chloroquine and mefloquine

chloroquine has been researched along with mefloquine in 568 studies

Research

Studies (568)

TimeframeStudies, this research(%)All Research%
pre-1990121 (21.30)18.7374
1990's176 (30.99)18.2507
2000's127 (22.36)29.6817
2010's125 (22.01)24.3611
2020's19 (3.35)2.80

Authors

AuthorsStudies
Alcorn, J; Auschwitz, JM; Das, U; Dimmock, JR; Hickman, MR; Leed, SE; Singh, RS1
Charman, SA; Chiu, FC; Chollet, J; Dong, Y; Katneni, K; Mannila, J; Morizzi, J; Ryan, E; Santo Tomas, J; Scheurer, C; Snyder, C; Steuten, J; Vennerstrom, JL; Wang, X; Wittlin, S1
Biamonte, MA; Le Roch, KG; Wanner, J1
Avery, VM; Sykes, ML1
Alcorn, J; Das, U; Dimmock, JR; Hickman, MR; Lee, PJ; Leed, SE; Roncal, N; Sciotti, RJ; Singh, RS1
Azam, A; Inam, A; Leite, AC; Macedo, TS; Moreira, DR; Siddiqui, SM; Soares, MB1
Avery, VM; Charman, SA; Chibale, K; Douelle, F; Duffy, S; Gonzàlez Cabrera, D; Le Manach, C; March, C; Nchinda, AT; Ryan, E; Street, LJ; Taylor, D; Waterson, D; White, KL; Wiesner, L; Wittlin, S; Witty, MJ; Younis, Y1
Bavari, S; Burnett, JC; Gomba, L; Konstantinović, J; Krstić, M; Nuss, JE; Opsenica, DM; Sciotti, RJ; Segan, S; Selaković, Z; Solaja, BA; Videnović, M; Zlatović, M1
Agnamey, P; Azas, N; Cohen, A; Daulouede, S; Del Favero, M; Farvacques, N; Guillon, J; Hutter, S; Le Pape, P; Mullié, C; Pagniez, F; Pinaud, N; Ronga, L; Savrimoutou, S; Sonnet, P; Soum, C; Vincendeau, P1
Arrendale, RF; Ballie, MT; Bushnev, AS; Culver, DG; Evers, TJ; Galinski, MR; Girard, KR; Holt, JJ; Howard, RB; Lapp, S; Liotta, DC; Menaldino, DS; Meyer, EV; Natchus, MG; Reddy, GP1
Abla, N; Besson, D; Bombrun, A; Brun, R; Burt, H; Georgi, K; Kaiser, M; Molette, J; Muzerelle, M; Nwaka, S; Routier, J; Scheer, A1
Avery, VM; Barth, S; Duffy, S; Frank, W; Geffken, D; Held, J; Kamber, J; Kuna, K; Kurz, T; Leven, M; Mordmüller, B; Sax, S; Siethoff, C; Tschan, S; Wittlin, S1
Blackie, MA; de Kock, C; Hamann, AR; Smith, PJ; van Otterlo, WA1
Akoto, M; Avery, VM; Duffy, S; Hagen, TJ; Helgren, TR; Igbinoba, O; Lee, P; Sciotti, RJ1
Bacher, A; Behrendt, C; Brücher, K; Fischer, M; Gräwert, T; Held, J; Illarionov, B; Konzuch, S; Kurz, T; Lienau, C; Maes, L; Mordmüller, B; Wittlin, S1
Brantner, A; Brun, R; Bucar, F; Faist, J; Gröblacher, B; Kaiser, M; Kalia, Y; Merino, V; Perozzo, R; Saf, R; Scapozza, L; Seebacher, W; Weis, R; Wolkinger, V1
Barros, MT; Faísca Phillips, AM; Murtinheira, F; Nogueira, F1
Angulo-Barturen, I; Bashyam, S; Birkholtz, LM; Botha, M; Brunschwig, C; Chibale, K; Churchyard, A; Coetzer, TL; Dhinakaran, R; Ferrer, S; Gonzàlez Cabrera, D; Han, Z; Jiménez-Díaz, MB; Lauterbach, S; Le Manach, C; Meister, S; Njoroge, M; Paquet, T; Reader, J; Santos Martínez, M; Street, LJ; Taylor, D; Waterson, D; Winzeler, EA; Wittlin, S; Witty, MJ1
Albuquerque, IS; Burojević, J; D'Alessandro, S; Djurković-Djaković, O; Konstantinović, J; Machado, M; Pecic, S; Prudêncio, M; Sciotti, RJ; Šolaja, BA; Srbljanović, J; Štajner, T; Taramelli, D; Terzić, N; Tot, M; Verbić, T; Zlatović, M1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Challal, S; de Queiroz E Silva, DMA; Dos Santos Filho, JM; Macedo, TS; Moreira, DRM; Queiroz, EF; Soares, MBP; Teixeira, HMP; Wolfender, JL1
Beswick, P; Choowongkomon, K; Chuckowree, I; Gleeson, MP; Hannongbua, S; Horata, N; Obounchoey, P; Phuangsawai, O; Ratanabunyong, S; Srisook, P; Suphakun, P; Tabtimmai, L; Ward, SE1
Angulo-Barturen, I; Antonova-Koch, Y; Bashyam, S; Birkholtz, LM; Botha, ME; Charman, SA; Chibale, K; Ferrer, S; Gonzàlez Cabrera, D; Han, Z; Jiménez-Díaz, MB; Lawrence, N; Le Manach, C; Martínez, MS; Meister, S; Nchinda, AT; Nondaba, SH; Paquet, T; Reader, J; Street, LJ; Taylor, D; Waterson, D; White, KL; Winzeler, EA; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, M1
Araújo, ADS; Barbosa-Lima, G; Bozza, PT; da Silva, ET; de Freitas, CS; de Souza, MVN; Marttorelli, A; Moraes, AM; Neto, JC; Souza, TML; Vieira, YR1
