chloroquine has been researched along with quinacrine in 337 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 253 (75.07) | 18.7374 |
1990's | 26 (7.72) | 18.2507 |
2000's | 32 (9.50) | 29.6817 |
2010's | 21 (6.23) | 24.3611 |
2020's | 5 (1.48) | 2.80 |
Authors | Studies |
---|---|
Denny, WA; Feigon, J; Kearns, DR; Leupin, W | 1 |
Chibale, K; Croft, SL; Fairlamb, AH; Haupt, H; Kendrick, H; Saravanamuthu, A; Yardley, V | 1 |
Elshorst, B; Fiebig, K; Griesinger, C; Grimme, S; Jacobs, DM; Vogtherr, M; Zahn, R | 1 |
Galanakis, D; Ganellin, CR | 1 |
Derisi, JL; Guy, RK; Liou, AP; Madrid, PB; Sherrill, J; Weisman, JL | 1 |
Bellocq, NC; Cheng, J; Davis, ME; Jensen, GS; Kulkarni, RP; Liu, A; Mishra, S; Pun, SH; Zeidan, R | 1 |
Harada, S; Huy, NT; Kamei, K; Maeda, A; Oida, T; Trang, DT; Uyen, DT | 1 |
Beauchene, J; Caffrey, CR; Cohen, FE; Debnath, A; Doyle, PS; Fafarman, AT; Fairlamb, AH; Kelly, B; Land, KM; May, BC; McKerrow, JH; Moll, H; Ponte-Sucre, A; Saravanamuthu, A; Schirmeister, T; Schreiber, K; Steverding, D; Swenerton, RK; Walshe, D; Weisman, JL; Zhou, YM; Zorn, JA | 1 |
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J | 1 |
Fitos, I; Mády, G; Visy, J; Zsila, F | 1 |
Acharya, BN; Kaushik, MP; Saraswat, D | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y | 1 |
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M | 1 |
Bolognesi, ML; Bongarzone, S; Brun, R; Cavalli, A; Lizzi, F; Luise Krauth-Siegel, R | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Glen, RC; Lowe, R; Mitchell, JB | 1 |
Baker, JR; Banaszak Holl, MM; Choi, SK; Harmon, A; Li, MH; Orr, BG; Plantinga, A; Sinniah, K; Witte, A | 1 |
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y | 1 |
Atzpodien, EA; Csato, M; Doessegger, L; Fischer, H; Lenz, B; Schmitt, G; Singer, T | 1 |
Almnayan, D; Lee, H; Solomon, VR | 1 |
Chen, Y; Feng, F; He, S; Jiang, X; Li, Q; Lu, X; Qu, W; Sun, H | 1 |
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P | 1 |
Bernatchez, JA; Li, J; Li, R; Luan, Y; Siqueira-Neto, JL; Tran, LT | 1 |
Byun, SY; Choi, I; Jeon, S; Kim, S; Ko, M; Lee, J; Park, S; Shum, D | 1 |
Kitagawa, T; Matsumoto, A; Terashima, I; Uesono, Y | 1 |
Lampen, JO; Traficante, LJ | 1 |
Rosenberg, LS; Schulman, SG | 1 |
Drenckhahn, D; Lüllmann-Rauch, R | 1 |
Blazsó, G; Kákár, T; Minker, E | 1 |
Cornelis, JJ; Hendrickx, B; Lakhanisky, T; Mouton, RF | 1 |
Frisch, W; Lüllmann-Rauch, R | 3 |
Calberg-Bacq, CM; Cannistraro, S; Piette, J; Van de Vorst, A | 1 |
Calberg-Bacq, CM; Piette, J; Van de Vorst, A | 1 |
Bychkov, MB | 1 |
Dubois, EL | 1 |
Davidson, MW; Jones, RL; Wilson, WD | 1 |
Matejka, Z; Minker, E | 2 |
Garfinkel, E; Hirschman, SZ | 1 |
Fossati, C | 1 |
Boykin, DW; Davidson, MW; Griggs, BG; Wilson, WD | 1 |
Mattock, NM; Peters, W | 1 |
Holbrook, DJ; Washington, ME; Wichard, LP | 1 |
Steigleder, GK | 1 |
Lot, TY | 3 |
Craig, JC; Kirby, GC; Shyamala, V; Warhurst, DC; Webster, RV | 1 |
Barr, R; Branstetter, BA; Crane, FL; Löw, H; Rajnicek, A | 1 |
Desbuquois, B; Dupuis, A; Janicot, M | 1 |
De Boeck, H; Maguire, PA; Sherman, IW; Zidovetzki, R | 1 |
Akera, T; Brody, TM; Ng, YC; Tona, L | 1 |
Kench, JG; Seale, JP; Temple, DM; Tennant, C | 1 |
Safa, AR; Spearman, T; Van Dyke, K; Ye, ZG | 1 |
Filippov, A; Kobrinsky, E; Porotikov, V; Saxon, M; Skatova, G | 1 |
Atiya, A; De Boeck, H; Sherman, IW; Zidovetzki, R | 1 |
Emerole, GO; Nashiru, TO; Thabrew, MI | 1 |
Lanciani, P | 1 |
Beck, WT; Cirtain, MC; Felsted, RL; Glover, CJ; Safa, AR | 1 |
Maroy, B | 1 |
Ha, SH; Shao, BR; Zhan, CQ | 1 |
Imamura, S; Miyachi, Y; Niwa, Y; Yoshioka, A | 1 |
Bell, AL; Betts, WH; Cleland, LG; French, JK; Hurst, NP; Nuki, G; O'Donnell, ML | 1 |
Chanthavanich, P; Edwards, G; Looareesuwan, S; Phillips, RE; Rodick, CL; Supanaranond, W; Warrell, DA | 1 |
Hauser, G; Jadali, F; Kiesel, L; Przylipiak, A; Rabe, T; Runnebaum, B | 1 |
Imamura, S; Miyachi, Y; Yoshioka, A | 1 |
Beck, WT; Pearce, HL; Zamora, JM | 1 |
Shao, BR; Xu, YQ | 1 |
Flayeh, KA | 1 |
Chander, A; Fisher, AB; Reicherter, J | 1 |
Komuniecki, PR; Whitten, JJ | 1 |
Au, AM; Chan, PH; Fishman, RA | 1 |
Ganster, HJ; Mehlhorn, H; Raether, W; Seidenath, H | 1 |
Creus, A; Marcos, R; Velázquez, A; Xamena, N | 1 |
Clark, SK | 1 |
Bohn, E; Hesse, B; Kunze, H; Löffler, BM | 1 |
Kern, HF; Pfab, R; Schachtschabel, DO | 1 |
Clark, JS; Jubb, SN; Maloney, PJ; Young, JM | 1 |
Holmes, J; Sapeika, N; Zwarenstein, H | 2 |
Chou, SC; Conklin, KA; Pan, HY | 1 |
Harinasuta, T; Suntharasamai, P; Viravan, C | 1 |
Chou, SC; Levy, MR | 1 |
Peters, W | 4 |
Boström, H; Whitehouse, MW | 1 |
Benex, J; Lamy, L | 1 |
Jarumilinta, R; Kradolfer, F; Sackmann, W | 1 |
Desmons, F; Gautier, G; Huriez, C | 1 |
Lie, SO; Schofield, B | 1 |
Cowey, FK; Whitehouse, MW | 1 |
Most, H | 1 |
Fain, JN; Pointer, RH | 1 |
Staiger, GR | 1 |
Hadwiger, LA | 1 |
Miller, A; Natsios, G; Smith, HC | 1 |
Abdel-Aziz, A; Idris, IB; Karrar, MA | 1 |
Brown, RK | 1 |
Olatunde, IA | 1 |
Allison, RG; Hahn, FE; Wolfe, AD | 1 |
Briesch, PE; Contacos, PG; Glew, RH; Krotoski, WA; Neva, FA | 1 |
Botha, D | 1 |
Chou, SC; Conklin, KA | 2 |
Gaudin, D; Gregg, RS; Yielding, KL | 1 |
Prasad, BN | 1 |
Sinohara, H | 1 |
Thomas, SC; Warhurst, DC | 1 |
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS | 1 |
Gärding, S; Gösta Henriksson, K; Larsson, JE | 1 |
Dawkins, AT; Stahler, N; Terzian, LA | 1 |
Modell, W | 1 |
Hunsicker, LG | 1 |
Lantz, CH; Saxe, LH; Szustkiewicz, C; Van Dyke, K | 1 |
Schmidt, LH | 1 |
Meier-Ruge, W | 1 |
Hall, SA | 1 |
Ciak, J; Hahn, FE | 1 |
Gorlin, RJ | 1 |
Cook, TM; Hahn, FE; Wolfe, AD | 1 |
Myint, UH; Win, UK | 1 |
Auckland, NL | 1 |
Brede, HD; de Klerk, JN; Groenewald, JH; Murphy, GP; Retief, CP; Schoonees, R; van Heerden, PD; van Zyl, JA; van Zyl, JJ; Weber, HW | 1 |
Brede, HD; de Klerk, JN; Groenewald, JH; Retief, CP; Schoonees, R; van Heerden, PD; van Zyl, JA; van Zyl, JJ; Weber, HW | 1 |
Brede, HD | 1 |
Barnes, MG; Polet, H | 1 |
Barr, CF; Polet, H | 1 |
Fink, E; Kretschmar, W | 1 |
Chou, SC; Conklin, KA; Heu, P | 1 |
Bruce-Chwatt, LJ | 2 |
Lantz, CH; Van Dyke, K | 1 |
Kochen, J; Roth, EF | 1 |
Brynolf, I | 1 |
Hahn, FE; O'Brien, RL; Olenick, JG | 1 |
Ball, EG; Markus, HB | 1 |
Cabanel, G; Chouteau, J; Marchal, A; Voog, R | 1 |
Cenedella, RJ; Saxe, LH; Van Dyke, K | 1 |
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K | 1 |
Polet, H | 1 |
Gregory, KG; Peters, W | 1 |
Nieper, HA | 1 |
Bishop, A | 1 |
Bengtsson, E | 1 |
Buchnícek, J; Turek, B | 1 |
Cheng, CC; Chien, PL | 1 |
Rockwell, DA | 1 |
Dodge, BG; Freeman, RG; Knox, JM | 1 |
Clancy, CF | 1 |
Schneider, MD | 1 |
Carr, RE; Henkind, P; Rothfield, N; Siegel, IM | 1 |
Ott, KJ | 1 |
Crim, JA; Gray, GD; Zeleznick, LD | 1 |
Hahn, FE; Macomber, PB; O'Brien, RL | 1 |
Banerjee, AK; Chowdhury, DS | 1 |
Hermann, P; Lefranc, E; Sourdille, P | 1 |
Mattila, M; Takki, S | 1 |
Reba, RC; Sheehy, TW | 1 |
Trager, W | 1 |
Purcell, WP; Singer, JA | 1 |
Famaey, JP; Fontaine, J; Ouedraogo, CO; Reuse, J | 1 |
Wolfe, MS | 1 |
Authi, KS; Traynor, JR | 1 |
Di Cerbo, A; Edelhoch, H; Nandi, PK | 1 |
Koranda, FC | 1 |
Trist, DG; Weatherall, M | 1 |
Doberstyn, EB | 1 |
Ferrante, A; Goh, DH | 1 |
Dubin, NH; Ghodgaonkar, RB; King, TM; Parmley, TH | 1 |
Harris, EJ; Jackson, MJ; Jones, DA | 1 |
Ioannides, C; Thabrew, MI | 1 |
Drenckhahn, D; Jacobi, B; Lüllmann-Rauch, R | 1 |
Hughes, GR; Lanham, JG | 1 |
Gould, S; Warhurst, DC | 1 |
Elgart, M; Isaacson, D; Turner, ML | 1 |
Ma, K; Sourkes, TL | 1 |
Berstein, GS; Trifunac, NP | 1 |
Kuye, JO; Walle, T; Wilson, MJ | 1 |
Izumi, F; Kobayashi, H; Sakurai, S; Wada, A; Yanagihara, N | 1 |
Tanenbaum, L; Tuffanelli, DL | 1 |
Andersson, A; Olsson, S; Tjälve, H | 1 |
Govitrapong, P; Jearnpipatkul, A; Panijpan, B; Wilairat, P; Yuthavong, Y | 1 |
Catt, KJ; Naor, Z | 1 |
Olansky, AJ | 1 |
Crescenzi, V; Delben, F; Giancotti, V; Quadrifoglio, F | 1 |
Biller, H; Hess, F; Leising, HB; Pfab, R; Schachtschabel, DO | 2 |
Bohn, E; Hesse, B; Kunze, H | 1 |
Bennett, T; Lot, TY | 1 |
Jones, RL; Keel, RA; Lanier, AC; Wilson, WD | 1 |
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B | 1 |
Brady, RO; Kusiak, JW; Quirk, JM | 1 |
Kádár, T; Matejka, Z; Minker, E | 1 |
Hodgson, LL; Morgan, EH; Quail, EA | 1 |
Cacoub, P; Frances, C; Godeau, P; Lipsker, D; Piette, JC | 1 |
Feldmann, R; Salomon, D; Saurat, JH | 1 |
Enomoto, K; Maeno, T | 1 |
Dutta, P; Karmali, R; Pinto, JT; Rivlin, RS | 1 |
Wallace, DJ | 1 |
Craig, JC; Scaria, PV; Shafer, RH | 1 |
Marcil, J; Ravindranath, N; Sairam, MR | 1 |
Lüllmann-Rauch, R; Pods, R; von Witzendorff, B | 1 |
Chen, SS; Jiang, MC; Lin, JK | 1 |
Croft, SL; Elueze, EI; Warhurst, DC | 1 |
Bächinger, HP; Hinrichs, DJ; Ignatushchenko, MV; Riscoe, MK; Winter, RW | 1 |
Dabancens, AO; Guerrero, AC; Zipper, JA | 1 |
Rynes, RI | 1 |
Horio, S; Ishida, Y; Moritoki, H; Nagare, T | 1 |
Loegering, DJ; Raley, MJ; Schwacha, MG | 1 |
Macfarlane, DE; Manzel, L | 2 |
Bondeson, J; Sundler, R | 1 |
Lehmann, P; Rönnau, AC; Ruzicka, T; Schuppe, HC; Specker, C; von Schmiedeberg, S | 1 |
Griffin, GE; Harrison, TS; Levitz, SM | 1 |
Cheng, SH; Przybylska, M; Song, A; Tousignant, JD; Wu, IH; Yew, NS; Zhao, H | 1 |
Vdovenko, AA; Williams, JE | 1 |
Piette, WW; Van Beek, MJ | 1 |
Rembao, D; Reyes, S; Sotelo, J | 1 |
Jjemba, PK | 1 |
ANSARI, AR; BRUMPT, LC; MAISON, E | 1 |
ROSENBAUM, S | 1 |
PASTOR BOTIJA, F | 1 |
BASU, PC; RAY, AP | 1 |
GONDARD, L | 1 |
DRIVER, IE; FARBER, EM | 1 |
KNOX, JM; LAMB, JH; MORGAN, RJ; SHELMIRE, B | 1 |
CAHN, MM; LEVY, EJ; SHAFFER, B | 2 |
FINN, OA; ROGERS, J | 1 |
CERTONCINY, A; FORESTIER, J | 1 |
VILANOVA, X | 1 |
BAYES, C; ESCARPENTER-ORIOL, J; GOMEZ, MS | 1 |
CHAMNARNKIT, C; CHETANASEN, S; SADUN, EH | 1 |
BORODA, C | 1 |
BRODTHAGEN, H | 1 |
BIGUET, J; BRETON, A; COUTELEN, F; DEBLOCK, S; DOBY, JM; MULLET, S | 1 |
CARRERAS BAYES, A; ESCARPENTER ORIOL, J; SARIOLS GOMEZ, M | 1 |
MARCHIONINI, A; THIES, W | 1 |
AZIMI-HAMID, A; TRONNIER, H | 1 |
CONNER, SK | 1 |
LANGLO, L | 1 |
CHRISTIANSEN, JV | 2 |
FLEISCHMAJER, R; REIN, CR | 1 |
ENGESET, A | 2 |
ANSELL, HB; APPEL, B; SCHIFF, B; TYE, MJ; WOLF, M | 1 |
FERNANDEZ NAFRIA, A | 1 |
KOCH, H; WISKEMANN, A | 1 |
VIDMAR-CVJETANOVIC, B | 1 |
ERLENDSSON, F | 1 |
ROBINSON, RC; SMITH, GC | 1 |
