chloroquine and quinacrine

chloroquine has been researched along with quinacrine in 337 studies

Research

Studies (337)

TimeframeStudies, this research(%)All Research%
pre-1990253 (75.07)18.7374
1990's26 (7.72)18.2507
2000's32 (9.50)29.6817
2010's21 (6.23)24.3611
2020's5 (1.48)2.80

Authors

AuthorsStudies
Denny, WA; Feigon, J; Kearns, DR; Leupin, W1
Chibale, K; Croft, SL; Fairlamb, AH; Haupt, H; Kendrick, H; Saravanamuthu, A; Yardley, V1
Elshorst, B; Fiebig, K; Griesinger, C; Grimme, S; Jacobs, DM; Vogtherr, M; Zahn, R1
Galanakis, D; Ganellin, CR1
Derisi, JL; Guy, RK; Liou, AP; Madrid, PB; Sherrill, J; Weisman, JL1
Bellocq, NC; Cheng, J; Davis, ME; Jensen, GS; Kulkarni, RP; Liu, A; Mishra, S; Pun, SH; Zeidan, R1
Harada, S; Huy, NT; Kamei, K; Maeda, A; Oida, T; Trang, DT; Uyen, DT1
Beauchene, J; Caffrey, CR; Cohen, FE; Debnath, A; Doyle, PS; Fafarman, AT; Fairlamb, AH; Kelly, B; Land, KM; May, BC; McKerrow, JH; Moll, H; Ponte-Sucre, A; Saravanamuthu, A; Schirmeister, T; Schreiber, K; Steverding, D; Swenerton, RK; Walshe, D; Weisman, JL; Zhou, YM; Zorn, JA1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Fitos, I; Mády, G; Visy, J; Zsila, F1
Acharya, BN; Kaushik, MP; Saraswat, D1
Lombardo, F; Obach, RS; Waters, NJ1
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Bolognesi, ML; Bongarzone, S; Brun, R; Cavalli, A; Lizzi, F; Luise Krauth-Siegel, R1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Glen, RC; Lowe, R; Mitchell, JB1
Baker, JR; Banaszak Holl, MM; Choi, SK; Harmon, A; Li, MH; Orr, BG; Plantinga, A; Sinniah, K; Witte, A1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Atzpodien, EA; Csato, M; Doessegger, L; Fischer, H; Lenz, B; Schmitt, G; Singer, T1
Almnayan, D; Lee, H; Solomon, VR1
Chen, Y; Feng, F; He, S; Jiang, X; Li, Q; Lu, X; Qu, W; Sun, H1
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P1
Bernatchez, JA; Li, J; Li, R; Luan, Y; Siqueira-Neto, JL; Tran, LT1
Byun, SY; Choi, I; Jeon, S; Kim, S; Ko, M; Lee, J; Park, S; Shum, D1
Kitagawa, T; Matsumoto, A; Terashima, I; Uesono, Y1
Lampen, JO; Traficante, LJ1
Rosenberg, LS; Schulman, SG1
Drenckhahn, D; Lüllmann-Rauch, R1
Blazsó, G; Kákár, T; Minker, E1
Cornelis, JJ; Hendrickx, B; Lakhanisky, T; Mouton, RF1
Frisch, W; Lüllmann-Rauch, R3
Calberg-Bacq, CM; Cannistraro, S; Piette, J; Van de Vorst, A1
Calberg-Bacq, CM; Piette, J; Van de Vorst, A1
Bychkov, MB1
Dubois, EL1
Davidson, MW; Jones, RL; Wilson, WD1
Matejka, Z; Minker, E2
Garfinkel, E; Hirschman, SZ1
Fossati, C1
Boykin, DW; Davidson, MW; Griggs, BG; Wilson, WD1
Mattock, NM; Peters, W1
Holbrook, DJ; Washington, ME; Wichard, LP1
Steigleder, GK1
Lot, TY3
Craig, JC; Kirby, GC; Shyamala, V; Warhurst, DC; Webster, RV1
Barr, R; Branstetter, BA; Crane, FL; Löw, H; Rajnicek, A1
Desbuquois, B; Dupuis, A; Janicot, M1
De Boeck, H; Maguire, PA; Sherman, IW; Zidovetzki, R1
Akera, T; Brody, TM; Ng, YC; Tona, L1
Kench, JG; Seale, JP; Temple, DM; Tennant, C1
Safa, AR; Spearman, T; Van Dyke, K; Ye, ZG1
Filippov, A; Kobrinsky, E; Porotikov, V; Saxon, M; Skatova, G1
Atiya, A; De Boeck, H; Sherman, IW; Zidovetzki, R1
Emerole, GO; Nashiru, TO; Thabrew, MI1
Lanciani, P1
Beck, WT; Cirtain, MC; Felsted, RL; Glover, CJ; Safa, AR1
Maroy, B1
Ha, SH; Shao, BR; Zhan, CQ1
Imamura, S; Miyachi, Y; Niwa, Y; Yoshioka, A1
Bell, AL; Betts, WH; Cleland, LG; French, JK; Hurst, NP; Nuki, G; O'Donnell, ML1
Chanthavanich, P; Edwards, G; Looareesuwan, S; Phillips, RE; Rodick, CL; Supanaranond, W; Warrell, DA1
Hauser, G; Jadali, F; Kiesel, L; Przylipiak, A; Rabe, T; Runnebaum, B1
Imamura, S; Miyachi, Y; Yoshioka, A1
Beck, WT; Pearce, HL; Zamora, JM1
Shao, BR; Xu, YQ1
Flayeh, KA1
Chander, A; Fisher, AB; Reicherter, J1
Komuniecki, PR; Whitten, JJ1
Au, AM; Chan, PH; Fishman, RA1
Ganster, HJ; Mehlhorn, H; Raether, W; Seidenath, H1
Creus, A; Marcos, R; Velázquez, A; Xamena, N1
Clark, SK1
Bohn, E; Hesse, B; Kunze, H; Löffler, BM1
Kern, HF; Pfab, R; Schachtschabel, DO1
Clark, JS; Jubb, SN; Maloney, PJ; Young, JM1
Holmes, J; Sapeika, N; Zwarenstein, H2
Chou, SC; Conklin, KA; Pan, HY1
Harinasuta, T; Suntharasamai, P; Viravan, C1
Chou, SC; Levy, MR1
Peters, W4
Boström, H; Whitehouse, MW1
Benex, J; Lamy, L1
Jarumilinta, R; Kradolfer, F; Sackmann, W1
Desmons, F; Gautier, G; Huriez, C1
Lie, SO; Schofield, B1
Cowey, FK; Whitehouse, MW1
Most, H1
Fain, JN; Pointer, RH1
Staiger, GR1
Hadwiger, LA1
Miller, A; Natsios, G; Smith, HC1
Abdel-Aziz, A; Idris, IB; Karrar, MA1
Brown, RK1
Olatunde, IA1
Allison, RG; Hahn, FE; Wolfe, AD1
Briesch, PE; Contacos, PG; Glew, RH; Krotoski, WA; Neva, FA1
Botha, D1
Chou, SC; Conklin, KA2
Gaudin, D; Gregg, RS; Yielding, KL1
Prasad, BN1
Sinohara, H1
Thomas, SC; Warhurst, DC1
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS1
Gärding, S; Gösta Henriksson, K; Larsson, JE1
Dawkins, AT; Stahler, N; Terzian, LA1
Modell, W1
Hunsicker, LG1
Lantz, CH; Saxe, LH; Szustkiewicz, C; Van Dyke, K1
Schmidt, LH1
Meier-Ruge, W1
Hall, SA1
Ciak, J; Hahn, FE1
Gorlin, RJ1
Cook, TM; Hahn, FE; Wolfe, AD1
Myint, UH; Win, UK1
Auckland, NL1
Brede, HD; de Klerk, JN; Groenewald, JH; Murphy, GP; Retief, CP; Schoonees, R; van Heerden, PD; van Zyl, JA; van Zyl, JJ; Weber, HW1
Brede, HD; de Klerk, JN; Groenewald, JH; Retief, CP; Schoonees, R; van Heerden, PD; van Zyl, JA; van Zyl, JJ; Weber, HW1
Brede, HD1
Barnes, MG; Polet, H1
Barr, CF; Polet, H1
Fink, E; Kretschmar, W1
Chou, SC; Conklin, KA; Heu, P1
Bruce-Chwatt, LJ2
Lantz, CH; Van Dyke, K1
Kochen, J; Roth, EF1
Brynolf, I1
Hahn, FE; O'Brien, RL; Olenick, JG1
Ball, EG; Markus, HB1
Cabanel, G; Chouteau, J; Marchal, A; Voog, R1
Cenedella, RJ; Saxe, LH; Van Dyke, K1
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K1
Polet, H1
Gregory, KG; Peters, W1
Nieper, HA1
Bishop, A1
Bengtsson, E1
Buchnícek, J; Turek, B1
Cheng, CC; Chien, PL1
Rockwell, DA1
Dodge, BG; Freeman, RG; Knox, JM1
Clancy, CF1
Schneider, MD1
Carr, RE; Henkind, P; Rothfield, N; Siegel, IM1
Ott, KJ1
Crim, JA; Gray, GD; Zeleznick, LD1
Hahn, FE; Macomber, PB; O'Brien, RL1
Banerjee, AK; Chowdhury, DS1
Hermann, P; Lefranc, E; Sourdille, P1
Mattila, M; Takki, S1
Reba, RC; Sheehy, TW1
Trager, W1
Purcell, WP; Singer, JA1
Famaey, JP; Fontaine, J; Ouedraogo, CO; Reuse, J1
Wolfe, MS1
Authi, KS; Traynor, JR1
Di Cerbo, A; Edelhoch, H; Nandi, PK1
Koranda, FC1
Trist, DG; Weatherall, M1
Doberstyn, EB1
Ferrante, A; Goh, DH1
Dubin, NH; Ghodgaonkar, RB; King, TM; Parmley, TH1
Harris, EJ; Jackson, MJ; Jones, DA1
Ioannides, C; Thabrew, MI1
Drenckhahn, D; Jacobi, B; Lüllmann-Rauch, R1
Hughes, GR; Lanham, JG1
Gould, S; Warhurst, DC1
Elgart, M; Isaacson, D; Turner, ML1
Ma, K; Sourkes, TL1
Berstein, GS; Trifunac, NP1
Kuye, JO; Walle, T; Wilson, MJ1
Izumi, F; Kobayashi, H; Sakurai, S; Wada, A; Yanagihara, N1
Tanenbaum, L; Tuffanelli, DL1
Andersson, A; Olsson, S; Tjälve, H1
Govitrapong, P; Jearnpipatkul, A; Panijpan, B; Wilairat, P; Yuthavong, Y1
Catt, KJ; Naor, Z1
Olansky, AJ1
Crescenzi, V; Delben, F; Giancotti, V; Quadrifoglio, F1
Biller, H; Hess, F; Leising, HB; Pfab, R; Schachtschabel, DO2
Bohn, E; Hesse, B; Kunze, H1
Bennett, T; Lot, TY1
Jones, RL; Keel, RA; Lanier, AC; Wilson, WD1
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B1
Brady, RO; Kusiak, JW; Quirk, JM1
Kádár, T; Matejka, Z; Minker, E1
Hodgson, LL; Morgan, EH; Quail, EA1
Cacoub, P; Frances, C; Godeau, P; Lipsker, D; Piette, JC1
Feldmann, R; Salomon, D; Saurat, JH1
Enomoto, K; Maeno, T1
Dutta, P; Karmali, R; Pinto, JT; Rivlin, RS1
Wallace, DJ1
Craig, JC; Scaria, PV; Shafer, RH1
Marcil, J; Ravindranath, N; Sairam, MR1
Lüllmann-Rauch, R; Pods, R; von Witzendorff, B1
Chen, SS; Jiang, MC; Lin, JK1
Croft, SL; Elueze, EI; Warhurst, DC1
Bächinger, HP; Hinrichs, DJ; Ignatushchenko, MV; Riscoe, MK; Winter, RW1
Dabancens, AO; Guerrero, AC; Zipper, JA1
Rynes, RI1
Horio, S; Ishida, Y; Moritoki, H; Nagare, T1
Loegering, DJ; Raley, MJ; Schwacha, MG1
Macfarlane, DE; Manzel, L2
Bondeson, J; Sundler, R1
Lehmann, P; Rönnau, AC; Ruzicka, T; Schuppe, HC; Specker, C; von Schmiedeberg, S1
Griffin, GE; Harrison, TS; Levitz, SM1
Cheng, SH; Przybylska, M; Song, A; Tousignant, JD; Wu, IH; Yew, NS; Zhao, H1
Vdovenko, AA; Williams, JE1
Piette, WW; Van Beek, MJ1
Rembao, D; Reyes, S; Sotelo, J1
Jjemba, PK1
ANSARI, AR; BRUMPT, LC; MAISON, E1
ROSENBAUM, S1
PASTOR BOTIJA, F1
BASU, PC; RAY, AP1
GONDARD, L1
DRIVER, IE; FARBER, EM1
KNOX, JM; LAMB, JH; MORGAN, RJ; SHELMIRE, B1
CAHN, MM; LEVY, EJ; SHAFFER, B2
FINN, OA; ROGERS, J1
CERTONCINY, A; FORESTIER, J1
VILANOVA, X1
BAYES, C; ESCARPENTER-ORIOL, J; GOMEZ, MS1
CHAMNARNKIT, C; CHETANASEN, S; SADUN, EH1
BORODA, C1
BRODTHAGEN, H1
BIGUET, J; BRETON, A; COUTELEN, F; DEBLOCK, S; DOBY, JM; MULLET, S1
CARRERAS BAYES, A; ESCARPENTER ORIOL, J; SARIOLS GOMEZ, M1
MARCHIONINI, A; THIES, W1
AZIMI-HAMID, A; TRONNIER, H1
CONNER, SK1
LANGLO, L1
CHRISTIANSEN, JV2
FLEISCHMAJER, R; REIN, CR1
ENGESET, A2
ANSELL, HB; APPEL, B; SCHIFF, B; TYE, MJ; WOLF, M1
FERNANDEZ NAFRIA, A1
KOCH, H; WISKEMANN, A1
VIDMAR-CVJETANOVIC, B1
ERLENDSSON, F1
ROBINSON, RC; SMITH, GC1
ANSELL, HB; APPEL, B; TYE, MJ; WHITE, H1
BROWNING, M; JONES, R; JONSSON, U; LESSNER, H; PRICE, CC; SEN, AK1
MARCIANO, MR; SHEARD, C1
HOJMAN, N; QUIROGA, FE; VAZQUEZ, HJ1
ABD-EL-GHAFFAR, V1
GROUNDS, JG1
GREWAL, RS; SHARMA, ML1
BEHRENDT, WA; URBAN, G1
BOCK, W; DOERDELMANN, P1
KURNICK, NB; RADCLIFFE, IE1
LEOVEY, A; NAGY, E1
FREDRIKSSON, T; LODIN, A; ROSENGREN, S1
SASLAW, S; SCHAEFER, J1
BONTOUX, D; GODEAU, P; LEVY, R; SIGUIER, F1
AMMA, MK; GUJRAL, ML; MISRA, N; SAREEN, K; VARMA, DR; VIJAYAMMA, N1
DARNET, C; LEBEURRE, R; VERHAEGHE, A1
EPSTEIN, JH; VANDENBERG, JJ; WRIGHT, WL1
KLINGMUELLER, G1
CONTACOS, PG; MILLAR, JW; STITCHER, JE; YOUNG, MD1
ABRAHAM, RK; DUBOIS, EI; TUFFANELLI, D1
HASERICK, JR1
ARORA, RB; LAL, A1
COATNEY, GR; CONTACOS, PG; LUNN, JS1
SAPP, OL1
BORC, K1
BOUMA, HG; DEVRIES, K; JANSZ, A; NIEWEG, HO1
RAAB, W1
SULLI, G; VARRONE, F1
BRACKEN, EC1
BOTTIROLI, JA; ROSENBERG, FJ1
ALVING, AS; BREWER, GJ; MILLAR, JW; POWELL, RD1
EYLES, DE; MONTGOMERY, R; SANDOSHAM, AA1
MATTILA, M1
DASHPUTRA, PG; DESHPANDE, VR; SHARMA, ML1
HELLERSTROEM, S1
FORBES, LS1
BRUCHACOVA, V; KRAJCI LAZARYOVA, M; NOVAK, A1
BETTLEY, FR1
MITCHELL, CL1
NEAL, RA1
HALSTEAD, SB; SADUN, EH1
CHANG, KC; CHIEN, TS; MENG, HY1
HERRMANN, WP; SCHULZ, KH1
STOUGHTON, RB1
THIES, W1
BRANDAO, N; DA FONSECA, A1
BALOGH, EE; NAGY, E1
REINERTSON, JW; THOMPSON, PE1
Bernhardt, I; Lang, HJ; Weiss, E1
Haystead, TA; Kwiek, JJ; Rudolph, J1
Bauer, S; Gellert, T; Lipford, GB; Luppa, P; Metzger, J; Rutz, M; Wagner, H1
Emerson, LR; Kuchler, K; Skillman, BC; Wirth, DF; Wolfger, H1
Forgac, M; Shao, E1
HANDFIELD-JONES, RP1
Tutor-Ureta, P; Yebra-Bango, M1
Benz, R; Orlik, F; Schiffler, B1
Pollaschek, C; Stuhlmeier, KM1
Colonna, M; Fuchs, A; Fung-Leung, WP; Gu, Y; Karlsson, L; Lai, KT; Rao, N; Sanjuan, MA; Sun, S1
Jailer, JW; Rosenfeld, M; Shannon, JA1
Boratyński, J; Lipka, D1
CRAIGE, B; PULLMAN, TN1
EYLES, DE; YOUNG, MD1
JAILER, JW; ZUBROD, CG1
Geng, Y; Klocke, BJ; Kohli, L; Roth, KA1
Baird, JK1
Bencina, M; Jerala, R; Jeras, M; Kuznik, A; Rozman, B; Svajger, U1
Chen, B; Coldham, I; Little, SM; Louth, JC; Thompson, MJ1
Albuquerque, I; Gomes, A; Gomes, P; Machado, M; Nogueira, F; Pérez, B; Prudêncio, M; Teixeira, C1
NAIR, CP; RAY, AP1
Gately, S; Gonzales, P; Goodall, ML; MacKeigan, JP; Martin, KR; Sepulveda, M; Wang, T1
Gomes, A; Gomes, P; Lobo, L; Machado, M; Nogueira, F; Prudêncio, M; Teixeira, C1
Bakardzhiev, I; Chokoeva, AA; Krasnaliev, I; Lotti, T; Tana, C; Tchernev, G; Wollina, U1
Barth, H; Benz, R; Kreidler, AM1
Marceau, F; Parks, A1
Carter, ER; Chiodini, PL; Hedley, L; Nabarro, LE1
Meggitt, SJ; Miller, JAL; Winn, RT1
Bensalem, J; Bryksin, V; Fourrier, C; Hattersley, K; Hein, LK; Sargeant, TJ1
Bottieau, E; Hatz, C; Kuenzli, E; Mechain, M; Mørch, K; Neumayr, A; Rothe, C; Schunk, M; Soriano Pérez, MJ; Sothmann, P; Sydow, V; Theunissen, C; Van Esbroeck, M1