Avery, VM; Buchholz, M; Delves, MJ; Duffy, S; Fischli, C; Held, J; Knaab, TC; Kuna, K; Kurz, T; Lehmann, U; Leven, M; Lungerich, B; Meister, S; Meitzner, D; Mordmüller, B; Stahlke, P; Winzeler, EA; Wittlin, S1
Feng, LS; Gao, C; Hu, YQ; Wu, X; Xu, L; Xu, Z; Zhang, S; Zhao, F1
Boddey, JA; Cowman, AF; Czabotar, PE; de Lezongard, RB; Hodder, AN; Jarman, KE; Jousset Sabroux, H; Nguyen, W; O'Neill, MT; Sleebs, BE; Thompson, JK1
Chu, XM; Gong, KK; Liang, LL; Liu, W; Sun, KL; Wang, C; Wang, WL1
Avery, VM; Baell, JB; Ban, K; Beveridge, JG; Blundell, S; Charman, SA; Chavchich, M; Chiu, FCK; Creek, D; Cuellar, ME; Dahlin, JL; Diab, S; Dingjan, T; Duffy, S; Edstein, MD; Ellis, K; Fletcher, S; Harjani, JR; Huang, F; Lucantoni, L; Marfurt, J; Noviyanti, R; Price, RN; Ralph, SA; Shi, DH; Strasser, JM; Teguh, S; Walters, MA; Wirjanata, G; Xue, L1
Aguiar, ACC; Boechat, N; Carvalho, AS; Coutinho, JP; da Silva, RMRJ; Gandi, MO; Krettli, AU; Mendonça, JS1
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P1
Azad, CS; Nainwal, LM; Narula, AK1
Bernatchez, JA; Li, J; Li, R; Luan, Y; Siqueira-Neto, JL; Tran, LT1
Baum, J; Bridgford, JL; Charman, SA; Churchyard, A; Crespo, B; Deni, I; Fidock, DA; Gahalawat, S; Gamo, FJ; Laleu, B; Lawong, A; Mittal, N; Mok, S; Niederstrasser, H; Okombo, J; Palmer, MJ; Phillips, MA; Posner, B; Ready, JM; Striepen, J; Winzeler, E; Wittlin, S; Yeo, T; Zhou, A1
Augereau, JM; Benoit-Vical, F; Deraeve, C; Jimenez, T; Mustière, R; Nguyen, M; Ouji, M1
Avery, VM; Challis, MP; Creek, DJ; De Paoli, A; Devine, SM; Kigotho, JK; MacRaild, CA; Norton, RS; Scammells, PJ; Siddiqui, G1
Agnamey, P; Azas, N; Cohen, A; Damiani, C; Dassonville-Klimpt, A; Dormoi, J; Guillon, J; Marchivie, M; Mullié, C; Pradines, B; Schneider, J; Sonnet, P; Taudon, N; Tisnerat, C; Totet, A1
Ghosh, SK; Sharma, VP; Yadav, RS1
Bunnag, D; Chindanond, D; Chittamas, S; Fernex, M; Harinasuta, T; Kristiansen, S; Malikul, S; Mittelholzer, ML; Sturchler, D1
Adio, RA; Dickschat, U; Mittelholzer, ML; Reber-Liske, R; Salako, LA; Sowunmi, A; Stürchler, D; Walker, O1
Rodríguez Rey, C1
Badoual, J1
Barnes, DA; Cowman, AF; Foote, SJ; Galatis, D; Kemp, DJ1
Bia, FJ1
Carbonaro, CA; Horowitz, H1
Collignon, PJ1
Brachman, PS; Kozarsky, PE; Metchock, B1
Bunnag, D; Chitamas, S; Harinasuta, T; Karbwang, J; Viravan, C1
Fadat, G; Gardon, J; Gazin, P; Hengy, C; Jambou, R; Louis, FJ; Louis, JP; Trebucq, A1
Cook, GC2
Bustos, MD; Ciceron, L; Danis, M; Gay, F; Gentilini, M; Pichet, C; Rojas-Rivero, L1
Currie, PF; Douglas, JG; Green, ST; Nathwani, D; Smith, NC1
Salako, LA; Sowunmi, A1
Bauchet, J; Hatin, I; Le Bras, J; Legros, F; Trape, JF1
Basco, LK; Bouchaud, O; Coulaud, JP; Farinotti, R; Gillotin, C; Gimenez, F; Le Bras, J; Rabenjarson, E; Ringwald, P1
Akintonwa, A; Orisakwe, OE1
Baudon, D; Cordoliani, G; Da Conceicao, S; Delolme, H; Doury, JC; Hovette, P; Lecamus, JL; Martet, G; Raphenon, G; Touze, JE1
Allaouchiche, B; Biron, F; Boibieux, A; Gaussorgues, P; Gerard-Boncompain, M; Peyramond, D; Robert, D; Salord, F; Sirodot, M1
Thomas, JE1
Trigg, PI1
Bocquet, JP; Taillan, F1
Carme, B1
Baird, JK; Bangs, MJ; Basri, H; Jones, TR; Ritonga, A1
Broderson, JR; Collins, WE; Ma, NS; Richardson, BB; Skinner, JC; Stanfill, PS1
Bergqvist, Y; Hellgren, U; Kihamia, CM; Rombo, L1
Ayivi, B; Bégué, P; Quinet, B; Ter Sakarian, M1
Boudreau, EF; Chaikummao, S; Pang, LW; Witayarut, C1
Bloland, P; Campbell, CC; Howell, BJ; Lackritz, EM; Lobel, HO1
Abua, JU; Lege-Oguntoye, L; Ogala, WN; Olurinola, PF; Slotboom, AB; Werblinska, B1
Sugioka, Y; Suzuki, M1
Brandicourt, O; Carme, B; Gay, F; Gentilini, M; Turk, P1
Bourdeau, EF; Childs, GE; Milhous, WK; Pang, L; Wimonwattratee, T1
Le Bras, M; Mazaudier, E; Raccurt, CP; Ripert, C; Schmitt, A1
Chakrabarti, NK; Nagaraj, C; Narasimham, MV1
Berger, M; Beytout, J; Cambon, M; Rey, M; Ringwald, P1
