choline and epibatidine

choline has been researched along with epibatidine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's8 (72.73)29.6817
2010's2 (18.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baydyuk, M; Davis, HE; Kellar, KJ; Wang, HP; Xiao, Y1
Frølund, B; Jensen, AA; Krogsgaard-Larsen, P; Liljefors, T1
Gurley, DA; Lanthorn, TH1
Markus, RP; Reno, LA; Santos, JM; Zago, W1
Matsumoto, A; Matsuyama, S1
Jones, IW; Pullar, IA; Rousseau, SJ; Wonnacott, S1
Grilli, M; Marchi, M; Parodi, M; Patti, L; Raiteri, L; Raiteri, M1
Hone, A; Innocent, N; Kimura, A; Livingstone, PD; McIntosh, JM; Whiteaker, P; Wonnacott, S; Young, T1
Gandía, L; García, AG; García-Eguiagaray, J; Tapia, L1
Abitbol, M; Ascher, P; Baud, F; Bernard, V; Cendelin, J; Farar, V; Fournet, V; Houze, P; Hrabovska, A; Klein, J; Krejci, E; Lamotte d'Incamps, B; Legrand, M; Leroy, J; Mohr, F; Myslivecek, J; Plaud, B; Tuma, J; Zimmermann, M1
He, YX; Qi, JS; Wu, MN; Zhang, H1

Reviews

1 review(s) available for choline and epibatidine

ArticleYear
Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Humans; Ligands; Mice; Mice, Knockout; Models, Molecular; Molecular Sequence Data; Nicotinic Agonists; Nicotinic Antagonists; Protein Conformation; Protein Subunits; Receptors, Nicotinic

2005

Other Studies

10 other study(ies) available for choline and epibatidine

ArticleYear
Pharmacology of the agonist binding sites of rat neuronal nicotinic receptor subtypes expressed in HEK 293 cells.
    Bioorganic & medicinal chemistry letters, 2004, Apr-19, Volume: 14, Issue:8

    Topics: Animals; Binding Sites; Binding, Competitive; Cell Line; Gene Expression; Humans; Neurons; Nicotinic Agonists; Protein Subunits; Rats; Receptors, Nicotinic; Transfection

2004
Nicotinic agonists competitively antagonize serotonin at mouse 5-HT3 receptors expressed in Xenopus oocytes.
    Neuroscience letters, 1998, May-15, Volume: 247, Issue:2-3

    Topics: Acetylcholine; Animals; Bacterial Toxins; Benzylidene Compounds; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Choline; Cyanobacteria Toxins; Dimethylphenylpiperazinium Iodide; DNA, Complementary; Female; Marine Toxins; Mice; Microcystins; Multigene Family; Nicotine; Nicotinic Agonists; Oocytes; Patch-Clamp Techniques; Pyridines; Receptors, Nicotinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Recombinant Fusion Proteins; Serotonin Antagonists; Structure-Activity Relationship; Xenopus laevis

1998
Melatonin nocturnal surge modulates nicotinic receptors and nicotine-induced [3H]glutamate release in rat cerebellum slices.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:2

    Topics: Adrenergic beta-Antagonists; alpha7 Nicotinic Acetylcholine Receptor; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Choline; Circadian Rhythm; Darkness; Glutamic Acid; In Vitro Techniques; Light; Male; Melatonin; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Propranolol; Pyridines; Rats; Rats, Wistar; Receptors, Nicotinic

2003
Epibatidine induces long-term potentiation (LTP) via activation of alpha4beta2 nicotinic acetylcholine receptors (nAChRs) in vivo in the intact mouse dentate gyrus: both alpha7 and alpha4beta2 nAChRs essential to nicotinic LTP.
    Journal of pharmacological sciences, 2003, Volume: 93, Issue:2

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Bridged Bicyclo Compounds, Heterocyclic; Choline; Dentate Gyrus; Drug Synergism; In Vitro Techniques; Long-Term Potentiation; Mecamylamine; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Receptors, Nicotinic