Reviews

27 review(s) available for chloroquine and quinacrine

ArticleYear
Design of Small Molecule Autophagy Modulators: A Promising Druggable Strategy.
    Journal of medicinal chemistry, 2018, 06-14, Volume: 61, Issue:11

    Topics: Animals; Autophagy; Drug Design; Humans; Small Molecule Libraries

2018
Drugs for the Treatment of Zika Virus Infection.
    Journal of medicinal chemistry, 2020, 01-23, Volume: 63, Issue:2

    Topics: Animals; Antiviral Agents; Drug Development; Drug Discovery; Humans; Viral Vaccines; Zika Virus; Zika Virus Infection

2020
Antimalarials in the management of discoid and systemic lupus erythematosus.
    Seminars in arthritis and rheumatism, 1978, Volume: 8, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Pigmentation Disorders; Quinacrine; Retinal Diseases; Vision Disorders

1978
[Treatment of intestinal parasitosis].
    La Clinica terapeutica, 1975, Oct-15, Volume: 75, Issue:1

    Topics: Amphotericin B; Anthelmintics; Bithionol; Cestode Infections; Chloroquine; Humans; Intestinal Diseases, Parasitic; Leishmaniasis; Malaria; Metronidazole; Nematode Infections; Quinacrine; Tetracycline; Thiabendazole

1975
Recent advances in antimalarial chemotherapy and drug resistance.
    Advances in parasitology, 1974, Volume: 12

    Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones

1974
Drug therapy. Treatment of common parasitic infections of man encountered in the United States. 2.
    The New England journal of medicine, 1972, Oct-05, Volume: 287, Issue:14

    Topics: Amebiasis; Amebicides; Anthelmintics; Antimalarials; Antimony; Benzenesulfonates; Chloroquine; Clonorchiasis; Clonorchis sinensis; Dysentery, Amebic; Giardiasis; Humans; Iodoquinol; Liver Abscess, Amebic; Malaria; Metronidazole; Niridazole; Protozoan Infections; Quinacrine; Schistosoma haematobium; Schistosoma mansoni; Schistosomiasis; Tartrates; Trematode Infections

1972
The present status of chloroquine in the drug treatment of malaria.
    The African journal of medical sciences, 1972, Volume: 3, Issue:1

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines

1972
Summary of recent abstracts. 3. Malaria. 2.
    Tropical diseases bulletin, 1972, Volume: 69, Issue:4

    Topics: Animals; Antimalarials; Birds; Chloroquine; Dapsone; Humans; India; Malaria; Malaria, Avian; Mammals; Naphthoquinones; Oxytetracycline; Plasmodium; Plasmodium falciparum; Quinacrine; Rats; Reptiles

1972
The pharmacology of the antimalarials. A rational approach to the therapy of resistant falciparum malaria.
    Archives of internal medicine, 1969, Volume: 123, Issue:6

    Topics: Amodiaquine; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Sulfadimethoxine; Sulfisoxazole

1969
Chemotherapy of the drug-resistant malarias.
    Annual review of microbiology, 1969, Volume: 23

    Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones

1969
Drug induced retinopathy.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1969, Volume: 158 Suppl

    Topics: Adsorption; Animals; Antineoplastic Agents; Chloroquine; Drug-Related Side Effects and Adverse Reactions; Eye Diseases; Humans; Pharmaceutical Preparations; Phenothiazines; Quinacrine; Quinolines; Retina; Retinal Pigments

1969
Malaria treatment and prevention. A review.
    East African medical journal, 1969, Volume: 46, Issue:10

    Topics: Adolescent; Adult; Africa, Eastern; Antimalarials; Biguanides; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Humans; Infant; Infant Mortality; Infant, Newborn; Malaria; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Quinacrine; Quinine; Quinolines; Sulfonamides

1969
Epidermolysis bullosa.
    Oral surgery, oral medicine, and oral pathology, 1971, Volume: 32, Issue:5

    Topics: Adrenal Cortex Hormones; Chloroquine; Epidermolysis Bullosa; Humans; Oral Manifestations; Quinacrine; Silver Nitrate; Skin Manifestations; Vitamins

1971
The treatment of intestinal protozoan infections.
    The Medical clinics of North America, 1982, Volume: 66, Issue:3

    Topics: Amebicides; Antimalarials; Antiprotozoal Agents; Balantidiasis; Chloroquine; Coccidiosis; Dientamoebiasis; Drug Combinations; Dysentery, Amebic; Emetine; Furans; Furazolidone; Giardiasis; Humans; Intestinal Diseases, Parasitic; Iodoquinol; Liver Abscess, Amebic; Metronidazole; Paromomycin; Quinacrine; Sulfamethoxazole; Tetracycline; Tinidazole; Trimethoprim; Trimethoprim, Sulfamethoxazole Drug Combination

1982
Antimalarials.
    Journal of the American Academy of Dermatology, 1981, Volume: 4, Issue:6

    Topics: Antimalarials; Chloroquine; DNA; Eye Diseases; Humans; Hydroxychloroquine; Quinacrine; RNA; Skin Diseases

1981
Resistance of Plasmodium falciparum.
    Experientia, 1984, Dec-15, Volume: 40, Issue:12

    Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America

1984
Antimalarial therapy in SLE.
    Clinics in rheumatic diseases, 1982, Volume: 8, Issue:1

    Topics: Antimalarials; Binding Sites; Chloroquine; Corneal Diseases; Dose-Response Relationship, Drug; Female; Humans; Hydroxychloroquine; Immune Tolerance; Inflammation; Kinetics; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Nucleoproteins; Photosensitivity Disorders; Pregnancy; Quinacrine; Retinal Diseases; Retinal Pigments; Skin Diseases; Virus Replication

1982
Anti-malarials in dermatology.
    International journal of dermatology, 1982, Volume: 21, Issue:7

    Topics: Absorption; Amodiaquine; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Female; Humans; Hydroxychloroquine; Quinacrine; Skin Diseases

1982
Antimalarial agents. Chloroquine, hydroxychloroquine, and quinacrine.
    Archives of dermatology, 1980, Volume: 116, Issue:5

    Topics: Abnormalities, Drug-Induced; Anti-Inflammatory Agents; Chloroquine; DNA; Eye Diseases; Female; Hematologic Diseases; Humans; Hydroxychloroquine; Immunosuppressive Agents; Male; Melanins; Neuromuscular Diseases; Porphyrias; Pregnancy; Quinacrine; Skin; Sunscreening Agents

1980
Antimalarials and ophthalmologic safety.
    Journal of the American Academy of Dermatology, 1982, Volume: 6, Issue:1

    Topics: Antimalarials; Arthritis, Rheumatoid; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Retinal Diseases

1982
Antimalarial agents and lupus.
    Rheumatic diseases clinics of North America, 1994, Volume: 20, Issue:1

    Topics: Antibodies, Antiphospholipid; Antimalarials; Chloroquine; Female; Humans; Hydroxychloroquine; Kidney Diseases; Lupus Erythematosus, Systemic; Neuromuscular Diseases; Pregnancy; Quinacrine

1994
Antimalarial drugs in the treatment of rheumatological diseases.
    British journal of rheumatology, 1997, Volume: 36, Issue:7

    Topics: Antimalarials; Chloroquine; Contraindications; Female; Humans; Hydroxychloroquine; Male; Pregnancy; Pregnancy Complications; Quinacrine; Rheumatic Diseases; Skin

1997
Antimalarials.
    Dermatologic clinics, 2001, Volume: 19, Issue:1

    Topics: Antimalarials; Chloroquine; Dermatologic Agents; Humans; Quinacrine; Skin Diseases

2001
[ANTIMALARIALS IN THE TREATMENT OF SKIN DISEASES].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 1963, Volume: 14

    Topics: Adrenal Cortex Hormones; Antimalarials; Chloroquine; Dermatology; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases

1963
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
    La Clinica terapeutica, 1963, Oct-31, Volume: 27

    Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus

1963
[Metalloproteinases. Structure and function].
    Postepy higieny i medycyny doswiadczalnej (Online), 2008, Jul-03, Volume: 62

    Topics: 4-Aminobenzoic Acid; Animals; Apoptosis; Arthritis; Autoimmune Diseases; Cell Movement; Chloroquine; Drug Combinations; Enzyme Activation; Extracellular Matrix; Humans; Matrix Metalloproteinase Inhibitors; Matrix Metalloproteinases; Membrane Proteins; Models, Molecular; Neoplasms; Neovascularization, Physiologic; Pantothenic Acid; Pyridoxine; Quinacrine; Tissue Inhibitor of Metalloproteinases

2008
Nitroimidazole-refractory giardiasis: a growing problem requiring rational solutions.
    Clinical microbiology and infection : the official publication of the European Society of Clinical Microbiology and Infectious Diseases, 2018, Volume: 24, Issue:1

    Topics: Albendazole; Antiprotozoal Agents; Chloroquine; Drug Resistance; Drug Therapy, Combination; Giardia lamblia; Giardiasis; Humans; Metronidazole; Quinacrine; Tinidazole; Treatment Failure

2018

Trials

5 trial(s) available for chloroquine and quinacrine

ArticleYear
[Delagil treatment of tumorous pleurisy].
    Voprosy onkologii, 1978, Volume: 24, Issue:2

    Topics: Chloroquine; Clinical Trials as Topic; Drug Evaluation; Humans; Injections; Pleura; Pleural Neoplasms; Pleurisy; Quinacrine

1978
The influence of ovarian hormones and of pregnancy on the action of some antimalarials on the isolated spontaneously contracting rat uterus.
    European journal of pharmacology, 1971, Volume: 16, Issue:2

    Topics: Antimalarials; Chloroquine; Clinical Trials as Topic; Drug Interactions; Estradiol; Female; Histamine H1 Antagonists; Hormones; Humans; Ovary; Progesterone; Proguanil; Quinacrine; Quinine; Uterus

1971
Renal allotransplantation in the baboon with chemical immunosuppression.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1968, Aug-17

    Topics: Animals; Azathioprine; Blood Cells; Blood Chemical Analysis; Blood Protein Electrophoresis; Chloroquine; Clinical Trials as Topic; Cyclophosphamide; Enzymes; Female; Glomerular Filtration Rate; Haplorhini; Hydrocortisone; Immunosuppressive Agents; Kidney Function Tests; Kidney Transplantation; Male; Quinacrine; Thalidomide; Transplantation, Homologous

1968
The effect of chemical immunosuppression in baboon allotransplantation: histopathological observations.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1968, Aug-17

    Topics: Animals; Azathioprine; Chloroquine; Clinical Trials as Topic; Cyclophosphamide; Haplorhini; Hydrocortisone; Immunosuppressive Agents; Kidney; Kidney Transplantation; Quinacrine; Renal Artery; Renal Veins; Thalidomide; Transplantation, Homologous

1968
The effect of chemical immunosuppression in baboon allotransplantation: serological observations.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1968, Aug-17

    Topics: Animals; Antibodies; Azathioprine; C-Reactive Protein; Chloroquine; Clinical Trials as Topic; Complement System Proteins; Cyclophosphamide; Haplorhini; Hemolysin Proteins; Humans; Hydrocortisone; Immunosuppressive Agents; Kidney Transplantation; Quinacrine; Rheumatoid Factor; Thalidomide; Transplantation, Homologous

1968

Other Studies

305 other study(ies) available for chloroquine and quinacrine

ArticleYear
Interactions of antitumor drugs with natural DNA: 1H NMR study of binding mode and kinetics.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Antineoplastic Agents; Base Composition; Chemical Phenomena; Chemistry; DNA; Hydrogen Bonding; Intercalating Agents; Kinetics; Magnetic Resonance Spectroscopy; Structure-Activity Relationship

1984
Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine.
    Bioorganic & medicinal chemistry letters, 2001, Oct-08, Volume: 11, Issue:19

    Topics: Animals; Antiprotozoal Agents; Leishmania; Parasitic Sensitivity Tests; Plasmodium; Quinacrine; Sulfonamides; Trypanosoma; Urea

2001
Antimalarial drug quinacrine binds to C-terminal helix of cellular prion protein.
    Journal of medicinal chemistry, 2003, Aug-14, Volume: 46, Issue:17

    Topics: Antimalarials; Binding Sites; Chloroquine; Humans; Magnetic Resonance Spectroscopy; Models, Molecular; Peptide Fragments; Phenothiazines; Prions; Protein Structure, Secondary; Quinacrine; Recombinant Proteins; Structure-Activity Relationship

2003
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
    Bioorganic & medicinal chemistry letters, 2004, Aug-02, Volume: 14, Issue:15

    Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated

2004
Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
    Bioorganic & medicinal chemistry letters, 2005, Feb-15, Volume: 15, Issue:4

    Topics: Aminoquinolines; Animals; Antimalarials; Chloroquine; Drug Resistance; Plasmodium falciparum; Structure-Activity Relationship

2005
Structure-function correlation of chloroquine and analogues as transgene expression enhancers in nonviral gene delivery.
    Journal of medicinal chemistry, 2006, Nov-02, Volume: 49, Issue:22

    Topics: Cell Line, Tumor; Chloroquine; Cyclodextrins; DNA; Drug Screening Assays, Antitumor; Electrophoretic Mobility Shift Assay; Gene Expression; Gene Transfer Techniques; HeLa Cells; Humans; Luciferases; Structure-Activity Relationship; Transgenes

2006
Simple colorimetric inhibition assay of heme crystallization for high-throughput screening of antimalarial compounds.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:1

    Topics: Animals; Antimalarials; Colorimetry; Crystallization; Drug Evaluation, Preclinical; Heme; Hemeproteins; Plasmodium falciparum; Polysorbates; Reproducibility of Results

2007
Bis-acridines as lead antiparasitic agents: structure-activity analysis of a discrete compound library in vitro.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:6

    Topics: Acridines; Animals; Antiparasitic Agents; Combinatorial Chemistry Techniques; Eukaryota; HL-60 Cells; Humans; Parasitic Sensitivity Tests; Plasmodium falciparum; Polyamines; Schistosoma mansoni; Structure-Activity Relationship; Trypanosoma brucei brucei

2007
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Selective plasma protein binding of antimalarial drugs to alpha1-acid glycoprotein.
    Bioorganic & medicinal chemistry, 2008, Apr-01, Volume: 16, Issue:7

    Topics: Antimalarials; Binding Sites; Chromatography, Affinity; Circular Dichroism; Humans; Molecular Structure; Orosomucoid; Protein Binding; Serum Albumin; Spectrophotometry; Stereoisomerism; Structure-Activity Relationship

2008
Pharmacophore based discovery of potential antimalarial agent targeting haem detoxification pathway.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:12

    Topics: Animals; Antimalarials; Drug Discovery; Heme; Isoniazid; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Small Molecule Libraries; Stereoisomerism

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Privileged structure-guided synthesis of quinazoline derivatives as inhibitors of trypanothione reductase.
    Bioorganic & medicinal chemistry letters, 2009, Jun-01, Volume: 19, Issue:11

