chloroquine and podophyllotoxin

chloroquine has been researched along with podophyllotoxin in 119 studies

Research

Studies (119)

TimeframeStudies, this research(%)All Research%
pre-19904 (3.36)18.7374
1990's0 (0.00)18.2507
2000's32 (26.89)29.6817
2010's75 (63.03)24.3611
2020's8 (6.72)2.80

Authors

AuthorsStudies
Croft, SL; Gamenara, D; Grady, S; Heinzen, H; Kendrick, H; Moyna, G; Moyna, P; Ren, H; Yardley, V1
Chibale, K; Croft, SL; Fairlamb, AH; Haupt, H; Kendrick, H; Saravanamuthu, A; Yardley, V1
Croft, SL; del Rayo Camacho, M; Kirby, GC; Marley, D; Phillipson, JD; Warhurst, DC1
Brun, R; Cimanga, K; Dommisse, R; Hostyn, S; Kaiser, M; Lemière, G; Maes, BU; Mátyus, P; Pieters, L; Van Miert, S; Vlietinck, A1
Bauer, H; Davioud-Charvet, E; Krauth-Siegel, RL; Lee, B; Melchers, J; Rattray, L; Ruppert, T; Yardley, V1
Alvarez, A; Atherton, R; Coro, J; Little, S; Pérez, R; Rodríguez, H; Súarez, M; Wharton, H; Yardley, V1
Brun, R; Gilbert, IH; Gonzalez-Pacanowska, D; Johansson, NG; Kaiser, M; Kasinathan, G; Leal, I; Musso-Buendia, A; Nguyen, C; Ruda, GF; Ruiz-Pérez, LM; Sahlberg, BL; Schipani, A1
Croft, SL; Gilbert, IH; Gonzalez-Pacanowska, D; Gros, L; Jimenez, CJ; Little, S; Lorente, SO; Rattray, L; Ruiz-Perez, LM; Wharton, H; Yardley, V1
Ahua, KM; Brun, R; Diallo, D; Hay, AE; Hostettmann, K; Ioset, JR1
Bakunov, SA; Bakunova, SM; Bridges, AS; Brun, R; Hall, JE; Jones, SK; Kumar, EV; Lombardy, RJ; Patrick, DA; Tidwell, RR; Wenzler, T; Zhirnov, O1
Bringmann, G; Brun, R; Kaiser, M; Neumann, S1
Bongard, E; Brown, DM; Loakes, D; Too, K; Vivas, L; Yardley, V1
Brun, R; Gunzenhauser, S; Senn, M; Séquin, U1
Bakunov, SA; Bakunova, SM; Barszcz, T; Brun, R; Hall, JE; Tidwell, RR; Wenzler, T; Werbovetz, KA1
Brun, R; Kaiser, M; Kuettel, S; Perozzo, R; Scapozza, L; Zambon, A1
Bringmann, G; Bruhn, T; Brun, R; Faber, JH; Gampe, CM; Gelhaus, C; Leippe, M; Mikyna, M; Reichert, M; Reichert, Y1
Aldana, I; Bongard, E; Burguete, A; Charnaud, S; Lima, LM; Monge, A; Perez-Silanes, S; Solano, B; Vicente, E; Villar, R; Vivas, L1
Becker, K; Davioud-Charvet, E; Friebolin, W; Furrer, J; Jannack, B; Lanzer, M; Oeser, T; Sanchez, CP; Wenzel, N; Yardley, V1
Arai, C; Brun, R; Ge, JF; Ihara, M; Kaiser, M; Wittlin, S1
Brun, R; Faist, J; Kaiser, M; Saf, R; Schlapper, C; Seebacher, W; Weis, R1
Brun, R; Kehraus, S; König, GM; Krick, A; Pontius, A1
Bakunov, SA; Bakunova, SM; Barszcz, T; Brun, R; Tidwell, RR; Wenzler, T; Werbovetz, KA2
Alp, M; Brun, R; Göker, H; Yildiz, S1
Becker, K; Fritz-Wolf, K; Hu, Y; Rahlfs, S; Sturm, N; Wittlin, S; Zimmermann, H1
Brun, R; Connolly, JD; Efange, SM; Hoye, TR; Makolo, FL; Mbah, JA; McAkam, T; Nelson, DP; Nyongbela, KD; Wirmum, CK; Wittlin, S1
Bakunov, SA; Bakunova, SM; Barszcz, T; Bridges, AS; Brun, R; Jones, SK; Kumar, EV; Ohemeng, KA; Patrick, DA; Tidwell, RR; Wenzler, T; Werbovetz, KA1
Baell, JB; Brun, R; Charman, WN; Fairlamb, AH; Holloway, GA; Kaiser, M; Kostewicz, E; Novello, PM; Parisot, JP; Richardson, J; Street, IP; Watson, KG1
Bakunov, SA; Bakunova, SM; Barzcz, T; Brun, R; Chen, H; Jones, SK; Kumar, EV; Patrick, DA; Tidwell, RR; Wenzler, T; Werbovetz, KA1
Bolognesi, ML; Bongarzone, S; Brun, R; Cavalli, A; Lizzi, F; Luise Krauth-Siegel, R1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Brun, R; Cos, P; Dhooghe, L; Dommisse, R; Hajós, G; Hostyn, S; Kaiser, M; Lemière, G; Maes, BU; Maes, L; Mátyus, P; Nagy, I; Pieters, L; Riedl, Z; Tapolcsányi, P; Van Baelen, G1
Bakunov, SA; Bakunova, SM; Brun, R; Ghebru, M; Tidwell, RR; Wenzler, T; Werbovetz, KA1
Brun, R; Lusvarghi, S; Mazzieri, MR; Pagliero, RJ; Pierini, AB1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Armstrong, T; Baell, JB; Holloway, GA; Novello, PM; Parisot, JP; Street, IP; Thompson, RC; Watson, KG1
Bauer, R; Brun, R; Gachet, MS; Kaiser, M; Kunert, O; Muñoz, RA; Schühly, W1
Amade, P; Cachet, N; Kaiser, M; Regalado, EL; Tasdemir, D; Thomas, OP1
Baumann, K; Bischof, SK; Bringmann, G; Brun, R; Dreher, J; Gulder, T; Kaiser, M; Moll, H; Müller, S; Stich, A; Winter, C1
Brun, R; Carballeira, NM; Herman, R; Kappe, SH; Lauinger, IL; Perozzo, R; Sanabria, D; Tarun, A; Tasdemir, D; Zloh, M1
Bourguet-Kondracki, ML; Copp, BR; Finlayson, R; Harper, JL; Kaiser, M; Page, MJ; Pearce, AN; Webb, VL1
Baragaña, B; Bosch-Navarrete, C; Brun, R; Gilbert, IH; González-Pacanowska, D; Johansson, NG; Kaiser, M; McCarthy, O; Roberts, SM; Sánchez, P; Whittingham, JL; Wilson, KS; Zhou, XX1
Bauer, R; Brun, R; Gachet, MS; Kaiser, M; Keller, W; Kunert, O; Muñoz, RA; Schuehly, W; Zehl, M1
Gerth, K; Jansen, R; Mohr, KI; Müller, R; Okanya, PW1
Charman, SA; Chibale, K; Fakorede, F; Gessner, RK; Gitari, PW; Hudson, A; Kaiser, M; Ndakala, AJ; October, N; Shackleford, DM; White, KL; Yeates, C1
Chibale, K; Feng, TS; Gut, J; Kumar, V; Mahajan, MP; Nasser, S; Raj, R; Rosenthal, PJ; Sachdeva, S; Singh, P; Vivas, L1
Chan, ST; Copp, BR; Kaiser, M; Page, MJ; Pearce, AN1
Brun, R; Ge, JF; Ihara, M; Kaiser, M; Liu, BQ; Shi, XL; Wittlin, S1
Anizon, F; Bouchikhi, F; Brun, R; Moreau, P1
Brun, R; Huang, TL; Kaiser, M; Mayence, A; Vanden Eynde, JJ; Yarlett, N1
Dürüst, Y; Kaiser, M; Karakuş, H; Tasdemir, D1
Boshoff, HI; Boyd, PD; Copp, BR; Kaiser, M; McCracken, ST1
Bettis, S; Brun, R; Fomovska, A; Huang, Q; Kaiser, M; Kozikowski, AP; McLeod, R; Mui, E; Pieroni, M; Stec, J; Witola, WH1
Agarwal, H; Bahar, M; Brun, R; Cason, E; Doskotch, RW; Drew, ME; Endeshaw, M; He, S; Kaiser, M; Kinghorn, AD; Li, C; Mahasenan, KV; Munde, M; Pandharkar, T; Werbovetz, KA; Wilson, WD; Zhu, X1
Copp, BR; Kaiser, M; Liew, LP1
Kaiser, M; McKeever, C; Rozas, I1
Barker, D; Rye, CE1
Andriamihaja, B; Bauer, JO; Lamshöft, M; Razakarivony, AA; Spiteller, M; Strohmann, C; Talontsi, FM1
El Sayed, I; Inokuchi, T; Kaiser, M; Lu, WJ; Maeda, T; Mei, ZW; Pang, CQ; Peng, W; Wang, L1
Campbell, M; Charman, SA; Gilbert, IH; Hudson, A; Kaiser, M; Katneni, K; Mital, A; Morizzi, J; Murugesan, D; Shackleford, DM; Yeates, C1
