Substances; Membrane Microdomains; Neoplasm Proteins; Phenotype; Phenylacetates; Prostaglandin D2; Protein Structure, Tertiary; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; RNA, Neoplasm; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Troglitazone; Tumor Cells, Cultured

2003
Regulation of retinoic acid receptor beta expression by peroxisome proliferator-activated receptor gamma ligands in cancer cells.
    Cancer research, 2003, Jul-01, Volume: 63, Issue:13

    Topics: Apoptosis; Benzoates; Breast Neoplasms; Cell Division; Female; Gene Expression Regulation, Neoplastic; Humans; Ligands; Lung Neoplasms; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoids; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Cells, Cultured

2003
Homocysteine mediated expression and secretion of monocyte chemoattractant protein-1 and interleukin-8 in human monocytes.
    Circulation research, 2003, Aug-22, Volume: 93, Issue:4

    Topics: Antioxidants; Cells, Cultured; Chemokine CCL2; Chromans; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Genistein; Homocysteine; Humans; Imidazoles; Indoles; Interleukin-8; Monocytes; Naphthalenes; Onium Compounds; Pyridines; Pyrrolidines; Reactive Oxygen Species; RNA, Messenger; Sulfonamides; Thiazoles; Thiazolidinediones; Thiocarbamates; Time Factors; Troglitazone; Tyrphostins

2003
Peroxisome proliferator-activated receptors alpha and gamma down-regulate allergic inflammation and eosinophil activation.
    The Journal of experimental medicine, 2003, Aug-04, Volume: 198, Issue:3

    Topics: Anilides; Animals; Asthma; Chemotaxis; Disease Models, Animal; DNA-Binding Proteins; Down-Regulation; Eosinophils; GATA3 Transcription Factor; Humans; Inflammation; Lung; Mice; Mice, Inbred BALB C; Mice, Knockout; Rats; Receptors, Cytoplasmic and Nuclear; Respiratory Hypersensitivity; Rosiglitazone; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors

2003
Oleoylethanolamide, an endogenous PPAR-alpha agonist, lowers body weight and hyperlipidemia in obese rats.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Animals; Body Weight; Butyrates; CD36 Antigens; Cholesterol; Coenzyme A Ligases; Eating; Endocannabinoids; Fatty Acid-Binding Proteins; Hepatocytes; Hyperlipidemias; Ion Channels; Liver; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mitochondrial Proteins; Obesity; Oleic Acids; Phenylurea Compounds; PPAR alpha; Pyrimidines; Rats; Rats, Inbred WF; Rats, Zucker; RNA, Messenger; Thiazoles; Thiazolidinediones; Triglycerides; Uncoupling Protein 2

2005
Inhibition of adult liver progenitor (oval) cell growth and viability by an agonist of the peroxisome proliferator activated receptor (PPAR) family member gamma, but not alpha or delta.
    Carcinogenesis, 2005, Volume: 26, Issue:10

    Topics: Animals; Cell Division; Cell Line; Cell Survival; Ethionine; Liver; Male; Mice; Mice, Inbred C57BL; PPAR alpha; PPAR gamma; Receptors, Cytoplasmic and Nuclear; Stem Cells; Thiazoles; Thiazolidinediones

2005
Mono(2-ethylhexyl)phthalate and mono-n-butyl phthalate activation of peroxisome proliferator activated-receptors alpha and gamma in breast.
    Toxicology letters, 2006, Jun-01, Volume: 163, Issue:3

    Topics: Breast Neoplasms; Butyrates; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Diethylhexyl Phthalate; Dose-Response Relationship, Drug; Female; Humans; Phenylurea Compounds; Phthalic Acids; Plasticizers; PPAR alpha; PPAR gamma; PPAR-beta; Statistics, Nonparametric; Thiazoles; Thiazolidinediones; Transfection

2006
Thiazolidinediones inhibit albumin uptake by proximal tubular cells through a mechanism independent of peroxisome proliferator activated receptor gamma.
    American journal of nephrology, 2006, Volume: 26, Issue:1