    Topics: Animals; Antiparasitic Agents; Cell Line; Computer Simulation; Drug Design; Enzyme Inhibitors; Glutathione Reductase; Humans; NADH, NADPH Oxidoreductases; Quinazolines; Rats; Structure-Activity Relationship; Trypanosoma cruzi

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Predicting phospholipidosis using machine learning.
    Molecular pharmaceutics, 2010, Oct-04, Volume: 7, Issue:5

    Topics: Animals; Artificial Intelligence; Databases, Factual; Drug Discovery; Humans; Lipidoses; Models, Biological; Phospholipids; Support Vector Machine

2010
Bioanalytical Screening of Riboflavin Antagonists for Targeted Drug Delivery - A Thermodynamic and Kinetic Study.
    ACS medicinal chemistry letters, 2011, May-12, Volume: 2, Issue:5

    Topics:

2011
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
In silico assay for assessing phospholipidosis potential of small druglike molecules: training, validation, and refinement using several data sets.
    Journal of medicinal chemistry, 2012, Jan-12, Volume: 55, Issue:1

    Topics: Animals; Cattle; Cells, Cultured; Computer Simulation; Cornea; Drug-Related Side Effects and Adverse Reactions; Fibroblasts; Lipidoses; Lysosomal Storage Diseases; Models, Molecular; Pharmaceutical Preparations; Phospholipids; Structure-Activity Relationship; Thermodynamics

2012
Design, synthesis and characterization of novel quinacrine analogs that preferentially kill cancer over non-cancer cells through the down-regulation of Bcl-2 and up-regulation of Bax and Bad.
    European journal of medicinal chemistry, 2017, Sep-08, Volume: 137

    Topics: Antineoplastic Agents; bcl-2-Associated X Protein; bcl-Associated Death Protein; Cell Death; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Down-Regulation; Drug Design; Drug Screening Assays, Antitumor; Humans; Molecular Structure; Proto-Oncogene Proteins c-bcl-2; Quinacrine; Structure-Activity Relationship; Up-Regulation

2017
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
    Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7

    Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship

2019
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.
    Antimicrobial agents and chemotherapy, 2020, 06-23, Volume: 64, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; Antiviral Agents; Betacoronavirus; Cell Line; Chlorocebus aethiops; Coronavirus Infections; COVID-19; Drug Evaluation, Preclinical; Drug Repositioning; Humans; Niclosamide; Pandemics; Pneumonia, Viral; Pregnenediones; SARS-CoV-2; Vero Cells

2020
Antimalarial Quinacrine and Chloroquine Lose Their Activity by Decreasing Cationic Amphiphilic Structure with a Slight Decrease in pH.
    Journal of medicinal chemistry, 2021, 04-08, Volume: 64, Issue:7

    Topics: Antifungal Agents; Cell Membrane; Chloroquine; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Molecular Structure; Monosaccharide Transport Proteins; Protons; Quinacrine; Saccharomyces cerevisiae; Surface-Active Agents

2021
Vesicle penicillinase of Bacillus licheniformis: existence of periplasmic-releasing factor(s).
    Journal of bacteriology, 1977, Volume: 129, Issue:1

    Topics: Bacillus; Chloroquine; Chromatography, Gel; Deoxycholic Acid; Hydrogen-Ion Concentration; Molecular Weight; Organoids; Penicillinase; Phenanthrolines; Phosphates; Protoplasts; Quinacrine

1977
Tautomerism of singly protonated chloroquine and quinacrine.
    Journal of pharmaceutical sciences, 1978, Volume: 67, Issue:12

    Topics: Chloroquine; Hydrogen-Ion Concentration; Kinetics; Quinacrine; Spectrophotometry; Spectrophotometry, Ultraviolet; Stereoisomerism

1978
Experimental myopathy induced by amphiphilic cationic compounds including several psychotropic drugs.
    Neuroscience, 1979, Volume: 4, Issue:4

    Topics: Amitriptyline; Animals; Chloroquine; Chlorphentermine; Chlorpromazine; Female; Imipramine; Iprindole; Male; Microscopy, Electron; Muscles; Muscular Diseases; Phentermine; Piperazines; Psychotropic Drugs; Quinacrine; Rats; Triparanol

1979
Inhibitory effect on gastric motility of chloroquine and mepacrine.
    Acta physiologica Academiae Scientiarum Hungaricae, 1978, Volume: 52, Issue:4

    Topics: Animals; Chloroquine; Depression, Chemical; Dose-Response Relationship, Drug; Female; Ganglionic Blockers; Gastrointestinal Motility; In Vitro Techniques; Parasympatholytics; Quinacrine; Rats; Sympathetic Nervous System; Sympatholytics

1978
A serological study of removal of UV-induced photoproducts in the DNA of Tetrahymena pyriformis GL: influence of caffeine, quinacrine and chloroquine.
    Photochemistry and photobiology, 1979, Volume: 29, Issue:4

    Topics: Animals; Caffeine; Chloroquine; DNA; DNA Repair; Immunologic Techniques; Photochemistry; Quinacrine; Tetrahymena pyriformis; Ultraviolet Rays

1979
Differential effects of chloroquine and of several other amphiphilic cationic drugs upon rat choroid plexus.
    Acta neuropathologica, 1979, May-15, Volume: 46, Issue:3

    Topics: Amitriptyline; Animals; Chloroquine; Chlorphentermine; Choroid Plexus; Clomipramine; Female; Hexestrol; Inclusion Bodies; Iprindole; Male; Microscopy, Electron; Quinacrine; Rats

1979
Photodynamic activity of dyes with different DNA binding properties I. free-radical induction in DNA.
    International journal of radiation biology and related studies in physics, chemistry, and medicine, 1978, Volume: 34, Issue:3

    Topics: Acridines; Binding Sites; Chloroquine; Coloring Agents; DNA; Ethidium; Free Radicals; Light; Proflavine; Pyronine; Quinacrine; Thioxanthenes

1978
Photodynamic activity of dyes with different DNA binding properties II. T4 phage inactivation.
    International journal of radiation biology and related studies in physics, chemistry, and medicine, 1978, Volume: 34, Issue:3

    Topics: Acridines; Binding Sites; Chloroquine; Coliphages; Coloring Agents; DNA, Viral; Ethidium; Light; Proflavine; Pyronine; Quinacrine; Thioxanthenes

1978
Comparative viscometric analysis of the interaction of chloroquine and quinacrine with superhelical and sonicated DNA.
    Biochimica et biophysica acta, 1979, Jan-26, Volume: 561, Issue:1

    Topics: Bacteriocin Plasmids; Chloroquine; DNA, Superhelical; Nucleic Acid Conformation; Quinacrine; Sonication; Viscosity

1979
Effect of mepacrine on gastric motility in the rat.
    Acta physiologica Academiae Scientiarum Hungaricae, 1979, Volume: 53, Issue:3

    Topics: Administration, Oral; Animals; Bencyclane; Chloroquine; Female; Gastric Emptying; Gastric Mucosa; Gastrointestinal Motility; Injections, Intraperitoneal; Papaverine; Quinacrine; Rats

1979
Inhibition of hepatitis B DNA polymerase by intercalating agents.
    Nature, 1978, Feb-16, Volume: 271, Issue:5646

    Topics: Chloroquine; Chlorpromazine; Drug Synergism; Ethidium; Hepatitis B; Hepatitis B virus; Humans; Indicators and Reagents; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine

1978
Molecular structural effects involved in the interaction of quinolinemethanolamines with DNA. Implications for antimalarial action.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:9

    Topics: Amino Alcohols; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; DNA; Drug Interactions; Piperidines; Quinacrine; Quinine; Quinolines

1977
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
    Annals of tropical medicine and parasitology, 1975, Volume: 69, Issue:3

    Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin

1975
Effect of nucleic-acid-binding compounds on the hydrolytic activity of various ribonucleases.
    European journal of biochemistry, 1975, Dec-15, Volume: 60, Issue:2

    Topics: Acridines; Aminoquinolines; Animals; Binding Sites; Cattle; Chloroquine; Ethidium; Kinetics; Pancreas; Primaquine; Proflavine; Protein Binding; Quinacrine; Ribonucleases; Spermidine; Spermine; Structure-Activity Relationship

1975
[Plaque-like form of cutaneous mucinosis (PGM) and reticular erythematous mucinosis (REM syndrome)].
    Zeitschrift fur Hautkrankheiten, 1975, Jan-01, Volume: 50, Issue:1

    Topics: Adult; Antimalarials; Chloroquine; Female; Humans; Methapyrilene; Quinacrine; Skin Diseases

1975
Smooth muscle sensitization and neuromuscular depression induced by chronic administration of antimalarial drugs.
    Physiology & behavior, 1992, Volume: 51, Issue:5

    Topics: Acetylcholine; Animals; Chickens; Chloroquine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Male; Muscle Contraction; Muscle, Smooth; Muscles; Neuromuscular Junction; Norepinephrine; Potassium Chloride; Quinacrine

1992
Antimalarial activity of optical isomers of quinacrine dihydrochloride against chloroquine-sensitive and -resistant Plasmodium falciparum in vitro.
    Biochemical pharmacology, 1991, Dec-11, Volume: 42 Suppl

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Plasmodium falciparum; Quinacrine; Stereoisomerism

1991
Chloroquine-sensitive transplasmalemma electron transport in Tetrahymena pyriformis: a hypothesis for control of parasite protozoa through transmembrane redox.
    Biochimica et biophysica acta, 1991, Jun-17, Volume: 1058, Issue:2

    Topics: Animals; Cell Wall; Chloroquine; Electron Transport; Ferricyanides; Hydrogen-Ion Concentration; Membrane Potentials; Oxidation-Reduction; Oxygen; Quinacrine; Tetrahymena pyriformis

1991
Degradation of insulin in isolated liver endosomes is functionally linked to ATP-dependent endosomal acidification.
    European journal of biochemistry, 1990, Oct-24, Volume: 193, Issue:2

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Cations; Chloroquine; Guanosine Triphosphate; Hydrogen-Ion Concentration; Inosine Triphosphate; Insulin; Liver; Male; Organelles; Quinacrine; Rats; Rats, Inbred Strains; Subcellular Fractions; Uridine Triphosphate

1990
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with lipids extracted from normal human erythrocytes.
    Molecular and biochemical parasitology, 1990, Jan-01, Volume: 38, Issue:1

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Deuterium; Erythrocytes; Humans; Magnetic Resonance Spectroscopy; Mefloquine; Membrane Lipids; Phosphatidylethanolamines; Phosphorus Isotopes; Quinacrine; Quinine

1990
Depressant effects of chloroquine on the isolated guinea-pig heart.
    European journal of pharmacology, 1990, Mar-27, Volume: 178, Issue:3

    Topics: Animals; Calcium; Chloroquine; Depression, Chemical; Electric Stimulation; Female; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Ouabain; Quinacrine

1990
The effects of non-steroidal inhibitors of phospholipase A2 on leukotriene and histamine release from human and guinea-pig lung.
    Prostaglandins, 1985, Volume: 30, Issue:2

    Topics: Animals; Calcimycin; Chloroquine; Guinea Pigs; Histamine Release; Humans; Lung; Ovalbumin; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; SRS-A

1985
3H-azidopine photoaffinity labeling of high molecular weight proteins in chloroquine resistant falciparum malaria.
    Biochemical and biophysical research communications, 1989, Jul-31, Volume: 162, Issue:2

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Chloroquine; Chlorpromazine; Dihydropyridines; Drug Resistance; Glycoproteins; Molecular Weight; Nicardipine; Photochemistry; Plasmodium falciparum; Proteins; Quinacrine; Reserpine; Trifluoperazine; Verapamil

1989
Ca2+-antagonistic properties of phospholipase A2 inhibitors, mepacrine and chloroquine.
    General physiology and biophysics, 1989, Volume: 8, Issue:2

    Topics: Animals; Calcium; Calcium Channel Blockers; Chloroquine; In Vitro Techniques; Membrane Potentials; Myocardium; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rana ridibunda

1989
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with dipalmitoylphosphatidylcholine bilayers.
    Molecular and biochemical parasitology, 1989, Volume: 35, Issue:3

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Mefloquine; Quinacrine; Quinine; Quinolines; Temperature

1989
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1985, Volume: 81, Issue:1

    Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains

1985
[Synthetic antimalarials in the therapy of rheumatoid arthritis: adverse effects and advantages].
    Minerva medica, 1985, Oct-06, Volume: 76, Issue:38

    Topics: Arthritis, Rheumatoid; Chloroquine; Drug Evaluation; Enzyme Inhibitors; Histamine H1 Antagonists; Humans; Hydroxychloroquine; Quinacrine; Time Factors

1985
Effects of indole alkaloids on multidrug resistance and labeling of P-glycoprotein by a photoaffinity analog of vinblastine.
    Biochemical and biophysical research communications, 1988, Jun-30, Volume: 153, Issue:3

    Topics: Affinity Labels; Alkaloids; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Survival; Chloroquine; Drug Interactions; Drug Resistance; Humans; Indoles; Leukemia; Membrane Glycoproteins; Photochemistry; Quinacrine; Quinine; Reserpine; Verapamil; Vinblastine; Vinca Alkaloids; Vindesine; Yohimbine

1988
[Effect of Collagenan on joint disease associated with collagenous colitis].
    Presse medicale (Paris, France : 1983), 1986, Nov-08, Volume: 15, Issue:39

    Topics: 4-Aminobenzoic Acid; Aminobenzoates; Chloroquine; Colitis; Collagen; Drug Combinations; Female; Humans; Joint Diseases; Middle Aged; Pantothenic Acid; Pyridoxine; Quinacrine

1986
[Evaluation of the phototoxicity of five antimalarial agents and praziquantel in mice].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1986, Volume: 7, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Female; Male; Mice; Naphthyridines; Photosensitivity Disorders; Praziquantel; Quinacrine; Quinazolines; Quinolines; Ultraviolet Rays

1986
Antioxidant action of antimalarials.
    Annals of the rheumatic diseases, 1986, Volume: 45, Issue:3

    Topics: Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Humans; Hydrogen Peroxide; Neutrophils; Oxygen; Quinacrine; Superoxides

1986
Differential effects of mepacrine, chloroquine and hydroxychloroquine on superoxide anion generation, phospholipid methylation and arachidonic acid release by human blood monocytes.
    Biochemical pharmacology, 1986, Sep-15, Volume: 35, Issue:18

    Topics: Arachidonic Acid; Arachidonic Acids; Calcimycin; Cell Survival; Chloroquine; Fluorides; Humans; Hydroxychloroquine; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Phospholipids; Quinacrine; Superoxides; Tetradecanoylphorbol Acetate; Zymosan

1986
Mepacrine accumulation during treatment of chloroquine-resistant falciparum malaria.
    Annals of tropical medicine and parasitology, 1988, Volume: 82, Issue:2

    Topics: Adolescent; Adult; Animals; Chloroquine; Drug Resistance; Female; Humans; Malaria; Male; Middle Aged; Plasmodium falciparum; Quinacrine

1988
Stimulation of luteinizing hormone release by melittin and phospholipase A2 in rat pituitary cells.
    Molecular and cellular endocrinology, 1987, Volume: 51, Issue:1-2

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bee Venoms; Cell Membrane; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Enzyme Activation; Female; Gonadotropin-Releasing Hormone; In Vitro Techniques; Luteinizing Hormone; Melitten; Phospholipases; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Quinacrine; Rats; Secretory Rate

1987
The mechanism of the inhibitory effects of antimalarials on UV-induced skin inflammation in mice.
    The Journal of dermatology, 1988, Volume: 15, Issue:2

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Chloroquine; Ear, External; Edema; Female; Inflammation; Mice; Mice, Inbred ICR; PUVA Therapy; Quinacrine; Skin; Ultraviolet Rays

1988
Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells.
    Molecular pharmacology, 1988, Volume: 33, Issue:4

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cell Line; Chemical Phenomena; Chemistry, Physical; Chloroquine; Computer Simulation; Doxorubicin; Drug Resistance; Humans; Leukemia; Naphthacenes; Podophyllotoxin; Quinacrine; Verapamil; Vinca Alkaloids

1988
[The mouse micronucleus test for mutagenicity of pyronaridine, chloroquine, quinacrine, primaquine, furapyrimidone and phenthiourezine].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1988, Volume: 6, Issue:4

    Topics: Animals; Anthelmintics; Antimalarials; Chloroquine; Filaricides; Male; Mice; Micronucleus Tests; Mutagenicity Tests; Naphthyridines; Nitrofurans; Piperazines; Primaquine; Quinacrine

1988
Spermidine oxidase activity in serum of normal and schizophrenic subjects.
    Clinical chemistry, 1988, Volume: 34, Issue:2

    Topics: Adult; Chloroquine; Female; Humans; Male; Middle Aged; Oxidoreductases Acting on CH-NH Group Donors; Polyamine Oxidase; Quality Control; Quinacrine; Reference Values; Schizophrenia; Substrate Specificity

1988
The in vitro pharmacology of chloroquine and quinacrine.
    Medical biology, 1986, Volume: 64, Issue:4

    Topics: Animals; Biological Transport, Active; Chickens; Chloroquine; Guanethidine; In Vitro Techniques; Male; Neurons; Nordefrin; Norepinephrine; Quinacrine

