chlorpheniramine and ebastine

chlorpheniramine has been researched along with ebastine in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's6 (66.67)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abou-Gharbia, M; Moyer, JA; Nielsen, ST; Patel, U; Webb, M1
Nagashima, R; Nishikawa, T; Tobita, M1
Sen, S; Sinha, N1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Arai, H; Fujii, T; Higuchi, M; Ido, T; Itoh, M; Iwata, R; Kano, M; Komemushi, S; Matsuda, M; Mizuki, Y; Okamura, N; Sasaki, H; Tagawa, M; Watanabe, T; Yanai, K1
Arai, H; Fujii, T; Higuchi, M; Itoh, M; Kano, M; Komemushi, S; Matsuda, M; Mizuki, Y; Okamura, N; Sasaki, H; Tagawa, M; Watanabe, T; Yanai, K1
Fujisaki, Y; Itoh, Y; Oishi, R1
Fukui, H; Izumi, N; Mizuguchi, H; Ogino, S; Umehara, H1
de Barrio, M; Fuentes, V; Herrero, T; Sánchez, I; Tornero, P; Zubeldia, J1

Trials

2 trial(s) available for chlorpheniramine and ebastine

ArticleYear
Neuroimaging of histamine H1-receptor occupancy in human brain by positron emission tomography (PET): a comparative study of ebastine, a second-generation antihistamine, and (+)-chlorpheniramine, a classical antihistamine.
    British journal of clinical pharmacology, 2001, Volume: 52, Issue:5

    Topics: Adult; Butyrophenones; Carbon Radioisotopes; Cerebral Cortex; Chlorpheniramine; Cross-Over Studies; Histamine H1 Antagonists; Humans; Male; Models, Biological; Piperidines; Receptors, Histamine H1; Single-Blind Method; Thalamus; Tomography, Emission-Computed; Treatment Outcome

2001
Differential cognitive effects of ebastine and (+)-chlorpheniramine in healthy subjects: correlation between cognitive impairment and plasma drug concentration.
    British journal of clinical pharmacology, 2002, Volume: 53, Issue:3

    Topics: Administration, Oral; Adult; Butyrophenones; Chlorpheniramine; Cognition; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Humans; Male; Piperidines; Reaction Time; Sleep; Stereoisomerism; Visual Perception

2002

Other Studies

7 other study(ies) available for chlorpheniramine and ebastine

ArticleYear
New antihistamines: substituted piperazine and piperidine derivatives as novel H1-antagonists.
    Journal of medicinal chemistry, 1995, Sep-29, Volume: 38, Issue:20

    Topics: Animals; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Male; Motor Activity; Piperazines; Piperidines; Rats; Structure-Activity Relationship

1995
A discriminant model constructed by the support vector machine method for HERG potassium channel inhibitors.
    Bioorganic & medicinal chemistry letters, 2005, Jun-02, Volume: 15, Issue:11

    Topics: Animals; CHO Cells; Cricetinae; Discriminant Analysis; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Potassium Channel Blockers; Potassium Channels, Voltage-Gated

2005
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
In vivo evidence for a lack of central effect of ebastine, an antihistaminic agent, in rats: a microdialysis study.
    Japanese journal of pharmacology, 2002, Volume: 90, Issue:4

    Topics: Animals; Butyrophenones; Chlorpheniramine; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Histamine H1 Antagonists; In Vitro Techniques; Male; Microdialysis; Nomifensine; Piperidines; Rats; Rats, Wistar

2002
Analysis of disease-dependent sedative profiles of H(1)-antihistamines by large-scale surveillance using the visual analog scale.
    Methods and findings in experimental and clinical pharmacology, 2008, Volume: 30, Issue:3

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Asthma; Butyrophenones; Cetirizine; Child; Chlorpheniramine; Dermatitis, Atopic; Dibenzazepines; Dibenzoxepins; Female; Histamine H1 Antagonists; Histamine H1 Antagonists, Non-Sedating; Humans; Imidazoles; Japan; Male; Middle Aged; Olopatadine Hydrochloride; Pain Measurement; Piperidines; Population Surveillance; Psychomotor Performance; Pyridines; Quality of Life; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Sleep Stages; Surveys and Questionnaires; Terfenadine; Urticaria

2008
Anaphylaxis to oral iron salts. desensitization protocol for tolerance induction.
    Journal of investigational allergology & clinical immunology, 2008, Volume: 18, Issue:4

    Topics: Aged; Anaphylaxis; Butyrophenones; Chlorpheniramine; Desensitization, Immunologic; Drug Hypersensitivity; Female; Ferrous Compounds; Histamine H1 Antagonists; Humans; Lactates; Piperidines

2008