ANSELL, HB; APPEL, B; TYE, MJ; WHITE, H | 1 |
BROWNING, M; JONES, R; JONSSON, U; LESSNER, H; PRICE, CC; SEN, AK | 1 |
MARCIANO, MR; SHEARD, C | 1 |
HOJMAN, N; QUIROGA, FE; VAZQUEZ, HJ | 1 |
ABD-EL-GHAFFAR, V | 1 |
GROUNDS, JG | 1 |
GREWAL, RS; SHARMA, ML | 1 |
BEHRENDT, WA; URBAN, G | 1 |
BOCK, W; DOERDELMANN, P | 1 |
KURNICK, NB; RADCLIFFE, IE | 1 |
LEOVEY, A; NAGY, E | 1 |
FREDRIKSSON, T; LODIN, A; ROSENGREN, S | 1 |
SASLAW, S; SCHAEFER, J | 1 |
BONTOUX, D; GODEAU, P; LEVY, R; SIGUIER, F | 1 |
AMMA, MK; GUJRAL, ML; MISRA, N; SAREEN, K; VARMA, DR; VIJAYAMMA, N | 1 |
DARNET, C; LEBEURRE, R; VERHAEGHE, A | 1 |
EPSTEIN, JH; VANDENBERG, JJ; WRIGHT, WL | 1 |
KLINGMUELLER, G | 1 |
CONTACOS, PG; MILLAR, JW; STITCHER, JE; YOUNG, MD | 1 |
ABRAHAM, RK; DUBOIS, EI; TUFFANELLI, D | 1 |
HASERICK, JR | 1 |
ARORA, RB; LAL, A | 1 |
COATNEY, GR; CONTACOS, PG; LUNN, JS | 1 |
SAPP, OL | 1 |
BORC, K | 1 |
BOUMA, HG; DEVRIES, K; JANSZ, A; NIEWEG, HO | 1 |
RAAB, W | 1 |
SULLI, G; VARRONE, F | 1 |
BRACKEN, EC | 1 |
BOTTIROLI, JA; ROSENBERG, FJ | 1 |
ALVING, AS; BREWER, GJ; MILLAR, JW; POWELL, RD | 1 |
EYLES, DE; MONTGOMERY, R; SANDOSHAM, AA | 1 |
MATTILA, M | 1 |
DASHPUTRA, PG; DESHPANDE, VR; SHARMA, ML | 1 |
HELLERSTROEM, S | 1 |
FORBES, LS | 1 |
BRUCHACOVA, V; KRAJCI LAZARYOVA, M; NOVAK, A | 1 |
BETTLEY, FR | 1 |
MITCHELL, CL | 1 |
NEAL, RA | 1 |
HALSTEAD, SB; SADUN, EH | 1 |
CHANG, KC; CHIEN, TS; MENG, HY | 1 |
HERRMANN, WP; SCHULZ, KH | 1 |
STOUGHTON, RB | 1 |
THIES, W | 1 |
BRANDAO, N; DA FONSECA, A | 1 |
BALOGH, EE; NAGY, E | 1 |
REINERTSON, JW; THOMPSON, PE | 1 |
Bernhardt, I; Lang, HJ; Weiss, E | 1 |
Haystead, TA; Kwiek, JJ; Rudolph, J | 1 |
Bauer, S; Gellert, T; Lipford, GB; Luppa, P; Metzger, J; Rutz, M; Wagner, H | 1 |
Emerson, LR; Kuchler, K; Skillman, BC; Wirth, DF; Wolfger, H | 1 |
Forgac, M; Shao, E | 1 |
HANDFIELD-JONES, RP | 1 |
Tutor-Ureta, P; Yebra-Bango, M | 1 |
Benz, R; Orlik, F; Schiffler, B | 1 |
Pollaschek, C; Stuhlmeier, KM | 1 |
Colonna, M; Fuchs, A; Fung-Leung, WP; Gu, Y; Karlsson, L; Lai, KT; Rao, N; Sanjuan, MA; Sun, S | 1 |
Jailer, JW; Rosenfeld, M; Shannon, JA | 1 |
Boratyński, J; Lipka, D | 1 |
CRAIGE, B; PULLMAN, TN | 1 |
EYLES, DE; YOUNG, MD | 1 |
JAILER, JW; ZUBROD, CG | 1 |
Geng, Y; Klocke, BJ; Kohli, L; Roth, KA | 1 |
Baird, JK | 1 |
Bencina, M; Jerala, R; Jeras, M; Kuznik, A; Rozman, B; Svajger, U | 1 |
Chen, B; Coldham, I; Little, SM; Louth, JC; Thompson, MJ | 1 |
Albuquerque, I; Gomes, A; Gomes, P; Machado, M; Nogueira, F; Pérez, B; Prudêncio, M; Teixeira, C | 1 |
NAIR, CP; RAY, AP | 1 |
Gately, S; Gonzales, P; Goodall, ML; MacKeigan, JP; Martin, KR; Sepulveda, M; Wang, T | 1 |
Gomes, A; Gomes, P; Lobo, L; Machado, M; Nogueira, F; Prudêncio, M; Teixeira, C | 1 |
Bakardzhiev, I; Chokoeva, AA; Krasnaliev, I; Lotti, T; Tana, C; Tchernev, G; Wollina, U | 1 |
Barth, H; Benz, R; Kreidler, AM | 1 |
Marceau, F; Parks, A | 1 |
Carter, ER; Chiodini, PL; Hedley, L; Nabarro, LE | 1 |
Meggitt, SJ; Miller, JAL; Winn, RT | 1 |
Bensalem, J; Bryksin, V; Fourrier, C; Hattersley, K; Hein, LK; Sargeant, TJ | 1 |
Bottieau, E; Hatz, C; Kuenzli, E; Mechain, M; Mørch, K; Neumayr, A; Rothe, C; Schunk, M; Soriano Pérez, MJ; Sothmann, P; Sydow, V; Theunissen, C; Van Esbroeck, M | 1 |
27 review(s) available for chloroquine and quinacrine
Article | Year |
---|---|
Design of Small Molecule Autophagy Modulators: A Promising Druggable Strategy.
Topics: Animals; Autophagy; Drug Design; Humans; Small Molecule Libraries | 2018 |
Drugs for the Treatment of Zika Virus Infection.
Topics: Animals; Antiviral Agents; Drug Development; Drug Discovery; Humans; Viral Vaccines; Zika Virus; Zika Virus Infection | 2020 |
Antimalarials in the management of discoid and systemic lupus erythematosus.
Topics: Animals; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Pigmentation Disorders; Quinacrine; Retinal Diseases; Vision Disorders | 1978 |
[Treatment of intestinal parasitosis].
Topics: Amphotericin B; Anthelmintics; Bithionol; Cestode Infections; Chloroquine; Humans; Intestinal Diseases, Parasitic; Leishmaniasis; Malaria; Metronidazole; Nematode Infections; Quinacrine; Tetracycline; Thiabendazole | 1975 |
Recent advances in antimalarial chemotherapy and drug resistance.
Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones | 1974 |
Drug therapy. Treatment of common parasitic infections of man encountered in the United States. 2.
Topics: Amebiasis; Amebicides; Anthelmintics; Antimalarials; Antimony; Benzenesulfonates; Chloroquine; Clonorchiasis; Clonorchis sinensis; Dysentery, Amebic; Giardiasis; Humans; Iodoquinol; Liver Abscess, Amebic; Malaria; Metronidazole; Niridazole; Protozoan Infections; Quinacrine; Schistosoma haematobium; Schistosoma mansoni; Schistosomiasis; Tartrates; Trematode Infections | 1972 |
The present status of chloroquine in the drug treatment of malaria.
Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines | 1972 |
Summary of recent abstracts. 3. Malaria. 2.
Topics: Animals; Antimalarials; Birds; Chloroquine; Dapsone; Humans; India; Malaria; Malaria, Avian; Mammals; Naphthoquinones; Oxytetracycline; Plasmodium; Plasmodium falciparum; Quinacrine; Rats; Reptiles | 1972 |
The pharmacology of the antimalarials. A rational approach to the therapy of resistant falciparum malaria.
Topics: Amodiaquine; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Sulfadimethoxine; Sulfisoxazole | 1969 |
Chemotherapy of the drug-resistant malarias.
Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones | 1969 |
Drug induced retinopathy.
Topics: Adsorption; Animals; Antineoplastic Agents; Chloroquine; Drug-Related Side Effects and Adverse Reactions; Eye Diseases; Humans; Pharmaceutical Preparations; Phenothiazines; Quinacrine; Quinolines; Retina; Retinal Pigments | 1969 |
Malaria treatment and prevention. A review.
Topics: Adolescent; Adult; Africa, Eastern; Antimalarials; Biguanides; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Humans; Infant; Infant Mortality; Infant, Newborn; Malaria; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Quinacrine; Quinine; Quinolines; Sulfonamides | 1969 |
Epidermolysis bullosa.
Topics: Adrenal Cortex Hormones; Chloroquine; Epidermolysis Bullosa; Humans; Oral Manifestations; Quinacrine; Silver Nitrate; Skin Manifestations; Vitamins | 1971 |
The treatment of intestinal protozoan infections.
Topics: Amebicides; Antimalarials; Antiprotozoal Agents; Balantidiasis; Chloroquine; Coccidiosis; Dientamoebiasis; Drug Combinations; Dysentery, Amebic; Emetine; Furans; Furazolidone; Giardiasis; Humans; Intestinal Diseases, Parasitic; Iodoquinol; Liver Abscess, Amebic; Metronidazole; Paromomycin; Quinacrine; Sulfamethoxazole; Tetracycline; Tinidazole; Trimethoprim; Trimethoprim, Sulfamethoxazole Drug Combination | 1982 |
Antimalarials.
Topics: Antimalarials; Chloroquine; DNA; Eye Diseases; Humans; Hydroxychloroquine; Quinacrine; RNA; Skin Diseases | 1981 |
Resistance of Plasmodium falciparum.
Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America | 1984 |
Antimalarial therapy in SLE.
Topics: Antimalarials; Binding Sites; Chloroquine; Corneal Diseases; Dose-Response Relationship, Drug; Female; Humans; Hydroxychloroquine; Immune Tolerance; Inflammation; Kinetics; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Nucleoproteins; Photosensitivity Disorders; Pregnancy; Quinacrine; Retinal Diseases; Retinal Pigments; Skin Diseases; Virus Replication | 1982 |
Anti-malarials in dermatology.
Topics: Absorption; Amodiaquine; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Female; Humans; Hydroxychloroquine; Quinacrine; Skin Diseases | 1982 |
Antimalarial agents. Chloroquine, hydroxychloroquine, and quinacrine.
Topics: Abnormalities, Drug-Induced; Anti-Inflammatory Agents; Chloroquine; DNA; Eye Diseases; Female; Hematologic Diseases; Humans; Hydroxychloroquine; Immunosuppressive Agents; Male; Melanins; Neuromuscular Diseases; Porphyrias; Pregnancy; Quinacrine; Skin; Sunscreening Agents | 1980 |
Antimalarials and ophthalmologic safety.
Topics: Antimalarials; Arthritis, Rheumatoid; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Retinal Diseases | 1982 |
Antimalarial agents and lupus.
Topics: Antibodies, Antiphospholipid; Antimalarials; Chloroquine; Female; Humans; Hydroxychloroquine; Kidney Diseases; Lupus Erythematosus, Systemic; Neuromuscular Diseases; Pregnancy; Quinacrine | 1994 |
Antimalarial drugs in the treatment of rheumatological diseases.
Topics: Antimalarials; Chloroquine; Contraindications; Female; Humans; Hydroxychloroquine; Male; Pregnancy; Pregnancy Complications; Quinacrine; Rheumatic Diseases; Skin | 1997 |
Antimalarials.
Topics: Antimalarials; Chloroquine; Dermatologic Agents; Humans; Quinacrine; Skin Diseases | 2001 |
[ANTIMALARIALS IN THE TREATMENT OF SKIN DISEASES].
Topics: Adrenal Cortex Hormones; Antimalarials; Chloroquine; Dermatology; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases | 1963 |
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus | 1963 |
[Metalloproteinases. Structure and function].
Topics: 4-Aminobenzoic Acid; Animals; Apoptosis; Arthritis; Autoimmune Diseases; Cell Movement; Chloroquine; Drug Combinations; Enzyme Activation; Extracellular Matrix; Humans; Matrix Metalloproteinase Inhibitors; Matrix Metalloproteinases; Membrane Proteins; Models, Molecular; Neoplasms; Neovascularization, Physiologic; Pantothenic Acid; Pyridoxine; Quinacrine; Tissue Inhibitor of Metalloproteinases | 2008 |
Nitroimidazole-refractory giardiasis: a growing problem requiring rational solutions.
Topics: Albendazole; Antiprotozoal Agents; Chloroquine; Drug Resistance; Drug Therapy, Combination; Giardia lamblia; Giardiasis; Humans; Metronidazole; Quinacrine; Tinidazole; Treatment Failure | 2018 |
5 trial(s) available for chloroquine and quinacrine
Article | Year |
---|---|
[Delagil treatment of tumorous pleurisy].
Topics: Chloroquine; Clinical Trials as Topic; Drug Evaluation; Humans; Injections; Pleura; Pleural Neoplasms; Pleurisy; Quinacrine | 1978 |
The influence of ovarian hormones and of pregnancy on the action of some antimalarials on the isolated spontaneously contracting rat uterus.
