Compounds > cholecystokinin (26-33), n-methyl-nle(28,31)-
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cholecystokinin (26-33), n-methyl-nle(28,31)- and sincalide

cholecystokinin (26-33), n-methyl-nle(28,31)- has been researched along with sincalide in 8 studies

Compound Research Comparison

Studies
(cholecystokinin (26-33), n-methyl-nle(28,31)-)		Trials
(cholecystokinin (26-33), n-methyl-nle(28,31)-)		Recent Studies (post-2010)
(cholecystokinin (26-33), n-methyl-nle(28,31)-)		Studies
(sincalide)		Trials
(sincalide)		Recent Studies (post-2010) (sincalide)
8004,01572533

Protein Interaction Comparison

ProteinTaxonomycholecystokinin (26-33), n-methyl-nle(28,31)- (IC50)sincalide (IC50)
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.0006
Cholecystokinin receptor type AHomo sapiens (human)0.0006
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.001
Gastrin/cholecystokinin type B receptorMus musculus (house mouse)0.0008
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.0004

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bergeron, F; Corringer, PJ; Ducos, B; Durieux, C; Roques, BP; Ruiz-Gayo, M1
Ayres, EA; Burks, TF; Fang, S; Hruby, VJ; Kramer, TH; Parkhurst, DN1
Bogert, CL; Fang, SN; Hruby, VJ; Knapp, RJ; Vaughn, LK; Yamamura, HI; Yamamura, MS1
Knapp, RJ; Malatynska, E; Stropova, D; Varga, E; Yamamura, HI1
Davis, TP; Fang, SN; Hruby, VJ; Knapp, RJ; Slaninova, J; Weber, SJ; Yamamura, HI1
Fang, S; Hruby, VJ; Knapp, RJ; Malatynska, E; Peterson, P; Smith, TL; Yamamura, HI; Zalewska, T1
Fang, S; Hashimoto, S; Hruby, VJ; Hunt, M; Knapp, RJ; Malatynska, E; Peterson, P; Wamsley, JK; Yamamura, HI; Zalewska, T1
Debonnel, G; Gronier, B1

Other Studies

8 other study(ies) available for cholecystokinin (26-33), n-methyl-nle(28,31)- and sincalide

ArticleYear
[3H]pBC 264, a suitable probe for studying cholecystokinin-B receptors: binding characteristics in rodent brains and comparison with [3H]SNF 8702.
    Molecular pharmacology, 1992, Volume: 41, Issue:6

    Topics: Amino Acid Sequence; Animals; Binding Sites; Brain; Cats; Cholecystokinin; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Mice; Molecular Sequence Data; Nucleotides; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide; Species Specificity; Tritium

1992
Antinociceptive and gastrointestinal transit effects of cholecystokinin (CCK-8) and related analogs of CCK-8 in the mouse.
    Proceedings of the Western Pharmacology Society, 1991, Volume: 34

    Topics: Amino Acid Sequence; Analgesics; Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Gastric Emptying; Gastrointestinal Transit; Indoles; Male; Mice; Mice, Inbred ICR; Molecular Sequence Data; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Peptide Fragments; Peptides; Phenylurea Compounds; Reaction Time; Receptors, Cholecystokinin; Sincalide

1991
A new, highly selective CCK-B receptor radioligand ([3H][N-methyl-Nle28,31]CCK26-33): evidence for CCK-B receptor heterogeneity.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Guanylyl Imidodiphosphate; Humans; Iodine Radioisotopes; Kinetics; Molecular Sequence Data; Peptide Fragments; Rats; Receptors, Cholecystokinin; Sincalide; Succinimides; Swine; Tritium

1990
The role of the Val353 residue in antagonist binding to rat CCK-B receptors.
    Neuroreport, 1995, Jun-19, Volume: 6, Issue:9

    Topics: Amino Acids; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Mutation; Peptide Fragments; Peptoids; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide; Valine

1995
[125I]SNF 8702: a selective radioligand for CCKB receptors.
    Peptides, 1995, Volume: 16, Issue:2

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Brain; Cell Membrane; Guinea Pigs; Iodine Radioisotopes; Isotope Labeling; Mice; Molecular Sequence Data; Organ Specificity; Pancreas; Peptide Fragments; Radioligand Assay; Receptors, Cholecystokinin; Sincalide; Species Specificity

1995
[N-methylnorleucine-(28,31)]cholecystokinin-(26-33) (SNF 8702) activity at a cloned rat CCKB receptor.
    European journal of pharmacology, 1994, Oct-14, Volume: 269, Issue:2

    Topics: Animals; Base Sequence; Calcium; Cell Line; Cloning, Molecular; DNA, Complementary; Ligands; Molecular Sequence Data; Peptide Fragments; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Cholecystokinin; Sincalide; Spectrometry, Fluorescence

1994
[3H]SNF8702 autoradiography of CCK-B receptors in guinea pig brain and studies with a cloned rat CCK-B receptor.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Animals; Autoradiography; Base Sequence; Brain; Cell Line; Cloning, Molecular; DNA Primers; Guinea Pigs; Molecular Sequence Data; Organ Specificity; Peptide Fragments; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Cholecystokinin; Recombinant Proteins; Sincalide; Transfection; Tritium

1994
CCKB receptors mediate CCK-8S-induced activation of dorsal hippocampus CA3 pyramidal neurons: an in vivo electrophysiological study in the rat.
    Synapse (New York, N.Y.), 1995, Volume: 21, Issue:2

    Topics: Animals; Electrophysiology; Hippocampus; Male; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide

1995