Hopfenmüller, W; Janitschke, K; Schultes, U; Weber, G; Weinke, T1
Bustos, MD; Danis, M; Diquet, B; Félix, R; Gay, F; Gentilini, M; Lyogoubi, A1
Eberlé, F; Gazin, P; Gelas, H; Hengy, C; Jambou, R; Kouka-Bemba, D1
Dutt, SC; Karmakar, P; Narasimham, MV; Sharma, RC1
Allen, MA; Bell, CA; Grogl, M; Hall, JE; Kyle, DE; Ohemeng, KA; Tidwell, RR1
Brandicourt, O; Carme, B; Gay, F; Gentilini, M; Le Bras, J; Mbitsi, A; Moudzeo, H; Ndounga, M; Sathounkazi, C1
Akogbeto, M; Chippaux, JP; Josse, R; Massougbodji, A; Sadeler, BC; Zohoun, T1
Broderson, JR; Collins, WE; Filipski, VK; Morris, CL; Ruebush, TK; Skinner, JC; Stanfill, PS1
Le Bras, J; Malhotra, K; Salmon, D; Vilde, JL1
De Boeck, H; Maguire, PA; Sherman, IW; Zidovetzki, R1
Go, ML; Lee, HS1
Andersen, BJ; Bygbjerg, IC; Pedersen, BK; Theander, TG1
Breckenridge, A1
Lapierre, J; Périn, M; Sureau, C1
Boudreau, EF; Childs, GE; Davidson, DE; Milhous, WK; Pang, L; Pooyindee, N; Wimonwattratee, T1
Afshar, A; Edrissian, GH; Emadi, AM; Ghorbani, M; Kanani, A; Mohsseni, G; Nasseri-Nejad, K; Satvat, MT1
Caligaris, S; Carosi, G; Castelli, F; Druilhe, P; Olliaro, P1
Abissègue, B; Garrigue, G; Gazin, P; Gelas, H; Ghogomu, NA; Hengy, C; Jambou, R; Kouka-Bemba, D; Le Bras, J1
Davis, DR; Lambros, C; Lewis, GE1
Chandrahas, RK; Choudhury, DS; Ghosh, SK; Ramanaiah, TV; Sharma, VP; Singh, N1
Gao, DQ; Liu, DQ; Liu, RJ; Qiu, CP; Ren, DX1
Andriamangatiana-Rason, MD; Coulanges, P; Deloron, P; Lepers, JP; Ramanamirija, JA1
Edrissian, GH1
Atiya, A; De Boeck, H; Sherman, IW; Zidovetzki, R1
Aderounmu, AF; Salako, LA; Simooya, OO1
Aina Adio, R; Fadeke Aderounmu, A; Laoye, AJ; Modupe Makinde, J; Salako, LA1
Bunnag, D; Harinasuta, T; Lasserre, R; Leimer, R; Vinijanont, S1
Diquet, B; Djibo, L; Druilhe, P; Felix, H; Jacquier, P1
Fadeke Aderounmu, A; Salako, LA1
Bunnag, D; Chittamas, S; Harinasuta, T; Looareesuwan, S; White, NJ1
Kollaritsch, H; Kollaritsch, R; Kremsner, P; Leimer, R; Mailer, H; Stemberger, H; Wiedermann, G1
Lwin, M; Zaw, M1
Walter, RD1
Bonnevie, O; Cordoliani, G; Dedet, JP; Germanetto, P; Le Bras, J1
Denis, MB; Giboda, M1
Brandicourt, O; Brasseur, P; Druilhe, P; Kouamouo, J; Moyou-Somo, R1
Bastien, P; Gentilini, M; Saliou, P1
Ihrahim, AM1
Brubaker, G; Draper, CC; Hills, M; Kilimali, VA1
Ali, S; Björkman, A; Lebbad, M; Warsame, M; Wernsdorfer, WH1
Druilhe, P; Gentilini, M; Stahel, E1
Kightlinger, LK; Kightlinger, MB1
Alpers, MP; Brabin, BJ; Eggelte, T; Klever, HJ; van der Kaay, HJ; Witte, AM1
Aderounmu, AF; Adio, RA; Laoye, JO; Makinde, JM; Salako, LA1
Bouchara, JP; Chabasse, D; De Gentile, L; Le Bras, J; Ligny, C; Rialland, X1
Rolfe, M1
Bellesi, N; Couto, AA; de Oliveira, SG; do Rosário, VE; Santos, MA1
Chanthavanich, P; Karbwang, J; Looareesuwan, S; Phillips, RE; Supanaranond, W; Turner, RC; Warrell, DA; White, NJ1
Ayub, M; Scott, TA1
Prapunwattana, P; Vanderkooi, G; Yuthavong, Y1
Babin-Chevaye, C; Labro, MT1
Chaumont, AJ; Kintz, P; Lamant, JM; Lugnier, AA; Mangin, P; Tracqui, A1
Childs, GE; Pooyindee, N; Wimonwattrawatee, T1
Boudreau, EF; Chen, C; Childs, GE; Häusler, B; Milhous, W; Pooyindee, N; Wimonwattrawatee, T1
Bugilimfura, L; Deloron, P; Neill, M; Ntilivamunda, A; Sexton, JD1
Ginsburg, H; Krugliak, M1
Burchard, GD; Winkler, E1
Björkman, A; Willcox, M1
Attanath, P; Chantavanich, P; Chongsuphajaisiddhi, T; Sabchareon, A; Sheth, UK; Singhasivanon, V; Wernsdorfer, WH1
Ho, KB; Mak, JW; Ramadas, M1
Long, GW; Mama, S; Ranoa, CP; Sangalang, RP; Sy, N1
Buck, RL; Long, GW; Ranoa, CP; Sangalang, RP; Sy, N; Watt, G1
Brockelman, CR; Bunnag, D; Satayavivad, J; Tan-ariya, P; Wongsawatkul, O1
Charmot, G; Le Bras, J; Simon, F1
Biaud, JM; Calmel, MB; Clausse, JL; Deloron, P; Hatin, I; Le Bras, J; Marchais, H; Porte, J; Ramanamirija, JA; Simon, F1
Fox, E; Khaliq, AA; Sarwar, M; Strickland, GT1
Huang, QL; Wu, Z; Zhang, KY; Zhou, JX1
Kuhlow, F; Walter, RD; Wittich, RM1