Topics: Antimalarials; Chloroquine; Clinical Trials as Topic; Drug Interactions; Estradiol; Female; Histamine H1 Antagonists; Hormones; Humans; Ovary; Progesterone; Proguanil; Quinacrine; Quinine; Uterus | 1971 |
Renal allotransplantation in the baboon with chemical immunosuppression.
Topics: Animals; Azathioprine; Blood Cells; Blood Chemical Analysis; Blood Protein Electrophoresis; Chloroquine; Clinical Trials as Topic; Cyclophosphamide; Enzymes; Female; Glomerular Filtration Rate; Haplorhini; Hydrocortisone; Immunosuppressive Agents; Kidney Function Tests; Kidney Transplantation; Male; Quinacrine; Thalidomide; Transplantation, Homologous | 1968 |
The effect of chemical immunosuppression in baboon allotransplantation: histopathological observations.
Topics: Animals; Azathioprine; Chloroquine; Clinical Trials as Topic; Cyclophosphamide; Haplorhini; Hydrocortisone; Immunosuppressive Agents; Kidney; Kidney Transplantation; Quinacrine; Renal Artery; Renal Veins; Thalidomide; Transplantation, Homologous | 1968 |
The effect of chemical immunosuppression in baboon allotransplantation: serological observations.
Topics: Animals; Antibodies; Azathioprine; C-Reactive Protein; Chloroquine; Clinical Trials as Topic; Complement System Proteins; Cyclophosphamide; Haplorhini; Hemolysin Proteins; Humans; Hydrocortisone; Immunosuppressive Agents; Kidney Transplantation; Quinacrine; Rheumatoid Factor; Thalidomide; Transplantation, Homologous | 1968 |
305 other study(ies) available for chloroquine and quinacrine
Article | Year |
---|---|
Interactions of antitumor drugs with natural DNA: 1H NMR study of binding mode and kinetics.
Topics: Antineoplastic Agents; Base Composition; Chemical Phenomena; Chemistry; DNA; Hydrogen Bonding; Intercalating Agents; Kinetics; Magnetic Resonance Spectroscopy; Structure-Activity Relationship | 1984 |
Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine.
Topics: Animals; Antiprotozoal Agents; Leishmania; Parasitic Sensitivity Tests; Plasmodium; Quinacrine; Sulfonamides; Trypanosoma; Urea | 2001 |
Antimalarial drug quinacrine binds to C-terminal helix of cellular prion protein.
Topics: Antimalarials; Binding Sites; Chloroquine; Humans; Magnetic Resonance Spectroscopy; Models, Molecular; Peptide Fragments; Phenothiazines; Prions; Protein Structure, Secondary; Quinacrine; Recombinant Proteins; Structure-Activity Relationship | 2003 |
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated | 2004 |
Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
Topics: Aminoquinolines; Animals; Antimalarials; Chloroquine; Drug Resistance; Plasmodium falciparum; Structure-Activity Relationship | 2005 |
Structure-function correlation of chloroquine and analogues as transgene expression enhancers in nonviral gene delivery.
Topics: Cell Line, Tumor; Chloroquine; Cyclodextrins; DNA; Drug Screening Assays, Antitumor; Electrophoretic Mobility Shift Assay; Gene Expression; Gene Transfer Techniques; HeLa Cells; Humans; Luciferases; Structure-Activity Relationship; Transgenes | 2006 |
Simple colorimetric inhibition assay of heme crystallization for high-throughput screening of antimalarial compounds.
Topics: Animals; Antimalarials; Colorimetry; Crystallization; Drug Evaluation, Preclinical; Heme; Hemeproteins; Plasmodium falciparum; Polysorbates; Reproducibility of Results | 2007 |
Bis-acridines as lead antiparasitic agents: structure-activity analysis of a discrete compound library in vitro.
Topics: Acridines; Animals; Antiparasitic Agents; Combinatorial Chemistry Techniques; Eukaryota; HL-60 Cells; Humans; Parasitic Sensitivity Tests; Plasmodium falciparum; Polyamines; Schistosoma mansoni; Structure-Activity Relationship; Trypanosoma brucei brucei | 2007 |
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase | 2008 |
Selective plasma protein binding of antimalarial drugs to alpha1-acid glycoprotein.
Topics: Antimalarials; Binding Sites; Chromatography, Affinity; Circular Dichroism; Humans; Molecular Structure; Orosomucoid; Protein Binding; Serum Albumin; Spectrophotometry; Stereoisomerism; Structure-Activity Relationship | 2008 |
Pharmacophore based discovery of potential antimalarial agent targeting haem detoxification pathway.
Topics: Animals; Antimalarials; Drug Discovery; Heme; Isoniazid; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Small Molecule Libraries; Stereoisomerism | 2008 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase | 2008 |
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship | 2008 |
Privileged structure-guided synthesis of quinazoline derivatives as inhibitors of trypanothione reductase.
Topics: Animals; Antiparasitic Agents; Cell Line; Computer Simulation; Drug Design; Enzyme Inhibitors; Glutathione Reductase; Humans; NADH, NADPH Oxidoreductases; Quinazolines; Rats; Structure-Activity Relationship; Trypanosoma cruzi | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
Topics: | 2008 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Predicting phospholipidosis using machine learning.
Topics: Animals; Artificial Intelligence; Databases, Factual; Drug Discovery; Humans; Lipidoses; Models, Biological; Phospholipids; Support Vector Machine | 2010 |
Bioanalytical Screening of Riboflavin Antagonists for Targeted Drug Delivery - A Thermodynamic and Kinetic Study.
Topics: | 2011 |
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites | 2011 |
In silico assay for assessing phospholipidosis potential of small druglike molecules: training, validation, and refinement using several data sets.
Topics: Animals; Cattle; Cells, Cultured; Computer Simulation; Cornea; Drug-Related Side Effects and Adverse Reactions; Fibroblasts; Lipidoses; Lysosomal Storage Diseases; Models, Molecular; Pharmaceutical Preparations; Phospholipids; Structure-Activity Relationship; Thermodynamics | 2012 |
Design, synthesis and characterization of novel quinacrine analogs that preferentially kill cancer over non-cancer cells through the down-regulation of Bcl-2 and up-regulation of Bax and Bad.
Topics: Antineoplastic Agents; bcl-2-Associated X Protein; bcl-Associated Death Protein; Cell Death; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Down-Regulation; Drug Design; Drug Screening Assays, Antitumor; Humans; Molecular Structure; Proto-Oncogene Proteins c-bcl-2; Quinacrine; Structure-Activity Relationship; Up-Regulation | 2017 |
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship | 2019 |
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.
Topics: Animals; Anti-Inflammatory Agents; Antiviral Agents; Betacoronavirus; Cell Line; Chlorocebus aethiops; Coronavirus Infections; COVID-19; Drug Evaluation, Preclinical; Drug Repositioning; Humans; Niclosamide; Pandemics; Pneumonia, Viral; Pregnenediones; SARS-CoV-2; Vero Cells | 2020 |
Antimalarial Quinacrine and Chloroquine Lose Their Activity by Decreasing Cationic Amphiphilic Structure with a Slight Decrease in pH.
Topics: Antifungal Agents; Cell Membrane; Chloroquine; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Molecular Structure; Monosaccharide Transport Proteins; Protons; Quinacrine; Saccharomyces cerevisiae; Surface-Active Agents | 2021 |
Vesicle penicillinase of Bacillus licheniformis: existence of periplasmic-releasing factor(s).
Topics: Bacillus; Chloroquine; Chromatography, Gel; Deoxycholic Acid; Hydrogen-Ion Concentration; Molecular Weight; Organoids; Penicillinase; Phenanthrolines; Phosphates; Protoplasts; Quinacrine | 1977 |
Tautomerism of singly protonated chloroquine and quinacrine.
Topics: Chloroquine; Hydrogen-Ion Concentration; Kinetics; Quinacrine; Spectrophotometry; Spectrophotometry, Ultraviolet; Stereoisomerism | 1978 |
Experimental myopathy induced by amphiphilic cationic compounds including several psychotropic drugs.
Topics: Amitriptyline; Animals; Chloroquine; Chlorphentermine; Chlorpromazine; Female; Imipramine; Iprindole; Male; Microscopy, Electron; Muscles; Muscular Diseases; Phentermine; Piperazines; Psychotropic Drugs; Quinacrine; Rats; Triparanol | 1979 |
Inhibitory effect on gastric motility of chloroquine and mepacrine.
Topics: Animals; Chloroquine; Depression, Chemical; Dose-Response Relationship, Drug; Female; Ganglionic Blockers; Gastrointestinal Motility; In Vitro Techniques; Parasympatholytics; Quinacrine; Rats; Sympathetic Nervous System; Sympatholytics | 1978 |
A serological study of removal of UV-induced photoproducts in the DNA of Tetrahymena pyriformis GL: influence of caffeine, quinacrine and chloroquine.
Topics: Animals; Caffeine; Chloroquine; DNA; DNA Repair; Immunologic Techniques; Photochemistry; Quinacrine; Tetrahymena pyriformis; Ultraviolet Rays | 1979 |
Differential effects of chloroquine and of several other amphiphilic cationic drugs upon rat choroid plexus.
Topics: Amitriptyline; Animals; Chloroquine; Chlorphentermine; Choroid Plexus; Clomipramine; Female; Hexestrol; Inclusion Bodies; Iprindole; Male; Microscopy, Electron; Quinacrine; Rats | 1979 |
Photodynamic activity of dyes with different DNA binding properties I. free-radical induction in DNA.
Topics: Acridines; Binding Sites; Chloroquine; Coloring Agents; DNA; Ethidium; Free Radicals; Light; Proflavine; Pyronine; Quinacrine; Thioxanthenes | 1978 |
Photodynamic activity of dyes with different DNA binding properties II. T4 phage inactivation.
Topics: Acridines; Binding Sites; Chloroquine; Coliphages; Coloring Agents; DNA, Viral; Ethidium; Light; Proflavine; Pyronine; Quinacrine; Thioxanthenes | 1978 |
Comparative viscometric analysis of the interaction of chloroquine and quinacrine with superhelical and sonicated DNA.
Topics: Bacteriocin Plasmids; Chloroquine; DNA, Superhelical; Nucleic Acid Conformation; Quinacrine; Sonication; Viscosity | 1979 |
Effect of mepacrine on gastric motility in the rat.
Topics: Administration, Oral; Animals; Bencyclane; Chloroquine; Female; Gastric Emptying; Gastric Mucosa; Gastrointestinal Motility; Injections, Intraperitoneal; Papaverine; Quinacrine; Rats | 1979 |
Inhibition of hepatitis B DNA polymerase by intercalating agents.
Topics: Chloroquine; Chlorpromazine; Drug Synergism; Ethidium; Hepatitis B; Hepatitis B virus; Humans; Indicators and Reagents; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine | 1978 |
Molecular structural effects involved in the interaction of quinolinemethanolamines with DNA. Implications for antimalarial action.
Topics: Amino Alcohols; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; DNA; Drug Interactions; Piperidines; Quinacrine; Quinine; Quinolines | 1977 |
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin | 1975 |
Effect of nucleic-acid-binding compounds on the hydrolytic activity of various ribonucleases.
Topics: Acridines; Aminoquinolines; Animals; Binding Sites; Cattle; Chloroquine; Ethidium; Kinetics; Pancreas; Primaquine; Proflavine; Protein Binding; Quinacrine; Ribonucleases; Spermidine; Spermine; Structure-Activity Relationship | 1975 |
[Plaque-like form of cutaneous mucinosis (PGM) and reticular erythematous mucinosis (REM syndrome)].
Topics: Adult; Antimalarials; Chloroquine; Female; Humans; Methapyrilene; Quinacrine; Skin Diseases | 1975 |
Smooth muscle sensitization and neuromuscular depression induced by chronic administration of antimalarial drugs.
Topics: Acetylcholine; Animals; Chickens; Chloroquine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Male; Muscle Contraction; Muscle, Smooth; Muscles; Neuromuscular Junction; Norepinephrine; Potassium Chloride; Quinacrine | 1992 |
Antimalarial activity of optical isomers of quinacrine dihydrochloride against chloroquine-sensitive and -resistant Plasmodium falciparum in vitro.
Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Plasmodium falciparum; Quinacrine; Stereoisomerism | 1991 |
Chloroquine-sensitive transplasmalemma electron transport in Tetrahymena pyriformis: a hypothesis for control of parasite protozoa through transmembrane redox.
Topics: Animals; Cell Wall; Chloroquine; Electron Transport; Ferricyanides; Hydrogen-Ion Concentration; Membrane Potentials; Oxidation-Reduction; Oxygen; Quinacrine; Tetrahymena pyriformis | 1991 |
Degradation of insulin in isolated liver endosomes is functionally linked to ATP-dependent endosomal acidification.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Cations; Chloroquine; Guanosine Triphosphate; Hydrogen-Ion Concentration; Inosine Triphosphate; Insulin; Liver; Male; Organelles; Quinacrine; Rats; Rats, Inbred Strains; Subcellular Fractions; Uridine Triphosphate | 1990 |
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with lipids extracted from normal human erythrocytes.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Deuterium; Erythrocytes; Humans; Magnetic Resonance Spectroscopy; Mefloquine; Membrane Lipids; Phosphatidylethanolamines; Phosphorus Isotopes; Quinacrine; Quinine | 1990 |
Depressant effects of chloroquine on the isolated guinea-pig heart.
Topics: Animals; Calcium; Chloroquine; Depression, Chemical; Electric Stimulation; Female; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Ouabain; Quinacrine | 1990 |
The effects of non-steroidal inhibitors of phospholipase A2 on leukotriene and histamine release from human and guinea-pig lung.
Topics: Animals; Calcimycin; Chloroquine; Guinea Pigs; Histamine Release; Humans; Lung; Ovalbumin; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; SRS-A | 1985 |
3H-azidopine photoaffinity labeling of high molecular weight proteins in chloroquine resistant falciparum malaria.
Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Chloroquine; Chlorpromazine; Dihydropyridines; Drug Resistance; Glycoproteins; Molecular Weight; Nicardipine; Photochemistry; Plasmodium falciparum; Proteins; Quinacrine; Reserpine; Trifluoperazine; Verapamil | 1989 |
Ca2+-antagonistic properties of phospholipase A2 inhibitors, mepacrine and chloroquine.
Topics: Animals; Calcium; Calcium Channel Blockers; Chloroquine; In Vitro Techniques; Membrane Potentials; Myocardium; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rana ridibunda | 1989 |
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with dipalmitoylphosphatidylcholine bilayers.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Mefloquine; Quinacrine; Quinine; Quinolines; Temperature | 1989 |
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains | 1985 |
[Synthetic antimalarials in the therapy of rheumatoid arthritis: adverse effects and advantages].