Egan, TJ; El Sayed, Iel T; Imai, K; Inokuchi, T; Kaiser, M; Lu, WJ; Mei, ZW; Wang, L; Wicht, KJ1
Arafa, RK; Boykin, DW; Brun, R; Ismail, MA; Jones, SK; Pandharkar, T; Patrick, DA; Tidwell, RR; Wenzler, T; Werbovetz, KA; Zhu, X1
Almohaywi, B; Avery, VM; Baell, JB; Campbell, M; Charman, SA; Ferrins, L; Hyland, C; Jones, AJ; Kaiser, M; Rahmani, R; Ryan, E; Smith, J; Sykes, ML; Teston, E; White, KL; Yin, J1
Bakunov, SA; Bakunova, SM; Barszcz, T; Boykin, DW; Brun, R; Jones, SK; Kumar, A; Patrick, DA; Tidwell, RR; Wenzler, T; Werbovetz, KA1
Bosch-Navarrete, C; Gilbert, IH; González-Pacanowska, D; Hampton, SE; Johansson, NG; Kahnberg, P; Kaiser, M; Recio, E; Schipani, A1
Brun, R; Harel, D; Prinz, H; Schepmann, D; Schmidt, TJ; Wünsch, B1
Belluti, F; Bisi, A; Bolognesi, ML; Brun, R; Cavalli, A; Colizzi, F; Gobbi, S; Kostrewa, D; Lauciello, L; Perozzo, R; Rampa, A; Recanatini, M; Scapozza, L1
Amewu, RK; Burrell-Saward, H; Chadwick, J; Hussain, A; Janneh, O; Miguel, C; O'Neill, PM; Panda, S; Rinki, R; Vivas, L; Ward, SA1
Bakunov, SA; Bakunova, SM; Brun, R; Patrick, DA; Tidwell, RR; Wenzler, T1
Batzer, A; Bode, HB; Chantratita, N; Grundmann, F; Kaiser, M; Kurz, M; Schiell, M; Thanwisai, A1
Anh Ngoc, T; Egan, TJ; Imai, K; Inokuchi, T; Kaiser, M; Kiguchi, R; Wang, MQ; Wang, N; Wicht, KJ1
Dardonville, C; Kaiser, M; Lagartera, L; Ríos Martínez, CH1
Chibale, K; Huang, J; Mahajan, A; Mekonnen, B; Meurillon, M; Naran, K; Sharma, RK; Tukulula, M; Warner, D1
Botta, B; Brun, R; Costi, R; De Vita, D; Di Santo, R; Friggeri, L; Kaiser, M; Moraca, F; Scipione, L; Tortorella, S; Zamperini, C1
Chibale, K; Gut, J; Njogu, PM; Rosenthal, PJ1
Andayi, WA; Chibale, K; Egan, TJ; Gut, J; Rosenthal, PJ1
Boykin, DW; Brun, R; Liu, ZY; Wenzler, T; Zhu, X1
Avery, VM; Baell, JB; Bergström, CA; Charman, SA; Ferrins, L; Gazdik, M; Jones, AJ; Kaiser, M; Rahmani, R; Ryan, E; Sykes, ML; Varghese, S; White, KL1
Bode, HB; Kaiser, M; Nollmann, FI; Reimer, D; Schultz, K1
Andricopulo, AD; Bwalya, AG; Carballeira, NM; Cordero-Maldonado, ML; Crawford, AD; Guido, RV; Itoe, MA; Kaiser, M; Mota, MM; Tasdemir, D1
Avery, VM; Barth, S; Duffy, S; Frank, W; Geffken, D; Held, J; Kamber, J; Kuna, K; Kurz, T; Leven, M; Mordmüller, B; Sax, S; Siethoff, C; Tschan, S; Wittlin, S1
Battistuzzi, G; Giannini, G1
Battistuzzi, G; Giannini, G; Vignola, D1
Dardonville, C; Kaiser, M; Montalvo-Quirós, S; Taladriz-Sender, A1
Bauer, JO; Happi, GM; Kouam, SF; Lamshöft, M; Spiteller, M; Strohmann, C; Talontsi, FM; Zühlke, S1
Gilbert, IH; Kaiser, M; Mital, A; Murugesan, D; Yeates, C1
Brun, R; Faist, J; Kaiser, M; Saf, R; Seebacher, W; Weis, R1
Brun, R; Göker, H; Kaiser, M; Karaaslan, C1
Faist, J; Hinteregger, C; Kaiser, M; Mäser, P; Saf, R; Seebacher, W; Weis, R1
Bringmann, G; Brun, R; Brünnert, D; Chatterjee, M; Efferth, T; Feineis, D; Kaiser, M; Li, J; Mudogo, V; Seo, EJ; Seupel, R1
Faist, J; Hochegger, P; Kaiser, M; Mäser, P; Saf, R; Seebacher, W; Weis, R2
Back, TG; Brun, R; Kaiser, M; Manivannan, S; Pastor, A; Snyder, FF; Tran, HA; Wen, X; Zheng, Z1
Barker, D; Bourguet-Kondracki, ML; Brunel, JM; Cadelis, MM; Copp, BR; Dubois, J; Kaiser, M1
Brun, R; Kaiser, M; Mazzieri, MR; Nieto, MJ; Pagliero, RJ1
Chianese, G; Erpenbeck, D; Kaiser, M; Luciano, P; Merten, C; Silber, J; Tasdemir, D; Topaloglu, B1
Copp, BR; Kaiser, M; Pearce, AN1
Awale, S; Bringmann, G; Bruhn, T; Brun, R; Feineis, D; Kaiser, M; Li, J; Mudogo, V; Seupel, R1
Alajlani, M; Bauer, R; Belaj, F; Brantner, A; Bucar, F; Faist, J; Hochegger, P; Kaiser, M; Kretschmer, N; Mäser, P; Mohsin, NU; Saf, R; Seebacher, W; Turek, I; Weis, R1
Bringmann, G; Brun, R; Efferth, T; Feineis, D; Kaiser, M; Mudogo, V; Seo, EJ; Tshitenge, DT1
Aliabadi, A; De Mieri, M; Ebrahimi, SN; Farimani, MM; Hamburger, M; Kaiser, M; Khodaei, B; Moradi, H1
Brun, R; Calvet, CM; Costi, R; De Leo, A; De Vita, D; Di Santo, R; Jennings, GK; Kaiser, M; Madia, VN; Mäser, P; Messore, A; Pescatori, L; Podust, LM; Saccoliti, F; Scipione, L; Tudino, V1
Bode, HB; Cai, X; Kaiser, M; Zhao, L1
Danton, O; Hamburger, M; Kaiser, M; Moridi Farimani, M; Nejad Ebrahimi, S; Neuburger, M; Potterat, O; Ramseyer, J; Salehi, P; Tabefam, M1
Battista, MR; Brun, R; Calvet, CM; Cirilli, R; Costi, R; De Leo, A; De Vita, D; Di Marco, A; Di Santo, R; Faggi, C; Jennings, GK; Kaiser, M; Madia, VN; Mäser, P; Messore, A; Pepe, G; Pescatori, L; Podust, LM; Saccoliti, F; Scipione, L; Summa, V; Tudino, V1
Awale, S; Bringmann, G; Bruhn, T; Brun, R; Feineis, D; Kaiser, M; Mudogo, V; Schmidt, D; Tshitenge, DT; Würthner, F1
Al-Harrasi, A; Babanezhad Harikandei, K; Bararjanian, M; Ebrahimi, SN; Kaiser, M; Salehi, P1
Awori, RM; Bode, HB; Groß, J; Kaiser, M; Opatz, T; Zhao, L1
Bucar, F; Kaiser, M; Kalt, MM; Ochensberger, S; Presser, A; Saf, R; Schuehly, W; Solnier, J1
Alajlani, M; Bauer, R; Belaj, F; Brantner, A; Dolensky, J; Hochegger, P; Kaiser, M; Kretschmer, N; Mäser, P; Mohsin, NU; Petritsch, M; Saf, R; Schühly, W; Seebacher, W; Weis, R1
Horiuchi, M; Ihara, M; Ikegami-Kawai, M; Itoh, I; Kaiser, M; Kojima, M; Miyagi, S; Mizukawa, Y; Nanga Chick, C; Sakanoue, S; Togashi, H; Tsubuki, M; Usuki, T1
Bringmann, G; Feineis, D; Kaiser, M; Lombe, BK; Mudogo, V1
Börgel, F; Jabor, VAP; Kaiser, M; Krauth-Siegel, RL; Lehmkuhl, K; Nonato, MC; Schepmann, D; Schmidt, TJ; Uth, JF; Wünsch, B1
Brun, R; Celik, I; Doganc, F; Eren, G; Goker, H; Kaiser, M1
Altucci, L; Benedetti, R; Brogi, S; Butini, S; Campiani, G; Carullo, G; Casagni, A; De Matteis, A; Díaz, JF; Federico, S; Galatello, P; Gemma, S; Ghanim, M; Ibrahim, O; Kelly, VP; Khan, T; Lamponi, S; Lucena-Agell, D; Magnano, S; McCabe, N; Nathwani, S; O'Sullivan, J; Papulino, C; Pozzetti, L; Ramunno, A; Relitti, N; Staiano, L; Turkington, R; Ulivieri, C; Valoti, M; Vanni, F; VanWemmel, R; Zisterer, D1
Beck, WT; Cirtain, MC; Danks, MK; Felsted, RL; Safa, AR; Suttle, DP; Trent, JM; Wolverton, JS1
Beck, WT; Pearce, HL; Zamora, JM1
Morgan, EH; Sorokin, LM; Yeoh, GC1
Arnold, AM; Whitehouse, JM1