Bendtzen, K; Bygbjerg, IC; Svenson, M; Theander, TG1
Armstead, A; Campbell, CC; Collins, WE; Milhous, WK; Roberts, JM1
Brandicourt, O; Brasseur, P; Danis, M; Druilhe, P; Kouamouo, J; Moyou, SR1
Ginsburg, H; Krugliak, M; Zarchin, S1
Denis, MB1
Andersen, BJ; Bygbjerg, IC; Flachs, H; Jepsen, S; Larsen, PB; Theander, TG1
Bonanni, LC; Geary, TG; Ginsburg, H; Jensen, JB1
Bhattacharya, DN; Hall, AP1
Brandicourt, O; Brasseur, P; Danis, M; Diouf, F; Druilhe, P; Gay, F; Kombila, MY; Kouamouo, J; Moyou, RS; Richard-Lenoble, D1
Delacollette, C; Hendrix, L; Mpungu, MT; Ngimbi, NP; Wery, M1
Liu, DQ; Liu, RJ; Qiu, CP; Ren, DX1
Rathaur, S; Walter, RD1
Gajanana, A; Sinha, S; Vasisth, S1
Back, DJ; Karbwang, J; Looareesuwan, S; Molyneux, ME; Nagachinta, B; Phillips, RE; Warrell, DA; Wattanagoon, Y1
Glasner, H; Landscheidt, H; Niklewski, G1
Alexander, BM; Bowdre, JH; Desjardins, RE; Oduola, AM; Weatherly, NF1
Boudreau, EF; Pang, LW; Pavanand, K; Webster, HK; Yongvanitchit, K1
Alcantara, AK; Buck, RL; Rodriguez, CS; Smrkovski, LL; Uylangco, CV1
Dixon, KE; Phintuyothin, P; Pitaktong, U1
Peters, W1
Arias, AE; Cortes, GT; Espinal, CA; Guerra, P1
Canfield, CJ; Cosgriff, TM; Pamplin, CL; Willet, GP1
Gluzman, IY; Krogstad, DJ; Schlesinger, PH1
Nguyen-Dinh, P1
Delacollette, C; Gregory, MG; Mpungu, MT; Ngimbi, NP; Wery, M1
Froeling, FM; Van der Kaay, HJ; Wernsdorfer, WH1
Coulanges, P; Deloron, P; Le Bras, J; Ramanamirija, JA1
Charmot, G; Dupont, B; Lapresle, C; Le Bras, J; Sansonetti, P1
Li, GD1
Hogerzeil, HV; Hogewoning, AA; van der Kaay, HJ; van Doorn, JW; Wernsdorfer, WH1
Danis, M; Gentilini, M1
Salako, LA1
Alcantara, AK; Cross, JH; Sangalang, RP; Uylangco, CV1
Bruce-Chwatt, LJ1
Mrema, JE; Rieckmann, KH1
Demel, RA; Ginsburg, H1
Ferrante, A; Goh, DH1
Deloron, P; Le Bras, J1
Bunnag, D; Harinasuta, T; Wernsdorfer, WH1
Beale, GH; Chutmongkonkul, M; Thaithong, S1
Andrieu, B; Coulaud, JP; Deloron, P; Le Bras, J; Ricour, A; Savel, J1
Kofi Ekue, JM; Rwabwogo-Atenyi, J; Sheth, UK; Ulrich, AM1
Prüfer, L; von Sonnenburg, F1
Burchard, GD; Dietrich, M; Horstmann, RD; Wernsdorfer, WH1
Chiodini, PL; Ellis, CJ1
Alpers, MP; Davidson, WL; Jolley, D; Knowles, G1
Coulanges, P; Deloron, P; Dourado, HV; Hartmann, JF; Larouze, B; Le Bras, J1
Bendle, MS; Das, M; Dutt, SC; Karmakar, P; Sharma, GK1
Rosário, VE; Vasconcelos, MA1
Akood, MA; Carlin, JM; Jensen, JB; Vande Waa, JA1
Coulanges, P; Coulaud, JP; Deloron, P; Le Bras, J1
Königk, E; Putfarken, B1
Dutta, P; Fitch, CD1
Andrieu, B; Deloron, P; Hartmann, JF; Le Bras, J1
Childs, GE; Davidson, DE; Klayman, DL; Lambros, C; Notsch, JD; Scovill, JP1
Abdel-Rasoul, S; Königk, E; Mirtsch, S; Putfarken, B1
Dutta, GP; Singh, PP1
Merkli, B; Peters, W; Richle, R1
Govitrapong, P; Jearnpipatkul, A; Panijpan, B; Wilairat, P; Yuthavong, Y1
Brockelman, CR; Monkolkeha, S; Tanariya, P1
Fernex, M1
Abdalla, RE; El Gaddal, AA; Kouznetsov, RL; Payne, D; Rooney, W; Wernsdorfer, WH1
Howells, RE; Judge, BM1
Sweeney, TR1
Alvar, J; Amela, C; Benito, A; Molina, R; Roche, J1
Crevoisier, C; Mittelholzer, ML; Peters, W; Robinson, BL; Stürchler, D1
Grisolia, CK; Takahashi, CS1
Lench, P1
Eichenlaub, D; Jelinek, T; Löscher, T; Schelbert, P1
Del Nero, L; Lamizana, L; Nebié, I; Pietra, V2
Knobloch, J1
Croft, A1
Deacon, HE; Freese, JA; Sharp, BL1
Hoffman, SL; Johnson, A; Koech, D; Oloo, AJ; Weiss, WR1
Armengaud, M; Piccoli, S; Picot, N1
Basco, LK; Le Bras, J; Makler, MM; Marquet, F1
Calvert, L; Raeside, F; Walker, E1
Chatnugrob, P; Eamsila, C; Lasserre, R; Mittelholzer, ML; Nopavong Na Ayuthya, A; Singharaj, P; Stürchler, D; Webster, HK; Yooyen, P1
Yang, H; Yang, P; Yang, Y1
Edwards, G; Ward, SA; Winstanley, PA1
Baric, RS; Bright, P; Handy, J; Peel, SA; Yount, B1
Aouba, A; Guiguemde, TR; Lamizana, L; Ouedraogo, JB1
Hovette, P; Martet, G; Merouze, F; Nicolas, P; Touze, JE1
Basco, LK; Le Bras, J3
Bailey D [corrected to Bradley, D]; Bradley, D; Warhurst, D1