1986
Degradation of dipalmitoyl phosphatidylcholine by isolated rat granular pneumocytes and reutilization for surfactant synthesis.
    The Journal of clinical investigation, 1987, Volume: 79, Issue:4

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Ammonium Chloride; Animals; Chloroquine; Choline; Liposomes; Lung; Methylamines; Organoids; Pulmonary Surfactants; Quinacrine; Rats

1987
Brugia pahangi: inhibition of protein synthesis.
    Experimental parasitology, 1987, Volume: 64, Issue:2

    Topics: Animals; Antimycin A; Brugia; Chloramphenicol; Chloroquine; Cyanides; Cycloheximide; Electron Transport; Lactates; Molecular Weight; Movement; Protein Biosynthesis; Protein Synthesis Inhibitors; Quinacrine

1987
Stimulation of phospholipase A2 activity by oxygen-derived free radicals in isolated brain capillaries.
    Journal of cellular biochemistry, 1985, Volume: 27, Issue:4

    Topics: Animals; Brain; Capillaries; Chloroquine; Fatty Acids; Fatty Acids, Unsaturated; Free Radicals; Oxygen; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains; Xanthine Oxidase

1985
The action of salinomycin-Na and lasalocid-Na on chloroquine- and mepacrine-resistant line of Plasmodium berghei K 173-strain in Wistar rats.
    Zeitschrift fur Parasitenkunde (Berlin, Germany), 1985, Volume: 71, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Cell Membrane; Chloroquine; Cytoplasm; Drug Resistance, Microbial; Lasalocid; Lethal Dose 50; Malaria; Male; Microscopy, Electron; Plasmodium berghei; Pyrans; Quinacrine; Rats; Rats, Inbred Strains; Time Factors

1985
Testing of chloroquine and quinacrine for mutagenicity in Drosophila melanogaster.
    Mutation research, 1985, Volume: 158, Issue:3

    Topics: Animals; Chloroquine; Drosophila melanogaster; Genes, Lethal; Genes, Recessive; Male; Mutagenicity Tests; Quinacrine; Sex Chromosome Aberrations

1985
Cutaneous lupus erythematosus. Recognition of its many forms.
    Postgraduate medicine, 1986, Volume: 79, Issue:5

    Topics: Adrenal Cortex Hormones; Adult; Chloroquine; Diagnosis, Differential; Female; Humans; Hydroxychloroquine; Infant, Newborn; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Male; Quinacrine; Sex Factors; Skin; Skin Diseases

1986
Effects of antimalarial drugs on phospholipase A and lysophospholipase activities in plasma membrane, mitochondrial, microsomal and cytosolic subcellular fractions of rat liver.
    Biochimica et biophysica acta, 1985, Jul-31, Volume: 835, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chloroquine; Cytosol; Endoplasmic Reticulum; Liver; Lysophospholipase; Male; Microsomes, Liver; Mitochondria, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1985
[Ultrastructural studies of the effect of x-rays and quinacrine (Atebrin) or chloroquine (Resochin)--alone or in combination--on Harding-Passey melanoma cells in monolayer culture].
    Strahlentherapie, 1985, Volume: 161, Issue:11

    Topics: Animals; Chloroquine; Combined Modality Therapy; In Vitro Techniques; Melanoma; Mice; Microscopy, Electron; Quinacrine; Radiation-Sensitizing Agents

1985
Pharmacological investigation of the mechanisms of platelet-activating factor induced mortality in the mouse.
    Prostaglandins, 1985, Volume: 30, Issue:4

    Topics: Anaphylaxis; Animals; Chloroquine; Chlortetracycline; Dexamethasone; Dose-Response Relationship, Drug; Female; Indomethacin; Injections, Intravenous; Male; Mice; Mice, Inbred DBA; Naproxen; Nicardipine; Nifedipine; Platelet Activating Factor; Pyrazoles; Quinacrine; Tetracycline; Verapamil

1985
Effect of quinoline, phthalazine and coumarin derivatives on the absorbance of NADPH.
    Research communications in chemical pathology and pharmacology, 1974, Volume: 7, Issue:1

    Topics: Chloroquine; Coumarins; Heterocyclic Compounds; Hydralazine; Indophenol; NADP; Novobiocin; Quinacrine; Quinidine; Quinine; Quinolines; Spectrophotometry; Warfarin

1974
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
    Pharmacology, 1974, Volume: 12, Issue:1

    Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides

1974
Chloroquine-resistant falciparum malaria in Thailand.
    Lancet (London, England), 1965, Oct-02, Volume: 2, Issue:7414

    Topics: Adolescent; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Humans; Infant; Malaria; Plasmodium falciparum; Quinacrine; Quinine; Thailand

1965
Activity and some properties of an acid proteinase from normal and Plasmodium berghei-infected red cells.
    The Journal of parasitology, 1973, Volume: 59, Issue:6

    Topics: Acid Phosphatase; Animals; Cell-Free System; Chloroquine; Dithiothreitol; Edetic Acid; Erythrocytes; Female; Hemoglobins; Hemolysis; Hydrogen-Ion Concentration; Malaria; Mice; Mice, Inbred BALB C; Peptide Hydrolases; Plasmodium berghei; Primaquine; Quinacrine; Rats; Solubility; Surface-Active Agents; Ultracentrifugation

1973
Biochemical properties of anti-inflammatory drugs. VI. The effects of chloroquine (resochin), mepacrine (quinacrine) and some of their potential metabolites on cartilage metabolism and oxidative phosphorylation.
    Biochemical pharmacology, 1965, Volume: 14, Issue:8

    Topics: Animals; Cartilage; Chloroquine; Glycosaminoglycans; Gold; Hydroxychloroquine; In Vitro Techniques; Indomethacin; Oxidative Phosphorylation; Polysaccharides; Quinacrine; Quinolines; Rats; Sulfates; Sulfur Isotopes; Thiosulfates

1965
[Use of a Dicrocoelium survival test in the study of the experimental activity of various chemical substances].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1967, Volume: 161, Issue:3

    Topics: Animals; Arsenicals; Chloroquine; Dicrocoelium; Piperazines; Quinacrine; Thiabendazole

1967
The amoebicidal, trichomonicidal, and antibacterial effects of niridazole in laboratory animals.
    Annals of the New York Academy of Sciences, 1969, Oct-06, Volume: 160, Issue:2

    Topics: Amebiasis; Amebicides; Amoeba; Animals; Anthelmintics; Antimony; Antiprotozoal Agents; Chloroquine; Clioquinol; Cricetinae; Dysentery, Bacillary; Emetine; Enterobacteriaceae Infections; Furazolidone; Imidazoles; Intestinal Diseases, Parasitic; Liver Abscess, Amebic; Metronidazole; Mice; Quinacrine; Salmonella Infections; Sulfonamides; Sulfones; Tartrates; Tetracycline; Thiazoles; Trichomonas Infections

1969
[Complications with synthetic antimalarials].
    Lille medical : journal de la Faculte de medecine et de pharmacie de l'Universite de Lille, 1969, Volume: 14, Issue:8

    Topics: Antimalarials; Asthenia; Central Nervous System Diseases; Chloroquine; Drug Eruptions; Eczema; Eye Diseases; Gastrointestinal Diseases; Hematologic Diseases; Humans; Lupus Erythematosus, Systemic; Pigmentation Disorders; Psoriasis; Quinacrine; Skin Diseases

1969
Inactivation of lysosomal function in normal cultured human fibroblasts by chloroquine.
    Biochemical pharmacology, 1973, Dec-01, Volume: 22, Issue:23

    Topics: Cell Survival; Cells, Cultured; Chloroquine; Fibroblasts; Glycosaminoglycans; Humans; Hydrogen-Ion Concentration; Lysosomes; Microscopy, Electron; Quinacrine; Quinine; Sulfur Radioisotopes; Time Factors

1973
Biochemical properties of anti-inflammatory drugs. VII. Inhibition of proteolytic enzymes in connective tissue by chloroquine (resochin) and related antimalarial antirheumatic drugs.
    Biochemical pharmacology, 1966, Volume: 15, Issue:8

    Topics: Acridines; Animals; Cartilage; Cattle; Chloroquine; Chondroitin; Connective Tissue; Hyaluronoglucosaminidase; Hydrogen-Ion Concentration; Hydroxychloroquine; Microbial Collagenase; Mucoproteins; Papain; Primaquine; Quaternary Ammonium Compounds; Quinacrine; Rabbits

1966
Response of isolated white fat cells to anti-malarial drugs.
    Biochemical pharmacology, 1973, Dec-01, Volume: 22, Issue:23

    Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Animals; Antimalarials; Bucladesine; Chloroquine; Drug Synergism; Fatty Acids, Nonesterified; Female; Glycerol; Norepinephrine; Primaquine; Proteins; Quinacrine; Quinidine; Rats; Theophylline; Triglycerides

1973
Light-microscopic demonstration of drug-induced myelin bodies in the liver of rats.
    Experientia, 1974, Apr-15, Volume: 30, Issue:4

    Topics: Animals; Chloroquine; Cytoplasmic Granules; Inclusion Bodies; Liver; Male; Microscopy; Microscopy, Fluorescence; Quinacrine; Triparanol

1974
Increased levels of pisatin and phenylalanine ammonia lyase activity in Pisum sativum treated with antihistaminic, antiviral, antimalarial, tranquilizing, or other drugs.
    Biochemical and biophysical research communications, 1972, Jan-14, Volume: 46, Issue:1

    Topics: Antidepressive Agents; Antitussive Agents; Antiviral Agents; Chloroquine; Deamination; Ethylamines; Fluorenes; Histamine H1 Antagonists; Imipramine; Ketones; Lectins; Leucine; Lyases; Parasympatholytics; Phenothiazines; Phenylalanine; Piperidines; Plant Lectins; Plant Proteins; Plants, Edible; Propantheline; Quinacrine; Stimulation, Chemical; Tranquilizing Agents; Trimeprazine

1972
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
    Biochemical pharmacology, 1971, Volume: 20, Issue:11

    Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes

1971
Discoid lupus erythematosus.
    Archives of dermatology, 1972, Volume: 105, Issue:5

    Topics: Adult; Antimalarials; Chloroquine; Color Vision Defects; Female; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Quinacrine; Retinal Diseases

1972
Labilizing action of intercalating drugs and dyes on bacterial ribosomes.
    Biochemistry, 1972, Apr-25, Volume: 11, Issue:9

    Topics: Acridines; Bacterial Proteins; Berberine Alkaloids; Carbon Isotopes; Centrifugation, Density Gradient; Chloroquine; Coloring Agents; Daunorubicin; Dioxoles; Escherichia coli; Ethidium; Hot Temperature; Lucanthone; Methylene Blue; Nucleoproteins; Phenanthridines; Phenylalanine; Quinacrine; Quinolines; Ribosomes; RNA, Ribosomal; Spectrometry, Fluorescence; Spermine; Tritium; Uridine

1972
Multidrug-resistant strain of Plasmodium falciparum from eastern Colombia.
    The Journal of infectious diseases, 1974, Volume: 129, Issue:4

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Colombia; Drug Combinations; Drug Resistance, Microbial; Female; Humans; Malaria; Male; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine

1974
Some pharmacological aspects of antimalarial drugs.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1974, Jun-15, Volume: 48, Issue:29

    Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim

1974
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
    The Journal of pharmacology and experimental therapeutics, 1972, Volume: 180, Issue:1

    Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine

1972
Inhibition of DNA repair replication by DNA binding drugs which sensitize cells to alkylating agents and X-rays.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1972, Volume: 141, Issue:2

    Topics: Alkylating Agents; Caffeine; Chloroquine; Cyanides; Cyclophosphamide; Dinitrophenols; DNA Repair; DNA Replication; Dose-Response Relationship, Radiation; Drug Combinations; Humans; Hydroxyurea; Injections, Intraperitoneal; Leukocyte Count; Lymphocytes; Protein Binding; Quinacrine; Quinolines; Radiation Effects; Radiation-Sensitizing Agents; Thymidine; Tritium; Ultraviolet Rays

1972
In vitro effect of drugs against pathogenic and non-pathogenic free-living amoebae and on anaerobic amoebae.
    Indian journal of experimental biology, 1972, Volume: 10, Issue:1

    Topics: Anaerobiosis; Animals; Biguanides; Chloroquine; Eukaryota; Metronidazole; Quinacrine

1972
Induction of enzymes in dormant spores of Aspergillus oryzae. IV. Effects of ethidium, aminoacridines, and related compounds.
    Biochimica et biophysica acta, 1973, Apr-11, Volume: 299, Issue:4

    Topics: Acridines; Alcohol Oxidoreductases; Amines; Aspergillus; Carbon Isotopes; Chloroquine; Enzyme Induction; Ethidium; Fungal Proteins; Glucose; Hydroquinones; Kinetics; Leucine; Oxygen Consumption; Phenanthridines; Phenothiazines; Quinacrine; Spores; Spores, Fungal; Sucrase

1973
Inhibitory effect of some quinoline, phthalazine, and coumarin derivatives on glucose-6-phosphate dehydrogenase in vitro.
    Research communications in chemical pathology and pharmacology, 1973, Volume: 6, Issue:2

    Topics: Binding, Competitive; Chloroquine; Coumarins; Glucosephosphate Dehydrogenase; Heterocyclic Compounds; Hydralazine; Isoniazid; Novobiocin; Phenazines; Phenelzine; Phenylhydrazines; Probenecid; Pyridines; Quinacrine; Quinidine; Quinine; Quinolines; Sulfanilamides; Warfarin; Yeasts

1973
Similarities between antimalarial schizontocides.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1973, Volume: 67, Issue:1

    Topics: Antimalarials; Binding Sites; Chloroquine; Quinacrine; Quinine; Structure-Activity Relationship

1973
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
    Gastroenterology, 1974, Volume: 66, Issue:5

    Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors

1974
[Chloroquine induced neuropathy].
    Lakartidningen, 1974, May-08, Volume: 71, Issue:19

    Topics: Administration, Oral; Chloroquine; Drug Combinations; Drug Therapy, Combination; Electromyography; Female; Humans; Leg; Middle Aged; Myotonic Dystrophy; Prednisolone; Quinacrine; Time Factors

1974
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones

1968
Malaria and victory in Vietnam. The first battle against drug-resistant malignant malaria is described.
    Science (New York, N.Y.), 1968, Dec-20, Volume: 162, Issue:3860

    Topics: Anopheles; Antimalarials; Chloroquine; Folic Acid Antagonists; Folic Acid Deficiency; History, 16th Century; History, 17th Century; History, 20th Century; Malaria; Military Medicine; Penicillin Resistance; Penicillins; Plasmodium falciparum; Pyrimidines; Quinacrine; Sulfonamides; Tropical Medicine; Vietnam

1968
Studies concerning the mechanism of action of antimalarial drugs. Inhibition of the incorporation of adenosine-8-3H into nucleic acids of Plasmodium berghei.
    Biochemical pharmacology, 1969, Volume: 18, Issue:6

    Topics: Animals; Antimalarials; Autoradiography; Chloroquine; DNA Nucleotidyltransferases; DNA Replication; Escherichia coli; Male; Methods; Nucleosides; Phenanthridines; Plasmodium; Quinacrine; Quinine; Rats; RNA; RNA Nucleotidyltransferases; Time Factors; Tritium

1969
The problems of drug-resistant pathogenic bacteria. Elimination of bacterial episomes by DNA-complexing compounds.
    Annals of the New York Academy of Sciences, 1971, Jun-11, Volume: 182

    Topics: Acridines; Carbon Isotopes; Centrifugation, Density Gradient; Cesium; Chloramphenicol; Chlorides; Chloroquine; DNA, Bacterial; Drug Resistance, Microbial; Escherichia coli; Genetics, Microbial; Kanamycin; Lactose; Methylene Blue; Phenanthridines; Quinacrine; Quinine; Rosaniline Dyes; Spermine; Thymidine

1971
Antibacterial nitroacridine, Nitroakridin 3582: binding to nucleic acids in vitro and effects on selected cell-free model systems of macromolecular biosynthesis.
    Journal of bacteriology, 1971, Volume: 108, Issue:3

    Topics: Acridines; Anti-Bacterial Agents; Binding Sites; Carbon Isotopes; Cell-Free System; Chloroquine; DNA Nucleotidyltransferases; DNA, Bacterial; Escherichia coli; Genetics, Microbial; Hot Temperature; Micrococcus; Models, Chemical; Nitro Compounds; Nucleic Acid Denaturation; Nucleic Acids; Phenanthridines; Phenylalanine; Polynucleotides; Protein Binding; Quinacrine; Ribosomes; RNA Nucleotidyltransferases; RNA, Bacterial; RNA, Transfer; Spectrophotometry; Templates, Genetic; Tritium

1971
The routine treatment of malaria.
    Tropical doctor, 1971, Volume: 1, Issue:4

    Topics: Acute Disease; Adolescent; Adult; Amodiaquine; Child; Child, Preschool; Chloroquine; Chronic Disease; Drug Resistance, Microbial; Female; Humans; Infant; Malaria; Male; Plasmodium falciparum; Quinacrine; Quinine; Sulfonamides