Reviews

1 review(s) available for chloroquine and podophyllotoxin

ArticleYear
Quest for a potent antimalarial drug lead: Synthesis and evaluation of 6,7-dimethoxyquinazoline-2,4-diamines.
    Bioorganic & medicinal chemistry, 2021, 03-01, Volume: 33

    Topics: Animals; Antimalarials; Dose-Response Relationship, Drug; Drug Discovery; Female; Malaria, Falciparum; Mice; Mice, Inbred ICR; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship

2021

Other Studies

118 other study(ies) available for chloroquine and podophyllotoxin

ArticleYear
Design, synthesis, and biological evaluation of a series of simple and novel potential antimalarial compounds.
    Bioorganic & medicinal chemistry letters, 2001, Jul-23, Volume: 11, Issue:14

    Topics: Animals; Antimalarials; Benzocycloheptenes; Drug Design; Nitrobenzenes; Oxazines; Plasmodium falciparum; Trypanosoma cruzi

2001
Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine.
    Bioorganic & medicinal chemistry letters, 2001, Oct-08, Volume: 11, Issue:19

    Topics: Animals; Antiprotozoal Agents; Leishmania; Parasitic Sensitivity Tests; Plasmodium; Quinacrine; Sulfonamides; Trypanosoma; Urea

2001
Assessment of the antiprotozoal activity of Galphimia glauca and the isolation of new nor-secofriedelanes and nor-friedelanes.
    Journal of natural products, 2002, Volume: 65, Issue:10

    Topics: Animals; Antiprotozoal Agents; Drug Screening Assays, Antitumor; Galphimia; Leishmania donovani; Plasmodium falciparum; Spectrum Analysis; Triterpenes; Trypanosoma brucei brucei; Tumor Cells, Cultured

2002
Isoneocryptolepine, a synthetic indoloquinoline alkaloid, as an antiplasmodial lead compound.
    Journal of natural products, 2005, Volume: 68, Issue:5

    Topics: Alkaloids; Animals; Antimalarials; Apocynaceae; Indole Alkaloids; Indoles; Molecular Structure; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2005
Irreversible inactivation of trypanothione reductase by unsaturated Mannich bases: a divinyl ketone as key intermediate.
    Journal of medicinal chemistry, 2005, Nov-17, Volume: 48, Issue:23

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chromatography, High Pressure Liquid; Dimethyl Sulfoxide; Drug Storage; Glutathione; Glutathione Reductase; Humans; Ketones; Leishmania donovani; Magnetic Resonance Spectroscopy; Mannich Bases; NADH, NADPH Oxidoreductases; Plasmodium falciparum; Spectrometry, Mass, Electrospray Ionization; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Thioredoxin-Disulfide Reductase; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2005
Alkyl-linked bis-THTT derivatives as potent in vitro trypanocidal agents.
    Bioorganic & medicinal chemistry letters, 2006, Mar-01, Volume: 16, Issue:5

    Topics: Alkylation; Animals; Carboxylic Acids; Leishmania donovani; Molecular Structure; Plasmodium falciparum; Structure-Activity Relationship; Thiadiazines; Trypanocidal Agents; Trypanosoma brucei rhodesiense

2006
Acyclic nucleoside analogues as inhibitors of Plasmodium falciparum dUTPase.
    Journal of medicinal chemistry, 2006, Jul-13, Volume: 49, Issue:14

    Topics: Animals; Antimalarials; Erythrocytes; Humans; In Vitro Techniques; Models, Molecular; Nucleosides; Plasmodium falciparum; Pyrophosphatases; Stereoisomerism; Structure-Activity Relationship; Trityl Compounds; Uracil

2006
Evaluation of azasterols as anti-parasitics.
    Journal of medicinal chemistry, 2006, Oct-05, Volume: 49, Issue:20

    Topics: Animals; Antimalarials; Azasteroids; Leishmania donovani; Methyltransferases; Plasmodium falciparum; Stereoisomerism; Sterols; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2006
Limonoid orthoacetates and antiprotozoal compounds from the roots of Pseudocedrela kotschyi.
    Journal of natural products, 2007, Volume: 70, Issue:1

    Topics: Animals; Antiprotozoal Agents; Leishmania donovani; Limonins; Mali; Meliaceae; Molecular Structure; Plant Roots; Plants, Medicinal; Plasmodium falciparum; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2007
Synthesis and in vitro antiprotozoal activities of dicationic 3,5-diphenylisoxazoles.
    Journal of medicinal chemistry, 2007, May-17, Volume: 50, Issue:10

    Topics: Animals; Antimalarials; Benzamidines; Cations; Cell Line; Combinatorial Chemistry Techniques; Isoxazoles; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense

2007
Synthesis and antiprotozoal activities of simplified analogs of naphthylisoquinoline alkaloids.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:1

    Topics: Alkaloids; Animals; Antiprotozoal Agents; Eukaryota; Isoquinolines; Myoblasts, Skeletal

2008
Anti-malarial activity of N6-modified purine analogues.
    Bioorganic & medicinal chemistry, 2007, Aug-15, Volume: 15, Issue:16

    Topics: Animals; Antimalarials; Male; Mice; Molecular Structure; Plasmodium falciparum; Purines; Structure-Activity Relationship

2007
Antiprotozoal polyacetylenes from the Tanzanian medicinal plant Cussonia zimmermannii.
    Journal of natural products, 2007, Volume: 70, Issue:10

    Topics: Animals; Antiprotozoal Agents; Araliaceae; Leishmania donovani; Molecular Structure; Plants, Medicinal; Plasmodium falciparum; Polyynes; Tanzania; Trypanosoma brucei rhodesiense

2007
Synthesis and in vitro antiprotozoal activity of bisbenzofuran cations.
    Journal of medicinal chemistry, 2007, Nov-15, Volume: 50, Issue:23

    Topics: Animals; Antimalarials; Benzofurans; Cations; Leishmania donovani; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense

2007
Synthesis and evaluation of antiparasitic activities of new 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine derivatives.
    Journal of medicinal chemistry, 2007, Nov-15, Volume: 50, Issue:23

    Topics: Animals; Antimalarials; Leishmania donovani; Morpholines; Plasmodium falciparum; Pyrazoles; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma

2007
Synthesis and pharmacological evaluation of fluorescent and photoactivatable analogues of antiplasmodial naphthylisoquinolines.
    Journal of medicinal chemistry, 2007, Nov-29, Volume: 50, Issue:24

    Topics: Alkaloids; Animals; Antimalarials; Fluorescent Dyes; Isoquinolines; Naphthalenes; Photoaffinity Labels; Plasmodium falciparum; Structure-Activity Relationship

2007
Synthesis and structure-activity relationship of 3-phenylquinoxaline 1,4-di-N-oxide derivatives as antimalarial agents.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:9

    Topics: Animals; Antimalarials; Cattle; Cell Survival; Drug Design; Humans; KB Cells; Plasmodium falciparum; Quinoxalines; Structure-Activity Relationship

2008
Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Animals; Antimalarials; Biological Transport; Cell Line, Tumor; Chloroquine; Drug Resistance; Drug Therapy, Combination; Glutathione Reductase; Humans; In Vitro Techniques; Malaria; Mice; Mice, Inbred BALB C; Naphthalenes; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2008
Synthesis and in vitro antiprotozoal activities of water-soluble, inexpensive 3,7-bis(dialkylamino)phenoxazin-5-ium derivatives.
    Journal of medicinal chemistry, 2008, Jun-26, Volume: 51, Issue:12

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Drug Resistance; Leishmania donovani; Oxazines; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrimethamine; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2008
Antiplasmodial and antitrypanosomal activities of aminobicyclo[2.2.2]octyl omega-aminoalkanoates.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:2

    Topics: Animals; Antiprotozoal Agents; Bridged Bicyclo Compounds; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense

2009
Antiprotozoal activities of heterocyclic-substituted xanthones from the marine-derived fungus Chaetomium sp.
    Journal of natural products, 2008, Volume: 71, Issue:9

    Topics: Animals; Antiprotozoal Agents; Bacillus megaterium; Chaetomium; Chlorella; Drug Screening Assays, Antitumor; Escherichia coli; Leishmania donovani; Marine Biology; Microbial Sensitivity Tests; Models, Molecular; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Trypanosoma cruzi; Xanthones

2008
Synthesis and antiprotozoal activity of cationic 2-phenylbenzofurans.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Animals; Antiprotozoal Agents; Benzofurans; Cations; Disease Models, Animal; Leishmania; Mice; Molecular Structure; Structure-Activity Relationship; Trypanosoma; Trypanosomiasis

2008
Synthesis and antiparasitic and antifungal evaluation of 2'-arylsubstituted-1H,1'H-[2,5']bisbenzimidazolyl-5-carboxamidines.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:5

    Topics: Amidines; Animals; Antifungal Agents; Antiparasitic Agents; Leishmania donovani; Microbial Sensitivity Tests; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Trypanosoma brucei brucei; Trypanosoma cruzi

2009
Compounds structurally related to ellagic acid show improved antiplasmodial activity.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:2

    Topics: Animals; Antimalarials; Cells, Cultured; Chloroquine; DNA, Complementary; Drug Resistance; Ellagic Acid; Glutathione Peroxidase; Glutathione Transferase; Heme; Humans; Kinetics; Plasmodium falciparum; Reverse Transcriptase Polymerase Chain Reaction

2009
Okundoperoxide, a bicyclic cyclofarnesylsesquiterpene endoperoxide from Scleria striatinux with antiplasmodial activity.
    Journal of natural products, 2009, Feb-27, Volume: 72, Issue:2

    Topics: Antimalarials; Chloroquine; Cyperaceae; Drug Resistance; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Plant Roots; Plants, Medicinal; Plasmodium falciparum; Sesquiterpenes; Stereoisomerism

2009
Structure-activity study of pentamidine analogues as antiprotozoal agents.
    Journal of medicinal chemistry, 2009, Apr-09, Volume: 52, Issue:7

    Topics: Animals; Antimalarials; Cadaverine; Drug Resistance; Female; Imidazoles; Leishmania donovani; Mice; Myoblasts; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosomiasis

2009
Trypanothione reductase high-throughput screening campaign identifies novel classes of inhibitors with antiparasitic activity.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:7

    Topics: Animals; Antiparasitic Agents; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Molecular Structure; NADH, NADPH Oxidoreductases; Structure-Activity Relationship; Trypanosoma; Trypanosomiasis

2009
Synthesis and antiprotozoal activities of dicationic bis(phenoxymethyl)benzenes, bis(phenoxymethyl)naphthalenes, and bis(benzyloxy)naphthalenes.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:9

    Topics: Animals; Antiprotozoal Agents; Benzene; Cell Survival; Leishmania donovani; Mice; Myoblasts; Naphthalenes; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2009
Privileged structure-guided synthesis of quinazoline derivatives as inhibitors of trypanothione reductase.
    Bioorganic & medicinal chemistry letters, 2009, Jun-01, Volume: 19, Issue:11

    Topics: Animals; Antiparasitic Agents; Cell Line; Computer Simulation; Drug Design; Enzyme Inhibitors; Glutathione Reductase; Humans; NADH, NADPH Oxidoreductases; Quinazolines; Rats; Structure-Activity Relationship; Trypanosoma cruzi

2009
Synthesis and antiprotozoal activity of pyridyl analogues of pentamidine.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Animals; Antiprotozoal Agents; Female; Leishmania donovani; Mice; Pentamidine; Plasmodium falciparum; Pyridines; Rats; Structure-Activity Relationship

2009
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Structure-activity relationship of antiparasitic and cytotoxic indoloquinoline alkaloids, and their tricyclic and bicyclic analogues.
    Bioorganic & medicinal chemistry, 2009, Oct-15, Volume: 17, Issue:20

    Topics: Animals; Antimalarials; Antineoplastic Agents; Indole Alkaloids; Mice; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2009
Synthesis and antiprotozoal activity of cationic 1,4-diphenyl-1H-1,2,3-triazoles.
    Journal of medicinal chemistry, 2010, Jan-14, Volume: 53, Issue:1

    Topics: Amidines; Animals; Antiprotozoal Agents; Cell Line; Cell Survival; Disease Models, Animal; Female; Leishmania donovani; Mice; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Stereoisomerism; Structure-Activity Relationship; Triazoles; Trypanosoma brucei rhodesiense

2010
Synthesis, stereoelectronic characterization and antiparasitic activity of new 1-benzenesulfonyl-2-methyl-1,2,3,4-tetrahydroquinolines.
    Bioorganic & medicinal chemistry, 2010, Jan-01, Volume: 18, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cell Line; Humans; Leishmania donovani; Models, Molecular; Parasitic Sensitivity Tests; Plasmodium falciparum; Protozoan Infections; Quinolines; Structure-Activity Relationship; Trypanosoma; Trypanosoma cruzi

2010
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Discovery of novel and potent benzhydryl-tropane trypanocides highly selective for Trypanosoma cruzi.
    Bioorganic & medicinal chemistry letters, 2010, Mar-15, Volume: 20, Issue:6

    Topics: Animals; Cell Line; Drug Discovery; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma cruzi

2010
Jacaranone-derived glucosidic esters from Jacaranda glabra and their activity against Plasmodium falciparum.
    Journal of natural products, 2010, Apr-23, Volume: 73, Issue:4

    Topics: Animals; Antimalarials; Benzoquinones; Ecuador; Esters; Glucosides; Myoblasts; Nuclear Magnetic Resonance, Biomolecular; Parasitic Sensitivity Tests; Phenylacetates; Plasmodium falciparum; Rats

2010
Antiprotozoal steroidal saponins from the marine sponge Pandaros acanthifolium.
    Journal of natural products, 2010, Aug-27, Volume: 73, Issue:8

    Topics: Animals; Antiprotozoal Agents; Leishmania donovani; Marine Biology; Nuclear Magnetic Resonance, Biomolecular; Oceans and Seas; Plasmodium falciparum; Porifera; Saponins; Steroids; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2010
QSAR guided synthesis of simplified antiplasmodial analogs of naphthylisoquinoline alkaloids.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Alkaloids; Animals; Antimalarials; Isoquinolines; Magnetic Resonance Spectroscopy; Models, Molecular; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Spectrometry, Mass, Electrospray Ionization; Spectroscopy, Fourier Transform Infrared