Casassus, P; Danis, M; Datry, A; Felix, H; Gay, F; Gentilini, M; Lortholary, O1
Huber, W; Hurt, N; Jaquet, C; Koella, JC; Mshinda, H; Tanner, M1
Cowman, AF; Karcz, S1
Bernard, KW; Campbell, CC; Eng, T; Hightower, AW; Lobel, HO; Miani, M1
DeFraites, RF; Hanson, RK; Sánchez, JL; Sharp, TW1
Fuchs, E; Funk, M; Naef, U; Nevill, C; Phillips-Howard, P; Schildknecht, J; Schlagenhauf, P; Steffen, R; Stürchler, D1
Allard, R; Gyorkos, TW; Milord, F1
Held, TK; Mansmann, U; Pohle, HD; Trautmann, M; Weinke, T1
Luxemburger, C; Nosten, F; ter Kuile, FO; White, NJ1
Basco, LK; Le Bras, J; Ramiliarisoa, O1
Aoki, M; Kamei, K; Miyashita, T; Nishiya, H; Ohyatsu, I; Ono, Y; Shibuya, T; Sugiyama, H; Tokumura, Y; Yamaguchi, M1
Fowler, VG; Irare, SG; Lemnge, M; Malecela, E; Mashaka, M; Mhina, J; Mtoi, R; Mtui, S1
Boudreau, E; Dausel, L; Hanson, R; Johnson, R; Novakowski, W; Redmond, D; Sanchez, J; Schuster, B1
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Ahmed, MA; Cox-Singh, J; Fatih, FA; Kocken, CH; Krishna, S; Pasini, EM; Siner, A; Singh, B; Staines, HM; Woon, LC1
Choi, AR; Kim, JH; Kim, YK; Yoon, S1
Chaijaroenkul, W; Muhamad, P; Na-Bangchang, K; Phompradit, P; Wisedpanichkij, R1
Eshleman, AJ; Hinrichs, DJ; Janowsky, A; Johnson, RA; Riscoe, MK; Smilkstein, MJ; Wolfrum, KM; Yang, J; Zabriskie, TM1
Aguiar, AC; Amaral, NS; De Marco, L; Krettli, AU; Pereira, DB1
David, K; Møller, CH1
Cui, L; Gupta, B; Miao, J; Sun, L; Wang, Z; Xu, S; Yang, Z1
Clark, J; Golenser, J; Guiguemde, WA; Guo, J; Guy, RK; Haynes, RK; Hunt, NH; Marciano, A1
Albrecht, L; Angerami, RN; Castiñeiras, CM; Costa, FT; Dos-Santos, JC; Garcia, MT; Lacerda, MV; Levy, CE; Lopes, SC; Moretti, ML1
Arboleda, M; Blair, S; Fernández, D; Garavito, G; Pabón, A; Segura, C1
Anstey, NM; Barber, BE; Dhanaraj, P; Grigg, MJ; Menon, J; Price, RN; Rajahram, G; von Seidlein, L; William, T; Yeo, TW1
Baret, E; Bercion, R; Camara, C; Diatta, B; Diémé, Y; Fall, B; Fall, KB; Fall, M; Mbaye, PS; Nakoulima, A; Pascual, A; Pradines, B; Wade, B; Wurtz, N1
Dahlstrom, S; Ferreira, PE; Franzén, O; Gil, JP; Lum, JK; Nosten, F; Osório, NS; Veiga, MI1
Bastiaens, GJ; Behet, MC; Bijker, EM; Graumans, W; Hermsen, CC; Obiero, JM; Sauerwein, RW; Schats, R; Scholzen, A; Teelen, K; van de Vegte-Bolmer, M; van Gemert, GJ; van Lieshout, L; Visser, LG1
Chandra, R; Dieng, Y; Djimdé, AA; Dunne, MW; Kain, KC; Mugyenyi, P; Mulenga, M; Oduro, AR; Ogutu, B; Robbins, J; Sagara, I; Sarkar, S; Sie, A; Tiono, AB; Wasunna, M1
Bijker, EM; Cockburn, I; Nganou-Makamdop, K; Sauerwein, RW; van Gemert, GJ; Zavala, F1
Buathong, N; Chanarat, N; Chann, S; Chaorattanakawee, S; Chuor, CM; Gosi, P; Heng, TK; Jacob, C; Kong, N; Kuntawunginn, W; Lanteri, CA; Lin, JT; Lon, C; Plowe, C; Prom, S; Saingam, P; Saunders, DL; Se, Y; Sea, D; Sriwichai, S; Sundrakes, S; Takala-Harrison, S; Tangthongchaiwiriya, K; Teja-Isavadharm, P; Tyner, SD; Yingyuen, K; Yom, Y1
Barnwell, JW; Goldman, I; Juma, E; Kariuki, S; Komino, F; Lucchi, NW; Okoth, SA; Onyona, P; Shi, YP; Udhayakumar, V; Wiegand, RE1
Cabrera, M; Cui, L1
Auburn, S; Handayuni, I; Marfurt, J; Noviyanti, R; Pava, Z; Poespoprodjo, JR; Price, RN; To, S; Trianty, L; Wirjanata, G1
Bannister-Tyrrell, M; Coosemans, M; d'Alessandro, U; Dierickx, S; Durnez, L; Erhart, A; Gerrets, R; Gryseels, C; Hausmann-Muela, S; Hoibak, S; Muela Ribera, J; Peeters Grietens, K; Phoeuk, P; Set, S; Sluydts, V; Suon, S; Tho, S; Trienekens, S; Uk, S1
Ramharter, M1
Anstey, NM; Barber, BE; Dhanaraj, P; Grigg, MJ; McCarthy, JS; Menon, J; Pasay, C; Price, RN; Rajahram, GS; von Seidlein, L; Wilkes, CS; William, T; Yeo, TW1
Anto, F; Ayanful-Torgby, R; Dery, V; Duah, NO; Matrevi, SA; Quashie, NB1
Akala, HM; Auschwitz, JM; Cheruiyot, AC; Gaona, HW; Hickman, MR; Johnson, JD; Kamau, E; Lee, PJ; Leed, SE; Murthy, T; Okello, CO; Talwar, M; Yeda, RA1
Bhardwaj, J; Goyal, M; Prakash, K; Puri, SK; Siddiqui, AJ; Soni, A1
