choline and vesamicol

choline has been researched along with vesamicol in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199010 (34.48)18.7374
1990's14 (48.28)18.2507
2000's5 (17.24)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Wagner, G; Walczok, A; Wessler, I1
Collier, B; Gomez, MV; Prado, MA1
Van der Kloot, W; Yu, SP1
Gildersleeve, DL; Jung, YW; Van Dort, ME; Wieland, DM1
Diebler, MF; Gaudry-Talarmain, YM; O'Regan, S1
Vizi, ES1
Collier, B; Mykita, S1
Suszkiw, JB; Toth, G1
Cabeza, R; Collier, B1
Carroll, PT; Ivy, MT1
Bahr, BA; Parsons, SM1
Johnson, GV; Jope, RS1
Collier, B; Welner, SA1
Meyer, EM; Otero, DH; Wilbekin, F1
Diebler, MF; Meunier, FM; O'Regan, S; Vyas, S1
Suidan, HS; Tolkovsky, AM1
Efange, SM; Khare, AB; Michelson, RH; Thomas, JR1
Nakamura, S; Ohno, T1
Bonanno, G; Fassio, A; Fontana, G; Marchi, M; Raiteri, M; Usai, C1
Balezina, OP; Naves, LA; Van der Kloot, W1
Naves, LA; Van der Kloot, W1
Fitzgerald, RS; Ishizawa, Y; Shirahata, M1
Kobayashi, H; Saitoh, S; Suzuki, T; Takeno, K; Watanabe, T; Yasufuku, T1
Eaton, BM; Sooranna, SR1
Auld, DS; Day, JC; Mennicken, F; Quirion, R2
Carroll, PT; Roghani, A1
Jin, H; Kopke, RD; Sha, D; Wu, JY1
Bravo, DT; Kolmakova, NG; Parsons, SM1

Other Studies

29 other study(ies) available for choline and vesamicol

ArticleYear
Suppression by cholinesterase inhibition of a Ca(2+)-independent efflux of [3H]acetylcholine from the neuromuscular junction of the isolated rat diaphragm.
    European journal of pharmacology, 1992, Oct-20, Volume: 221, Issue:2-3

    Topics: Acetylcholine; Animals; Calcium; Choline; Cholinesterase Inhibitors; Diaphragm; Female; In Vitro Techniques; Male; Neuromuscular Junction; Physostigmine; Piperidines; Potassium Chloride; Rats; Rats, Sprague-Dawley; Tritium

1992
Mobilization of the readily releasable pool of acetylcholine from a sympathetic ganglion by tityustoxin in the presence of vesamicol.
    Journal of neurochemistry, 1992, Volume: 59, Issue:2

    Topics: Acetylcholine; Animals; Cats; Choline; Electric Stimulation; Female; Ganglia, Sympathetic; Male; Neuromuscular Depolarizing Agents; Piperidines; Scorpion Venoms; Tritium

1992
Increasing quantal size at the mouse neuromuscular junction and the role of choline.
    The Journal of physiology, 1991, Volume: 433

    Topics: Acetylcholine; Animals; Anura; Choline; Curare; Electric Stimulation; Female; Hormones; Hypertonic Solutions; In Vitro Techniques; Kinetics; Male; Mice; Models, Neurological; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Piperidines; Sodium; Species Specificity; Synapses

1991
A radiotracer for mapping cholinergic neurons of the brain.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:8

    Topics: Acetylcholine; Animals; Brain; Cerebellum; Cerebral Cortex; Choline; Corpus Striatum; Female; Iodine Radioisotopes; Kinetics; Mice; Molecular Structure; Neurons; Phencyclidine; Piperidines; Stereoisomerism; Tetrahydronaphthalenes; Tritium

1990
Compared effects of two vesicular acetylcholine uptake blockers, AH5183 and cetiedil, on cholinergic functions in Torpedo synaptosomes: acetylcholine synthesis, choline transport, vesicular uptake, and evoked acetylcholine release.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Acetylcholine; Animals; Azepines; Biological Transport; Calcimycin; Choline; Electric Organ; Hydrogen-Ion Concentration; Kinetics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo

1989
In favour of the vesicular hypothesis: neurochemical evidence that vesamicol (AH5183) inhibits stimulation-evoked release of acetylcholine from neuromuscular junction.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Acetylcholine; Animals; Calcium; Choline; Diaphragm; Electric Stimulation; In Vitro Techniques; Male; Mice; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Phencyclidine; Phrenic Nerve; Piperidines

1989
Acetylcholine synthesis by a sympathetic ganglion in the presence of 2-(4-phenylpiperidino)cyclohexanol (AH5183) and picrylsulfonic acid.
    Journal of neurochemistry, 1989, Volume: 52, Issue:6

    Topics: Acetylcholine; Animals; Cats; Choline; Drug Combinations; Electric Stimulation; Female; Ganglia, Sympathetic; Male; Neuromuscular Depolarizing Agents; Nitrobenzenes; Osmolar Concentration; Phencyclidine; Piperidines; Trinitrobenzenesulfonic Acid

1989
Storage and release of acetylcholine in rat cortical synaptosomes: effects of D,L-2-(4-phenylpiperidino)cyclohexanol (AH5183).
    Brain research, 1986, Oct-29, Volume: 386, Issue:1-2

    Topics: Acetylcholine; Animals; Calcium; Cerebral Cortex; Choline; Cholinergic Fibers; Phencyclidine; Piperidines; Potassium; Rats; Synaptic Transmission; Synaptosomes

1986
Acetylcholine mobilization in a sympathetic ganglion in the presence and absence of 2-(4-phenylpiperidino)cyclohexanol (AH5183).
    Journal of neurochemistry, 1988, Volume: 50, Issue:1

    Topics: Acetylcholine; Animals; Black Widow Spider; Cats; Choline; Electric Stimulation; Female; Ganglia, Sympathetic; Kinetics; Male; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Spider Venoms; Tritium

1988
Effect of 2-(4-phenylpiperidino)cyclohexanol (AH 5183) on the veratridine-induced increase in acetylcholine synthesis by rat hippocampal tissue.
    Journal of neurochemistry, 1988, Volume: 51, Issue:3

    Topics: Acetylcholine; Animals; Choline; Choline O-Acetyltransferase; Hippocampus; Isotonic Solutions; L-Lactate Dehydrogenase; Male; Naphthylvinylpyridine; Octoxynol; Phencyclidine; Piperidines; Polyethylene Glycols; Rats; Rats, Inbred Strains; Solubility; Subcellular Fractions; Veratridine; Veratrine

1988
Demonstration of a receptor in Torpedo synaptic vesicles for the acetylcholine storage blocker L-trans-2-(4-phenyl[3,4-3H]-piperidino) cyclohexanol.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:7

    Topics: Acetylcholine; Animals; Binding, Competitive; Choline; Electric Organ; Kinetics; Phencyclidine; Piperidines; Receptors, Drug; Stereoisomerism; Synaptic Vesicles; Torpedo

1986
Quinacrine and 2-(4-phenylpiperidino)cyclohexanol (AH5183) inhibit acetylcholine release and synthesis in rat brain slices.
    Molecular pharmacology, 1986, Volume: 29, Issue:1

    Topics: Acetylcholine; Animals; Biological Transport; Brain; Choline; In Vitro Techniques; Kinetics; Male; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Potassium; Quinacrine; Rats; Rats, Inbred Strains

1986
Accumulation, acetylation, and releasability of diethylhomocholine from a sympathetic ganglion.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Acetylation; Acetylcholine; Animals; Calcium; Cats; Choline; Electric Stimulation; Female; Ganglia, Sympathetic; Magnesium; Male; Neuromuscular Depolarizing Agents; Phencyclidine; Physostigmine; Piperidines

1985
Effects of 4-(2-hydroxyethyl)-1-piperazine-ethanesulfonic acid (AH5183) on rat cortical synaptosome choline uptake, acetylcholine storage and release.
    Brain research, 1985, Dec-16, Volume: 359, Issue:1-2

    Topics: Acetylcholine; Animals; Cerebral Cortex; Choline; In Vitro Techniques; Male; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Synaptosomes