2010
2-Hexadecynoic acid inhibits plasmodial FAS-II enzymes and arrests erythrocytic and liver stage Plasmodium infections.
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Alkynes; Antimalarials; Binding Sites; Cell Line, Tumor; Computer Simulation; Erythrocytes; Fatty Acid Synthase, Type II; Fatty Acids, Unsaturated; Humans; Kinetics; Liver; Malaria, Falciparum; Plasmodium falciparum; Protozoan Proteins

2010
Didemnidines A and B, indole spermidine alkaloids from the New Zealand ascidian Didemnum sp.
    Journal of natural products, 2011, Apr-25, Volume: 74, Issue:4

    Topics: Animals; Antiprotozoal Agents; Indole Alkaloids; Leishmania donovani; Molecular Structure; New Zealand; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Spermidine; Structure-Activity Relationship; Trypanosoma; Urochordata

2011
β-Branched acyclic nucleoside analogues as inhibitors of Plasmodium falciparum dUTPase.
    Bioorganic & medicinal chemistry, 2011, Apr-01, Volume: 19, Issue:7

    Topics: Antimalarials; Deoxyuridine; Enzyme Inhibitors; Humans; Models, Molecular; Plasmodium falciparum; Pyrophosphatases; Structure-Activity Relationship

2011
Antiparasitic compounds from Cupania cinerea with activities against Plasmodium falciparum and Trypanosoma brucei rhodesiense.
    Journal of natural products, 2011, Apr-25, Volume: 74, Issue:4

    Topics: Animals; Antiprotozoal Agents; Cells, Cultured; Crystallography, X-Ray; Diterpenes; Ecuador; Glycosides; Hexanes; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Polycyclic Sesquiterpenes; Rats; Sapindaceae; Sesquiterpenes; Triterpenes; Trypanosoma brucei rhodesiense

2011
Marinoquinolines A-F, pyrroloquinolines from Ohtaekwangia kribbensis (Bacteroidetes).
    Journal of natural products, 2011, Apr-25, Volume: 74, Issue:4

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antimalarials; Antineoplastic Agents; Bacteroidetes; Drug Screening Assays, Antitumor; Female; Humans; India; Inhibitory Concentration 50; Microbial Sensitivity Tests; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Pyrroles; Quinolines

2011
Antimalarial pyrido[1,2-a]benzimidazoles.
    Journal of medicinal chemistry, 2011, Jul-14, Volume: 54, Issue:13

    Topics: Administration, Oral; Animals; Antimalarials; Benzimidazoles; Drug Resistance, Multiple; Humans; In Vitro Techniques; Injections, Intraperitoneal; L Cells; Malaria; Male; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Pyridines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

2011
Antiplasmodial and cytotoxicity evaluation of 3-functionalized 2-azetidinone derivatives.
    Bioorganic & medicinal chemistry letters, 2011, Aug-01, Volume: 21, Issue:15

    Topics: Antimalarials; Azetidines; beta-Lactams; Cell Line, Tumor; Humans; Plasmodium falciparum; Triazoles

2011
Antimalarial β-carbolines from the New Zealand ascidian Pseudodistoma opacum.
    Journal of natural products, 2011, Sep-23, Volume: 74, Issue:9

    Topics: Animals; Antimalarials; Carbolines; Chloroquine; Drug Resistance; Molecular Structure; New Zealand; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Stereoisomerism; Urochordata

2011
Synthesis and in vitro antiprotozoal activities of 5-phenyliminobenzo[a]phenoxazine derivatives.
    Bioorganic & medicinal chemistry letters, 2011, Oct-01, Volume: 21, Issue:19

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Drug Design; Inhibitory Concentration 50; Leishmania donovani; Malaria; Models, Chemical; Molecular Structure; Myoblasts; Oxazines; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyridinium Compounds; Rats; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2011
Biological evaluation of glycosyl-isoindigo derivatives against the pathogenic agents of tropical diseases (malaria, Chagas disease, leishmaniasis and human African trypanosomiasis).
    Bioorganic & medicinal chemistry letters, 2011, Nov-01, Volume: 21, Issue:21

    Topics: Animals; Antiprotozoal Agents; Drug Evaluation, Preclinical; Humans; Protozoan Infections

2011
Bis(oxyphenylene)benzimidazoles: a novel class of anti-Plasmodium falciparum agents.
    Bioorganic & medicinal chemistry, 2011, Dec-15, Volume: 19, Issue:24

    Topics: Animals; Antimalarials; Benzimidazoles; Cell Line; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats

2011
Synthesis and anti-protozoal activity of novel dihydropyrrolo[3,4-d][1,2,3]triazoles.
    European journal of medicinal chemistry, 2012, Volume: 48

    Topics: Animals; Antiprotozoal Agents; Cell Line; Eukaryota; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Molecular Structure; Oxadiazoles; Protozoan Infections; Pyrroles; Rats; Spectrometry, Mass, Electrospray Ionization; Spectroscopy, Fourier Transform Infrared; Structure-Activity Relationship; Triazoles

2012
Synthesis and antimalarial and antituberculosis activities of a series of natural and unnatural 4-methoxy-6-styryl-pyran-2-ones, dihydro analogues and photo-dimers.
    Bioorganic & medicinal chemistry, 2012, Feb-15, Volume: 20, Issue:4

    Topics: Antimalarials; Antitubercular Agents; Coumarins; Dimerization; Fatty Acids, Monounsaturated; Inhibitory Concentration 50; Leishmania donovani; Light; Molecular Structure; Plasmodium falciparum; Pyrones

2012
Synthesis, biological evaluation, and structure-activity relationships of N-benzoyl-2-hydroxybenzamides as agents active against P. falciparum (K1 strain), Trypanosomes, and Leishmania.
    Journal of medicinal chemistry, 2012, Apr-12, Volume: 55, Issue:7

    Topics: Antimalarials; Benzamides; Imides; Leishmania donovani; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2012
8,8-dialkyldihydroberberines with potent antiprotozoal activity.
    Journal of natural products, 2013, Mar-22, Volume: 76, Issue:3

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Berberine Alkaloids; Crystallography, X-Ray; Female; Inhibitory Concentration 50; Leishmania donovani; Mice; Mice, Inbred BALB C; Parasitic Sensitivity Tests; Plasmodium falciparum; Trypanosoma

2013
Discovery and preliminary structure-activity relationship analysis of 1,14-sperminediphenylacetamides as potent and selective antimalarial lead compounds.
    Bioorganic & medicinal chemistry letters, 2013, Jan-15, Volume: 23, Issue:2

    Topics: Acetamides; Animals; Antimalarials; Drug Discovery; Inhibitory Concentration 50; Malaria; Molecular Structure; Plasmodium falciparum; Spermine; Structure-Activity Relationship

2013
Aminoalkyl derivatives of guanidine diaromatic minor groove binders with antiprotozoal activity.
    Journal of medicinal chemistry, 2013, Feb-14, Volume: 56, Issue:3

    Topics: Animals; Antiprotozoal Agents; Guanidine; Nucleic Acid Denaturation; Plasmodium falciparum; Trypanosoma brucei rhodesiense

2013
Asymmetric synthesis and anti-protozoal activity of the 8,4'-oxyneolignans virolin, surinamensin and analogues.
    European journal of medicinal chemistry, 2013, Volume: 60

    Topics: Anisoles; Antiprotozoal Agents; Leishmania donovani; Lignans; Molecular Conformation; Parasitic Sensitivity Tests; Plasmodium falciparum

2013
Antibacterial and antiplasmodial constituents of Beilschmiedia cryptocaryoides.
    Journal of natural products, 2013, Jan-25, Volume: 76, Issue:1

    Topics: Acinetobacter calcoaceticus; Anti-Bacterial Agents; Antimalarials; Chloroquine; Drug Resistance; Escherichia coli; Lauraceae; Madagascar; Microbial Sensitivity Tests; Molecular Conformation; Plant Bark; Plasmodium falciparum; Pseudomonas stutzeri

