Page last updated: 2024-09-03

cholestyramine resin and sertraline

cholestyramine resin has been researched along with sertraline in 5 studies

Compound Research Comparison

Studies
(cholestyramine resin)
Trials
(cholestyramine resin)
Recent Studies (post-2010)
(cholestyramine resin)
Studies
(sertraline)
Trials
(sertraline)
Recent Studies (post-2010) (sertraline)
2,6693421903,4801,0281,329

Protein Interaction Comparison

ProteinTaxonomycholestyramine resin (IC50)sertraline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.083
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)0.9848
Muscarinic acetylcholine receptor M2Homo sapiens (human)2.7675
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.6309
Cytochrome P450 3A4Homo sapiens (human)0.8
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.5073
Alpha-2A adrenergic receptorHomo sapiens (human)0.2888
Cytochrome P450 2D6Homo sapiens (human)1.4
Muscarinic acetylcholine receptor M1Homo sapiens (human)1.2882
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)8.3173
Alpha-2B adrenergic receptorHomo sapiens (human)0.1814
Alpha-2C adrenergic receptorHomo sapiens (human)4.477
DRattus norvegicus (Norway rat)0.26
D(3) dopamine receptorRattus norvegicus (Norway rat)0.26
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.8783
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.825
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.26
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.7409
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.083
D(4) dopamine receptorRattus norvegicus (Norway rat)0.26
3-oxo-5-alpha-steroid 4-dehydrogenase 2Homo sapiens (human)0.8
Sodium-dependent serotonin transporterHomo sapiens (human)0.0016
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.1743
Melanocortin receptor 5Homo sapiens (human)4.598
Cytochrome P450 2C19Homo sapiens (human)0.655
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.3935
D(2) dopamine receptorRattus norvegicus (Norway rat)0.26
Sodium-dependent dopamine transporter Homo sapiens (human)0.2175
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)8.3173
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)8.3173
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.0697
TransporterRattus norvegicus (Norway rat)0.26

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Drolz, A; Fuhrmann, V; Trauner, M1
Beuers, U; Bolier, R; Oude Elferink, RP1
Mittal, A1
Debray, D; Gonzales, E; Thébaut, A1
Carrion, AF; Levy, C; Rosen, JD1

Reviews

5 review(s) available for cholestyramine resin and sertraline

ArticleYear
Extracorporeal artificial liver support systems in the management of intractable cholestatic pruritus.
    Liver international : official journal of the International Association for the Study of the Liver, 2011, Volume: 31 Suppl 3

    Topics: Cholestasis; Cholestyramine Resin; Humans; Lysophospholipids; Opioid Peptides; Plasmapheresis; Pruritus; Renal Dialysis; Rifampin; Sertraline; Sorption Detoxification; Ursodeoxycholic Acid

2011
Advances in pathogenesis and treatment of pruritus.
    Clinics in liver disease, 2013, Volume: 17, Issue:2

    Topics: Animals; Anion Exchange Resins; Antibiotics, Antitubercular; Bile Acids and Salts; Cholestasis; Cholestyramine Resin; Humans; Lysophospholipids; Narcotic Antagonists; Pregnane X Receptor; Pruritus; Receptors, Steroid; Rifampin; Selective Serotonin Reuptake Inhibitors; Sertraline; Signal Transduction

2013
Cholestatic Itch Management.
    Current problems in dermatology, 2016, Volume: 50

    Topics: Anion Exchange Resins; Cholagogues and Choleretics; Cholestasis; Cholestyramine Resin; Humans; Lysophospholipids; Naltrexone; Narcotic Antagonists; Plasmapheresis; Pregnane X Receptor; Pruritus; Receptors, Steroid; Rifampin; Selective Serotonin Reuptake Inhibitors; Sertraline; Ultraviolet Therapy; Ursodeoxycholic Acid

2016
[Physiopathology and management of cholestatic pruritus in children].
    Archives de pediatrie : organe officiel de la Societe francaise de pediatrie, 2017, Volume: 24, Issue:7

    Topics: Anion Exchange Resins; Biliary Tract Surgical Procedures; Child; Cholagogues and Choleretics; Cholestasis; Cholestyramine Resin; Chronic Disease; Cytochrome P-450 CYP3A Inducers; Humans; Liver Transplantation; Narcotic Antagonists; Pruritus; Rifampin; Selective Serotonin Reuptake Inhibitors; Sertraline; Sorption Detoxification; Ursodeoxycholic Acid

2017
Understanding and Treating Pruritus in Primary Biliary Cholangitis.
    Clinics in liver disease, 2018, Volume: 22, Issue:3

    Topics: Anion Exchange Resins; Bile Acids and Salts; Cholestyramine Resin; Drainage; Filtration; Humans; Liver Cirrhosis, Biliary; Lysophospholipids; Narcotic Antagonists; Opioid Peptides; Phosphoric Diester Hydrolases; Plasmapheresis; Pruritus; Receptors, Opioid; Rifampin; Selective Serotonin Reuptake Inhibitors; Serotonin; Sertraline; Substance P

2018