Groger, M; Lötsch, F; Ramharter, M; Rehman, K; Sauerzopf, U; Veletzky, L1
Anstey, NM; Auburn, S; Barber, BE; Edstein, MD; Grigg, MJ; Menon, J; Price, RN; Rajahram, GS; Wilkes, CS; William, T; Yeo, TW1
Amalvict, R; Benoit, N; Diatta, B; Diawara, S; Diémé, Y; Fall, B; Fall, M; Gendrot, M; Madamet, M; Nakoulima, A; Pradines, B; Wade, B; Wade, KA1
Cabral, L; Cristiano, ML; Lobo, L; Nogueira, F; Sousa, Bd1
Muhamad, P; Na-Bangchang, K; Phompradit, P; Thiengsusuk, A1
Liu, XJ; Peng, HJ; Wei, HX; Xia, J; Zhou, LJ1
Amalvict, R; Benoit, N; Briolant, S; Diatta, B; Diawara, S; Diémé, Y; Fall, B; Fall, M; Gendrot, M; Kounta, MB; Madamet, M; Nakoulima, A; Pradines, B; Wade, B; Wade, KA1
Ataide, R; Beeson, JG; Boel, M; Drew, D; Fowkes, FJI; McGready, R; McLean, ARD; Nosten, F; Simpson, JA; Tsuboi, T1
Agnamey, P; Azas, N; Bentzinger, G; Cohen, A; Dassonville-Klimpt, A; Guillon, J; Hutter, S; Jonet, A; Moreau, S; Mullie, C; Savrimoutou, S; Schneider, J; Sonnet, P; Taudon, N1
Byaruhanga, O; Ceja, FG; Conrad, MD; Cooper, RA; Katairo, T; Nsobya, SL; Rasmussen, SA; Rosenthal, PJ; Tumwebaze, PK1
Maayan, N; Pace, C; Saunders, R; Sinclair, D; Tickell-Painter, M1
Annan, K; Ansah, C; Forkuo, AD; Gyan, B; Mancama, D; Mensah, KB; Theron, A; Wright, CW1
Choi, L; Garner, P; Gelband, H; Graves, PM1
Avery, SV; Islahudin, F; Lakhani, DH; Tindall, SM; Ting, KN; Vallières, C1
Ahmed, AM; Dang, TN; Dat, TV; Egan, TJ; Elhady, MT; Fukuda, M; Giang, HTN; Hirayama, K; Huy, NT; Huynh, LK; Kamel, MG; Kaneko, O; Mizukami, S; Mizuta, S; Mosaddeque, F; Tanaka, Y; Teklemichael, AA; Toan, DV; Vuong, NL1
Agarwal, P; Anvikar, AR; Pillai, CR; Srivastava, K1
Fairley, JK; Gutman, JR; Tan, KR; Wang, M1
Churcher, ZR; Johnson, PE; Slavkovic, S1
Horii, T; Tougan, T; Toya, Y; Uchihashi, K1
Banic, DM; Baptista, BO; Bianco-Junior, C; Carvalho, LJM; Cassiano, GC; Daniel-Ribeiro, CT; de Oliveira-Ferreira, J; Lima-Junior, JDC; Machado, RLD; Perce-Da-Silva, DS; Pratt-Riccio, LR; Riccio, EKP; Storti-Melo, LM; Torres, VR; Totino, PRR1
Brett-Major, D; Fraser, J; Hickey, PW; Mitra, I; Riddle, MS; Tribble, DR1
Gutman, JR; McKinney, KL; Tan, KR; Wu, HM1
Bah, S; Dabitao, D; Dama, S; Diakité, M; Diakité, SAS; Doumbia, S; Doumbouya, M; Guindo, MA; Keita, B; Konaté, DS; Sangaré, M; Sanogo, I; Traoré, K1
Boonyuen, U; Day, NPJ; Dondorp, AM; Imwong, M; Nosten, F; Pimpat, Y; Pukrittayakamee, S; Saralamba, N; Smithuis, F1
Bensalem, J; Bryksin, V; Fourrier, C; Hattersley, K; Hein, LK; Sargeant, TJ1
Anywar, DA; Auma, MA; Balikagala, B; Emoto, S; Fukuda, N; Hashimoto, M; Hirai, M; Horii, T; Ikeda, M; Kataoka, M; Katuro, OT; Kimura, E; Mita, T; Mori, T; Obwoya, PS; Odongo-Aginya, EI; Ogwang, M; Opio, W; Palacpac, NMQ; Sakurai-Yatsushiro, M; Sekihara, M; Tachibana, SI; Yamauchi, M; Yatsushiro, S1
Ahmad, SS; Rahi, M; Ranjan, V; Sharma, A1
Jongwutiwes, S; Kuamsab, N; Pattanawong, U; Putaporntip, C; Rojrung, R; Seethamchai, S; Weng Cheng, C; Yanmanee, S1
Barreto-Vieira, DF; Blanco, C; Bou-Habib, DC; Bozza, PT; Chaves, OA; Da Silva, APD; da Silva, CS; da Silva, MAN; Dias, SSG; Ferreira, AC; Fintelman-Rodrigues, N; Mattos, M; Miranda, MD; Owen, A; Paccanaro, A; Pereira-Dutra, F; Rajoli, RKR; Sacramento, CQ; Santos, SS; Soares, VC; Souza, TML; Temerozo, JR; Torres, M1
Corry, B; Martin, RE; Richards, SN; Shafik, SH1
Boroujeni, SS; Dehpour, AR; Jafari, RM; Karimi, E; Maleki, A; Mohammadi, P; Sabzevari, O; Shafaroodi, H; Solaimanian, S1
Iwanaga, S; Kamchonwongpaisan, S; Kubota, R; Nishi, T; Shinzawa, N; Srichairatanakool, S; Syafruddin, D; Uthaipibull, C; Yuda, M1
Bifani, P; Blackman, MJ; Christensen, P; Chua, ACY; Dhingra, SK; Fidock, DA; Kaneko, O; Kyle, DE; Lee, MCS; Matheson, J; Moon, RW; Racklyeft, A; Remmert, C; Rénia, L; Russell, B; Snounou, G; Suwanarusk, R; Ward, KE1
Bajpai, S; Banerjee, S; Kushwaha, R; Mandal, A; Mandal, AA; Yadav, AK1