1971
Drugs for petit mal.
    Canadian Medical Association journal, 1965, Sep-25, Volume: 93, Issue:13

    Topics: Acetazolamide; Amphetamine; Anticonvulsants; Barbiturates; Child; Child, Preschool; Chlordiazepoxide; Chloroquine; Epilepsy, Absence; Ethosuximide; Humans; Meprobamate; Quinacrine; Succinimides; Trimethadione

1965
The influence of methylene blue on the pentose phosphate pathway in erythrocytes of monkeys infected with Plasmodium knowlesi.
    The Journal of laboratory and clinical medicine, 1969, Volume: 74, Issue:1

    Topics: Animals; Carbon Isotopes; Chloroquine; DNA; Erythrocytes; Glucose; Haplorhini; Isoleucine; Malaria; Methylene Blue; Orotic Acid; Pentosephosphates; Plasmodium; Protein Biosynthesis; Quinacrine; Quinine; RNA; Tritium

1969
Uptake of chloroquine-3-H3 by plasmodium knowlesi in vitro.
    The Journal of pharmacology and experimental therapeutics, 1969, Volume: 168, Issue:1

    Topics: Albumins; Animals; Chloroquine; Cyanates; Dinitrophenols; Erythrocytes; Fluorides; Glucose; Haplorhini; In Vitro Techniques; Iodoacetates; Lysosomes; Malaria; Pinocytosis; Plasmodium; Quinacrine; Quinine; Temperature; Time Factors; Tritium

1969
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1970, Volume: 21, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors

1970
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
    Biochemical pharmacology, 1971, Volume: 20, Issue:8

    Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents

1971
The role of drugs in a malaria program.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Malaria; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Recurrence; Sulfonamides; Sulfones; Trimethoprim

1972
Studies concerning the mechanism of action of antimalarial drugs. II. Inhibition of the incorporation of adenosine-5'-monophosphate- 3 H into nucleic acids of erythrocyte-free malarial parasites.
    Biochemical pharmacology, 1971, Volume: 20, Issue:6

    Topics: Adenine Nucleotides; Adenosine; Adenosine Monophosphate; Amodiaquine; Animals; Antimalarials; Chloroquine; DNA; Erythrocytes; Methods; Naphthalenes; Phenanthridines; Plasmodium; Proguanil; Quinacrine; Quinine; Rats; RNA; Saponins; Triazines; Trimethoprim; Tritium

1971
Acridine orange potentiation of actinomycin D uptake and activity.
    Science (New York, N.Y.), 1971, Nov-12, Volume: 174, Issue:4010

    Topics: Acridines; Animals; Autoradiography; Chloroquine; Dactinomycin; DNA; Drug Synergism; Freezing; Humans; In Vitro Techniques; Lymphocytes; Male; Mice; Organ Size; Protein Binding; Quinacrine; Spleen; Tritium; Vibration

1971
Pigmentation of the hard and solf palate in a patient with rheumatoid arthritis treated with an antimalarial (triquin).
    Svensk tandlakare tidskrift. Swedish dental journal, 1970, Volume: 63, Issue:9

    Topics: Arthritis, Rheumatoid; Biopsy; Chloroquine; Female; Humans; Middle Aged; Palate; Pigmentation Disorders; Quinacrine; Time Factors

1970
Reactions of quinine, chloroquine, and quinacrine with DNA and their effects on the DNA and RNA polymerase reactions.
    Proceedings of the National Academy of Sciences of the United States of America, 1966, Volume: 55, Issue:6

    Topics: Chemical Phenomena; Chemistry; Chloroquine; DNA; Escherichia coli; Nucleotidyltransferases; Quinacrine; Quinine; Spermine

1966
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
    Biochimica et biophysica acta, 1969, Dec-17, Volume: 187, Issue:4

    Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats

1969
[Asthma therapy with a combination of synthetic antimalarials (83 cases)].
    La Presse medicale, 1969, Dec-13, Volume: 77, Issue:53

    Topics: Adolescent; Adult; Aged; Asthma; Chloroquine; Drug Synergism; Electrocardiography; Eosinophilia; Eye Manifestations; Glucocorticoids; Humans; Middle Aged; Pyridoxine; Quinacrine; Sympathomimetics; Vitamin B Complex

1969
An automated method of mass drug testing applied to screening for antimalarial activity.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones

1970
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium

1970
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
    The Journal of pharmacology and experimental therapeutics, 1970, Volume: 173, Issue:1

    Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium

1970
Antimalarials: effects on in vivo and in vitro protein synthesis.
    Science (New York, N.Y.), 1970, Dec-11, Volume: 170, Issue:3963

    Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
The chemotherapy of rodent malaria. XII. Substituted tetrahydrofurans, a new chemical family of antimalarials. The action of 2-(p-chlorophenyl)-2-(4-piperidyl)-tetrahydrofuran against Plasmodium berghei and Plasmodium chabaudi.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:2

    Topics: Aminobenzoates; Animals; Antimalarials; Chloroquine; Diet; Drug Resistance, Microbial; Drug Synergism; Folic Acid; Furans; Mice; Piperidines; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1970
[Cytostatic effect of resochin and atebrin (compare same journal 20 (N.F.) 28: 1591 (1969))].
    Die Medizinische Welt, 1970, May-30, Volume: 22

    Topics: Animals; Antineoplastic Agents; Chloroquine; Humans; Neoplasms; Neoplasms, Experimental; Quinacrine

1970
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
    Parasitology, 1967, Volume: 57, Issue:4

    Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines

1967
[Tropical diseases treated at Roslagstulls Hospital].
    Lakartidningen, 1967, Sep-20, Volume: 64, Issue:38

    Topics: Adolescent; Adult; Aged; Amebiasis; Anti-Bacterial Agents; Antimony; Child; Chloroquine; Diethylcarbamazine; Female; Filariasis; Giardiasis; Hospitals, General; Humans; Malaria; Male; Middle Aged; Quinacrine; Schistosomiasis; Sweden

1967
The inhibitory effect of mepacrine and chloroquine on the photodynamic action.
    Arzneimittel-Forschung, 1967, Volume: 17, Issue:6

    Topics: Animals; Chloroquine; Depression, Chemical; Light; Methylene Blue; Quinacrine; Tetrahymena

1967
Synthesis and antimalarial evaluation of some 1,7-nephthyridines and 2,9-diazaanthracenes.
    Journal of medicinal chemistry, 1968, Volume: 11, Issue:1

    Topics: Animals; Benzene Derivatives; Chloroquine; Malaria; Methods; Mice; Naphthyridines; Quinacrine

1968
Psychiatric complications with chloroquine and quinacrine.
    The American journal of psychiatry, 1968, Volume: 124, Issue:9

    Topics: Anti-Inflammatory Agents; Chloroquine; Humans; Malaria; Malingering; Psychoses, Substance-Induced; Quinacrine; Suicide; United States

1968
Erythema dyschromicum perstans.
    Archives of dermatology, 1968, Volume: 97, Issue:3

    Topics: Adolescent; Adult; Biopsy; Blood Cell Count; Blood Sedimentation; Child, Preschool; Chloroquine; Erythema; Feces; Female; Humans; Hydroquinones; Hydroxychloroquine; Male; Middle Aged; Parasitic Diseases; Prednisone; Quinacrine; Steroids; Syphilis Serodiagnosis; Triamcinolone

1968
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
    The American journal of tropical medicine and hygiene, 1968, Volume: 17, Issue:3

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena

1968
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
Ocular toxicity of antimalarial drugs. Long-term follow-up.
    American journal of ophthalmology, 1968, Volume: 66, Issue:4

    Topics: Adolescent; Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Electrooculography; Electroretinography; Eye Diseases; Follow-Up Studies; Fundus Oculi; Humans; Hydroxychloroquine; Light; Lupus Erythematosus, Systemic; Macula Lutea; Middle Aged; Ophthalmoscopy; Quinacrine; Retinitis; Vision Tests; Visual Fields

1968
The Plasmodium chabaudi-mouse system in chemotherapy studies.
    Experimental parasitology, 1969, Volume: 24, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Injections, Intravenous; Malaria; Male; Mice; Plasmodium; Primaquine; Quinacrine

1969
Immunosuppression by compounds which complex with deoxyribonucleic acid.
    Biochemical pharmacology, 1969, Volume: 18, Issue:8

    Topics: Acridines; Alcohols; Animals; Antibody Formation; Chloroquine; Coloring Agents; DNA; Erythrocytes; Female; Fishes; Immunosuppressive Agents; Male; Methods; Mice; Protein Binding; Quinacrine; Quinolines; Sheep; Spleen; Splenomegaly; Transplantation Immunology; Transplantation, Homologous

1969
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1965
Chloroquine: physiological basis of drug resistance in Plasmodium berghei.
    Science (New York, N.Y.), 1966, Jun-03, Volume: 152, Issue:3727

    Topics: Animals; Carbon Isotopes; Chloroquine; Drug Resistance, Microbial; Erythrocytes; In Vitro Techniques; Liver; Malaria; Male; Mice; Plasmodium; Quinacrine; Quinine; Radiometry; Spleen

1966
Mepacrine and chloroquine in vitiligo.
    Bulletin of the Calcutta School of Tropical Medicine, 1966, Volume: 14, Issue:1

    Topics: Chloroquine; Female; Humans; Male; Quinacrine; Vitiligo

1966
[Ocular accidents from synthetic antimalarials (apropos of 4 new cases)].
    Bulletin des societes d'ophtalmologie de France, 1966, Volume: 66, Issue:11

    Topics: Adolescent; Antimalarials; Child; Chloroquine; Electroretinography; Eye Diseases; Humans; Quinacrine

1966
Metabolic effects of anthelmintic drugs on the cat's tapeworm in vitro.
    Annales medicinae experimentalis et biologiae Fenniae, 1966, Volume: 44, Issue:3

    Topics: Animals; Anthelmintics; Cats; Cestoda; Chloroquine; Glycolysis; In Vitro Techniques; Plant Extracts; Plants, Medicinal; Quinacrine; Resins, Plant; Respiration

1966
Treatment of chloroquine-resistant Plasmodium falciparum infections in Vietnam.
    Annals of internal medicine, 1967, Volume: 66, Issue:3

    Topics: Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Vietnam

1967
The different effects of antimalarial drugs on Plasmodium lophurae developing intracellularly and extracellularly in vitro.
    The American journal of tropical medicine and hygiene, 1967, Volume: 16, Issue:1

    Topics: Animals; Chloroquine; In Vitro Techniques; Malaria, Avian; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine

1967
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
    Journal of medicinal chemistry, 1967, Volume: 10, Issue:5

    Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA

1967
An analysis of the inhibitory effects of quinine and mepacrine in the guinea-pig isolated ileum.
    The Journal of pharmacy and pharmacology, 1980, Volume: 32, Issue:4

    Topics: Animals; Chloroquine; Depression, Chemical; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Prostaglandin Antagonists; Prostaglandins E; Quinacrine; Quinine

1980
Stimulation of polymorphonuclear leucocyte phospholipase A2 activity by chloroquine and mepacrine.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:11

    Topics: Animals; Ascitic Fluid; Chloroquine; Escherichia coli; Female; In Vitro Techniques; Neutrophils; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rabbits

1982
Interaction of basic compounds with coated vesicles.
    Biochemistry, 1984, Dec-04, Volume: 23, Issue:25

    Topics: Alkanesulfonates; Alkanesulfonic Acids; Amines; Animals; Brain; Buffers; Cattle; Centrifugation, Density Gradient; Chloroquine; Clathrin; Coated Pits, Cell-Membrane; Diamines; Endosomes; Hydrogen-Ion Concentration; Light; Morpholines; Polyamines; Quinacrine; Scattering, Radiation

1984
Inhibition of lymphocyte transformation by mepacrine and chloroquine.
    The Journal of pharmacy and pharmacology, 1981, Volume: 33, Issue:7

    Topics: 1-Methyl-3-isobutylxanthine; Cells, Cultured; Chloroquine; Humans; In Vitro Techniques; Leucine; Lymphocyte Activation; Phytohemagglutinins; Quinacrine; Thymidine; Uridine

1981
The effect of anti-malarial drugs on human natural killer cells in vitro.
    Parasite immunology, 1984, Volume: 6, Issue:6

    Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines

1984
Comparative effects of intrauterine instillation of analogues of quinacrine and tetracycline on uterine morphology in the rat.
    Contraception, 1984, Volume: 29, Issue:6

    Topics: Animals; Chloroquine; Demeclocycline; Doxycycline; Female; Primaquine; Quinacrine; Rats; Rats, Inbred Strains; Sodium Chloride; Tetracycline; Tetracyclines; Trimethoprim; Uterus

1984
Inhibition of lipid peroxidation in muscle homogenates by phospholipase A2 inhibitors.
    Bioscience reports, 1984, Volume: 4, Issue:7

    Topics: Animals; Chloroquine; Chlorpromazine; Dibucaine; Female; Free Radicals; In Vitro Techniques; Iron; Lipid Peroxides; Mice; Muscles; Phospholipases; Phospholipases A; Phospholipases A2; Procaine; Quinacrine; Tetracaine

1984
Inhibition of rat hepatic mixed function oxidases by antimalarial drugs: selectivity for cytochromes P-450 and P-448.
    Chemico-biological interactions, 1984, Volume: 51, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Cytochromes; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases; Oxidoreductases, N-Demethylating; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1984
Corneal lipidosis in rats treated with amphiphilic cationic drugs.
    Arzneimittel-Forschung, 1983, Volume: 33, Issue:6

    Topics: Animals; Cations; Chloroquine; Chlorphentermine; Corneal Diseases; Female; Iprindole; Lipidoses; Male; Quinacrine; Rats; Rats, Inbred Strains; Tamoxifen

1983
The chemotherapy of rodent malaria XXXIII. The activity of chloroquine and related blood schizontocides and of some analogues in drug-induced pigment clumping.
    Annals of tropical medicine and parasitology, 1982, Volume: 76, Issue:3

    Topics: Amodiaquine; Animals; Chloroquine; Cyclic N-Oxides; Dose-Response Relationship, Drug; Erythrocytes; Pigmentation; Plasmodium berghei; Quinacrine

1982
Inhibition of diamine oxidase by antimalarial drugs.
    Agents and actions, 1980, Volume: 10, Issue:5

    Topics: Amine Oxidase (Copper-Containing); Amodiaquine; Animals; Antimalarials; Chloroquine; In Vitro Techniques; Intestine, Small; Male; Putrescine; Quinacrine; Rats

1980
Inhibition of the metabolism and motility of human spermatozoa by various alkaloids.
    Contraception, 1982, Volume: 25, Issue:1

    Topics: Antimalarials; Carbon Dioxide; Chloroquine; Emetine; Humans; Lactates; Lactic Acid; Male; Quinacrine; Quinine; Sperm Motility; Spermatozoa

1982
Gas chromatographic analysis of chloroquine after a unique reaction with chloroformates.
    Journal of chromatography, 1983, Feb-11, Volume: 272, Issue:2

    Topics: Aminoquinolines; Chemical Phenomena; Chemistry; Chloroquine; Chromatography, Gas; Humans; Mass Spectrometry; Phosgene; Quinacrine

1983
Suppression by phospholipase A2 inhibitors of secretion of catecholamines from isolated adrenal medullary cells by suppression of cellular calcium uptake.
    Biochemical pharmacology, 1983, Apr-01, Volume: 32, Issue:7

    Topics: Acetophenones; Adrenal Medulla; Animals; Calcium; Carbachol; Catecholamines; Cattle; Chloroquine; Dose-Response Relationship, Drug; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Quinine

1983
The uptake of 14C-chloroquine by mouse pancreatic islets in vitro.
    Acta pharmacologica et toxicologica, 1980, Volume: 47, Issue:1

    Topics: Absorption; Animals; Chloroquine; Chlorpromazine; Desipramine; Glucose; Hydrogen-Ion Concentration; Imipramine; Islets of Langerhans; Lidocaine; Mice; Nicotine; Nitrogen; Ouabain; Quinacrine; Temperature

1980
Binding of antimalarial drugs to hemozoin from Plasmodium berghei.
    Experientia, 1980, Sep-15, Volume: 36, Issue:9

    Topics: Animals; Antimalarials; Chloroquine; Heme; Hemeproteins; Mefloquine; Methemoglobin; Pigments, Biological; Piperidines; Plasmodium berghei; Protein Binding; Protoporphyrins; Quinacrine; Quinolines; Spectrophotometry

1980
Mechanism of action of gonadotropin-releasing hormone. Involvement of phospholipid turnover in luteinizing hormone release.
    The Journal of biological chemistry, 1981, Mar-10, Volume: 256, Issue:5

    Topics: Animals; Arachidonic Acids; Calcium; Cells, Cultured; Chloroquine; Female; Gonadotropin-Releasing Hormone; Indomethacin; Kinetics; Luteinizing Hormone; Phospholipases A; Phospholipases A2; Pituitary Gland; Quinacrine; Rats

1981
Comparative microcalorimetric dilatometric analysis of the interactions of quinacrine, chloroquine, and ethidium bromide with DNA.
    Biopolymers, 1982, Volume: 21, Issue:2

