cholic acid and int-777

cholic acid has been researched along with int-777 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Auwerx, J; Gioiello, A; Macchiarulo, A; Natalini, B; Pastorini, E; Pellicciari, R; Pruzanski, M; Roda, A; Rosatelli, E; Sardella, R; Schoonjans, K; Thomas, C1
Adorini, L; Colliva, C; Gioiello, A; Macchiarulo, A; Nuti, R; Pellicciari, R; Pruzanski, M; Rizzo, G; Roda, A; Sabbatini, P; Venturoni, F1
Auwerx, J; De Franco, F; Ferrari, C; Giacchè, N; Gioiello, A; Macchiarulo, A; Nuti, R; Pellicciari, R; Pols, TW; Pruzanski, M; Schoonjans, K; Thomas, C1
Carotti, A; Colliva, C; De Franco, F; Filipponi, P; Franco, P; Gadaleta, RM; Gioiello, A; Macchiarulo, A; Moschetta, A; Mostarda, S; Passeri, D; Pellicciari, R; Roda, A1

Other Studies

4 other study(ies) available for cholic acid and int-777

ArticleYear
Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesity.
    Journal of medicinal chemistry, 2009, Dec-24, Volume: 52, Issue:24

    Topics: Animals; Chlorocebus aethiops; CHO Cells; Cholic Acids; COS Cells; Cricetinae; Cricetulus; Diabetes Mellitus; Humans; Obesity; Rats; Receptors, G-Protein-Coupled; Stereoisomerism

2009
Avicholic Acid: A Lead Compound from Birds on the Route to Potent TGR5 Modulators.
    ACS medicinal chemistry letters, 2012, Apr-12, Volume: 3, Issue:4

    Topics:

2012
Probing the Binding Site of Bile Acids in TGR5.
    ACS medicinal chemistry letters, 2013, Dec-12, Volume: 4, Issue:12

    Topics:

2013
Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders.
    Journal of medicinal chemistry, 2016, Oct-13, Volume: 59, Issue:19

    Topics:

2016