Topics: Arthritis, Rheumatoid; Chloroquine; Drug Evaluation; Enzyme Inhibitors; Histamine H1 Antagonists; Humans; Hydroxychloroquine; Quinacrine; Time Factors | 1985 |
Effects of indole alkaloids on multidrug resistance and labeling of P-glycoprotein by a photoaffinity analog of vinblastine.
Topics: Affinity Labels; Alkaloids; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Survival; Chloroquine; Drug Interactions; Drug Resistance; Humans; Indoles; Leukemia; Membrane Glycoproteins; Photochemistry; Quinacrine; Quinine; Reserpine; Verapamil; Vinblastine; Vinca Alkaloids; Vindesine; Yohimbine | 1988 |
[Effect of Collagenan on joint disease associated with collagenous colitis].
Topics: 4-Aminobenzoic Acid; Aminobenzoates; Chloroquine; Colitis; Collagen; Drug Combinations; Female; Humans; Joint Diseases; Middle Aged; Pantothenic Acid; Pyridoxine; Quinacrine | 1986 |
[Evaluation of the phototoxicity of five antimalarial agents and praziquantel in mice].
Topics: Animals; Antimalarials; Chloroquine; Female; Male; Mice; Naphthyridines; Photosensitivity Disorders; Praziquantel; Quinacrine; Quinazolines; Quinolines; Ultraviolet Rays | 1986 |
Antioxidant action of antimalarials.
Topics: Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Humans; Hydrogen Peroxide; Neutrophils; Oxygen; Quinacrine; Superoxides | 1986 |
Differential effects of mepacrine, chloroquine and hydroxychloroquine on superoxide anion generation, phospholipid methylation and arachidonic acid release by human blood monocytes.
Topics: Arachidonic Acid; Arachidonic Acids; Calcimycin; Cell Survival; Chloroquine; Fluorides; Humans; Hydroxychloroquine; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Phospholipids; Quinacrine; Superoxides; Tetradecanoylphorbol Acetate; Zymosan | 1986 |
Mepacrine accumulation during treatment of chloroquine-resistant falciparum malaria.
Topics: Adolescent; Adult; Animals; Chloroquine; Drug Resistance; Female; Humans; Malaria; Male; Middle Aged; Plasmodium falciparum; Quinacrine | 1988 |
Stimulation of luteinizing hormone release by melittin and phospholipase A2 in rat pituitary cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bee Venoms; Cell Membrane; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Enzyme Activation; Female; Gonadotropin-Releasing Hormone; In Vitro Techniques; Luteinizing Hormone; Melitten; Phospholipases; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Quinacrine; Rats; Secretory Rate | 1987 |
The mechanism of the inhibitory effects of antimalarials on UV-induced skin inflammation in mice.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Chloroquine; Ear, External; Edema; Female; Inflammation; Mice; Mice, Inbred ICR; PUVA Therapy; Quinacrine; Skin; Ultraviolet Rays | 1988 |
Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells.
Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cell Line; Chemical Phenomena; Chemistry, Physical; Chloroquine; Computer Simulation; Doxorubicin; Drug Resistance; Humans; Leukemia; Naphthacenes; Podophyllotoxin; Quinacrine; Verapamil; Vinca Alkaloids | 1988 |
[The mouse micronucleus test for mutagenicity of pyronaridine, chloroquine, quinacrine, primaquine, furapyrimidone and phenthiourezine].
Topics: Animals; Anthelmintics; Antimalarials; Chloroquine; Filaricides; Male; Mice; Micronucleus Tests; Mutagenicity Tests; Naphthyridines; Nitrofurans; Piperazines; Primaquine; Quinacrine | 1988 |
Spermidine oxidase activity in serum of normal and schizophrenic subjects.
Topics: Adult; Chloroquine; Female; Humans; Male; Middle Aged; Oxidoreductases Acting on CH-NH Group Donors; Polyamine Oxidase; Quality Control; Quinacrine; Reference Values; Schizophrenia; Substrate Specificity | 1988 |
The in vitro pharmacology of chloroquine and quinacrine.
Topics: Animals; Biological Transport, Active; Chickens; Chloroquine; Guanethidine; In Vitro Techniques; Male; Neurons; Nordefrin; Norepinephrine; Quinacrine | 1986 |
Degradation of dipalmitoyl phosphatidylcholine by isolated rat granular pneumocytes and reutilization for surfactant synthesis.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Ammonium Chloride; Animals; Chloroquine; Choline; Liposomes; Lung; Methylamines; Organoids; Pulmonary Surfactants; Quinacrine; Rats | 1987 |
Brugia pahangi: inhibition of protein synthesis.
Topics: Animals; Antimycin A; Brugia; Chloramphenicol; Chloroquine; Cyanides; Cycloheximide; Electron Transport; Lactates; Molecular Weight; Movement; Protein Biosynthesis; Protein Synthesis Inhibitors; Quinacrine | 1987 |
Stimulation of phospholipase A2 activity by oxygen-derived free radicals in isolated brain capillaries.
Topics: Animals; Brain; Capillaries; Chloroquine; Fatty Acids; Fatty Acids, Unsaturated; Free Radicals; Oxygen; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains; Xanthine Oxidase | 1985 |
The action of salinomycin-Na and lasalocid-Na on chloroquine- and mepacrine-resistant line of Plasmodium berghei K 173-strain in Wistar rats.
Topics: Animals; Anti-Bacterial Agents; Cell Membrane; Chloroquine; Cytoplasm; Drug Resistance, Microbial; Lasalocid; Lethal Dose 50; Malaria; Male; Microscopy, Electron; Plasmodium berghei; Pyrans; Quinacrine; Rats; Rats, Inbred Strains; Time Factors | 1985 |
Testing of chloroquine and quinacrine for mutagenicity in Drosophila melanogaster.
Topics: Animals; Chloroquine; Drosophila melanogaster; Genes, Lethal; Genes, Recessive; Male; Mutagenicity Tests; Quinacrine; Sex Chromosome Aberrations | 1985 |
Cutaneous lupus erythematosus. Recognition of its many forms.
Topics: Adrenal Cortex Hormones; Adult; Chloroquine; Diagnosis, Differential; Female; Humans; Hydroxychloroquine; Infant, Newborn; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Male; Quinacrine; Sex Factors; Skin; Skin Diseases | 1986 |
Effects of antimalarial drugs on phospholipase A and lysophospholipase activities in plasma membrane, mitochondrial, microsomal and cytosolic subcellular fractions of rat liver.
Topics: Animals; Antimalarials; Cell Membrane; Chloroquine; Cytosol; Endoplasmic Reticulum; Liver; Lysophospholipase; Male; Microsomes, Liver; Mitochondria, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1985 |
[Ultrastructural studies of the effect of x-rays and quinacrine (Atebrin) or chloroquine (Resochin)--alone or in combination--on Harding-Passey melanoma cells in monolayer culture].
Topics: Animals; Chloroquine; Combined Modality Therapy; In Vitro Techniques; Melanoma; Mice; Microscopy, Electron; Quinacrine; Radiation-Sensitizing Agents | 1985 |
Pharmacological investigation of the mechanisms of platelet-activating factor induced mortality in the mouse.
Topics: Anaphylaxis; Animals; Chloroquine; Chlortetracycline; Dexamethasone; Dose-Response Relationship, Drug; Female; Indomethacin; Injections, Intravenous; Male; Mice; Mice, Inbred DBA; Naproxen; Nicardipine; Nifedipine; Platelet Activating Factor; Pyrazoles; Quinacrine; Tetracycline; Verapamil | 1985 |
Effect of quinoline, phthalazine and coumarin derivatives on the absorbance of NADPH.
Topics: Chloroquine; Coumarins; Heterocyclic Compounds; Hydralazine; Indophenol; NADP; Novobiocin; Quinacrine; Quinidine; Quinine; Quinolines; Spectrophotometry; Warfarin | 1974 |
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides | 1974 |
Chloroquine-resistant falciparum malaria in Thailand.
Topics: Adolescent; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Humans; Infant; Malaria; Plasmodium falciparum; Quinacrine; Quinine; Thailand | 1965 |
Activity and some properties of an acid proteinase from normal and Plasmodium berghei-infected red cells.
Topics: Acid Phosphatase; Animals; Cell-Free System; Chloroquine; Dithiothreitol; Edetic Acid; Erythrocytes; Female; Hemoglobins; Hemolysis; Hydrogen-Ion Concentration; Malaria; Mice; Mice, Inbred BALB C; Peptide Hydrolases; Plasmodium berghei; Primaquine; Quinacrine; Rats; Solubility; Surface-Active Agents; Ultracentrifugation | 1973 |
Biochemical properties of anti-inflammatory drugs. VI. The effects of chloroquine (resochin), mepacrine (quinacrine) and some of their potential metabolites on cartilage metabolism and oxidative phosphorylation.
Topics: Animals; Cartilage; Chloroquine; Glycosaminoglycans; Gold; Hydroxychloroquine; In Vitro Techniques; Indomethacin; Oxidative Phosphorylation; Polysaccharides; Quinacrine; Quinolines; Rats; Sulfates; Sulfur Isotopes; Thiosulfates | 1965 |
[Use of a Dicrocoelium survival test in the study of the experimental activity of various chemical substances].
Topics: Animals; Arsenicals; Chloroquine; Dicrocoelium; Piperazines; Quinacrine; Thiabendazole | 1967 |
The amoebicidal, trichomonicidal, and antibacterial effects of niridazole in laboratory animals.
Topics: Amebiasis; Amebicides; Amoeba; Animals; Anthelmintics; Antimony; Antiprotozoal Agents; Chloroquine; Clioquinol; Cricetinae; Dysentery, Bacillary; Emetine; Enterobacteriaceae Infections; Furazolidone; Imidazoles; Intestinal Diseases, Parasitic; Liver Abscess, Amebic; Metronidazole; Mice; Quinacrine; Salmonella Infections; Sulfonamides; Sulfones; Tartrates; Tetracycline; Thiazoles; Trichomonas Infections | 1969 |
[Complications with synthetic antimalarials].
Topics: Antimalarials; Asthenia; Central Nervous System Diseases; Chloroquine; Drug Eruptions; Eczema; Eye Diseases; Gastrointestinal Diseases; Hematologic Diseases; Humans; Lupus Erythematosus, Systemic; Pigmentation Disorders; Psoriasis; Quinacrine; Skin Diseases | 1969 |
Inactivation of lysosomal function in normal cultured human fibroblasts by chloroquine.
Topics: Cell Survival; Cells, Cultured; Chloroquine; Fibroblasts; Glycosaminoglycans; Humans; Hydrogen-Ion Concentration; Lysosomes; Microscopy, Electron; Quinacrine; Quinine; Sulfur Radioisotopes; Time Factors | 1973 |
Biochemical properties of anti-inflammatory drugs. VII. Inhibition of proteolytic enzymes in connective tissue by chloroquine (resochin) and related antimalarial antirheumatic drugs.
Topics: Acridines; Animals; Cartilage; Cattle; Chloroquine; Chondroitin; Connective Tissue; Hyaluronoglucosaminidase; Hydrogen-Ion Concentration; Hydroxychloroquine; Microbial Collagenase; Mucoproteins; Papain; Primaquine; Quaternary Ammonium Compounds; Quinacrine; Rabbits | 1966 |
Response of isolated white fat cells to anti-malarial drugs.
Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Animals; Antimalarials; Bucladesine; Chloroquine; Drug Synergism; Fatty Acids, Nonesterified; Female; Glycerol; Norepinephrine; Primaquine; Proteins; Quinacrine; Quinidine; Rats; Theophylline; Triglycerides | 1973 |
Light-microscopic demonstration of drug-induced myelin bodies in the liver of rats.
Topics: Animals; Chloroquine; Cytoplasmic Granules; Inclusion Bodies; Liver; Male; Microscopy; Microscopy, Fluorescence; Quinacrine; Triparanol | 1974 |
Increased levels of pisatin and phenylalanine ammonia lyase activity in Pisum sativum treated with antihistaminic, antiviral, antimalarial, tranquilizing, or other drugs.
Topics: Antidepressive Agents; Antitussive Agents; Antiviral Agents; Chloroquine; Deamination; Ethylamines; Fluorenes; Histamine H1 Antagonists; Imipramine; Ketones; Lectins; Leucine; Lyases; Parasympatholytics; Phenothiazines; Phenylalanine; Piperidines; Plant Lectins; Plant Proteins; Plants, Edible; Propantheline; Quinacrine; Stimulation, Chemical; Tranquilizing Agents; Trimeprazine | 1972 |
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes | 1971 |
Discoid lupus erythematosus.
Topics: Adult; Antimalarials; Chloroquine; Color Vision Defects; Female; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Quinacrine; Retinal Diseases | 1972 |
Labilizing action of intercalating drugs and dyes on bacterial ribosomes.
Topics: Acridines; Bacterial Proteins; Berberine Alkaloids; Carbon Isotopes; Centrifugation, Density Gradient; Chloroquine; Coloring Agents; Daunorubicin; Dioxoles; Escherichia coli; Ethidium; Hot Temperature; Lucanthone; Methylene Blue; Nucleoproteins; Phenanthridines; Phenylalanine; Quinacrine; Quinolines; Ribosomes; RNA, Ribosomal; Spectrometry, Fluorescence; Spermine; Tritium; Uridine | 1972 |
Multidrug-resistant strain of Plasmodium falciparum from eastern Colombia.
Topics: Adolescent; Adult; Antimalarials; Chloroquine; Colombia; Drug Combinations; Drug Resistance, Microbial; Female; Humans; Malaria; Male; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine | 1974 |
Some pharmacological aspects of antimalarial drugs.
Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim | 1974 |
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine | 1972 |
Inhibition of DNA repair replication by DNA binding drugs which sensitize cells to alkylating agents and X-rays.
Topics: Alkylating Agents; Caffeine; Chloroquine; Cyanides; Cyclophosphamide; Dinitrophenols; DNA Repair; DNA Replication; Dose-Response Relationship, Radiation; Drug Combinations; Humans; Hydroxyurea; Injections, Intraperitoneal; Leukocyte Count; Lymphocytes; Protein Binding; Quinacrine; Quinolines; Radiation Effects; Radiation-Sensitizing Agents; Thymidine; Tritium; Ultraviolet Rays | 1972 |
In vitro effect of drugs against pathogenic and non-pathogenic free-living amoebae and on anaerobic amoebae.
Topics: Anaerobiosis; Animals; Biguanides; Chloroquine; Eukaryota; Metronidazole; Quinacrine | 1972 |
Induction of enzymes in dormant spores of Aspergillus oryzae. IV. Effects of ethidium, aminoacridines, and related compounds.
Topics: Acridines; Alcohol Oxidoreductases; Amines; Aspergillus; Carbon Isotopes; Chloroquine; Enzyme Induction; Ethidium; Fungal Proteins; Glucose; Hydroquinones; Kinetics; Leucine; Oxygen Consumption; Phenanthridines; Phenothiazines; Quinacrine; Spores; Spores, Fungal; Sucrase | 1973 |
Inhibitory effect of some quinoline, phthalazine, and coumarin derivatives on glucose-6-phosphate dehydrogenase in vitro.