2003
Presynaptic alpha7 and non-alpha7 nicotinic acetylcholine receptors modulate [3H]d-aspartate release from rat frontal cortex in vitro.
    Neuropharmacology, 2005, Volume: 49, Issue:1

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Animals, Newborn; Aspartic Acid; Azetidines; Bacterial Toxins; Bridged Bicyclo Compounds, Heterocyclic; Bungarotoxins; Calcium; Choline; Cyanobacteria Toxins; Dicarboxylic Acids; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Frontal Lobe; Immunohistochemistry; In Vitro Techniques; Male; Marine Toxins; Mecamylamine; Microcystins; Microscopy, Confocal; Neurotransmitter Uptake Inhibitors; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Phosphopyruvate Hydratase; Potassium Chloride; Pyridines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Presynaptic; Synaptosomes; Time Factors; Tritium; Tropanes

2005
P2X(7) receptors exert a permissive role on the activation of release-enhancing presynaptic alpha7 nicotinic receptors co-existing on rat neocortex glutamatergic terminals.
    Neuropharmacology, 2006, Volume: 50, Issue:6

    Topics: Adenosine Triphosphate; alpha7 Nicotinic Acetylcholine Receptor; Analysis of Variance; Animals; Aspartic Acid; Bridged Bicyclo Compounds, Heterocyclic; Bungarotoxins; Choline; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; Enzyme Activation; Glutamic Acid; In Vitro Techniques; Magnesium; Male; Neocortex; Nicotine; Nicotinic Agonists; Presynaptic Terminals; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Time Factors; Tritium

2006
Alpha-conotoxin Arenatus IB[V11L,V16D] [corrected] is a potent and selective antagonist at rat and human native alpha7 nicotinic acetylcholine receptors.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:2

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Calcium; Choline; Conotoxins; Dopamine; Humans; Isoxazoles; Male; Nicotinic Antagonists; PC12 Cells; Phenylurea Compounds; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Spiro Compounds

2008
Preconditioning stimuli that augment chromaffin cell secretion.
    American journal of physiology. Cell physiology, 2009, Volume: 296, Issue:4

    Topics: Acetylcholine; Adrenal Glands; Animals; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Catecholamines; Cattle; Cells, Cultured; Choline; Chromaffin Cells; Dose-Response Relationship, Drug; Mecamylamine; Methacholine Chloride; Muscarinic Agonists; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Potassium; Pyridines; Receptors, Muscarinic; Receptors, Nicotinic; Sympathetic Nervous System; Time Factors

2009
Near-complete adaptation of the PRiMA knockout to the lack of central acetylcholinesterase.
    Journal of neurochemistry, 2012, Volume: 122, Issue:5

    Topics: Acetylcholine; Acetylcholinesterase; Adaptation, Physiological; Animals; Animals, Newborn; Body Temperature; Brain; Bridged Bicyclo Compounds, Heterocyclic; Bungarotoxins; Choline; Cholinergic Agents; Cholinesterase Inhibitors; Collagen; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Exploratory Behavior; Gait; Gene Expression Regulation; In Vitro Techniques; Maze Learning; Membrane Potentials; Membrane Proteins; Mice; Mice, Knockout; Microdialysis; Motor Activity; Muscarinic Antagonists; Muscle Proteins; Nails, Ingrown; Neostigmine; Nerve Tissue Proteins; Neurons; Pirenzepine; Protein Binding; Pyridines; Radioisotopes; Receptors, Muscarinic; Rotarod Performance Test; Scopolamine; Spinal Cord; Statistics, Nonparametric; Tritium

2012
Amyloid β-protein suppressed nicotinic acetylcholine receptor-mediated currents in acutely isolated rat hippocampal CA1 pyramidal neurons.
    Synapse (New York, N.Y.), 2013, Volume: 67, Issue:1

    Topics: Amyloid beta-Peptides; Animals; Bridged Bicyclo Compounds, Heterocyclic; CA1 Region, Hippocampal; Choline; Membrane Potentials; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Pyramidal Cells; Pyridines; Rats; Rats, Wistar; Receptors, Nicotinic

2013