Reviews

66 review(s) available for chloroquine and mefloquine

ArticleYear
Recent advances in malaria drug discovery.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure

2013
Approaches to protozoan drug discovery: phenotypic screening.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Drug Discovery; Humans; Molecular Structure; Neglected Diseases; Phenotype; Plasmodium falciparum; Protozoan Infections; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma cruzi

2013
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Quinoline hybrids and their antiplasmodial and antimalarial activities.
    European journal of medicinal chemistry, 2017, Oct-20, Volume: 139

    Topics: Antimalarials; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2017
Triazole derivatives and their antiplasmodial and antimalarial activities.
    European journal of medicinal chemistry, 2019, Mar-15, Volume: 166

    Topics: Animals; Antimalarials; Humans; Parasitic Sensitivity Tests; Plasmodium; Triazoles

2019
New dimensions in the field of antimalarial research against malaria resurgence.
    European journal of medicinal chemistry, 2019, Nov-01, Volume: 181

    Topics: Animals; Antimalarials; Artemisinins; Drug Resistance; Humans; Malaria; Plasmodium falciparum

2019
Drugs for the Treatment of Zika Virus Infection.
    Journal of medicinal chemistry, 2020, 01-23, Volume: 63, Issue:2

    Topics: Animals; Antiviral Agents; Drug Development; Drug Discovery; Humans; Viral Vaccines; Zika Virus; Zika Virus Infection

2020
Trends and controversies in the prophylaxis and treatment of malaria.
    Infectious agents and disease, 1992, Volume: 1, Issue:2

    Topics: Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine

1992
Plasmodium falciparum malaria in pregnancy: a review.
    British journal of obstetrics and gynaecology, 1992, Volume: 99, Issue:2

    Topics: Animals; Chloroquine; Critical Care; Female; Humans; Immunocompromised Host; Malaria, Falciparum; Mefloquine; Pregnancy; Pregnancy Complications, Infectious

1992
Risks and benefits of prophylactic antimalarial drugs.
    BMJ (Clinical research ed.), 1989, Oct-28, Volume: 299, Issue:6707

    Topics: Antimalarials; Chloroquine; Humans; Malaria; Mefloquine; Proguanil; Risk Factors

1989
The problem of drug resistance in malaria.
    Parasitology, 1985, Volume: 90 ( Pt 4)

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dapsone; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance, Microbial; Humans; India; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
Pharmacokinetics of antimalarial drugs: their therapeutic and toxicological implications.
    Annali dell'Istituto superiore di sanita, 1985, Volume: 21, Issue:3

    Topics: Adult; Amodiaquine; Animals; Antimalarials; Child; Chloroquine; Dapsone; Drug Combinations; Drug Resistance, Microbial; Half-Life; Humans; Kinetics; Male; Mefloquine; Mice; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Quinolines; Sulfadoxine; Sulfalene

