Page last updated: 2024-09-02

ci 988 and chlordiazepoxide

ci 988 has been researched along with chlordiazepoxide in 5 studies

Compound Research Comparison

Studies
(ci 988)
Trials
(ci 988)
Recent Studies (post-2010)
(ci 988)
Studies
(chlordiazepoxide)
Trials
(chlordiazepoxide)
Recent Studies (post-2010) (chlordiazepoxide)
1478143,962385104

Protein Interaction Comparison

ProteinTaxonomyci 988 (IC50)chlordiazepoxide (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.216
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)1.1
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.216
Histamine H1 receptorHomo sapiens (human)1.795
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.216
GABA theta subunitRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.216

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barrett, JE; Powell, KR1
Field, MJ; Hughes, J; Lewis, AS; Singh, L; Woodruff, GN1
Boyce, S; Rupniak, NM; Webb, JK1
Birkemo, LS; Ervin, GN; Johnson, MF; Mosher, JT1
Brown, P; Field, M; Hinks, GL; Hughes, J; Poat, JA1

Other Studies

5 other study(ies) available for ci 988 and chlordiazepoxide

ArticleYear
Evaluation of the effects of PD 134308 (CI-988), a CCK-B antagonist, on the punished responding of squirrel monkeys.
    Neuropeptides, 1991, Volume: 19 Suppl

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Chlordiazepoxide; Electroshock; Indoles; Male; Meglumine; Punishment; Receptors, Cholecystokinin; Saimiri

1991
Evidence for an involvement of the brain cholecystokinin B receptor in anxiety.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, Feb-15, Volume: 88, Issue:4

    Topics: Animals; Anxiety; Benzodiazepinones; Cerebral Ventricles; Ceruletide; Chlordiazepoxide; Cholecystokinin; Devazepide; Indoles; Injections, Intraventricular; Male; Meglumine; Pentagastrin; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin

1991
Inhibition of pentagastrin-induced pressor response in conscious rats by the CCK-B receptor antagonist CI-988 and chlordiazepoxide.
    Regulatory peptides, 1996, Jan-16, Volume: 61, Issue:1

    Topics: Animals; Blood Pressure; Carbolines; Chlordiazepoxide; Hormone Antagonists; Indoles; Male; Meglumine; Pentagastrin; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin

1996
Several roles of CCKA and CCKB receptor subtypes in CCK-8-induced and LiCl-induced taste aversion conditioning.
    Peptides, 1996, Volume: 17, Issue:3

    Topics: Animals; Benzodiazepinones; Chlordiazepoxide; Conditioning, Psychological; Devazepide; Dose-Response Relationship, Drug; Hormone Antagonists; Indoles; Lithium Chloride; Male; Meglumine; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Taste

1996
The anxiolytics CI-988 and chlordiazepoxide fail to reduce immediate early gene mRNA stimulation following exposure to the rat elevated X-maze.
    European journal of pharmacology, 1996, Sep-26, Volume: 312, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Chlordiazepoxide; Gene Expression Regulation; Genes, Immediate-Early; Indoles; Male; Meglumine; Rats; RNA, Messenger; Transcriptional Activation

1996