    Topics: Calorimetry; Chemistry Techniques, Analytical; Chloroquine; DNA; Ethidium; Osmolar Concentration; Quinacrine; Thermodynamics

1982
[Influence of x-rays and quinacrine (atebrine) or chloroquine (resochine)--alone or in combination--on growth and melanin formation of Harding-Passey melanoma cells in monolayer culture].
    Strahlentherapie, 1982, Volume: 158, Issue:7

    Topics: Cell Survival; Cells, Cultured; Chloroquine; Dose-Response Relationship, Radiation; Melanins; Melanoma; Neoplasms, Experimental; Quinacrine

1982
Effects of antimalarial drugs on several rat-liver lysosomal enzymes involved in phosphatidylethanolamine catabolism.
    Biochimica et biophysica acta, 1982, Oct-14, Volume: 713, Issue:1

    Topics: Animals; Antimalarials; Carboxylic Ester Hydrolases; Chloroquine; Dose-Response Relationship, Drug; Liver; Lysophospholipase; Lysosomes; Male; Monoacylglycerol Lipases; Phosphatidylethanolamines; Phospholipases; Phospholipases A; Phospholipases A1; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1982
Comparison of the effects of chloroquine quinacrine and quinidine on autonomic neuroeffector mechanisms.
    Medical biology, 1982, Volume: 60, Issue:6

    Topics: Animals; Autonomic Nervous System; Chickens; Chloroquine; Electric Stimulation; Female; Indomethacin; Male; Mice; Norepinephrine; Quinacrine; Quinidine; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Tetrodotoxin

1982
The effect of ionic strength on DNA-ligand unwinding angles for acridine and quinoline derivatives.
    Nucleic acids research, 1980, Apr-11, Volume: 8, Issue:7

    Topics: Aminacrine; Aminoacridines; Animals; Cattle; Chemical Phenomena; Chemistry; Chloroquine; DNA; Ethidium; Kinetics; Molecular Conformation; Nucleic Acid Conformation; Osmolar Concentration; Quinacrine; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Thymus Gland; Viscosity

1980
Effects of several lipidosis-inducing drugs upon the area postrema and adjacent medullary nuclei of adult rats. II. Axonal alternations.
    Acta neuropathologica, 1981, Volume: 53, Issue:1

    Topics: Animals; Axons; Chloroquine; Chlorphentermine; Medulla Oblongata; Microscopy, Electron; Perhexiline; Piperidines; Quinacrine; Rats

1981
Pharmacological basis of dosage form of two antimalarials: chloroquine and mepacrine.
    Acta physiologica Academiae Scientiarum Hungaricae, 1981, Volume: 57, Issue:2

    Topics: Administration, Oral; Animals; Chloroquine; Duodenum; Female; Gastric Emptying; Gastric Mucosa; Infusions, Parenteral; Injections, Intraperitoneal; Intubation, Gastrointestinal; Quinacrine; Rats; Rats, Inbred Strains

1981
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
    Medical microbiology and immunology, 1980, Volume: 168, Issue:1

    Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine

1980
Factors that influence the uptake of beta-hexosaminidase A by rat peritoneal macrophages.
    Biochemical and biophysical research communications, 1980, May-14, Volume: 94, Issue:1

    Topics: Acetylglucosaminidase; Ammonium Chloride; Animals; Biological Transport; Chloroquine; Colchicine; Cytochalasin B; Female; Glycoproteins; Hexosaminidases; Humans; Kinetics; Macrophages; Methylamines; Phagocytosis; Placenta; Pregnancy; Quinacrine; Rats

1980
Effect of chloroquine and mepacrine on the spontaneous and evoked movements of the rat portal vein.
    Acta physiologica Academiae Scientiarum Hungaricae, 1980, Volume: 55, Issue:1

    Topics: Animals; Chloroquine; Dose-Response Relationship, Drug; Epinephrine; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Parasympatholytics; Parasympathomimetics; Phentolamine; Portal Vein; Quinacrine; Rats

1980
[Intensification of the inhibitory effect of X-rays on the growth of Ehrlich ascites tumor cells in monolayer culture by quinacrine (atebrine) or chloroquine (resochine) (author's transl)].
    Strahlentherapie, 1980, Volume: 156, Issue:8

    Topics: Animals; Carcinoma, Ehrlich Tumor; Cell Division; Cells, Cultured; Chloroquine; Quinacrine; Radiotherapy Dosage

1980
Effects of several lipidosis-including drugs upon the area postrema and adjacent medullary nuclei of adult rats. I. Alterations is perikarya and dendrites.
    Acta neuropathologica, 1980, Volume: 52, Issue:3

    Topics: Animals; Blood-Brain Barrier; Brain Diseases; Chloroquine; Chlorphentermine; Female; Lipidoses; Male; Medulla Oblongata; Microscopy, Electron; Perhexiline; Piperidines; Quinacrine; Rats; Time Factors

1980
Receptor-independent uptake of transferrin-bound iron by reticulocytes.
    Archives of biochemistry and biophysics, 1994, Volume: 308, Issue:1

    Topics: Animals; Biological Transport; Cations; Chloroquine; Cytosol; Dicumarol; Edetic Acid; Egtazic Acid; Endocytosis; Erythrocyte Membrane; Heme; In Vitro Techniques; Iodine Radioisotopes; Iron; Iron Radioisotopes; Kinetics; Quinacrine; Rabbits; Receptors, Transferrin; Reticulocytes; Transferrin; Tretinoin

1994
Chloroquine-quinacrine association in resistant cutaneous lupus.
    Dermatology (Basel, Switzerland), 1995, Volume: 190, Issue:3

    Topics: Adult; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Male; Middle Aged; Quinacrine

1995
The association of the two antimalarials chloroquine and quinacrine for treatment-resistant chronic and subacute cutaneous lupus erythematosus.
    Dermatology (Basel, Switzerland), 1994, Volume: 189, Issue:4

    Topics: Adult; Aged; Chloroquine; Drug Combinations; Drug Tolerance; Female; Humans; Hydroxychloroquine; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Male; Middle Aged; Quinacrine; Vision Disorders

1994
Effects of vesicular acetylcholine uptake blockers on frequency augmentation-potentiation in frog neuromuscular transmission.
    Neuroscience, 1994, Volume: 59, Issue:2

    Topics: Acetylcholine; Animals; Antidepressive Agents; Azepines; Chloroquine; Ethacridine; Evoked Potentials; In Vitro Techniques; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Piperidines; Pyrilamine; Quinacrine; Ranidae; Regression Analysis; Synaptic Transmission

1994
The effects of chronic administration of chloroquine and quinacrine on the response of normal and denervated smooth muscle to agonist drugs.
    Physiology & behavior, 1993, Volume: 54, Issue:2

    Topics: Acetylcholine; Age Factors; Animals; Atropine; Chickens; Chloroquine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Male; Muscle, Smooth; Neurotransmitter Agents; Norepinephrine; Potassium Chloride; Pyrilamine; Quinacrine; Serotonin; Synaptic Transmission

1993
Enhanced growth of mammary adenocarcinoma in rats by chloroquine and quinacrine.
    Cancer letters, 1994, Jan-30, Volume: 76, Issue:2-3

    Topics: Adenocarcinoma; Animals; Body Weight; Cell Division; Chloroquine; Dinoprostone; Erythrocytes; Female; Glutathione; Mammary Neoplasms, Experimental; Neoplasm Transplantation; Oxygen; Quinacrine; Rats; Rats, Inbred F344; Riboflavin; Riboflavin Deficiency; Stimulation, Chemical; Stress, Physiological

1994
Differential binding of the enantiomers of chloroquine and quinacrine to polynucleotides: implications for stereoselective metabolism.
    Biopolymers, 1993, Volume: 33, Issue:6

    Topics: Chloroquine; Polynucleotides; Quinacrine; Stereoisomerism

1993
Cytotoxic activity of lutropin-gelonin conjugate in mouse Leydig tumor cells: potentiation of the hormonotoxin activity by different drugs.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:1

    Topics: Animals; Antineoplastic Agents; Chloroquine; Drug Screening Assays, Antitumor; Drug Synergism; Leydig Cell Tumor; Leydig Cells; Luteinizing Hormone; Male; Mice; Monensin; Neoplasm Proteins; Plant Proteins; Progesterone; Protein Synthesis Inhibitors; Quinacrine; Receptors, LH; Ribosome Inactivating Proteins, Type 1; Testicular Neoplasms; Tumor Cells, Cultured; Verapamil

1993
The antimalarials quinacrine and chloroquine induce weak lysosomal storage of sulphated glycosaminoglycans in cell culture and in vivo.
    Toxicology, 1996, Jun-17, Volume: 110, Issue:1-3

    Topics: Animals; Anti-Inflammatory Agents; Antimalarials; beta-N-Acetylhexosaminidases; Cattle; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Female; Fibroblasts; Glycosaminoglycans; Histocytochemistry; Lipidoses; Liver; Lysosomes; Microscopy, Electron; Microscopy, Fluorescence; Mucopolysaccharidoses; Quinacrine; Rats; Rats, Wistar; Structure-Activity Relationship; Sulfates; Tilorone

1996
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
    Biochemical and biophysical research communications, 1996, Sep-04, Volume: 226, Issue:1

    Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication

1996
Activity of pyronaridine and mepacrine against twelve strains of Plasmodium falciparum in vitro.
    The Journal of antimicrobial chemotherapy, 1996, Volume: 37, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Mefloquine; Naphthyridines; Plasmodium falciparum; Quinacrine; Quinine

1996
Xanthones as antimalarial agents; studies of a possible mode of action.
    FEBS letters, 1997, Jun-02, Volume: 409, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Heme; Humans; Plasmodium falciparum; Polymers; Primaquine; Quinacrine; Structure-Activity Relationship; Xanthenes; Xanthones

1997
Opposing effects of quinacrine and chloroquine on the development of TA3 transplanted tumors in mice.
    Biological research, 1995, Volume: 28, Issue:3

    Topics: Animals; Antineoplastic Agents; Cell Division; Chloroquine; Male; Mice; Neoplasm Transplantation; Quinacrine

1995
Interaction of local anaesthetics with histamine H1 receptors in guinea-pig ileum.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: Anesthetics, Local; Animals; Binding, Competitive; Chloroquine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Isotope Labeling; Male; Muscle Contraction; Muscle, Smooth; Procaine; Pyrilamine; Quinacrine; Receptors, Histamine H1; Structure-Activity Relationship; Tetracaine

1997
Lysosomotropic agents ameliorate macrophage dysfunction following the phagocytosis of IgG-coated erythrocytes: a role for lipid peroxidation.
    Inflammation, 1997, Volume: 21, Issue:6

    Topics: Ammonium Chloride; Animals; Chloroquine; Erythrocytes; Immunoglobulin G; Lipid Peroxidation; Macrophage Activation; Macrophages, Peritoneal; Methylamines; Phagocytosis; Quinacrine; Rats; Rats, Sprague-Dawley

1997
CpG-oligodeoxynucleotide supports growth of IL-6-dependent 7TD1 murine hybridoma cells.
    Life sciences, 1998, Volume: 62, Issue:1

    Topics: Animals; Antimalarials; Cell Count; Cell Division; Chloroquine; Dose-Response Relationship, Drug; Hybridomas; Interleukin-6; Mice; Oligodeoxyribonucleotides; Quinacrine

1998
Antimalarial drugs inhibit phospholipase A2 activation and induction of interleukin 1beta and tumor necrosis factor alpha in macrophages: implications for their mode of action in rheumatoid arthritis.
    General pharmacology, 1998, Volume: 30, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Eicosanoids; Female; Interleukin-1; Macrophages, Peritoneal; Mice; Phospholipases A; Phospholipases A2; Quinacrine; Tumor Necrosis Factor-alpha

1998
Antagonism of immunostimulatory CpG-oligodeoxynucleotides by quinacrine, chloroquine, and structurally related compounds.
    Journal of immunology (Baltimore, Md. : 1950), 1998, Feb-01, Volume: 160, Issue:3

    Topics: Acids; Adjuvants, Immunologic; Animals; Apoptosis; Binding, Competitive; Biological Transport; Cell Division; Cell Line; Chloroquine; CpG Islands; Drug Resistance, Multiple; Humans; Immunosuppressive Agents; Intercalating Agents; Interleukin-6; Kinetics; Leukocytes, Mononuclear; Lipopolysaccharides; Mice; Oligodeoxyribonucleotides; Quinacrine; Structure-Activity Relationship; Thionucleotides

1998
[Combination of antimalarial drugs mepacrine and chloroquine in therapy refractory cutaneous lupus erythematosus].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 2000, Volume: 51, Issue:2

    Topics: Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Facial Dermatoses; Female; Humans; Lupus Erythematosus, Discoid; Quinacrine

2000
Conditional lethality of the diprotic weak bases chloroquine and quinacrine against Cryptococcus neoformans.
    The Journal of infectious diseases, 2000, Volume: 182, Issue:1

    Topics: Anti-Bacterial Agents; Antifungal Agents; Cell Division; Chloroquine; Cryptococcus neoformans; Drug Combinations; Enzyme Inhibitors; Macrolides; Microbial Sensitivity Tests; Quinacrine

2000
Reduced inflammatory response to plasmid DNA vectors by elimination and inhibition of immunostimulatory CpG motifs.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2000, Volume: 1, Issue:3

    Topics: Administration, Intranasal; Animals; Antimalarials; Bronchoalveolar Lavage Fluid; Chloroquine; CpG Islands; Cytokines; DNA, Bacterial; Gene Transfer Techniques; Genetic Vectors; Inflammation; Interleukin-12; Lipids; Lung; Mice; Mice, Inbred BALB C; Mutagenesis, Site-Directed; Plasmids; Quinacrine; Sequence Deletion; Spleen

2000
Blastocystis hominis: neutral red supravital staining and its application to in vitro drug sensitivity testing.
    Parasitology research, 2000, Volume: 86, Issue:7

    Topics: Amebicides; Animals; Blastocystis hominis; Chloroquine; Coloring Agents; Humans; Metronidazole; Neutral Red; Nitro Compounds; Parasitic Sensitivity Tests; Paromomycin; Quinacrine; Staining and Labeling; Sulfamethoxazole; Tetracycline; Thiazoles; Trimethoprim

2000
The antimalarials quinacrine and chloroquine potentiate the transplacental carcinogenic effect of ethylnitrosourea on ependymal cells.
    Brain tumor pathology, 2001, Volume: 18, Issue:2

    Topics: Animals; Antimalarials; Brain Neoplasms; Carcinogens; Chloroquine; Drug Synergism; Ependyma; Ependymoma; Ethylnitrosourea; Female; Glial Fibrillary Acidic Protein; Immunoenzyme Techniques; Male; Pregnancy; Prenatal Exposure Delayed Effects; Quinacrine; Rats; Rats, Wistar; Spinal Cord Neoplasms; Synaptophysin

2001
The effect of chloroquine, quinacrine, and metronidazole on both soybean plants and soil microbiota.
    Chemosphere, 2002, Volume: 46, Issue:7

    Topics: Animals; Anti-Bacterial Agents; Antimalarials; Bacteria; Chloroquine; Eukaryota; Glycine max; Metronidazole; Plant Roots; Population Dynamics; Quinacrine; Soil Microbiology

2002
[The treatment of giardiasis; nivaquine or quinacrine].
    Archives des maladies de l'appareil digestif et des maladies de la nutrition, 1952, Volume: 41, Issue:4

    Topics: Chloroquine; Giardiasis; Quinacrine; Quinolines

1952
Enteritis due to flagellata in children.
    Harefuah, 1952, Apr-15, Volume: 42, Issue:8

    Topics: Child; Chloroquine; Enteritis; Giardiasis; Humans; Infant; Quinacrine

1952
[Case of malaria due to Plasmodium falciparum resistant to quinacrine and to quinine and treated with nivaquine].
    La Medicina colonial, 1952, Volume: 20, Issue:5

    Topics: Chloroquine; Humans; Malaria; Plasmodium falciparum; Quinacrine; Quinine

1952
Screening of antimalarials against P. gallinaceum in chicks.
    Indian journal of malariology, 1952, Volume: 6, Issue:2

    Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Chickens; Chloroquine; Malaria; Proguanil; Quinacrine; Quinine; Sulfadiazine

1952
[Superiority of premaline over quinacrine and nivaquine in the treatment of lambliasis].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1953, Volume: 46, Issue:1

    Topics: Aminoquinolines; Chloroquine; Giardiasis; Humans; Quinacrine; Quinolines

1953
Atabrine and chloroquine in the treatment of chronic discoid lupus erythematosus.
    Stanford medical bulletin, 1953, Volume: 11, Issue:3

    Topics: Chloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1953
Light sensitive eruptions treated with atabrine and chloroquine.
    The Journal of investigative dermatology, 1954, Volume: 22, Issue:1

    Topics: Chloroquine; Dermatitis; Light; Quinacrine

1954
The use of chloroquine diphosphate (aralen) and quinacrine (atabrine) hydrochloride in the prevention of polymorphorus light eruptions.
    The Journal of investigative dermatology, 1954, Volume: 22, Issue:2