1985
A Ewing's sarcoma cell line showing some, but not all, of the traits of a cholinergic neuron.
    Journal of neurochemistry, 1995, Volume: 64, Issue:1

    Topics: Acetylcholine; Adult; Calcium-Binding Proteins; Choline; Choline O-Acetyltransferase; Cholinergic Fibers; Humans; Male; Membrane Glycoproteins; Nerve Tissue Proteins; Neuromuscular Depolarizing Agents; Neurons; Piperidines; Proteolipids; RNA, Messenger; Sarcoma, Ewing; Synaptotagmin I; Synaptotagmins; Tritium; Tumor Cells, Cultured; Tyrosine 3-Monooxygenase

1995
Sympathetic neurons expressing cholinergic properties are poised to allocate choline symmetrically between acetylcholine and the phosphatidylcholine-generating pathway in growing neurites.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:3

    Topics: Acetylcholine; Animals; Animals, Newborn; Biological Transport; Cells, Cultured; Choline; Choline O-Acetyltransferase; Ganglia, Sympathetic; Kinetics; Meglumine; Neurites; Neuromuscular Depolarizing Agents; Neurons; Organ Culture Techniques; Phosphatidylcholines; Piperidines; Potassium; Rats; Time Factors; Tritium

1993
Synthesis and tissue distribution of (m-[125I]iodobenzyl)trozamicol ([125I]MIBT): potential radioligand for mapping central cholinergic innervation.
    Journal of medicinal chemistry, 1993, Jun-11, Volume: 36, Issue:12

    Topics: Animals; Autoradiography; Brain; Cerebellum; Cerebral Cortex; Choline; Corpus Striatum; Iodine Radioisotopes; Iodobenzenes; Isotope Labeling; Kinetics; Male; Molecular Structure; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Tissue Distribution

1993
Spatial learning impairment in aged rats: comparing between aged basal forebrain lesioned and normal aged rats.
    Behavioural brain research, 1995, Volume: 70, Issue:1

    Topics: Acetylcholinesterase; Aging; Animals; Aziridines; Cerebral Cortex; Choline; Choline O-Acetyltransferase; Coloring Agents; Kinetics; Male; Maze Learning; Neuromuscular Blocking Agents; Piperidines; Prosencephalon; Rats; Rats, Inbred F344; Space Perception

1995
Role of external and internal calcium on heterocarrier-mediated transmitter release.
    Journal of neurochemistry, 1996, Volume: 66, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Carrier Proteins; Chelating Agents; Choline; Clonidine; Dopamine; Dopamine Agonists; Egtazic Acid; Ergolines; GABA Modulators; Hippocampus; Male; Muscarinic Agonists; Neostriatum; Neuromuscular Depolarizing Agents; Neurons; Neurotransmitter Agents; Norepinephrine; Oxotremorine; Piperidines; Presynaptic Terminals; Quinpirole; Rats; Rats, Sprague-Dawley; Synaptosomes; Tritium; Yohimbine

1996
Monoethylcholine as a false transmitter precursor at the frog and mouse neuromuscular junctions.
    Brain research, 1996, Aug-19, Volume: 730, Issue:1-2

    Topics: Animals; Choline; Cholinesterase Inhibitors; Edrophonium; Electric Stimulation; Hemicholinium 3; Methylamines; Mice; Mice, Inbred Strains; Neostigmine; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Neurotransmitter Agents; Neurotransmitter Uptake Inhibitors; Piperidines; Prodrugs; Rana pipiens

1996
Transmitter packaging at frog neuromuscular junctions exposed to anticholinesterases; the role of second-stage acetylcholine loading.
    Journal of neurophysiology, 1996, Volume: 76, Issue:4

    Topics: Acetylcholine; Analysis of Variance; Animals; Choline; Cholinesterase Inhibitors; Motor Endplate; Neostigmine; Neuromuscular Depolarizing Agents; Piperidines; Rana pipiens

1996
The presynaptic component of a cholinergic mechanism in the carotid body chemotransduction of hypoxia in the cat.
    Advances in experimental medicine and biology, 1996, Volume: 410