Topics: Binding, Competitive; Chloroquine; Coumarins; Glucosephosphate Dehydrogenase; Heterocyclic Compounds; Hydralazine; Isoniazid; Novobiocin; Phenazines; Phenelzine; Phenylhydrazines; Probenecid; Pyridines; Quinacrine; Quinidine; Quinine; Quinolines; Sulfanilamides; Warfarin; Yeasts | 1973 |
Similarities between antimalarial schizontocides.
Topics: Antimalarials; Binding Sites; Chloroquine; Quinacrine; Quinine; Structure-Activity Relationship | 1973 |
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors | 1974 |
[Chloroquine induced neuropathy].
Topics: Administration, Oral; Chloroquine; Drug Combinations; Drug Therapy, Combination; Electromyography; Female; Humans; Leg; Middle Aged; Myotonic Dystrophy; Prednisolone; Quinacrine; Time Factors | 1974 |
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones | 1968 |
Malaria and victory in Vietnam. The first battle against drug-resistant malignant malaria is described.
Topics: Anopheles; Antimalarials; Chloroquine; Folic Acid Antagonists; Folic Acid Deficiency; History, 16th Century; History, 17th Century; History, 20th Century; Malaria; Military Medicine; Penicillin Resistance; Penicillins; Plasmodium falciparum; Pyrimidines; Quinacrine; Sulfonamides; Tropical Medicine; Vietnam | 1968 |
Studies concerning the mechanism of action of antimalarial drugs. Inhibition of the incorporation of adenosine-8-3H into nucleic acids of Plasmodium berghei.
Topics: Animals; Antimalarials; Autoradiography; Chloroquine; DNA Nucleotidyltransferases; DNA Replication; Escherichia coli; Male; Methods; Nucleosides; Phenanthridines; Plasmodium; Quinacrine; Quinine; Rats; RNA; RNA Nucleotidyltransferases; Time Factors; Tritium | 1969 |
The problems of drug-resistant pathogenic bacteria. Elimination of bacterial episomes by DNA-complexing compounds.
Topics: Acridines; Carbon Isotopes; Centrifugation, Density Gradient; Cesium; Chloramphenicol; Chlorides; Chloroquine; DNA, Bacterial; Drug Resistance, Microbial; Escherichia coli; Genetics, Microbial; Kanamycin; Lactose; Methylene Blue; Phenanthridines; Quinacrine; Quinine; Rosaniline Dyes; Spermine; Thymidine | 1971 |
Antibacterial nitroacridine, Nitroakridin 3582: binding to nucleic acids in vitro and effects on selected cell-free model systems of macromolecular biosynthesis.
Topics: Acridines; Anti-Bacterial Agents; Binding Sites; Carbon Isotopes; Cell-Free System; Chloroquine; DNA Nucleotidyltransferases; DNA, Bacterial; Escherichia coli; Genetics, Microbial; Hot Temperature; Micrococcus; Models, Chemical; Nitro Compounds; Nucleic Acid Denaturation; Nucleic Acids; Phenanthridines; Phenylalanine; Polynucleotides; Protein Binding; Quinacrine; Ribosomes; RNA Nucleotidyltransferases; RNA, Bacterial; RNA, Transfer; Spectrophotometry; Templates, Genetic; Tritium | 1971 |
The routine treatment of malaria.
Topics: Acute Disease; Adolescent; Adult; Amodiaquine; Child; Child, Preschool; Chloroquine; Chronic Disease; Drug Resistance, Microbial; Female; Humans; Infant; Malaria; Male; Plasmodium falciparum; Quinacrine; Quinine; Sulfonamides | 1971 |
Drugs for petit mal.
Topics: Acetazolamide; Amphetamine; Anticonvulsants; Barbiturates; Child; Child, Preschool; Chlordiazepoxide; Chloroquine; Epilepsy, Absence; Ethosuximide; Humans; Meprobamate; Quinacrine; Succinimides; Trimethadione | 1965 |
The influence of methylene blue on the pentose phosphate pathway in erythrocytes of monkeys infected with Plasmodium knowlesi.
Topics: Animals; Carbon Isotopes; Chloroquine; DNA; Erythrocytes; Glucose; Haplorhini; Isoleucine; Malaria; Methylene Blue; Orotic Acid; Pentosephosphates; Plasmodium; Protein Biosynthesis; Quinacrine; Quinine; RNA; Tritium | 1969 |
Uptake of chloroquine-3-H3 by plasmodium knowlesi in vitro.
Topics: Albumins; Animals; Chloroquine; Cyanates; Dinitrophenols; Erythrocytes; Fluorides; Glucose; Haplorhini; In Vitro Techniques; Iodoacetates; Lysosomes; Malaria; Pinocytosis; Plasmodium; Quinacrine; Quinine; Temperature; Time Factors; Tritium | 1969 |
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors | 1970 |
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents | 1971 |
The role of drugs in a malaria program.
Topics: Amodiaquine; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Malaria; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Recurrence; Sulfonamides; Sulfones; Trimethoprim | 1972 |
Studies concerning the mechanism of action of antimalarial drugs. II. Inhibition of the incorporation of adenosine-5'-monophosphate- 3 H into nucleic acids of erythrocyte-free malarial parasites.
Topics: Adenine Nucleotides; Adenosine; Adenosine Monophosphate; Amodiaquine; Animals; Antimalarials; Chloroquine; DNA; Erythrocytes; Methods; Naphthalenes; Phenanthridines; Plasmodium; Proguanil; Quinacrine; Quinine; Rats; RNA; Saponins; Triazines; Trimethoprim; Tritium | 1971 |
Acridine orange potentiation of actinomycin D uptake and activity.
Topics: Acridines; Animals; Autoradiography; Chloroquine; Dactinomycin; DNA; Drug Synergism; Freezing; Humans; In Vitro Techniques; Lymphocytes; Male; Mice; Organ Size; Protein Binding; Quinacrine; Spleen; Tritium; Vibration | 1971 |
Pigmentation of the hard and solf palate in a patient with rheumatoid arthritis treated with an antimalarial (triquin).
Topics: Arthritis, Rheumatoid; Biopsy; Chloroquine; Female; Humans; Middle Aged; Palate; Pigmentation Disorders; Quinacrine; Time Factors | 1970 |
Reactions of quinine, chloroquine, and quinacrine with DNA and their effects on the DNA and RNA polymerase reactions.
Topics: Chemical Phenomena; Chemistry; Chloroquine; DNA; Escherichia coli; Nucleotidyltransferases; Quinacrine; Quinine; Spermine | 1966 |
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats | 1969 |
[Asthma therapy with a combination of synthetic antimalarials (83 cases)].
Topics: Adolescent; Adult; Aged; Asthma; Chloroquine; Drug Synergism; Electrocardiography; Eosinophilia; Eye Manifestations; Glucocorticoids; Humans; Middle Aged; Pyridoxine; Quinacrine; Sympathomimetics; Vitamin B Complex | 1969 |
An automated method of mass drug testing applied to screening for antimalarial activity.
Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones | 1970 |
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium | 1970 |
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium | 1970 |
Antimalarials: effects on in vivo and in vitro protein synthesis.
Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena | 1970 |
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines | 1970 |
The chemotherapy of rodent malaria. XII. Substituted tetrahydrofurans, a new chemical family of antimalarials. The action of 2-(p-chlorophenyl)-2-(4-piperidyl)-tetrahydrofuran against Plasmodium berghei and Plasmodium chabaudi.
Topics: Aminobenzoates; Animals; Antimalarials; Chloroquine; Diet; Drug Resistance, Microbial; Drug Synergism; Folic Acid; Furans; Mice; Piperidines; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines | 1970 |
[Cytostatic effect of resochin and atebrin (compare same journal 20 (N.F.) 28: 1591 (1969))].
Topics: Animals; Antineoplastic Agents; Chloroquine; Humans; Neoplasms; Neoplasms, Experimental; Quinacrine | 1970 |
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines | 1967 |
[Tropical diseases treated at Roslagstulls Hospital].
Topics: Adolescent; Adult; Aged; Amebiasis; Anti-Bacterial Agents; Antimony; Child; Chloroquine; Diethylcarbamazine; Female; Filariasis; Giardiasis; Hospitals, General; Humans; Malaria; Male; Middle Aged; Quinacrine; Schistosomiasis; Sweden | 1967 |
The inhibitory effect of mepacrine and chloroquine on the photodynamic action.
Topics: Animals; Chloroquine; Depression, Chemical; Light; Methylene Blue; Quinacrine; Tetrahymena | 1967 |
Synthesis and antimalarial evaluation of some 1,7-nephthyridines and 2,9-diazaanthracenes.
Topics: Animals; Benzene Derivatives; Chloroquine; Malaria; Methods; Mice; Naphthyridines; Quinacrine | 1968 |
Psychiatric complications with chloroquine and quinacrine.
Topics: Anti-Inflammatory Agents; Chloroquine; Humans; Malaria; Malingering; Psychoses, Substance-Induced; Quinacrine; Suicide; United States | 1968 |
Erythema dyschromicum perstans.
Topics: Adolescent; Adult; Biopsy; Blood Cell Count; Blood Sedimentation; Child, Preschool; Chloroquine; Erythema; Feces; Female; Humans; Hydroquinones; Hydroxychloroquine; Male; Middle Aged; Parasitic Diseases; Prednisone; Quinacrine; Steroids; Syphilis Serodiagnosis; Triamcinolone | 1968 |
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena | 1968 |
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine | 1968 |
Ocular toxicity of antimalarial drugs. Long-term follow-up.
Topics: Adolescent; Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Electrooculography; Electroretinography; Eye Diseases; Follow-Up Studies; Fundus Oculi; Humans; Hydroxychloroquine; Light; Lupus Erythematosus, Systemic; Macula Lutea; Middle Aged; Ophthalmoscopy; Quinacrine; Retinitis; Vision Tests; Visual Fields | 1968 |
The Plasmodium chabaudi-mouse system in chemotherapy studies.
Topics: Animals; Antimalarials; Chloroquine; Injections, Intravenous; Malaria; Male; Mice; Plasmodium; Primaquine; Quinacrine | 1969 |
Immunosuppression by compounds which complex with deoxyribonucleic acid.
Topics: Acridines; Alcohols; Animals; Antibody Formation; Chloroquine; Coloring Agents; DNA; Erythrocytes; Female; Fishes; Immunosuppressive Agents; Male; Methods; Mice; Protein Binding; Quinacrine; Quinolines; Sheep; Spleen; Splenomegaly; Transplantation Immunology; Transplantation, Homologous | 1969 |
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines | 1965 |
Chloroquine: physiological basis of drug resistance in Plasmodium berghei.
Topics: Animals; Carbon Isotopes; Chloroquine; Drug Resistance, Microbial; Erythrocytes; In Vitro Techniques; Liver; Malaria; Male; Mice; Plasmodium; Quinacrine; Quinine; Radiometry; Spleen | 1966 |
Mepacrine and chloroquine in vitiligo.
Topics: Chloroquine; Female; Humans; Male; Quinacrine; Vitiligo | 1966 |
[Ocular accidents from synthetic antimalarials (apropos of 4 new cases)].
Topics: Adolescent; Antimalarials; Child; Chloroquine; Electroretinography; Eye Diseases; Humans; Quinacrine | 1966 |
Metabolic effects of anthelmintic drugs on the cat's tapeworm in vitro.
Topics: Animals; Anthelmintics; Cats; Cestoda; Chloroquine; Glycolysis; In Vitro Techniques; Plant Extracts; Plants, Medicinal; Quinacrine; Resins, Plant; Respiration | 1966 |
Treatment of chloroquine-resistant Plasmodium falciparum infections in Vietnam.
Topics: Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Vietnam | 1967 |
The different effects of antimalarial drugs on Plasmodium lophurae developing intracellularly and extracellularly in vitro.
Topics: Animals; Chloroquine; In Vitro Techniques; Malaria, Avian; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine | 1967 |
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA | 1967 |
An analysis of the inhibitory effects of quinine and mepacrine in the guinea-pig isolated ileum.
Topics: Animals; Chloroquine; Depression, Chemical; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Prostaglandin Antagonists; Prostaglandins E; Quinacrine; Quinine | 1980 |
Stimulation of polymorphonuclear leucocyte phospholipase A2 activity by chloroquine and mepacrine.
Topics: Animals; Ascitic Fluid; Chloroquine; Escherichia coli; Female; In Vitro Techniques; Neutrophils; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rabbits | 1982 |
Interaction of basic compounds with coated vesicles.
Topics: Alkanesulfonates; Alkanesulfonic Acids; Amines; Animals; Brain; Buffers; Cattle; Centrifugation, Density Gradient; Chloroquine; Clathrin; Coated Pits, Cell-Membrane; Diamines; Endosomes; Hydrogen-Ion Concentration; Light; Morpholines; Polyamines; Quinacrine; Scattering, Radiation | 1984 |
Inhibition of lymphocyte transformation by mepacrine and chloroquine.
Topics: 1-Methyl-3-isobutylxanthine; Cells, Cultured; Chloroquine; Humans; In Vitro Techniques; Leucine; Lymphocyte Activation; Phytohemagglutinins; Quinacrine; Thymidine; Uridine | 1981 |
The effect of anti-malarial drugs on human natural killer cells in vitro.
Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines | 1984 |
Comparative effects of intrauterine instillation of analogues of quinacrine and tetracycline on uterine morphology in the rat.
Topics: Animals; Chloroquine; Demeclocycline; Doxycycline; Female; Primaquine; Quinacrine; Rats; Rats, Inbred Strains; Sodium Chloride; Tetracycline; Tetracyclines; Trimethoprim; Uterus | 1984 |
Inhibition of lipid peroxidation in muscle homogenates by phospholipase A2 inhibitors.
Topics: Animals; Chloroquine; Chlorpromazine; Dibucaine; Female; Free Radicals; In Vitro Techniques; Iron; Lipid Peroxides; Mice; Muscles; Phospholipases; Phospholipases A; Phospholipases A2; Procaine; Quinacrine; Tetracaine | 1984 |
Inhibition of rat hepatic mixed function oxidases by antimalarial drugs: selectivity for cytochromes P-450 and P-448.
Topics: Animals; Antimalarials; Chloroquine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Cytochromes; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases; Oxidoreductases, N-Demethylating; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1984 |
Corneal lipidosis in rats treated with amphiphilic cationic drugs.
Topics: Animals; Cations; Chloroquine; Chlorphentermine; Corneal Diseases; Female; Iprindole; Lipidoses; Male; Quinacrine; Rats; Rats, Inbred Strains; Tamoxifen | 1983 |
The chemotherapy of rodent malaria XXXIII. The activity of chloroquine and related blood schizontocides and of some analogues in drug-induced pigment clumping.