    Topics: Albumins; Anilides; Animals; Cells, Cultured; Cholesterol; Chromans; Farnesol; Kidney Tubules, Proximal; Ligands; Mevalonic Acid; Opossums; Polyisoprenyl Phosphates; PPAR gamma; Rosiglitazone; Thiazoles; Thiazolidinediones; Thiazolidines; Troglitazone

2006
Inhibitory effect of meloxicam, a selective cyclooxygenase-2 inhibitor, and ciglitazone, a peroxisome proliferator-activated receptor gamma ligand, on the growth of human ovarian cancers.
    Cancer, 2007, Aug-15, Volume: 110, Issue:4

    Topics: Animals; Apoptosis; Ascites; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dinoprostone; Female; Humans; Immunohistochemistry; Intramolecular Oxidoreductases; Meloxicam; Mice; Mice, Inbred BALB C; Mice, Nude; Ovarian Neoplasms; Peritoneal Neoplasms; PPAR gamma; Prostaglandin-E Synthases; Survival Analysis; Thiazines; Thiazoles; Thiazolidinediones; Vascular Endothelial Growth Factor A; Xenograft Model Antitumor Assays

2007
PPAR and LXR activators regulate ABCA12 expression in human keratinocytes.
    The Journal of investigative dermatology, 2008, Volume: 128, Issue:1

    Topics: ATP-Binding Cassette Transporters; Cells, Cultured; DNA-Binding Proteins; Dose-Response Relationship, Drug; Epidermis; Gene Expression Regulation; Humans; Keratinocytes; Liver X Receptors; Orphan Nuclear Receptors; Permeability; Peroxisome Proliferator-Activated Receptors; Receptors, Calcitriol; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones

2008
Peroxisome proliferator-activated receptor-gamma and retinoid X receptor agonists synergistically suppress proliferation of immortalized endometrial stromal cells.
    Fertility and sterility, 2009, Volume: 91, Issue:5 Suppl

    Topics: Cell Division; Cell Line; Endometrium; Estradiol; Female; Humans; Nicotinic Acids; PPAR gamma; Progesterone; Retinoid X Receptors; Stromal Cells; Tetrahydronaphthalenes; Tetrazolium Salts; Thiazoles; Thiazolidinediones

2009
Peroxisome-proliferator-activated receptors γ and β/δ mediate vascular endothelial growth factor production in colorectal tumor cells.
    Journal of cancer research and clinical oncology, 2011, Volume: 137, Issue:1

    Topics: Cell Line, Tumor; Colorectal Neoplasms; Cyclooxygenase 2; Humans; Peroxisome Proliferator-Activated Receptors; PPAR delta; PPAR gamma; PPAR-beta; RNA, Messenger; Thiazoles; Thiazolidinediones; Vascular Endothelial Growth Factor A

2011
The use of rat lens explant cultures to study the mechanism of drug-induced cataractogenesis.
    Toxicological sciences : an official journal of the Society of Toxicology, 2012, Volume: 126, Issue:1

    Topics: Acetates; Animals; Cataract; Cell Survival; Eye Proteins; Gene Expression Profiling; Gene Expression Regulation; Lens, Crystalline; Male; Oligonucleotide Array Sequence Analysis; Oxidative Stress; PPAR delta; Rats; Rats, Wistar; RNA, Messenger; Thiazoles; Thiazolidinediones; Tissue Culture Techniques

2012
Study of the interactions between Edaglitazone and Ciglitazone with PPARγ and their antiplatelet profile.
    Life sciences, 2017, Oct-01, Volume: 186

    Topics: Binding Sites; Blood Platelets; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Healthy Volunteers; Humans; Ligands; Molecular Docking Simulation; Molecular Structure; Oxazoles; Platelet Aggregation; Platelet Aggregation Inhibitors; PPAR gamma; Protein Binding; Thiazoles; Thiazolidinediones

2017