2013
Synthesis and in vitro antimalarial testing of neocryptolepines: SAR study for improved activity by introduction and modifications of side chains at C2 and C11 on indolo[2,3-b]quinolines.
    Journal of medicinal chemistry, 2013, Feb-28, Volume: 56, Issue:4

    Topics: Alkaloids; Animals; Antimalarials; Cell Line; Chloroquine; Drug Resistance; Indoles; Malaria; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolines; Rats; Structure-Activity Relationship

2013
Discovery and structure-activity relationships of pyrrolone antimalarials.
    Journal of medicinal chemistry, 2013, Apr-11, Volume: 56, Issue:7

    Topics: Animals; Antimalarials; Cell Line; Drug Discovery; Magnetic Resonance Spectroscopy; Mass Spectrometry; Plasmodium falciparum; Pyrroles; Rats; Structure-Activity Relationship

2013
Synthesis and antimalarial testing of neocryptolepine analogues: addition of ester function in SAR study of 2,11-disubstituted indolo[2,3-b]quinolines.
    European journal of medicinal chemistry, 2013, Volume: 64

    Topics: Alkaloids; Animals; Antimalarials; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Indoles; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Rats; Structure-Activity Relationship

2013
Synthesis and antiprotozoal activity of dicationic m-terphenyl and 1,3-dipyridylbenzene derivatives.
    Journal of medicinal chemistry, 2013, Jul-11, Volume: 56, Issue:13

    Topics: Animals; Antiprotozoal Agents; Benzene; Chagas Disease; Female; Leishmania donovani; Mice; Mice, Inbred Strains; Models, Chemical; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyridines; Structure-Activity Relationship; Terphenyl Compounds; Trypanosoma cruzi

2013
3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis.
    European journal of medicinal chemistry, 2013, Volume: 66

    Topics: Anilides; Animals; Humans; Mice; Myoblasts, Skeletal; Rats; Species Specificity; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2013
Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives.
    European journal of medicinal chemistry, 2013, Volume: 67

    Topics: Animals; Antiprotozoal Agents; Dose-Response Relationship, Drug; Leishmania donovani; Mice; Molecular Structure; Myoblasts; Parasitic Sensitivity Tests; Pentamidine; Phenyl Ethers; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis

2013
Investigation of acyclic uridine amide and 5'-amido nucleoside analogues as potential inhibitors of the Plasmodium falciparum dUTPase.
    Bioorganic & medicinal chemistry, 2013, Sep-15, Volume: 21, Issue:18

    Topics: Amides; Antimalarials; Enzyme Inhibitors; Kinetics; Nucleosides; Plasmodium falciparum; Protein Binding; Protozoan Proteins; Pyrophosphatases; Uridine

2013
Natural product derived antiprotozoal agents: synthesis, biological evaluation, and structure-activity relationships of novel chromene and chromane derivatives.
    Journal of medicinal chemistry, 2013, Sep-26, Volume: 56, Issue:18

    Topics: Antiprotozoal Agents; Biological Products; Chemistry Techniques, Synthetic; Chromans; Inhibitory Concentration 50; Structure-Activity Relationship

2013
Design, synthesis, and biological and crystallographic evaluation of novel inhibitors of Plasmodium falciparum enoyl-ACP-reductase (PfFabI).
    Journal of medicinal chemistry, 2013, Oct-10, Volume: 56, Issue:19

    Topics: Animals; Antimalarials; Cell Line; Coumarins; Crystallography, X-Ray; Drug Design; Drug Resistance, Multiple; Enoyl-(Acyl-Carrier-Protein) Reductase (NADH); Molecular Docking Simulation; Plasmodium falciparum; Protein Binding; Protein Conformation; Structure-Activity Relationship

2013
Synthesis and evaluation of the antimalarial, anticancer, and caspase 3 activities of tetraoxane dimers.
    Bioorganic & medicinal chemistry, 2013, Dec-01, Volume: 21, Issue:23

    Topics: Antimalarials; Antineoplastic Agents; Caspase 3; Cell Line, Tumor; Dimerization; Humans; Malaria, Falciparum; Neoplasms; Plasmodium falciparum; Tetraoxanes

2013
Antiprotozoal activity of dicationic 3,5-diphenylisoxazoles, their prodrugs and aza-analogues.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Animals; Antiprotozoal Agents; Isoxazoles; Mice; Molecular Structure; Plasmodium falciparum; Prodrugs; Structure-Activity Relationship; Trypanosomiasis, African

2014
Antiparasitic chaiyaphumines from entomopathogenic Xenorhabdus sp. PB61.4.
    Journal of natural products, 2014, Apr-25, Volume: 77, Issue:4

    Topics: Animals; Antiparasitic Agents; Bacillus subtilis; Depsipeptides; Escherichia coli; Humans; Inhibitory Concentration 50; Micrococcus luteus; Molecular Structure; Nematoda; Nuclear Magnetic Resonance, Biomolecular; Parasitic Sensitivity Tests; Plasmodium falciparum; Saccharomyces cerevisiae; Thailand; Trypanosoma brucei rhodesiense; Trypanosoma cruzi; Xenorhabdus

2014
Synthesis, β-haematin inhibition, and in vitro antimalarial testing of isocryptolepine analogues: SAR study of indolo[3,2-c]quinolines with various substituents at C2, C6, and N11.
    Bioorganic & medicinal chemistry, 2014, May-01, Volume: 22, Issue:9

    Topics: Animals; Antimalarials; Cell Line; Cell Survival; Hemin; Humans; Indole Alkaloids; Indoles; Mice; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quinolines; Rats; Structure-Activity Relationship

2014
Antiprotozoal activity and DNA binding of N-substituted N-phenylbenzamide and 1,3-diphenylurea bisguanidines.
    European journal of medicinal chemistry, 2014, Jun-23, Volume: 81

    Topics: Animals; Antiparasitic Agents; Benzamides; Binding Sites; Cell Line; Cell Survival; Disease Models, Animal; DNA; Dose-Response Relationship, Drug; Female; Guanidines; Mice; Mice, Inbred Strains; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Surface Plasmon Resonance; Trypanosoma brucei rhodesiense; Trypanosomiasis, African; Urea

2014
Synthesis and antiplasmodial and antimycobacterial evaluation of new nitroimidazole and nitroimidazooxazine derivatives.
    ACS medicinal chemistry letters, 2013, Jan-10, Volume: 4, Issue:1

    Topics:

2013
New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.
    ACS medicinal chemistry letters, 2013, Jun-13, Volume: 4, Issue:6

    Topics:

2013
Design, Synthesis, and Antiplasmodial Activity of Hybrid Compounds Based on (2R,3S)-N-Benzoyl-3-phenylisoserine.
    ACS medicinal chemistry letters, 2013, Jul-11, Volume: 4, Issue:7

    Topics:

2013
Synthesis, Antiplasmodial Activity, and β-Hematin Inhibition of Hydroxypyridone-Chloroquine Hybrids.
    ACS medicinal chemistry letters, 2013, Jul-11, Volume: 4, Issue:7

    Topics:

2013
Synthesis and antiparasitic activity of new bis-arylimidamides: DB766 analogs modified in the terminal groups.
    European journal of medicinal chemistry, 2014, Aug-18, Volume: 83

    Topics: Amides; Animals; Antiparasitic Agents; Cell Line; Chemistry Techniques, Synthetic; Leishmania; Plasmodium falciparum; Rats; Trypanosoma

2014
Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei.
    Journal of medicinal chemistry, 2014, Aug-14, Volume: 57, Issue:15

    Topics: Animals; Benzamides; Cell Line; HEK293 Cells; Humans; Microsomes, Liver; Myoblasts; Pyridines; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense

2014
Xenortide Biosynthesis by Entomopathogenic Xenorhabdus nematophila.
    Journal of natural products, 2014, Aug-22, Volume: 77, Issue:8

    Topics: Chromatography, High Pressure Liquid; Dipeptides; Leishmania; Molecular Structure; Multigene Family; Nuclear Magnetic Resonance, Biomolecular; Parasitic Sensitivity Tests; Plasmodium falciparum; Trypanosoma brucei brucei; Tryptamines; Xenorhabdus

2014
2-Octadecynoic acid as a dual life stage inhibitor of Plasmodium infections and plasmodial FAS-II enzymes.
    Bioorganic & medicinal chemistry letters, 2014, Sep-01, Volume: 24, Issue:17