Topics: Amodiaquine; Animals; Chloroquine; Cyclic N-Oxides; Dose-Response Relationship, Drug; Erythrocytes; Pigmentation; Plasmodium berghei; Quinacrine | 1982 |
Inhibition of diamine oxidase by antimalarial drugs.
Topics: Amine Oxidase (Copper-Containing); Amodiaquine; Animals; Antimalarials; Chloroquine; In Vitro Techniques; Intestine, Small; Male; Putrescine; Quinacrine; Rats | 1980 |
Inhibition of the metabolism and motility of human spermatozoa by various alkaloids.
Topics: Antimalarials; Carbon Dioxide; Chloroquine; Emetine; Humans; Lactates; Lactic Acid; Male; Quinacrine; Quinine; Sperm Motility; Spermatozoa | 1982 |
Gas chromatographic analysis of chloroquine after a unique reaction with chloroformates.
Topics: Aminoquinolines; Chemical Phenomena; Chemistry; Chloroquine; Chromatography, Gas; Humans; Mass Spectrometry; Phosgene; Quinacrine | 1983 |
Suppression by phospholipase A2 inhibitors of secretion of catecholamines from isolated adrenal medullary cells by suppression of cellular calcium uptake.
Topics: Acetophenones; Adrenal Medulla; Animals; Calcium; Carbachol; Catecholamines; Cattle; Chloroquine; Dose-Response Relationship, Drug; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Quinine | 1983 |
The uptake of 14C-chloroquine by mouse pancreatic islets in vitro.
Topics: Absorption; Animals; Chloroquine; Chlorpromazine; Desipramine; Glucose; Hydrogen-Ion Concentration; Imipramine; Islets of Langerhans; Lidocaine; Mice; Nicotine; Nitrogen; Ouabain; Quinacrine; Temperature | 1980 |
Binding of antimalarial drugs to hemozoin from Plasmodium berghei.
Topics: Animals; Antimalarials; Chloroquine; Heme; Hemeproteins; Mefloquine; Methemoglobin; Pigments, Biological; Piperidines; Plasmodium berghei; Protein Binding; Protoporphyrins; Quinacrine; Quinolines; Spectrophotometry | 1980 |
Mechanism of action of gonadotropin-releasing hormone. Involvement of phospholipid turnover in luteinizing hormone release.
Topics: Animals; Arachidonic Acids; Calcium; Cells, Cultured; Chloroquine; Female; Gonadotropin-Releasing Hormone; Indomethacin; Kinetics; Luteinizing Hormone; Phospholipases A; Phospholipases A2; Pituitary Gland; Quinacrine; Rats | 1981 |
Comparative microcalorimetric dilatometric analysis of the interactions of quinacrine, chloroquine, and ethidium bromide with DNA.
Topics: Calorimetry; Chemistry Techniques, Analytical; Chloroquine; DNA; Ethidium; Osmolar Concentration; Quinacrine; Thermodynamics | 1982 |
[Influence of x-rays and quinacrine (atebrine) or chloroquine (resochine)--alone or in combination--on growth and melanin formation of Harding-Passey melanoma cells in monolayer culture].
Topics: Cell Survival; Cells, Cultured; Chloroquine; Dose-Response Relationship, Radiation; Melanins; Melanoma; Neoplasms, Experimental; Quinacrine | 1982 |
Effects of antimalarial drugs on several rat-liver lysosomal enzymes involved in phosphatidylethanolamine catabolism.
Topics: Animals; Antimalarials; Carboxylic Ester Hydrolases; Chloroquine; Dose-Response Relationship, Drug; Liver; Lysophospholipase; Lysosomes; Male; Monoacylglycerol Lipases; Phosphatidylethanolamines; Phospholipases; Phospholipases A; Phospholipases A1; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1982 |
Comparison of the effects of chloroquine quinacrine and quinidine on autonomic neuroeffector mechanisms.
Topics: Animals; Autonomic Nervous System; Chickens; Chloroquine; Electric Stimulation; Female; Indomethacin; Male; Mice; Norepinephrine; Quinacrine; Quinidine; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Tetrodotoxin | 1982 |
The effect of ionic strength on DNA-ligand unwinding angles for acridine and quinoline derivatives.
Topics: Aminacrine; Aminoacridines; Animals; Cattle; Chemical Phenomena; Chemistry; Chloroquine; DNA; Ethidium; Kinetics; Molecular Conformation; Nucleic Acid Conformation; Osmolar Concentration; Quinacrine; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Thymus Gland; Viscosity | 1980 |
Effects of several lipidosis-inducing drugs upon the area postrema and adjacent medullary nuclei of adult rats. II. Axonal alternations.
Topics: Animals; Axons; Chloroquine; Chlorphentermine; Medulla Oblongata; Microscopy, Electron; Perhexiline; Piperidines; Quinacrine; Rats | 1981 |
Pharmacological basis of dosage form of two antimalarials: chloroquine and mepacrine.
Topics: Administration, Oral; Animals; Chloroquine; Duodenum; Female; Gastric Emptying; Gastric Mucosa; Infusions, Parenteral; Injections, Intraperitoneal; Intubation, Gastrointestinal; Quinacrine; Rats; Rats, Inbred Strains | 1981 |
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine | 1980 |
Factors that influence the uptake of beta-hexosaminidase A by rat peritoneal macrophages.
Topics: Acetylglucosaminidase; Ammonium Chloride; Animals; Biological Transport; Chloroquine; Colchicine; Cytochalasin B; Female; Glycoproteins; Hexosaminidases; Humans; Kinetics; Macrophages; Methylamines; Phagocytosis; Placenta; Pregnancy; Quinacrine; Rats | 1980 |
Effect of chloroquine and mepacrine on the spontaneous and evoked movements of the rat portal vein.
Topics: Animals; Chloroquine; Dose-Response Relationship, Drug; Epinephrine; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Parasympatholytics; Parasympathomimetics; Phentolamine; Portal Vein; Quinacrine; Rats | 1980 |
[Intensification of the inhibitory effect of X-rays on the growth of Ehrlich ascites tumor cells in monolayer culture by quinacrine (atebrine) or chloroquine (resochine) (author's transl)].
Topics: Animals; Carcinoma, Ehrlich Tumor; Cell Division; Cells, Cultured; Chloroquine; Quinacrine; Radiotherapy Dosage | 1980 |
Effects of several lipidosis-including drugs upon the area postrema and adjacent medullary nuclei of adult rats. I. Alterations is perikarya and dendrites.
Topics: Animals; Blood-Brain Barrier; Brain Diseases; Chloroquine; Chlorphentermine; Female; Lipidoses; Male; Medulla Oblongata; Microscopy, Electron; Perhexiline; Piperidines; Quinacrine; Rats; Time Factors | 1980 |
Receptor-independent uptake of transferrin-bound iron by reticulocytes.
Topics: Animals; Biological Transport; Cations; Chloroquine; Cytosol; Dicumarol; Edetic Acid; Egtazic Acid; Endocytosis; Erythrocyte Membrane; Heme; In Vitro Techniques; Iodine Radioisotopes; Iron; Iron Radioisotopes; Kinetics; Quinacrine; Rabbits; Receptors, Transferrin; Reticulocytes; Transferrin; Tretinoin | 1994 |
Chloroquine-quinacrine association in resistant cutaneous lupus.
Topics: Adult; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Male; Middle Aged; Quinacrine | 1995 |
The association of the two antimalarials chloroquine and quinacrine for treatment-resistant chronic and subacute cutaneous lupus erythematosus.
Topics: Adult; Aged; Chloroquine; Drug Combinations; Drug Tolerance; Female; Humans; Hydroxychloroquine; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Male; Middle Aged; Quinacrine; Vision Disorders | 1994 |
Effects of vesicular acetylcholine uptake blockers on frequency augmentation-potentiation in frog neuromuscular transmission.
Topics: Acetylcholine; Animals; Antidepressive Agents; Azepines; Chloroquine; Ethacridine; Evoked Potentials; In Vitro Techniques; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Piperidines; Pyrilamine; Quinacrine; Ranidae; Regression Analysis; Synaptic Transmission | 1994 |
The effects of chronic administration of chloroquine and quinacrine on the response of normal and denervated smooth muscle to agonist drugs.
Topics: Acetylcholine; Age Factors; Animals; Atropine; Chickens; Chloroquine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Male; Muscle, Smooth; Neurotransmitter Agents; Norepinephrine; Potassium Chloride; Pyrilamine; Quinacrine; Serotonin; Synaptic Transmission | 1993 |
Enhanced growth of mammary adenocarcinoma in rats by chloroquine and quinacrine.
Topics: Adenocarcinoma; Animals; Body Weight; Cell Division; Chloroquine; Dinoprostone; Erythrocytes; Female; Glutathione; Mammary Neoplasms, Experimental; Neoplasm Transplantation; Oxygen; Quinacrine; Rats; Rats, Inbred F344; Riboflavin; Riboflavin Deficiency; Stimulation, Chemical; Stress, Physiological | 1994 |
Differential binding of the enantiomers of chloroquine and quinacrine to polynucleotides: implications for stereoselective metabolism.
Topics: Chloroquine; Polynucleotides; Quinacrine; Stereoisomerism | 1993 |
Cytotoxic activity of lutropin-gelonin conjugate in mouse Leydig tumor cells: potentiation of the hormonotoxin activity by different drugs.
Topics: Animals; Antineoplastic Agents; Chloroquine; Drug Screening Assays, Antitumor; Drug Synergism; Leydig Cell Tumor; Leydig Cells; Luteinizing Hormone; Male; Mice; Monensin; Neoplasm Proteins; Plant Proteins; Progesterone; Protein Synthesis Inhibitors; Quinacrine; Receptors, LH; Ribosome Inactivating Proteins, Type 1; Testicular Neoplasms; Tumor Cells, Cultured; Verapamil | 1993 |
The antimalarials quinacrine and chloroquine induce weak lysosomal storage of sulphated glycosaminoglycans in cell culture and in vivo.
Topics: Animals; Anti-Inflammatory Agents; Antimalarials; beta-N-Acetylhexosaminidases; Cattle; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Female; Fibroblasts; Glycosaminoglycans; Histocytochemistry; Lipidoses; Liver; Lysosomes; Microscopy, Electron; Microscopy, Fluorescence; Mucopolysaccharidoses; Quinacrine; Rats; Rats, Wistar; Structure-Activity Relationship; Sulfates; Tilorone | 1996 |
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication | 1996 |
Activity of pyronaridine and mepacrine against twelve strains of Plasmodium falciparum in vitro.
Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Mefloquine; Naphthyridines; Plasmodium falciparum; Quinacrine; Quinine | 1996 |
Xanthones as antimalarial agents; studies of a possible mode of action.
Topics: Animals; Antimalarials; Chloroquine; Heme; Humans; Plasmodium falciparum; Polymers; Primaquine; Quinacrine; Structure-Activity Relationship; Xanthenes; Xanthones | 1997 |
Opposing effects of quinacrine and chloroquine on the development of TA3 transplanted tumors in mice.
Topics: Animals; Antineoplastic Agents; Cell Division; Chloroquine; Male; Mice; Neoplasm Transplantation; Quinacrine | 1995 |
Interaction of local anaesthetics with histamine H1 receptors in guinea-pig ileum.
Topics: Anesthetics, Local; Animals; Binding, Competitive; Chloroquine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Isotope Labeling; Male; Muscle Contraction; Muscle, Smooth; Procaine; Pyrilamine; Quinacrine; Receptors, Histamine H1; Structure-Activity Relationship; Tetracaine | 1997 |
Lysosomotropic agents ameliorate macrophage dysfunction following the phagocytosis of IgG-coated erythrocytes: a role for lipid peroxidation.
Topics: Ammonium Chloride; Animals; Chloroquine; Erythrocytes; Immunoglobulin G; Lipid Peroxidation; Macrophage Activation; Macrophages, Peritoneal; Methylamines; Phagocytosis; Quinacrine; Rats; Rats, Sprague-Dawley | 1997 |
CpG-oligodeoxynucleotide supports growth of IL-6-dependent 7TD1 murine hybridoma cells.
Topics: Animals; Antimalarials; Cell Count; Cell Division; Chloroquine; Dose-Response Relationship, Drug; Hybridomas; Interleukin-6; Mice; Oligodeoxyribonucleotides; Quinacrine | 1998 |
Antimalarial drugs inhibit phospholipase A2 activation and induction of interleukin 1beta and tumor necrosis factor alpha in macrophages: implications for their mode of action in rheumatoid arthritis.
Topics: Animals; Antimalarials; Chloroquine; Eicosanoids; Female; Interleukin-1; Macrophages, Peritoneal; Mice; Phospholipases A; Phospholipases A2; Quinacrine; Tumor Necrosis Factor-alpha | 1998 |
Antagonism of immunostimulatory CpG-oligodeoxynucleotides by quinacrine, chloroquine, and structurally related compounds.
Topics: Acids; Adjuvants, Immunologic; Animals; Apoptosis; Binding, Competitive; Biological Transport; Cell Division; Cell Line; Chloroquine; CpG Islands; Drug Resistance, Multiple; Humans; Immunosuppressive Agents; Intercalating Agents; Interleukin-6; Kinetics; Leukocytes, Mononuclear; Lipopolysaccharides; Mice; Oligodeoxyribonucleotides; Quinacrine; Structure-Activity Relationship; Thionucleotides | 1998 |
[Combination of antimalarial drugs mepacrine and chloroquine in therapy refractory cutaneous lupus erythematosus].
Topics: Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Facial Dermatoses; Female; Humans; Lupus Erythematosus, Discoid; Quinacrine | 2000 |
Conditional lethality of the diprotic weak bases chloroquine and quinacrine against Cryptococcus neoformans.
Topics: Anti-Bacterial Agents; Antifungal Agents; Cell Division; Chloroquine; Cryptococcus neoformans; Drug Combinations; Enzyme Inhibitors; Macrolides; Microbial Sensitivity Tests; Quinacrine | 2000 |
Reduced inflammatory response to plasmid DNA vectors by elimination and inhibition of immunostimulatory CpG motifs.
Topics: Administration, Intranasal; Animals; Antimalarials; Bronchoalveolar Lavage Fluid; Chloroquine; CpG Islands; Cytokines; DNA, Bacterial; Gene Transfer Techniques; Genetic Vectors; Inflammation; Interleukin-12; Lipids; Lung; Mice; Mice, Inbred BALB C; Mutagenesis, Site-Directed; Plasmids; Quinacrine; Sequence Deletion; Spleen | 2000 |
Blastocystis hominis: neutral red supravital staining and its application to in vitro drug sensitivity testing.
Topics: Amebicides; Animals; Blastocystis hominis; Chloroquine; Coloring Agents; Humans; Metronidazole; Neutral Red; Nitro Compounds; Parasitic Sensitivity Tests; Paromomycin; Quinacrine; Staining and Labeling; Sulfamethoxazole; Tetracycline; Thiazoles; Trimethoprim | 2000 |
The antimalarials quinacrine and chloroquine potentiate the transplacental carcinogenic effect of ethylnitrosourea on ependymal cells.