    Topics: Biomedical Research; Chloroquine; Light; Lupus Erythematosus, Systemic; Quinacrine; Sunlight

1954
Synthetic antimalarial drugs in chronic discoid lupus erythematosus and light eruptions.
    A.M.A. archives of dermatology and syphilology, 1954, Volume: 70, Issue:1

    Topics: Antimalarials; Chloroquine; Light; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases; Sunlight

1954
[Serological research in chronic inflammatory rheumatism; study of antistreptolysin O].
    Revue du rhumatisme et des maladies osteo-articulaires, 1954, Volume: 21, Issue:5

    Topics: Antistreptolysin; Arthritis, Rheumatoid; Chloroquine; Chronic Disease; Humans; Quinacrine; Research; Rheumatic Fever

1954
[Atebrine and chloroquine/resochin therapy of lupus erythematous and dermatoses due to photosensitivity].
    Klinische Wochenschrift, 1954, Oct-01, Volume: 32, Issue:37-38

    Topics: Chloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases

1954
[Atebrin and resochin treatment in progressive chronic polyarthritis].
    Die Medizinische, 1955, Aug-06, Issue:31-32

    Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine

1955
Studies on the treatment of Opisthorchis viverrini in human infections with quinacrine hydrochloride and chloroquine phosphate.
    The American journal of tropical medicine and hygiene, 1955, Volume: 4, Issue:6

    Topics: Animals; Chloroquine; Infections; Opisthorchis; Quinacrine

1955
Treatment on malaria with single doses of mepacrine, chloroquine and amodiaquin.
    The West African medical journal, 1955, Volume: 4, Issue:3

    Topics: Amodiaquine; Antimalarials; Chloroquine; Humans; Malaria; Quinacrine

1955
Mepacrine and chloroquine in the treatment of rosacea.
    The British journal of dermatology, 1955, Volume: 67, Issue:12

    Topics: Chloroquine; Humans; Quinacrine; Rosacea

1955
[Comparative study of the effect of quinacrine, nivaquine B and C on giardiasis].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1955, Volume: 48, Issue:3

    Topics: Chloroquine; Giardiasis; Humans; Quinacrine; Quinolines

1955
[Antimalarial drugs in therapy of chronic evolutive polyarthritis].
    Revista espanola de reumatismo y enfermedades osteoarticulares, 1955, Volume: 6, Issue:2

    Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine

1955
[Lupus erythematosus, etiology, pathogenesis and therapy].
    Munchener medizinische Wochenschrift (1950), 1956, Mar-09, Volume: 98, Issue:10

    Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine

1956
[Reaction of the human skin to ultraviolet rays. 10. Effects of atebrin and resochin on skin sensitivity].
    Zeitschrift fur Haut- und Geschlechtskrankheiten, 1957, Jan-01, Volume: 22, Issue:1

    Topics: Chloroquine; Humans; Quinacrine; Skin; Skin Physiological Phenomena; Sunlight; Ultraviolet Rays

1957
Systemic lupus erythematosus; a report on twelve cases treated with quinacrine (atabrine) and chloroquine (aralen).
    Annals of the rheumatic diseases, 1957, Volume: 16, Issue:1

    Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine

1957
The efficiency of local application of chloroquine and mepacrine in preventing the effects of ultraviolet rays on human skin.
    Acta dermato-venereologica, 1957, Volume: 37, Issue:1

    Topics: Chloroquine; Humans; Quinacrine; Skin; Ultraviolet Rays

1957
Treatment of lupus erythematosus with chloroquine; therapeutic results and a comparison of the value of chloroquine and mepacrine.
    The British journal of dermatology, 1957, Volume: 69, Issue:5

    Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1957
The treatment of lupus erythematosus and lymphocytic infiltration of the skin with A.P.A. 5533.
    The British journal of dermatology, 1957, Volume: 69, Issue:5

    Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin; Skin Diseases

1957
[Quinacrine & chloroquine in asthma therapy].
    Nordisk medicin, 1957, Oct-03, Volume: 58, Issue:40

    Topics: Asthma; Chloroquine; Disease; Peritoneal Diseases; Peritoneum; Quinacrine

1957
[Chloroquine therapy of lupus erythematosus; comparative effectivity of chloroquine and mepacrine].
    Ugeskrift for laeger, 1957, Oct-17, Volume: 119, Issue:42

    Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Quinacrine

1957
Treatment of chronic lupus erythematosus: effectiveness of plaquenil and APA (Aralen 65 mg., plaquenil 50 mg., Atabrine 25 mg.) as compared with Aralen, with observations on side-reactions and toxicity; report and presentation of unusual cases.
    A.M.A. archives of dermatology, 1958, Volume: 77, Issue:4

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1958
Treatment of rheumatoid arthritis with quinacrine and chloroquine.
    Acta rheumatologica Scandinavica, 1958, Volume: 4, Issue:1

    Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine

1958
[Experimental malaria: Plasmodium berghei].
    La Medicina tropical, 1958, Volume: 31, Issue:2

    Topics: Chloroquine; Malaria; Plasmodium berghei; Quinacrine; Quinine

1958
[Experimental & clinical studies on the mechanism of action of atabrine & resochin in chronic lupus erythematosus].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 1958, Volume: 9, Issue:5

    Topics: Biomedical Research; Chloroquine; Lupus Erythematosus, Systemic; Quinacrine

1958
[Atabrine and resohine therapy of lupus erythematosus].
    Radovi Medicinskog faculteta u Zagrebu, 1957, Volume: 3

    Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine

1957
[Long term treatment of rheumatoid arthritis with mepacrine & chloroquine].
    Ugeskrift for laeger, 1958, Jun-19, Volume: 120, Issue:25

    Topics: Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Long-Term Care; Quinacrine

1958
Triquin in the treatment of discoid lupus erythematosus and light sensitive eruptions.
    Bulletin of the School of Medicine (Baltimore, Md.), 1958, Volume: 43, Issue:4

    Topics: Chloroquine; Exanthema; Humans; Light; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases

1958
Lupus erythematosus treated with a combination of quinacrine, hydroxychloroquine and chloroquine.
    The New England journal of medicine, 1959, Jan-08, Volume: 260, Issue:2

    Topics: Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1959
Initial clinical trial of the nitrogen mustard analogues of chloroquine and quinacrine; a preliminary report.
    Annals of the New York Academy of Sciences, 1958, Apr-24, Volume: 68, Issue:3

    Topics: Chloroquine; Humans; Mechlorethamine; Nitrogen Mustard Compounds; Quinacrine

1958
The use of triquin in the treatment of discoid lupus erythematosus and some other skin conditions.
    A.M.A. archives of dermatology, 1959, Volume: 79, Issue:6

    Topics: Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine; Skin Diseases

1959
[Observations on quinacrine & chloroquine in the treatment of petit mal; preliminary report].
    La Semana medica, 1959, Jan-15, Volume: 114, Issue:3

    Topics: Chloroquine; Epilepsy; Epilepsy, Absence; Quinacrine

1959
Successful treatment of hepatic and splenic amebic abscesses with atabrine after failure of emetine, chloroquine and terramycin.
    The Journal of the Egyptian Medical Association, 1960, Volume: 43

    Topics: Amebiasis; Chloroquine; Disease; Dysentery, Amebic; Emetine; Humans; Liver Abscess; Oxytetracycline; Quinacrine; Spleen

1960
Single dose treatment of malaria with amodiaquin chloroquine and mepacrine in a semi-immune poplation.
    East African medical journal, 1960, Volume: 37

    Topics: Amodiaquine; Antimalarials; Chloroquine; Humans; Malaria; Quinacrine

1960
Action of quinine, qunidine mepacrine and chloroquine on the skeletal muscle.
    The Indian journal of medical research, 1960, Volume: 48

    Topics: Antimalarials; Chloroquine; Humans; Muscle, Skeletal; Muscles; Quinacrine; Quinine

1960
[Discolorations of atabrine and resochin solutions by autogenous, reducing substances after UV irradiation].
    Naunyn-Schmiedebergs Archiv fur experimentelle Pathologie und Pharmakologie, 1960, Volume: 238

    Topics: Chloroquine; Quinacrine; Solutions; Ultraviolet Rays

1960
[Modification of Rh antigen-antibody reactions].
    Archiv fur Gynakologie, 1962, Volume: 197

    Topics: Antigen-Antibody Reactions; Aspirin; Chloroquine; Humans; Phenylbutazone; Quinacrine

1962
Reaction between DNA and quinacrine and other antimalarials.
    The Journal of laboratory and clinical medicine, 1962, Volume: 60

    Topics: Antimalarials; Chloroquine; DNA; Quinacrine; Quinidine; Quinine

1962
[Skin symptoms caused by synthetic antimalarials].
    Dermatologica, 1963, Volume: 126

    Topics: Antimalarials; Chloroquine; Drug Eruptions; Humans; Quinacrine

1963
[Treatment of discoid lupus erythematosus, polymorphous photodermatosis and rosacea with Triquin--a combination of 3 anti-malarials].
    Svenska lakartidningen, 1962, Oct-04, Volume: 59

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Photosensitivity Disorders; Quinacrine; Rosacea

1962
In vivo and in vitro effects of antimalarials on Histoplasma capsulatum.
    Antibiotics & chemotherapy (Northfield, Ill.), 1962, Volume: 12

    Topics: Amodiaquine; Antimalarials; Chloroquine; Histoplasma; Humans; In Vitro Techniques; Primaquine; Quinacrine

1962
[Therapeutic use of 22/360 (Collagenan) during various collagen diseases].
    La semaine des hopitaux : organe fonde par l'Association d'enseignement medical des hopitaux de Paris, 1963, Mar-14, Volume: 39

    Topics: 4-Aminobenzoic Acid; Antimalarials; Chloroquine; Collagen Diseases; Drug Combinations; Humans; Pantothenic Acid; Pyridoxine; Quinacrine; Vitamin B Complex

1963
Oral contraceptives. VII. Antimalarials as antifertility agents.
    Indian journal of physiology and pharmacology, 1962, Volume: 6

    Topics: Amodiaquine; Antimalarials; Chloroquine; Contraceptive Agents; Contraceptives, Oral; Female; Humans; Proguanil; Pyrimethamine; Quinacrine

1962
[Report on the use, in the treatment of chronic evolutive polyarthritis, of a drug combining notably 2 synthetic antimalarials].
    Revue du rhumatisme et des maladies osteo-articulaires, 1963, Volume: 30

    Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Humans; Quinacrine

1963
SOLAR URTICARIA.
    Archives of dermatology, 1963, Volume: 88

    Topics: Chloroquine; Dermatitis, Phototoxic; Humans; Photosensitivity Disorders; Porphyrins; Pregnancy; Quinacrine; Toxicology; Urticaria

1963
[ON DARK PIGMENTATIONS DUE TO ATABRINE AND AMODIAQUINE].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 1963, Volume: 14

    Topics: Amodiaquine; Chloroquine; Pigmentation; Pigmentation Disorders; Quinacrine; Toxicology

1963
DRUG RESISTANCE IN PLASMODIUM FALCIPARUM FROM THAILAND.
    The American journal of tropical medicine and hygiene, 1963, Volume: 12

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand

1963
PIGMENTATION FROM ANTIMALARIAL THERAPY. ITS POSSIBLE RELATIONSHIP TO THE OCULAR LESIONS.
    Archives of dermatology, 1963, Volume: 88

    Topics: Antimalarials; Arthritis; Arthritis, Rheumatoid; Chloroquine; Cornea; Eye; Eye Manifestations; Histocytochemistry; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Photomicrography; Pigmentation; Pigmentation Disorders; Quinacrine; Retina; Toxicology

1963
LUPUS ERYTHEMATOSUS--A CLINICAL QUIZ. A SERIES OF DIAGNOSTIC AND THERAPEUTIC PROBLEMS.
    Skin, 1963, Volume: 2

    Topics: Chloroquine; Diagnosis; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1963
POLYMORPHOUS LIGHT ERUPTION. A TEN-YEAR FOLLOW-UP AND EVALUATION.
    Archives of dermatology, 1963, Volume: 88

    Topics: Chloroquine; Dermatitis, Phototoxic; Follow-Up Studies; Humans; Hydroxychloroquine; Lupus Erythematosus, Systemic; Photosensitivity Disorders; Prurigo; Quinacrine; Seasons; Sunlight

1963
ANTIMALARIAL DRUGS ON THE AUTOMATICITY OF SINO-AURICULAR AND ATRIO-VENTRICULAR NODES.
    The Indian journal of medical research, 1963, Volume: 51

    Topics: Administration, Intravenous; Amodiaquine; Animals; Anti-Arrhythmia Agents; Antimalarials; Atrioventricular Node; Atropine; Chloroquine; Dogs; Heart Conduction System; Humans; Hydroxychloroquine; Hypotension; Injections, Intravenous; Primaquine; Quinacrine; Quinidine; Research; Statistics as Topic

1963
DRUG-RESISTANT FALCIPARUM MALARIA FROM CAMBODIA AND MALAYA.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1963, Volume: 57

    Topics: Animals; Cambodia; Chloroquine; Culicidae; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Malaria, Falciparum; Malaysia; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine

1963
TOXIC PSYCHOSIS DUE TO QUINARCRINE AND CHLOROQUINE.
    JAMA, 1964, Feb-01, Volume: 187

    Topics: Amebiasis; Chloroquine; Giardiasis; Humans; Psychoses, Substance-Induced; Psychotic Disorders; Quinacrine; Toxicology; Trichomonas Infections

1964
[CHRONIC DISCOID ERYTHEMATOSUS (REPORT ON 69 CASES OVER A PERIOD OF 6 YEARS FROM THE VIEWPOINT OF OPTIMUM THERAPY)].
    Ceskoslovenska dermatologie, 1963, Volume: 38

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Quinacrine

1963
HAEMATOLOGICAL SIDE-EFFECTS OF SOME ANTI-RHEUMATIC DRUGS.
    Annals of the rheumatic diseases, 1963, Volume: 22

    Topics: Aminopyrine; Antirheumatic Agents; Aspirin; Blood Platelets; Chloroquine; Colchicine; Complement Fixation Tests; Drug Hypersensitivity; Gold; Humans; Hydroxychloroquine; Meprobamate; Phenacetin; Phenylbutazone; Probenecid; Purpura; Purpura, Thrombocytopenic; Quinacrine; Rheumatic Diseases; Splenectomy; Toxicology

1963
ANTIHELMINTHIC THERAPY: A SIMPLIFIED APPROACH.
    Southern medical journal, 1964, Volume: 57

    Topics: Amebiasis; Anthelmintics; Ascariasis; Chloroquine; Dysentery, Amebic; Giardiasis; Hookworm Infections; Humans; Oxytetracycline; Quinacrine; Strongyloidiasis; Trichinellosis

1964
ANTIMALARIALS AND OTHER ANTICONVULSANT DRUGS: PREDICTIVE VALIDITY OF LABORATORY TESTS.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1964, Volume: 115

    Topics: Animals; Anticonvulsants; Antimalarials; Chloroquine; Electric Stimulation; Hydroxychloroquine; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Phenytoin; Quinacrine; Research; Seizures

1964
STUDIES ON A STRAIN OF CHLOROQUINE-RESISTANT PLASMODIUM FALCIPARUM FROM THAILAND.
    Bulletin of the World Health Organization, 1964, Volume: 30

    Topics: Amodiaquine; Antimalarials; Asia, Southeastern; Biomedical Research; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Hydroxychloroquine; Malaria; Malaria, Falciparum; Pharmacology; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand

1964
DRUG-RESISTANCE IN FALCIPARUM MALARIA IN SOUTH-EAST ASIA.
    The Medical journal of Malaya, 1964, Volume: 18

    Topics: Adolescent; Asia, Southeastern; Child; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Drug Therapy; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Statistics as Topic; Toxicology

1964
[MODERN ANTHELMINTIC DRUGS].
    Suomen laakarilehti. Finlands lakartidning, 1964, Jun-01, Volume: 19

    Topics: Anthelmintics; Chemical Phenomena; Chemistry; Chloroquine; Diethylcarbamazine; Dithiazanine; Dryopteris; Gentian Violet; Humans; Niclosamide; Piperazines; Pyrvinium Compounds; Quinacrine

1964
ANTIHISTAMINIC ACTION OF ANTIMALARIALS.
    Indian journal of physiology and pharmacology, 1963, Volume: 7

    Topics: Acetylcholine; Animals; Antimalarials; Blood Pressure; Blood Pressure Determination; Capillary Permeability; Chloroquine; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Muscle, Smooth; Pharmacology; Quinacrine; Quinine; Research

1963
[PSORIASIS AND ITS TREATMENT IN THE LIGHT OF A NEW EXPERIENCE].
    Svenska lakartidningen, 1964, Jul-01, Volume: 61

    Topics: Chloroquine; Fluocinolone Acetonide; Humans; Light; Psoriasis; Quinacrine

1964
THE EFFECT OF CERTAIN SUBSTANCES AGAINST ECHINOCOCCUS GRANULOSUS AND TAENIA HYDATIGENA INFECTIONS IN DOGS.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Animals; Anthelmintics; Benzimidazoles; Chloroquine; Dithiazanine; Dog Diseases; Dogs; Echinococcosis; Echinococcus granulosus; England; Fascioliasis; Hexachlorophene; Hexylresorcinol; Iodoquinol; Niclosamide; Piperazines; Protozoan Infections; Quinacrine; Taenia; Thiabendazole