    Topics: Acetyl Coenzyme A; Acetylcholine; Animals; Azepines; Carotid Body; Carrier Proteins; Cats; Cell Hypoxia; Choline; Choline O-Acetyltransferase; Enzyme Inhibitors; Glossopharyngeal Nerve; Hemicholinium 3; Hypoxia; Membrane Transport Proteins; Models, Neurological; Naphthylvinylpyridine; Nerve Tissue Proteins; Piperidines; Pyridines; Receptors, Presynaptic; Signal Transduction; Synaptic Vesicles

1996
Effects of systemic administration of 2-(4-phenyl-piperidino)-cyclohexanol (vesamicol) and an organophosphate DDVP on the cholinergic system in brain regions of rats.
    Brain research bulletin, 1997, Volume: 43, Issue:1

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Brain; Choline; Choline O-Acetyltransferase; Dichlorvos; Injections, Intraperitoneal; Male; Neuromuscular Depolarizing Agents; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Subcellular Fractions

1997
Regulation of the choline transport system in superfused microcarrier cultures of BeWo cells.
    Placenta, 1998, Volume: 19, Issue:8

    Topics: Bethanechol; Biological Transport; Choline; Choriocarcinoma; Drug Carriers; Female; Hemicholinium 3; Humans; Microvilli; Naphthalenes; Neostigmine; Nicotine; Physostigmine; Piperidines; Quaternary Ammonium Compounds; Trophoblasts; Tumor Cells, Cultured; Uterine Neoplasms

1998
Pharmacological characterization of endogenous acetylcholine release from primary septal cultures.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:2

    Topics: Acetylcholine; Animals; Cells, Cultured; Choline; Choline O-Acetyltransferase; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Muscarinic Agonists; Neuromuscular Depolarizing Agents; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Rats; Septum of Brain; Time Factors; Veratridine

2000
Neurotrophins differentially enhance acetylcholine release, acetylcholine content and choline acetyltransferase activity in basal forebrain neurons.
    Journal of neurochemistry, 2001, Volume: 77, Issue:1

    Topics: Acetylcholine; Animals; Biological Transport; Calcium Channel Blockers; Carrier Proteins; Cells, Cultured; Choline; Choline O-Acetyltransferase; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Membrane Transport Proteins; Nerve Growth Factors; Neuromuscular Depolarizing Agents; Neurons; Piperidines; Potassium; Prosencephalon; Rats; Rats, Sprague-Dawley; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

2001
Analysis of uptake and release of newly synthesized acetylcholine in PC12 cells overexpressing the rat vesicular acetylcholine transporter (VAChT).
    Brain research. Molecular brain research, 2002, Apr-30, Volume: 100, Issue:1-2

    Topics: Acetates; Acetylcholine; Animals; Brain Chemistry; Carbon Radioisotopes; Carrier Proteins; Central Nervous System; Choline; Choline O-Acetyltransferase; Clone Cells; Cloning, Molecular; Gene Expression Regulation; Membrane Potentials; Membrane Transport Proteins; Neuromuscular Depolarizing Agents; PC12 Cells; Piperidines; Potassium; Presynaptic Terminals; Rats; Subcellular Fractions; Synaptic Membranes; Synaptic Transmission; Synaptic Vesicles; Transfection; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

2002
Choline acetyltransferase: regulation and coupling with protein kinase and vesicular acetylcholine transporter on synaptic vesicles.
    Neurochemical research, 2004, Volume: 29, Issue:1

    Topics: Adenosine Triphosphate; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Choline; Choline O-Acetyltransferase; Enzyme Activation; Enzyme Inhibitors; Gramicidin; Membrane Transport Proteins; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Swine; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

2004
Choline is transported by vesicular acetylcholine transporter.
    Journal of neurochemistry, 2004, Volume: 91, Issue:3

    Topics: Acetylcholine; Animals; Binding, Competitive; Biological Transport; Carbon Radioisotopes; Choline; Intracellular Membranes; Membrane Transport Proteins; PC12 Cells; Piperidines; Quaternary Ammonium Compounds; Radioligand Assay; Rats; Subcellular Fractions; Tritium; Vesicular Acetylcholine Transport Proteins

2004