    Topics: Animals; Antimalarials; Cell Line, Tumor; Dose-Response Relationship, Drug; Fatty Acid Synthase, Type II; Fatty Acids, Unsaturated; Humans; Malaria; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship; Zebrafish

2014
Blood schizontocidal and gametocytocidal activity of 3-hydroxy-N'-arylidenepropanehydrazonamides: a new class of antiplasmodial compounds.
    Journal of medicinal chemistry, 2014, Oct-09, Volume: 57, Issue:19

    Topics: Animals; Antimalarials; Chloroquine; Malaria; Mice; Parasitemia; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium berghei; Plasmodium falciparum; Rats; Structure-Activity Relationship

2014
Exploring in vitro and in vivo Hsp90 inhibitors activity against human protozoan parasites.
    Bioorganic & medicinal chemistry letters, 2015, Feb-01, Volume: 25, Issue:3

    Topics: Animals; Antiprotozoal Agents; Cell Line, Tumor; Disease Models, Animal; HSP90 Heat-Shock Proteins; Humans; Mice; Parasitemia; Plasmodium falciparum; Protein Binding; Rats; Triazoles; Trypanosoma brucei rhodesiense

2015
Hydroxamic acid based histone deacetylase inhibitors with confirmed activity against the malaria parasite.
    Bioorganic & medicinal chemistry letters, 2015, Feb-01, Volume: 25, Issue:3

    Topics: Animals; Antimalarials; Cell Line, Tumor; Dipeptides; Disease Models, Animal; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Hydroxamic Acids; Malaria; Mice; Parasites; Plasmodium falciparum; Protein Isoforms

2015
Antiprotozoal activity and DNA binding of dicationic acridones.
    Journal of medicinal chemistry, 2015, Feb-26, Volume: 58, Issue:4

    Topics: Acridines; Acridones; Antiprotozoal Agents; Binding Sites; Cations; DNA; Dose-Response Relationship, Drug; Leishmania donovani; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2015
Antiplasmodial and Cytotoxic Triterpenoids from the Bark of the Cameroonian Medicinal Plant Entandrophragma congoënse.
    Journal of natural products, 2015, Apr-24, Volume: 78, Issue:4

    Topics: Animals; Antimalarials; Cameroon; Chloroquine; Disease Resistance; Erythrocytes; Meliaceae; Molecular Structure; Muscle, Skeletal; Nuclear Magnetic Resonance, Biomolecular; Parasitic Sensitivity Tests; Plant Bark; Plant Stems; Plants, Medicinal; Plasmodium falciparum; Rats; Triterpenes

2015
Discovery and optimisation studies of antimalarial phenotypic hits.
    European journal of medicinal chemistry, 2015, Oct-20, Volume: 103

    Topics: Animals; Antimalarials; Cell Line; Cell Survival; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Discovery; Humans; Malaria; Mice; Microsomes, Liver; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Rats; Solubility; Structure-Activity Relationship

2015
Antiprotozoal activity of bicycles featuring a dimethylamino group at their bridgehead.
    Bioorganic & medicinal chemistry, 2016, 08-15, Volume: 24, Issue:16

    Topics: Animals; Antiprotozoal Agents; Bridged Bicyclo Compounds; Cells, Cultured; Plasmodium falciparum; Rats; Spectrum Analysis; Structure-Activity Relationship; Trypanosoma brucei rhodesiense

2016
Synthesis and potent antiprotozoal activity of mono/di amidino 2-anilinobenzimidazoles versus Plasmodium falciparum and Trypanosoma brucei rhodesiense.
    Bioorganic & medicinal chemistry, 2016, 09-15, Volume: 24, Issue:18

    Topics: Aniline Compounds; Animals; Antiprotozoal Agents; Benzimidazoles; Cell Line; Humans; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2016
New derivatives of 7-chloroquinolin-4-amine with antiprotozoal activity.
    Bioorganic & medicinal chemistry, 2017, 02-01, Volume: 25, Issue:3

    Topics: Aminoquinolines; Animals; Antiprotozoal Agents; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense

2017
Dioncophyllines C
    Journal of natural products, 2017, 02-24, Volume: 80, Issue:2

    Topics: Alkaloids; Antimalarials; Antineoplastic Agents; Humans; Isoquinolines; Magnoliopsida; Molecular Structure; Multiple Myeloma; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Structure-Activity Relationship

2017
New derivatives of quinoline-4-carboxylic acid with antiplasmodial activity.
    Bioorganic & medicinal chemistry, 2017, 04-01, Volume: 25, Issue:7

    Topics: Animals; Antimalarials; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Spectrum Analysis; Structure-Activity Relationship

2017
Synthesis and activity of nucleoside-based antiprotozoan compounds.
    Bioorganic & medicinal chemistry, 2017, 04-01, Volume: 25, Issue:7

    Topics: Animals; Antiprotozoal Agents; Carbon-13 Magnetic Resonance Spectroscopy; Inhibitory Concentration 50; Leishmania donovani; Plasmodium falciparum; Proton Magnetic Resonance Spectroscopy; Spectrophotometry, Infrared; Trypanosoma brucei brucei; Trypanosoma cruzi

2017
Structure-activity relationship studies on thiaplidiaquinones A and B as novel inhibitors of Plasmodium falciparum and farnesyltransferase.
    Bioorganic & medicinal chemistry, 2017, 08-15, Volume: 25, Issue:16

    Topics: Animals; Anti-Bacterial Agents; Antimalarials; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Farnesyltranstransferase; Microbial Sensitivity Tests; Molecular Structure; Plasmodium falciparum; Rats; Staphylococcus; Structure-Activity Relationship; Terpenes

2017
Lead selection of antiparasitic compounds from a focused library of benzenesulfonyl derivatives of heterocycles.
    Bioorganic & medicinal chemistry letters, 2017, 09-01, Volume: 27, Issue:17

    Topics: Animals; Antiparasitic Agents; Benzyl Compounds; Dose-Response Relationship, Drug; Heterocyclic Compounds; Leishmania donovani; Molecular Structure; Myoblasts; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2017
Antiprotozoal Linear Furanosesterterpenoids from the Marine Sponge Ircinia oros.
    Journal of natural products, 2017, 09-22, Volume: 80, Issue:9

    Topics: Animals; Antiprotozoal Agents; Furans; Magnetic Resonance Spectroscopy; Molecular Structure; Porifera; Sesquiterpenes; Spectroscopy, Fourier Transform Infrared

2017
Synthesis and antimalarial evaluation of artesunate-polyamine and trioxolane-polyamine conjugates.
    European journal of medicinal chemistry, 2017, Nov-10, Volume: 140

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Humans; Polyamines; Rats; Spectrum Analysis; Structure-Activity Relationship

2017
Jozilebomines A and B, Naphthylisoquinoline Dimers from the Congolese Liana Ancistrocladus ileboensis, with Antiausterity Activities against the PANC-1 Human Pancreatic Cancer Cell Line.
    Journal of natural products, 2017, 10-27, Volume: 80, Issue:10

    Topics: Algorithms; Alkaloids; Animals; Antimalarials; Antineoplastic Agents, Phytogenic; Congo; Drug Screening Assays, Antitumor; HeLa Cells; Humans; Isoquinolines; Leishmania donovani; Magnoliopsida; Molecular Structure; Naphthalenes; Nuclear Magnetic Resonance, Biomolecular; Pancreatic Neoplasms; Plasmodium falciparum; Rats; Trypanosoma brucei rhodesiense; Trypanosoma cruzi; Tumor Cells, Cultured

2017
Synthesis of new 1-benzyl tetrahydropyridinylidene ammonium salts and their antimicrobial and anticellular activities.
    European journal of medicinal chemistry, 2018, Jan-01, Volume: 143

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Antineoplastic Agents; Antiprotozoal Agents; Bacteria; Benzyl Compounds; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Mice; Microbial Sensitivity Tests; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyridines; Quaternary Ammonium Compounds; Rats; Saccharomyces cerevisiae; Salts; Structure-Activity Relationship; Trypanosoma brucei rhodesiense

2018
Mbandakamine-Type Naphthylisoquinoline Dimers and Related Alkaloids from the Central African Liana Ancistrocladus ealaensis with Antiparasitic and Antileukemic Activities.
    Journal of natural products, 2018, 04-27, Volume: 81, Issue:4