1964
[APROPOS OF LAMBLIASIS IN CHILDHOOD].
    Bratislavske lekarske listy, 1964, Aug-15, Volume: 44

    Topics: Acridines; Adolescent; Child; Chloroquine; Drug Therapy; Giardiasis; Humans; Quinacrine; Quinolines

1964
CHILBLAIN LUPUS ERYTHEMATOSUS.
    Proceedings of the Royal Society of Medicine, 1964, Volume: 57

    Topics: Chilblains; Chloroquine; Fluocinolone Acetonide; Frostbite; Humans; Hydroxychloroquine; Hypothyroidism; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Niacinamide; Quinacrine; Telangiectasis; Triamcinolone

1964
THE ABSENCE OF ANTICONVULSANT PROPERTIES OF QUINACRINE AND CHLOROQUINE IN MICE.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1964, Volume: 116

    Topics: Anticonvulsants; Chloroquine; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Quinacrine; Research; Seizures; Toxicology

1964
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology

1964
ALIMENTARY HYPERSENSITIVITY INDUCED BY GIARDIA LAMBLIA; REPORT OF A CASE OF ACUTE MEAT INTOLERANCE.
    Annals of internal medicine, 1965, Volume: 62

    Topics: Abdomen; Abdomen, Acute; Chloroquine; Drug Therapy; Food Hypersensitivity; Giardia lamblia; Giardiasis; Humans; Meat; Pathology; Quinacrine

1965
PLEUROPULMONARY AMEBIASIS. CLINICAL ANALYSIS OF 64 CASES.
    Chinese medical journal (Peking, China : 1932), 1965, Volume: 84

    Topics: Amebiasis; Chloroquine; Diagnosis, Differential; Drainage; Drug Therapy; Emetine; Empyema; Humans; Liver Abscess; Liver Abscess, Amebic; Lung Abscess; Lung Diseases, Parasitic; Pathology; Pleural Effusion; Pleurisy; Prognosis; Quinacrine; Radiography, Thoracic

1965
[ALLERGIC CONTACT ECZEMA CAUSED BY RESOCHIN].
    Dermatologica, 1965, Volume: 130

    Topics: Chloroquine; Dermatitis; Dermatitis, Allergic Contact; Dermatitis, Contact; Quinacrine; Skin Tests; Toxicology

1965
Treatment of chronic lupus erythematosus with atabrine and chloroquine.
    The Illinois medical journal, 1955, Volume: 107, Issue:6

    Topics: Chloroquine; Lupus Erythematosus, Systemic; Quinacrine

1955
[Recent experience in the treatment of erythematodes chronicus discoides with atebrin and resochin, with special reference to local and combined therapeutic methods].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 1955, Volume: 6, Issue:5

    Topics: Chloroquine; Combined Modality Therapy; Erythema; Humans; Quinacrine

1955
[Treatment of chronic lupus erythematosus with synthetic antimalarials: quinacrine and chloroquine].
    Actas dermo-sifiliograficas, 1955, Volume: 46, Issue:6

    Topics: Antimalarials; Chloroquine; Humans; Lupus Erythematosus, Systemic; Quinacrine

1955
Clinical findings for the treatment of Mucha-Habermann disease (parapsoriasis varioliformis) with acridine and chinoline derivatives.
    Dermatologica, 1959, Volume: 118

    Topics: Acridines; Chloroquine; Humans; Parapsoriasis; Pityriasis Lichenoides; Quinacrine

1959
Evaluation of synthetic anti-malarial drugs in children from a hyperendemic area in West Africa.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1951, Volume: 44, Issue:5

    Topics: Africa, Western; Antimalarials; Child; Chloroquine; Humans; Malaria; Quinacrine

1951
Chemotherapy of amebic hepatitis in hamsters with emetine, chloroquine, amodiaquin (camoquin), quinacrine and other drugs.
    The American journal of tropical medicine and hygiene, 1951, Volume: 31, Issue:6

    Topics: Amebiasis; Amodiaquine; Chloroquine; Dysentery, Amebic; Emetine; Hepatitis; Liver Diseases; Quinacrine

1951
Inhibitors of the K+(Na+)/H+ exchanger of human red blood cells.
    Bioelectrochemistry (Amsterdam, Netherlands), 2004, Volume: 62, Issue:2

    Topics: Chloroquine; Dose-Response Relationship, Drug; Erythrocytes; Humans; Osmolar Concentration; Potassium; Potassium-Hydrogen Antiporters; Quinacrine; Sodium-Hydrogen Exchangers

2004
Kinetic mechanism of quinone oxidoreductase 2 and its inhibition by the antimalarial quinolines.
    Biochemistry, 2004, Apr-20, Volume: 43, Issue:15

    Topics: Antimalarials; Binding, Competitive; Chloroquine; Copper; Humans; Kinetics; Niacinamide; Oxidation-Reduction; Primaquine; Quinacrine; Quinolines; Quinone Reductases; Recombinant Proteins; Spectrophotometry; Substrate Specificity; Zinc

2004
Toll-like receptor 9 binds single-stranded CpG-DNA in a sequence- and pH-dependent manner.
    European journal of immunology, 2004, Volume: 34, Issue:9

    Topics: Amino Acid Sequence; Binding Sites; Cell Line; Chloroquine; CpG Islands; DNA, Single-Stranded; Humans; Hydrogen-Ion Concentration; Membrane Glycoproteins; Molecular Sequence Data; Quinacrine; Receptors, Cell Surface; Toll-Like Receptor 2; Toll-Like Receptor 9; Toll-Like Receptors

2004
The sensitivities of yeast strains deficient in PDR ABC transporters, to quinoline-ring antimalarial drugs.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:6

    Topics: Antimalarials; ATP-Binding Cassette Transporters; Chloroquine; Cycloheximide; Drug Resistance, Multiple, Fungal; Gene Deletion; Genes, Fungal; Mefloquine; Mutation; Quinacrine; Quinidine; Quinine; Saccharomyces cerevisiae; Transcription, Genetic

2004
Involvement of the nonhomologous region of subunit A of the yeast V-ATPase in coupling and in vivo dissociation.
    The Journal of biological chemistry, 2004, Nov-19, Volume: 279, Issue:47

    Topics: Adenosine Triphosphate; Blotting, Western; Catalysis; Chloroquine; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Epitopes; Escherichia coli; Genetic Vectors; Glucose; Hydrogen-Ion Concentration; Immunoprecipitation; Mutation; Plasmids; Protein Binding; Protein Structure, Tertiary; Protons; Quinacrine; Saccharomyces cerevisiae; Time Factors; Vacuolar Proton-Translocating ATPases; Vacuoles

2004
Chloroquine, proguanil, mepacrine and quinine in the treatment of malaria caused by Plasmodium falciparum.
    Annals of tropical medicine and parasitology, 1949, Volume: 43, Issue:3-4

    Topics: Chloroquine; Humans; Malaria; Plasmodium falciparum; Proguanil; Quinacrine; Quinine

1949
[Systemic lupus erythematosus therapy. Antimalarials in inflammatory diseases].
    Revista clinica espanola, 2004, Volume: 204, Issue:11

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Lupus Erythematosus, Systemic; Quinacrine

2004
Anthrax toxin protective antigen: inhibition of channel function by chloroquine and related compounds and study of binding kinetics using the current noise analysis.
    Biophysical journal, 2005, Volume: 88, Issue:3

    Topics: Algorithms; Antigens, Bacterial; Bacterial Toxins; Binding Sites; Chloroquine; Fluphenazine; Ion Channel Gating; Ion Channels; Lipid Bilayers; Permeability; Quinacrine; Recombinant Proteins

2005
Quinacrine but not chloroquine inhibits PMA induced upregulation of matrix metalloproteinases in leukocytes: quinacrine acts at the transcriptional level through a PLA2-independent mechanism.
    The Journal of rheumatology, 2006, Volume: 33, Issue:3

    Topics: Antigens, Human Platelet; Antirheumatic Agents; Cell Survival; Chloroquine; Dose-Response Relationship, Drug; Gene Expression Regulation, Enzymologic; Humans; Leukocytes, Mononuclear; Matrix Metalloproteinases; Phorbol Esters; Quinacrine; RNA, Messenger; Transcription, Genetic; Up-Regulation

2006
CpG-induced tyrosine phosphorylation occurs via a TLR9-independent mechanism and is required for cytokine secretion.
    The Journal of cell biology, 2006, Mar-27, Volume: 172, Issue:7

    Topics: Actin Cytoskeleton; Adaptor Proteins, Signal Transducing; Androstadienes; Animals; Antigens, CD; Cell Adhesion; Cell Line, Tumor; Cell Membrane; Chloroquine; CpG Islands; Cytokines; Cytoskeleton; Dendritic Cells; Humans; I-kappa B Proteins; Interferon-alpha; Interleukin-6; Intracellular Signaling Peptides and Proteins; Macrophages; Mice; Mice, Knockout; Models, Biological; Monocytes; Myeloid Differentiation Factor 88; NF-KappaB Inhibitor alpha; Oligodeoxyribonucleotides; Phosphorylation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-hck; Pyrazoles; Pyrimidines; Quinacrine; RNA, Small Interfering; src-Family Kinases; Syk Kinase; Toll-Like Receptor 9; Tyrosine; Wortmannin

2006
THE INFLUENCE OF ORALLY ADMINISTERED ALKALI AND ACID ON THE RENAL EXCRETION OF QUINACRINE, CHLOROQUINE AND SANTOQUINE.
    The Journal of clinical investigation, 1947, Volume: 26, Issue:6

    Topics: Alkalies; Chloroquine; Fluids and Secretions; Humans; Quinacrine; Renal Elimination

1947
Comparison of chloroquine, quinacrine (atabrine) and quinine in the treatment of acute attacks of sporozoite-induced vivax malaria, Chesson strain.
    The Journal of clinical investigation, 1948, Volume: 27, Issue:3 Pt1

    Topics: Animals; Behavior, Animal; Chloroquine; Humans; Malaria, Vivax; Quinacrine; Quinine; Sporozoites

1948
The efficacy of chloroquine, quinacrine, quinine and totaquine in the treatment of Plasmodium malariae infections (quartan malaria).
    The American journal of tropical medicine and hygiene, 1948, Volume: 28, Issue:1

    Topics: Chloroquine; Humans; Malaria; Plasmodium malariae; Quinacrine; Quinine

1948
Effect of acidosis and anoxia on the concentration of quinacrine and chloroquine in blood.
    The Journal of pharmacology and experimental therapeutics, 1948, Volume: 92, Issue:3

    Topics: Acidosis; Chloroquine; Hypoxia; Quinacrine

1948
Chloroquine-induced autophagic vacuole accumulation and cell death in glioma cells is p53 independent.
    Neuro-oncology, 2010, Volume: 12, Issue:5

    Topics: Antineoplastic Agents; Autophagy; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Chloroquine; Glioma; Humans; Immunohistochemistry; Mefloquine; Quinacrine; Tumor Suppressor Protein p53; Vacuoles

2010
Resistance to chloroquine unhinges vivax malaria therapeutics.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:5

    Topics: Aminoquinolines; Antimalarials; Chloroquine; Drug Interactions; Drug Resistance; Humans; Malaria, Vivax; Plasmodium vivax; Primaquine; Quinacrine

2011
Mechanism of endosomal TLR inhibition by antimalarial drugs and imidazoquinolines.
    Journal of immunology (Baltimore, Md. : 1950), 2011, Apr-15, Volume: 186, Issue:8

    Topics: Animals; Antimalarials; Binding, Competitive; Cell Line; Cells, Cultured; Chloroquine; Culture Media; Cytokines; Endosomes; HEK293 Cells; Humans; Hydrogen-Ion Concentration; Imidazoles; Nucleic Acids; Quinacrine; Quinolines; Serum; Toll-Like Receptor 3; Toll-Like Receptor 7; Toll-Like Receptor 8; Toll-Like Receptor 9; Toll-Like Receptors; Transfection

2011
2,4-diarylthiazole antiprion compounds as a novel structural class of antimalarial leads.
    Bioorganic & medicinal chemistry letters, 2011, Jun-15, Volume: 21, Issue:12

    Topics: Antimalarials; Chloroquine; Mefloquine; Molecular Structure; Plasmodium falciparum; Prions; Quinacrine; Structure-Activity Relationship; Thiazoles

2011
N-cinnamoylation of antimalarial classics: quinacrine analogues with decreased toxicity and dual-stage activity.
    ChemMedChem, 2014, Volume: 9, Issue:2

    Topics: Antimalarials; Cell Line; Chloroquine; Drug Design; Drug Resistance; Humans; Malaria; Plasmodium berghei; Plasmodium falciparum; Quinacrine

2014
Suppressive action of mepacrine, aphacrine, chloroquin, camoquin and proguanil against P. knowlesi in S. rhesus monkeys.
    Indian journal of malariology, 1950, Volume: 4, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Humans; Macaca mulatta; Malaria; Proguanil; Quinacrine

1950
Synthesis of improved lysomotropic autophagy inhibitors.
    Journal of medicinal chemistry, 2015, Apr-09, Volume: 58, Issue:7

    Topics: Antineoplastic Agents; Autophagy; Cell Line; Cell Survival; Chemistry Techniques, Synthetic; Chloroquine; Drug Evaluation, Preclinical; Humans; Lysosomes; Microtubule-Associated Proteins; Quinacrine; Structure-Activity Relationship

2015
N-Cinnamoylation of Antimalarial Classics: Effects of Using Acyl Groups Other than Cinnamoyl toward Dual-Stage Antimalarials.
    ChemMedChem, 2015, Volume: 10, Issue:8

    Topics: Antimalarials; Cell Survival; Chloroquine; Cinnamates; Hep G2 Cells; Humans; Life Cycle Stages; Plasmodium berghei; Plasmodium falciparum; Quinacrine; Structure-Activity Relationship

2015
Unilateral unique Lupus tumidus: pathogenetic mystery and diagnostic problem.
    Wiener medizinische Wochenschrift (1946), 2016, Volume: 166, Issue:7-8

    Topics: Adrenal Cortex Hormones; Adult; Azathioprine; Biopsy; Chloroquine; Combined Modality Therapy; Dapsone; Diagnosis, Differential; Humans; Hydroxychloroquine; Lasers, Dye; Lupus Erythematosus, Discoid; Male; Ointments; Quinacrine; Skin; Sunscreening Agents; Tacrolimus

2016
Chloroquine derivatives block the translocation pores and inhibit cellular entry of Clostridium botulinum C2 toxin and Bacillus anthracis lethal toxin.
    Archives of toxicology, 2017, Volume: 91, Issue:3

    Topics: Antigens, Bacterial; Bacterial Toxins; Biological Transport; Botulinum Toxins; Cell Membrane; Chloroquine; Fluphenazine; HeLa Cells; Humans; Lipid Bilayers; Primaquine; Quinacrine

2017
Lysosomotropic cationic drugs induce cytostatic and cytotoxic effects: Role of liposolubility and autophagic flux and antagonism by cholesterol ablation.
    Toxicology and applied pharmacology, 2016, 08-15, Volume: 305

    Topics: Amiodarone; Anticholesteremic Agents; Autophagy; beta-Cyclodextrins; Cell Line, Tumor; Cell Proliferation; Cells, Cultured; Chloroquine; Cholesterol; Cytostatic Agents; Cytotoxins; Human Umbilical Vein Endothelial Cells; Humans; Hydroxychloroquine; Lidocaine; Lovastatin; Lysosomes; Microtubule-Associated Proteins; Poly (ADP-Ribose) Polymerase-1; Procainamide; Quinacrine

2016
Is chloroquine neuromyotoxicity in a patient with refractory discoid lupus erythematosus potentiated by concomitant use of mepacrine?
    Clinical and experimental dermatology, 2018, Volume: 43, Issue:8

    Topics: Antimalarials; Chloroquine; Drug Therapy, Combination; Extremities; Female; Humans; Lupus Erythematosus, Discoid; Middle Aged; Muscle Weakness; Paresthesia; Quinacrine

2018
Comparison of chloroquine-like molecules for lysosomal inhibition and measurement of autophagic flux in the brain.
    Biochemical and biophysical research communications, 2021, 01-01, Volume: 534

    Topics: Animals; Autophagy; Brain; Chloroquine; Drug Evaluation, Preclinical; Female; HeLa Cells; Humans; Lysosomes; Macrolides; Male; Mefloquine; Mice, Inbred C57BL; Mice, Transgenic; Microtubule-Associated Proteins; Promazine; Quinacrine; Trifluoperazine

2021
Efficacy and Tolerability of Quinacrine Monotherapy and Albendazole Plus Chloroquine Combination Therapy in Nitroimidazole-Refractory Giardiasis: A TropNet Study.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2021, 10-20, Volume: 73, Issue:8

    Topics: Albendazole; Antiprotozoal Agents; Chloroquine; Giardia lamblia; Giardiasis; Humans; Nitroimidazoles; Prospective Studies; Quinacrine

2021