Topics: Animals; Antimalarials; Brain Neoplasms; Carcinogens; Chloroquine; Drug Synergism; Ependyma; Ependymoma; Ethylnitrosourea; Female; Glial Fibrillary Acidic Protein; Immunoenzyme Techniques; Male; Pregnancy; Prenatal Exposure Delayed Effects; Quinacrine; Rats; Rats, Wistar; Spinal Cord Neoplasms; Synaptophysin | 2001 |
The effect of chloroquine, quinacrine, and metronidazole on both soybean plants and soil microbiota.
Topics: Animals; Anti-Bacterial Agents; Antimalarials; Bacteria; Chloroquine; Eukaryota; Glycine max; Metronidazole; Plant Roots; Population Dynamics; Quinacrine; Soil Microbiology | 2002 |
[The treatment of giardiasis; nivaquine or quinacrine].
Topics: Chloroquine; Giardiasis; Quinacrine; Quinolines | 1952 |
Enteritis due to flagellata in children.
Topics: Child; Chloroquine; Enteritis; Giardiasis; Humans; Infant; Quinacrine | 1952 |
[Case of malaria due to Plasmodium falciparum resistant to quinacrine and to quinine and treated with nivaquine].
Topics: Chloroquine; Humans; Malaria; Plasmodium falciparum; Quinacrine; Quinine | 1952 |
Screening of antimalarials against P. gallinaceum in chicks.
Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Chickens; Chloroquine; Malaria; Proguanil; Quinacrine; Quinine; Sulfadiazine | 1952 |
[Superiority of premaline over quinacrine and nivaquine in the treatment of lambliasis].
Topics: Aminoquinolines; Chloroquine; Giardiasis; Humans; Quinacrine; Quinolines | 1953 |
Atabrine and chloroquine in the treatment of chronic discoid lupus erythematosus.
Topics: Chloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1953 |
Light sensitive eruptions treated with atabrine and chloroquine.
Topics: Chloroquine; Dermatitis; Light; Quinacrine | 1954 |
The use of chloroquine diphosphate (aralen) and quinacrine (atabrine) hydrochloride in the prevention of polymorphorus light eruptions.
Topics: Biomedical Research; Chloroquine; Light; Lupus Erythematosus, Systemic; Quinacrine; Sunlight | 1954 |
Synthetic antimalarial drugs in chronic discoid lupus erythematosus and light eruptions.
Topics: Antimalarials; Chloroquine; Light; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases; Sunlight | 1954 |
[Serological research in chronic inflammatory rheumatism; study of antistreptolysin O].
Topics: Antistreptolysin; Arthritis, Rheumatoid; Chloroquine; Chronic Disease; Humans; Quinacrine; Research; Rheumatic Fever | 1954 |
[Atebrine and chloroquine/resochin therapy of lupus erythematous and dermatoses due to photosensitivity].
Topics: Chloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases | 1954 |
[Atebrin and resochin treatment in progressive chronic polyarthritis].
Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine | 1955 |
Studies on the treatment of Opisthorchis viverrini in human infections with quinacrine hydrochloride and chloroquine phosphate.
Topics: Animals; Chloroquine; Infections; Opisthorchis; Quinacrine | 1955 |
Treatment on malaria with single doses of mepacrine, chloroquine and amodiaquin.
Topics: Amodiaquine; Antimalarials; Chloroquine; Humans; Malaria; Quinacrine | 1955 |
Mepacrine and chloroquine in the treatment of rosacea.
Topics: Chloroquine; Humans; Quinacrine; Rosacea | 1955 |
[Comparative study of the effect of quinacrine, nivaquine B and C on giardiasis].
Topics: Chloroquine; Giardiasis; Humans; Quinacrine; Quinolines | 1955 |
[Antimalarial drugs in therapy of chronic evolutive polyarthritis].
Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine | 1955 |
[Lupus erythematosus, etiology, pathogenesis and therapy].
Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine | 1956 |
[Reaction of the human skin to ultraviolet rays. 10. Effects of atebrin and resochin on skin sensitivity].
Topics: Chloroquine; Humans; Quinacrine; Skin; Skin Physiological Phenomena; Sunlight; Ultraviolet Rays | 1957 |
Systemic lupus erythematosus; a report on twelve cases treated with quinacrine (atabrine) and chloroquine (aralen).
Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine | 1957 |
The efficiency of local application of chloroquine and mepacrine in preventing the effects of ultraviolet rays on human skin.
Topics: Chloroquine; Humans; Quinacrine; Skin; Ultraviolet Rays | 1957 |
Treatment of lupus erythematosus with chloroquine; therapeutic results and a comparison of the value of chloroquine and mepacrine.
Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1957 |
The treatment of lupus erythematosus and lymphocytic infiltration of the skin with A.P.A. 5533.
Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin; Skin Diseases | 1957 |
[Quinacrine & chloroquine in asthma therapy].
Topics: Asthma; Chloroquine; Disease; Peritoneal Diseases; Peritoneum; Quinacrine | 1957 |
[Chloroquine therapy of lupus erythematosus; comparative effectivity of chloroquine and mepacrine].
Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Quinacrine | 1957 |
Treatment of chronic lupus erythematosus: effectiveness of plaquenil and APA (Aralen 65 mg., plaquenil 50 mg., Atabrine 25 mg.) as compared with Aralen, with observations on side-reactions and toxicity; report and presentation of unusual cases.
Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1958 |
Treatment of rheumatoid arthritis with quinacrine and chloroquine.
Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine | 1958 |
[Experimental malaria: Plasmodium berghei].
Topics: Chloroquine; Malaria; Plasmodium berghei; Quinacrine; Quinine | 1958 |
[Experimental & clinical studies on the mechanism of action of atabrine & resochin in chronic lupus erythematosus].
Topics: Biomedical Research; Chloroquine; Lupus Erythematosus, Systemic; Quinacrine | 1958 |
[Atabrine and resohine therapy of lupus erythematosus].
Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine | 1957 |
[Long term treatment of rheumatoid arthritis with mepacrine & chloroquine].
Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Long-Term Care; Quinacrine | 1958 |
Triquin in the treatment of discoid lupus erythematosus and light sensitive eruptions.
Topics: Chloroquine; Exanthema; Humans; Light; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases | 1958 |
Lupus erythematosus treated with a combination of quinacrine, hydroxychloroquine and chloroquine.
Topics: Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1959 |
Initial clinical trial of the nitrogen mustard analogues of chloroquine and quinacrine; a preliminary report.
Topics: Chloroquine; Humans; Mechlorethamine; Nitrogen Mustard Compounds; Quinacrine | 1958 |
The use of triquin in the treatment of discoid lupus erythematosus and some other skin conditions.
Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases | 1959 |
[Observations on quinacrine & chloroquine in the treatment of petit mal; preliminary report].
Topics: Chloroquine; Epilepsy; Epilepsy, Absence; Quinacrine | 1959 |
Successful treatment of hepatic and splenic amebic abscesses with atabrine after failure of emetine, chloroquine and terramycin.
Topics: Amebiasis; Chloroquine; Disease; Dysentery, Amebic; Emetine; Humans; Liver Abscess; Oxytetracycline; Quinacrine; Spleen | 1960 |
Single dose treatment of malaria with amodiaquin chloroquine and mepacrine in a semi-immune poplation.
Topics: Amodiaquine; Antimalarials; Chloroquine; Humans; Malaria; Quinacrine | 1960 |
Action of quinine, qunidine mepacrine and chloroquine on the skeletal muscle.
Topics: Antimalarials; Chloroquine; Humans; Muscle, Skeletal; Muscles; Quinacrine; Quinine | 1960 |
[Discolorations of atabrine and resochin solutions by autogenous, reducing substances after UV irradiation].
Topics: Chloroquine; Quinacrine; Solutions; Ultraviolet Rays | 1960 |
[Modification of Rh antigen-antibody reactions].
Topics: Antigen-Antibody Reactions; Aspirin; Chloroquine; Humans; Phenylbutazone; Quinacrine | 1962 |
Reaction between DNA and quinacrine and other antimalarials.
Topics: Antimalarials; Chloroquine; DNA; Quinacrine; Quinidine; Quinine | 1962 |
[Skin symptoms caused by synthetic antimalarials].
Topics: Antimalarials; Chloroquine; Drug Eruptions; Humans; Quinacrine | 1963 |
[Treatment of discoid lupus erythematosus, polymorphous photodermatosis and rosacea with Triquin--a combination of 3 anti-malarials].
Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Photosensitivity Disorders; Quinacrine; Rosacea | 1962 |
In vivo and in vitro effects of antimalarials on Histoplasma capsulatum.
Topics: Amodiaquine; Antimalarials; Chloroquine; Histoplasma; Humans; In Vitro Techniques; Primaquine; Quinacrine | 1962 |
[Therapeutic use of 22/360 (Collagenan) during various collagen diseases].
Topics: 4-Aminobenzoic Acid; Antimalarials; Chloroquine; Collagen Diseases; Drug Combinations; Humans; Pantothenic Acid; Pyridoxine; Quinacrine; Vitamin B Complex | 1963 |
Oral contraceptives. VII. Antimalarials as antifertility agents.
Topics: Amodiaquine; Antimalarials; Chloroquine; Contraceptive Agents; Contraceptives, Oral; Female; Humans; Proguanil; Pyrimethamine; Quinacrine | 1962 |
[Report on the use, in the treatment of chronic evolutive polyarthritis, of a drug combining notably 2 synthetic antimalarials].
Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine | 1963 |
SOLAR URTICARIA.
Topics: Chloroquine; Dermatitis, Phototoxic; Humans; Photosensitivity Disorders; Porphyrins; Pregnancy; Quinacrine; Toxicology; Urticaria | 1963 |
[ON DARK PIGMENTATIONS DUE TO ATABRINE AND AMODIAQUINE].
Topics: Amodiaquine; Chloroquine; Pigmentation; Pigmentation Disorders; Quinacrine; Toxicology | 1963 |
DRUG RESISTANCE IN PLASMODIUM FALCIPARUM FROM THAILAND.
Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand | 1963 |
PIGMENTATION FROM ANTIMALARIAL THERAPY. ITS POSSIBLE RELATIONSHIP TO THE OCULAR LESIONS.
Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Cornea; Eye; Eye Manifestations; Histocytochemistry; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Photomicrography; Pigmentation; Pigmentation Disorders; Quinacrine; Retina; Toxicology | 1963 |
LUPUS ERYTHEMATOSUS--A CLINICAL QUIZ. A SERIES OF DIAGNOSTIC AND THERAPEUTIC PROBLEMS.
Topics: Chloroquine; Diagnosis; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1963 |
POLYMORPHOUS LIGHT ERUPTION. A TEN-YEAR FOLLOW-UP AND EVALUATION.
Topics: Chloroquine; Dermatitis, Phototoxic; Follow-Up Studies; Humans; Hydroxychloroquine; Lupus Erythematosus, Systemic; Photosensitivity Disorders; Prurigo; Quinacrine; Seasons; Sunlight | 1963 |
ANTIMALARIAL DRUGS ON THE AUTOMATICITY OF SINO-AURICULAR AND ATRIO-VENTRICULAR NODES.
Topics: Administration, Intravenous; Amodiaquine; Animals; Anti-Arrhythmia Agents; Antimalarials; Atrioventricular Node; Atropine; Chloroquine; Dogs; Heart Conduction System; Humans; Hydroxychloroquine; Hypotension; Injections, Intravenous; Primaquine; Quinacrine; Quinidine; Research; Statistics as Topic | 1963 |
DRUG-RESISTANT FALCIPARUM MALARIA FROM CAMBODIA AND MALAYA.
Topics: Animals; Cambodia; Chloroquine; Culicidae; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Malaria, Falciparum; Malaysia; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine | 1963 |
TOXIC PSYCHOSIS DUE TO QUINARCRINE AND CHLOROQUINE.
Topics: Amebiasis; Chloroquine; Giardiasis; Humans; Psychoses, Substance-Induced; Psychotic Disorders; Quinacrine; Toxicology; Trichomonas Infections | 1964 |
[CHRONIC DISCOID ERYTHEMATOSUS (REPORT ON 69 CASES OVER A PERIOD OF 6 YEARS FROM THE VIEWPOINT OF OPTIMUM THERAPY)].
Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine | 1963 |
HAEMATOLOGICAL SIDE-EFFECTS OF SOME ANTI-RHEUMATIC DRUGS.
Topics: Aminopyrine; Antirheumatic Agents; Aspirin; Blood Platelets; Chloroquine; Colchicine; Complement Fixation Tests; Drug Hypersensitivity; Gold; Humans; Hydroxychloroquine; Meprobamate; Phenacetin; Phenylbutazone; Probenecid; Purpura; Purpura, Thrombocytopenic; Quinacrine; Rheumatic Diseases; Splenectomy; Toxicology | 1963 |
ANTIHELMINTHIC THERAPY: A SIMPLIFIED APPROACH.
Topics: Amebiasis; Anthelmintics; Ascariasis; Chloroquine; Dysentery, Amebic; Giardiasis; Hookworm Infections; Humans; Oxytetracycline; Quinacrine; Strongyloidiasis; Trichinellosis | 1964 |
ANTIMALARIALS AND OTHER ANTICONVULSANT DRUGS: PREDICTIVE VALIDITY OF LABORATORY TESTS.
Topics: Animals; Anticonvulsants; Antimalarials; Chloroquine; Electric Stimulation; Hydroxychloroquine; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Phenytoin; Quinacrine; Research; Seizures | 1964 |
STUDIES ON A STRAIN OF CHLOROQUINE-RESISTANT PLASMODIUM FALCIPARUM FROM THAILAND.
Topics: Amodiaquine; Antimalarials; Asia, Southeastern; Biomedical Research; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Hydroxychloroquine; Malaria; Malaria, Falciparum; Pharmacology; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand | 1964 |
DRUG-RESISTANCE IN FALCIPARUM MALARIA IN SOUTH-EAST ASIA.
Topics: Adolescent; Asia, Southeastern; Child; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Drug Therapy; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Statistics as Topic; Toxicology | 1964 |
[MODERN ANTHELMINTIC DRUGS].
Topics: Anthelmintics; Chemical Phenomena; Chemistry; Chloroquine; Diethylcarbamazine; Dithiazanine; Dryopteris; Gentian Violet; Humans; Niclosamide; Piperazines; Pyrvinium Compounds; Quinacrine | 1964 |
ANTIHISTAMINIC ACTION OF ANTIMALARIALS.
Topics: Acetylcholine; Animals; Antimalarials; Blood Pressure; Blood Pressure Determination; Capillary Permeability; Chloroquine; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Muscle, Smooth; Pharmacology; Quinacrine; Quinine; Research | 1963 |
[PSORIASIS AND ITS TREATMENT IN THE LIGHT OF A NEW EXPERIENCE].