    Topics: Africa, Central; Alkaloids; Antimalarials; Antineoplastic Agents, Phytogenic; Antiparasitic Agents; Caryophyllales; Cell Line, Tumor; Humans; Isoquinolines; Naphthalenes; Plasmodium falciparum; Quinolines

2018
Phytochemical Study of Salvia leriifolia Roots: Rearranged Abietane Diterpenoids with Antiprotozoal Activity.
    Journal of natural products, 2018, 06-22, Volume: 81, Issue:6

    Topics: Abietanes; Antimalarials; Antiprotozoal Agents; Inhibitory Concentration 50; Leishmania donovani; Parasitic Sensitivity Tests; Phytochemicals; Plant Extracts; Plant Roots; Plasmodium falciparum; Salvia; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2018
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents.
    European journal of medicinal chemistry, 2018, Aug-05, Volume: 156

    Topics: Animals; Antiprotozoal Agents; Cell Line; Chagas Disease; Female; Humans; Imidazoles; Inhibitory Concentration 50; Leishmania donovani; Leishmaniasis, Visceral; Malaria, Falciparum; Mice; Mice, Inbred BALB C; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi; Trypanosomiasis, African

2018
Methionine-Containing Rhabdopeptide/Xenortide-like Peptides from Heterologous Expression of the Biosynthetic Gene Cluster kj12ABC in Escherichia coli.
    Journal of natural products, 2018, 10-26, Volume: 81, Issue:10

    Topics: Amino Acids; Animals; Antineoplastic Agents; Antiparasitic Agents; Escherichia coli; Methionine; Multigene Family; Oligopeptides; Parasites; Rats; Xenorhabdus

2018
Antiprotozoal Isoprenoids from Salvia hydrangea.
    Journal of natural products, 2018, 12-28, Volume: 81, Issue:12

    Topics: Animals; Antiprotozoal Agents; Cell Line; Leishmania donovani; Magnetic Resonance Spectroscopy; Molecular Structure; Plasmodium falciparum; Rats; Salvia; Spectrum Analysis; Terpenes; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2018
Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents.
    Journal of medicinal chemistry, 2019, 02-14, Volume: 62, Issue:3

    Topics: Animals; Antiprotozoal Agents; Cytochrome P-450 Enzyme Inhibitors; Drug Design; Drug Evaluation, Preclinical; Humans; Imidazoles; Parasitic Sensitivity Tests; Trypanosoma

2019
Synthesis and structure-activity relationships for new 6-fluoroquinoline derivatives with antiplasmodial activity.
    Bioorganic & medicinal chemistry, 2019, 05-15, Volume: 27, Issue:10

    Topics: Animals; Antimalarials; Cell Line; Cell Survival; Disease Models, Animal; Drug Resistance; Malaria; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2019
Ealamines A-H, a Series of Naphthylisoquinolines with the Rare 7,8'-Coupling Site, from the Congolese Liana
    Journal of natural products, 2019, 11-22, Volume: 82, Issue:11

    Topics: Animals; Antineoplastic Agents, Phytogenic; Antiprotozoal Agents; Caryophyllales; Drug Screening Assays, Antitumor; Humans; Isoquinolines; Leishmania; Molecular Structure; Naphthalenes; Pancreatic Neoplasms; Plant Components, Aerial; Plant Leaves; Plasmodium; Rats; Trypanosoma

2019
Synthesis, in-vitro antiprotozoal activity and molecular docking study of isothiocyanate derivatives.
    Bioorganic & medicinal chemistry, 2020, 01-01, Volume: 28, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Isothiocyanates; Leishmania donovani; Molecular Docking Simulation; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2020
Structure, Biosynthesis, and Bioactivity of Photoditritide from
    Journal of natural products, 2019, 12-27, Volume: 82, Issue:12

    Topics: Anti-Bacterial Agents; Antiprotozoal Agents; Microbial Sensitivity Tests; Micrococcus luteus; Molecular Structure; Photorhabdus; Spectrum Analysis; Trypanosoma brucei rhodesiense

2019
Palladium-catalysed synthesis of arylnaphthoquinones as antiprotozoal and antimycobacterial agents.
    European journal of medicinal chemistry, 2020, Dec-01, Volume: 207

    Topics: Anti-Bacterial Agents; Antiprotozoal Agents; Catalysis; Chemistry Techniques, Synthetic; Mycobacterium smegmatis; Palladium; Plasmodium falciparum; Quinones; Trypanosoma brucei rhodesiense

2020
Preparation of new 1,3-dibenzyl tetrahydropyridinylidene ammonium salts and their antimicrobial and anticellular activities.
    European journal of medicinal chemistry, 2021, Jan-15, Volume: 210

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Antimalarials; Antineoplastic Agents; Candida albicans; Cell Line; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Epidermis; Escherichia coli; Female; Humans; Mice; Microbial Sensitivity Tests; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Pseudomonas aeruginosa; Quaternary Ammonium Compounds; Rats; Salts; Staphylococcus aureus; Structure-Activity Relationship

2021
Spirombandakamine A
    Journal of natural products, 2021, 04-23, Volume: 84, Issue:4

    Topics: Alkaloids; Animals; Antiprotozoal Agents; Caryophyllales; Cell Line; Democratic Republic of the Congo; Isoquinolines; Molecular Structure; Phytochemicals; Plant Leaves; Plasmodium falciparum; Rats; Trypanosoma brucei rhodesiense

2021
Synthesis and Biological Evaluation of Natural-Product-Inspired, Aminoalkyl-Substituted 1-Benzopyrans as Novel Antiplasmodial Agents.
    Journal of medicinal chemistry, 2021, 05-13, Volume: 64, Issue:9

    Topics: Alkylation; Animals; Antimalarials; Benzopyrans; Biological Products; Biomimetic Materials; Chemistry Techniques, Synthetic; Erythrocytes; Kinetics; Mice; Plasmodium; Structure-Activity Relationship

2021
Synthesis, in vitro antiprotozoal activity, molecular docking and molecular dynamics studies of some new monocationic guanidinobenzimidazoles.
    European journal of medicinal chemistry, 2021, Oct-05, Volume: 221

    Topics: Antiprotozoal Agents; Benzimidazoles; Cations; Dose-Response Relationship, Drug; Guanidine; Leishmania donovani; Models, Molecular; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2021
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy.
    European journal of medicinal chemistry, 2022, May-05, Volume: 235

    Topics: Antineoplastic Agents; Apoptosis; Autophagy; Carcinoma, Squamous Cell; Cell Line, Tumor; Humans; Microtubules; Mouth Neoplasms

2022
Pharmacological, molecular, and cytogenetic analysis of "atypical" multidrug-resistant human leukemic cells.
    Cancer research, 1987, Oct-15, Volume: 47, Issue:20

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Chloroquine; Chromosome Banding; Chromosomes, Human, Pair 13; Colchicine; Dactinomycin; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Leukemia; Membrane Glycoproteins; Molecular Weight; Podophyllotoxin; Teniposide; Tumor Cells, Cultured; Verapamil; Vinblastine; Vinca Alkaloids

1987
Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells.
    Molecular pharmacology, 1988, Volume: 33, Issue:4

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cell Line; Chemical Phenomena; Chemistry, Physical; Chloroquine; Computer Simulation; Doxorubicin; Drug Resistance; Humans; Leukemia; Naphthacenes; Podophyllotoxin; Quinacrine; Verapamil; Vinca Alkaloids

1988
Transferrin endocytosis and iron uptake in developing myogenic cells in culture: effects of microtubular and metabolic inhibitors, sulphydryl reagents and lysosomotrophic agents.
    Journal of cellular physiology, 1988, Volume: 137, Issue:3

    Topics: 2,4-Dinitrophenol; Ammonium Chloride; Animals; Antimycin A; Azides; Cells, Cultured; Chick Embryo; Chloroquine; Colchicine; Dinitrophenols; Endocytosis; Iron; Methylamines; Muscles; Podophyllotoxin; Sodium Azide; Sulfhydryl Reagents; Transferrin; Vinblastine

1988
Interaction of VP16-213 with the DNA repair antagonist chloroquine.
    Cancer chemotherapy and pharmacology, 1982, Volume: 7, Issue:2-3

    Topics: Animals; Chloroquine; DNA Repair; Drug Interactions; Etoposide; Female; Lymphoma; Mice; Mice, Inbred CBA; Neoplasms, Experimental; Podophyllotoxin; Vincristine

1982