Topics: Chloroquine; Fluocinolone Acetonide; Humans; Light; Psoriasis; Quinacrine | 1964 |
THE EFFECT OF CERTAIN SUBSTANCES AGAINST ECHINOCOCCUS GRANULOSUS AND TAENIA HYDATIGENA INFECTIONS IN DOGS.
Topics: Animals; Anthelmintics; Benzimidazoles; Chloroquine; Dithiazanine; Dog Diseases; Dogs; Echinococcosis; Echinococcus granulosus; England; Fascioliasis; Hexachlorophene; Hexylresorcinol; Iodoquinol; Niclosamide; Piperazines; Protozoan Infections; Quinacrine; Taenia; Thiabendazole | 1964 |
[APROPOS OF LAMBLIASIS IN CHILDHOOD].
Topics: Acridines; Adolescent; Child; Chloroquine; Drug Therapy; Giardiasis; Humans; Quinacrine; Quinolines | 1964 |
CHILBLAIN LUPUS ERYTHEMATOSUS.
Topics: Chilblains; Chloroquine; Fluocinolone Acetonide; Frostbite; Humans; Hydroxychloroquine; Hypothyroidism; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Niacinamide; Quinacrine; Telangiectasis; Triamcinolone | 1964 |
THE ABSENCE OF ANTICONVULSANT PROPERTIES OF QUINACRINE AND CHLOROQUINE IN MICE.
Topics: Anticonvulsants; Chloroquine; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Quinacrine; Research; Seizures; Toxicology | 1964 |
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology | 1964 |
ALIMENTARY HYPERSENSITIVITY INDUCED BY GIARDIA LAMBLIA; REPORT OF A CASE OF ACUTE MEAT INTOLERANCE.
Topics: Abdomen; Abdomen, Acute; Chloroquine; Drug Therapy; Food Hypersensitivity; Giardia lamblia; Giardiasis; Humans; Meat; Pathology; Quinacrine | 1965 |
PLEUROPULMONARY AMEBIASIS. CLINICAL ANALYSIS OF 64 CASES.
Topics: Amebiasis; Chloroquine; Diagnosis, Differential; Drainage; Drug Therapy; Emetine; Empyema; Humans; Liver Abscess; Liver Abscess, Amebic; Lung Abscess; Lung Diseases, Parasitic; Pathology; Pleural Effusion; Pleurisy; Prognosis; Quinacrine; Radiography, Thoracic | 1965 |
[ALLERGIC CONTACT ECZEMA CAUSED BY RESOCHIN].
Topics: Chloroquine; Dermatitis; Dermatitis, Allergic Contact; Dermatitis, Contact; Quinacrine; Skin Tests; Toxicology | 1965 |
Treatment of chronic lupus erythematosus with atabrine and chloroquine.
Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine | 1955 |
[Recent experience in the treatment of erythematodes chronicus discoides with atebrin and resochin, with special reference to local and combined therapeutic methods].
Topics: Chloroquine; Combined Modality Therapy; Erythema; Humans; Quinacrine | 1955 |
[Treatment of chronic lupus erythematosus with synthetic antimalarials: quinacrine and chloroquine].
Topics: Antimalarials; Chloroquine; Humans; Lupus Erythematosus, Systemic; Quinacrine | 1955 |
Clinical findings for the treatment of Mucha-Habermann disease (parapsoriasis varioliformis) with acridine and chinoline derivatives.
Topics: Acridines; Chloroquine; Humans; Parapsoriasis; Pityriasis Lichenoides; Quinacrine | 1959 |
Evaluation of synthetic anti-malarial drugs in children from a hyperendemic area in West Africa.
Topics: Africa, Western; Antimalarials; Child; Chloroquine; Humans; Malaria; Quinacrine | 1951 |
Chemotherapy of amebic hepatitis in hamsters with emetine, chloroquine, amodiaquin (camoquin), quinacrine and other drugs.
Topics: Amebiasis; Amodiaquine; Chloroquine; Dysentery, Amebic; Emetine; Hepatitis; Liver Diseases; Quinacrine | 1951 |
Inhibitors of the K+(Na+)/H+ exchanger of human red blood cells.
Topics: Chloroquine; Dose-Response Relationship, Drug; Erythrocytes; Humans; Osmolar Concentration; Potassium; Potassium-Hydrogen Antiporters; Quinacrine; Sodium-Hydrogen Exchangers | 2004 |
Kinetic mechanism of quinone oxidoreductase 2 and its inhibition by the antimalarial quinolines.
Topics: Antimalarials; Binding, Competitive; Chloroquine; Copper; Humans; Kinetics; Niacinamide; Oxidation-Reduction; Primaquine; Quinacrine; Quinolines; Quinone Reductases; Recombinant Proteins; Spectrophotometry; Substrate Specificity; Zinc | 2004 |
Toll-like receptor 9 binds single-stranded CpG-DNA in a sequence- and pH-dependent manner.
Topics: Amino Acid Sequence; Binding Sites; Cell Line; Chloroquine; CpG Islands; DNA, Single-Stranded; Humans; Hydrogen-Ion Concentration; Membrane Glycoproteins; Molecular Sequence Data; Quinacrine; Receptors, Cell Surface; Toll-Like Receptor 2; Toll-Like Receptor 9; Toll-Like Receptors | 2004 |
The sensitivities of yeast strains deficient in PDR ABC transporters, to quinoline-ring antimalarial drugs.
Topics: Antimalarials; ATP-Binding Cassette Transporters; Chloroquine; Cycloheximide; Drug Resistance, Multiple, Fungal; Gene Deletion; Genes, Fungal; Mefloquine; Mutation; Quinacrine; Quinidine; Quinine; Saccharomyces cerevisiae; Transcription, Genetic | 2004 |
Involvement of the nonhomologous region of subunit A of the yeast V-ATPase in coupling and in vivo dissociation.
Topics: Adenosine Triphosphate; Blotting, Western; Catalysis; Chloroquine; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Epitopes; Escherichia coli; Genetic Vectors; Glucose; Hydrogen-Ion Concentration; Immunoprecipitation; Mutation; Plasmids; Protein Binding; Protein Structure, Tertiary; Protons; Quinacrine; Saccharomyces cerevisiae; Time Factors; Vacuolar Proton-Translocating ATPases; Vacuoles | 2004 |
Chloroquine, proguanil, mepacrine and quinine in the treatment of malaria caused by Plasmodium falciparum.
Topics: Chloroquine; Humans; Malaria; Plasmodium falciparum; Proguanil; Quinacrine; Quinine | 1949 |
[Systemic lupus erythematosus therapy. Antimalarials in inflammatory diseases].
Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Systemic; Quinacrine | 2004 |
Anthrax toxin protective antigen: inhibition of channel function by chloroquine and related compounds and study of binding kinetics using the current noise analysis.
Topics: Algorithms; Antigens, Bacterial; Bacterial Toxins; Binding Sites; Chloroquine; Fluphenazine; Ion Channel Gating; Ion Channels; Lipid Bilayers; Permeability; Quinacrine; Recombinant Proteins | 2005 |
Quinacrine but not chloroquine inhibits PMA induced upregulation of matrix metalloproteinases in leukocytes: quinacrine acts at the transcriptional level through a PLA2-independent mechanism.
Topics: Antigens, Human Platelet; Antirheumatic Agents; Cell Survival; Chloroquine; Dose-Response Relationship, Drug; Gene Expression Regulation, Enzymologic; Humans; Leukocytes, Mononuclear; Matrix Metalloproteinases; Phorbol Esters; Quinacrine; RNA, Messenger; Transcription, Genetic; Up-Regulation | 2006 |
CpG-induced tyrosine phosphorylation occurs via a TLR9-independent mechanism and is required for cytokine secretion.
Topics: Actin Cytoskeleton; Adaptor Proteins, Signal Transducing; Androstadienes; Animals; Antigens, CD; Cell Adhesion; Cell Line, Tumor; Cell Membrane; Chloroquine; CpG Islands; Cytokines; Cytoskeleton; Dendritic Cells; Humans; I-kappa B Proteins; Interferon-alpha; Interleukin-6; Intracellular Signaling Peptides and Proteins; Macrophages; Mice; Mice, Knockout; Models, Biological; Monocytes; Myeloid Differentiation Factor 88; NF-KappaB Inhibitor alpha; Oligodeoxyribonucleotides; Phosphorylation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-hck; Pyrazoles; Pyrimidines; Quinacrine; RNA, Small Interfering; src-Family Kinases; Syk Kinase; Toll-Like Receptor 9; Tyrosine; Wortmannin | 2006 |
THE INFLUENCE OF ORALLY ADMINISTERED ALKALI AND ACID ON THE RENAL EXCRETION OF QUINACRINE, CHLOROQUINE AND SANTOQUINE.
Topics: Alkalies; Chloroquine; Fluids and Secretions; Humans; Quinacrine; Renal Elimination | 1947 |
Comparison of chloroquine, quinacrine (atabrine) and quinine in the treatment of acute attacks of sporozoite-induced vivax malaria, Chesson strain.
Topics: Animals; Behavior, Animal; Chloroquine; Humans; Malaria, Vivax; Quinacrine; Quinine; Sporozoites | 1948 |
The efficacy of chloroquine, quinacrine, quinine and totaquine in the treatment of Plasmodium malariae infections (quartan malaria).
Topics: Chloroquine; Humans; Malaria; Plasmodium malariae; Quinacrine; Quinine | 1948 |
Effect of acidosis and anoxia on the concentration of quinacrine and chloroquine in blood.
Topics: Acidosis; Chloroquine; Hypoxia; Quinacrine | 1948 |
Chloroquine-induced autophagic vacuole accumulation and cell death in glioma cells is p53 independent.
Topics: Antineoplastic Agents; Autophagy; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Chloroquine; Glioma; Humans; Immunohistochemistry; Mefloquine; Quinacrine; Tumor Suppressor Protein p53; Vacuoles | 2010 |
Resistance to chloroquine unhinges vivax malaria therapeutics.
Topics: Aminoquinolines; Antimalarials; Chloroquine; Drug Interactions; Drug Resistance; Humans; Malaria, Vivax; Plasmodium vivax; Primaquine; Quinacrine | 2011 |
Mechanism of endosomal TLR inhibition by antimalarial drugs and imidazoquinolines.
Topics: Animals; Antimalarials; Binding, Competitive; Cell Line; Cells, Cultured; Chloroquine; Culture Media; Cytokines; Endosomes; HEK293 Cells; Humans; Hydrogen-Ion Concentration; Imidazoles; Nucleic Acids; Quinacrine; Quinolines; Serum; Toll-Like Receptor 3; Toll-Like Receptor 7; Toll-Like Receptor 8; Toll-Like Receptor 9; Toll-Like Receptors; Transfection | 2011 |
2,4-diarylthiazole antiprion compounds as a novel structural class of antimalarial leads.
Topics: Antimalarials; Chloroquine; Mefloquine; Molecular Structure; Plasmodium falciparum; Prions; Quinacrine; Structure-Activity Relationship; Thiazoles | 2011 |
N-cinnamoylation of antimalarial classics: quinacrine analogues with decreased toxicity and dual-stage activity.
Topics: Antimalarials; Cell Line; Chloroquine; Drug Design; Drug Resistance; Humans; Malaria; Plasmodium berghei; Plasmodium falciparum; Quinacrine | 2014 |
Suppressive action of mepacrine, aphacrine, chloroquin, camoquin and proguanil against P. knowlesi in S. rhesus monkeys.
Topics: Amodiaquine; Animals; Chloroquine; Humans; Macaca mulatta; Malaria; Proguanil; Quinacrine | 1950 |
Synthesis of improved lysomotropic autophagy inhibitors.
Topics: Antineoplastic Agents; Autophagy; Cell Line; Cell Survival; Chemistry Techniques, Synthetic; Chloroquine; Drug Evaluation, Preclinical; Humans; Lysosomes; Microtubule-Associated Proteins; Quinacrine; Structure-Activity Relationship | 2015 |
N-Cinnamoylation of Antimalarial Classics: Effects of Using Acyl Groups Other than Cinnamoyl toward Dual-Stage Antimalarials.
Topics: Antimalarials; Cell Survival; Chloroquine; Cinnamates; Hep G2 Cells; Humans; Life Cycle Stages; Plasmodium berghei; Plasmodium falciparum; Quinacrine; Structure-Activity Relationship | 2015 |
Unilateral unique Lupus tumidus: pathogenetic mystery and diagnostic problem.
Topics: Adrenal Cortex Hormones; Adult; Azathioprine; Biopsy; Chloroquine; Combined Modality Therapy; Dapsone; Diagnosis, Differential; Humans; Hydroxychloroquine; Lasers, Dye; Lupus Erythematosus, Discoid; Male; Ointments; Quinacrine; Skin; Sunscreening Agents; Tacrolimus | 2016 |
Chloroquine derivatives block the translocation pores and inhibit cellular entry of Clostridium botulinum C2 toxin and Bacillus anthracis lethal toxin.
Topics: Antigens, Bacterial; Bacterial Toxins; Biological Transport; Botulinum Toxins; Cell Membrane; Chloroquine; Fluphenazine; HeLa Cells; Humans; Lipid Bilayers; Primaquine; Quinacrine | 2017 |
Lysosomotropic cationic drugs induce cytostatic and cytotoxic effects: Role of liposolubility and autophagic flux and antagonism by cholesterol ablation.
Topics: Amiodarone; Anticholesteremic Agents; Autophagy; beta-Cyclodextrins; Cell Line, Tumor; Cell Proliferation; Cells, Cultured; Chloroquine; Cholesterol; Cytostatic Agents; Cytotoxins; Human Umbilical Vein Endothelial Cells; Humans; Hydroxychloroquine; Lidocaine; Lovastatin; Lysosomes; Microtubule-Associated Proteins; Poly (ADP-Ribose) Polymerase-1; Procainamide; Quinacrine | 2016 |
Is chloroquine neuromyotoxicity in a patient with refractory discoid lupus erythematosus potentiated by concomitant use of mepacrine?
Topics: Antimalarials; Chloroquine; Drug Therapy, Combination; Extremities; Female; Humans; Lupus Erythematosus, Discoid; Middle Aged; Muscle Weakness; Paresthesia; Quinacrine | 2018 |
Comparison of chloroquine-like molecules for lysosomal inhibition and measurement of autophagic flux in the brain.
Topics: Animals; Autophagy; Brain; Chloroquine; Drug Evaluation, Preclinical; Female; HeLa Cells; Humans; Lysosomes; Macrolides; Male; Mefloquine; Mice, Inbred C57BL; Mice, Transgenic; Microtubule-Associated Proteins; Promazine; Quinacrine; Trifluoperazine | 2021 |
Efficacy and Tolerability of Quinacrine Monotherapy and Albendazole Plus Chloroquine Combination Therapy in Nitroimidazole-Refractory Giardiasis: A TropNet Study.
Topics: Albendazole; Antiprotozoal Agents; Chloroquine; Giardia lamblia; Giardiasis; Humans; Nitroimidazoles; Prospective Studies; Quinacrine | 2021 |