1985
[Progress in immunodiagnosis and chemotherapy of protozoan infections].
    Der Internist, 1983, Volume: 24, Issue:11

    Topics: Amebiasis; Animals; Antibodies; Babesiosis; Chloroquine; Drug Resistance, Microbial; Giardiasis; Humans; Leishmaniasis; Malaria; Mefloquine; Pneumocystis; Pneumonia, Pneumocystis; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Quinolines; Serologic Tests; Sulfadoxine; Tetracycline; Toxoplasmosis; Trypanosomiasis

1983
[Urgent need for new antimalarias (author's transl)].
    Schweizerische Rundschau fur Medizin Praxis = Revue suisse de medecine Praxis, 1981, Jun-02, Volume: 70, Issue:23

    Topics: Antimalarials; Biological Availability; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Humans; Immunotherapy; Mefloquine; Piperidines; Pyrimethamine; Quinolines; Sulfadoxine; World Health Organization

1981
The present status of malaria chemotherapy: mefloquine, a novel antimalarial.
    Medicinal research reviews, 1981,Fall, Volume: 1, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Aotus trivirgatus; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dogs; Drug Therapy, Combination; Erythrocytes; Female; Humans; Lethal Dose 50; Macaca mulatta; Malaria; Male; Mefloquine; Mice; Plasmodium berghei; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Protein Conformation; Pyrimethamine; Quinolines; Rats; Stereoisomerism; Swine

1981
Clinical pharmacokinetics in the treatment of tropical diseases. Some applications and limitations.
    Clinical pharmacokinetics, 1994, Volume: 27, Issue:2

    Topics: Chloroquine; Diethylcarbamazine; Drug Resistance; Echinococcosis; Filariasis; Humans; Malaria; Mefloquine; Pharmacokinetics; Phenanthrenes; Pyrimethamine; Quinine; Sulfadoxine; Tropical Medicine

1994
Drug resistance and the P-glycoprotein homologues of Plasmodium falciparum.
    Seminars in cell biology, 1993, Volume: 4, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Chloroquine; Drug Resistance; Gene Expression; Mefloquine; Membrane Glycoproteins; Phenotype; Protozoan Proteins

1993
[Malaria: the most important emergency in subjects returning from the tropics].
    Schweizerische medizinische Wochenschrift, 1993, May-01, Volume: 123, Issue:17

    Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Emergencies; Humans; Malaria; Malaria, Falciparum; Mefloquine; Plasmodium; Pyrimethamine; Quinidine; Quinine; Sulfadoxine

1993
Prophylaxis against malaria for travellers from the United Kingdom. Malaria Reference Laboratory and the Ross Institute.
    BMJ (Clinical research ed.), 1993, May-08, Volume: 306, Issue:6887

    Topics: Animals; Child; Child, Preschool; Chloroquine; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Proguanil; Travel

1993
Quinoline antimalarials: mechanisms of action and resistance.
    International journal for parasitology, 1997, Volume: 27, Issue:2

    Topics: Animals; Antimalarials; Blood Proteins; Chloroquine; Drug Resistance; Erythrocytes; Hemoglobins; Humans; Mefloquine; Membrane Proteins; Plasmodium; Quinine; Quinolines

1997
[The treatment of malaria].
    Nederlands tijdschrift voor geneeskunde, 1997, Sep-13, Volume: 141, Issue:37

    Topics: Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Female; Humans; Infant, Newborn; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Phenanthrenes; Pregnancy; Primaquine

1997
Malaria prevention in travelers.
    American family physician, 1999, May-01, Volume: 59, Issue:9

    Topics: Animals; Antimalarials; Bedding and Linens; Chloroquine; Doxycycline; Humans; Malaria; Malaria, Falciparum; Mefloquine; Patient Education as Topic; Plasmodium falciparum; Primaquine; Proguanil; Protective Clothing; Teaching Materials; Travel

1999
[Neurological toxicity of antifungal and antiprotozoal drugs].
    Ryoikibetsu shokogun shirizu, 1999, Issue:27 Pt 2

    Topics: Amphotericin B; Antifungal Agents; Antimalarials; Antiprotozoal Agents; Antitrichomonal Agents; Central Nervous System Diseases; Chloroquine; Humans; Mefloquine; Metronidazole; Quinine

1999
Comparative efficacy and safety of chloroquine and alternative antimalarial drugs: a meta-analysis from six African countries.
    East African medical journal, 1999, Volume: 76, Issue:6

    Topics: Africa, Eastern; Africa, Western; Amodiaquine; Antimalarials; Chloroquine; Drug Combinations; Drug Costs; Humans; Malaria; Mefloquine; Patient Selection; Phenanthrenes; Pyrimethamine; Quinine; Safety; Sulfadoxine; Treatment Outcome

1999
[Malaria in Norway--diagnosis, treatment and prevention].
    Tidsskrift for den Norske laegeforening : tidsskrift for praktisk medicin, ny raekke, 2000, May-30, Volume: 120, Issue:14

    Topics: Antimalarials; Chloroquine; Humans; Insect Bites and Stings; Malaria; Malaria, Falciparum; Mefloquine; Norway; Practice Guidelines as Topic; Primaquine; Travel

2000
Combination therapy for malaria in Africa: hype or hope?
    Bulletin of the World Health Organization, 2000, Volume: 78, Issue:12

    Topics: Africa; Antimalarials; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Cross-Cultural Comparison; Half-Life; Humans; Insecticide Resistance; Malaria; Mefloquine; Pyrimethamine; Self Medication; Sesquiterpenes; Sulfadoxine; Thailand

2000
Antimalarial chemoprophylaxis in infants and children.
    Paediatric drugs, 2001, Volume: 3, Issue:2

    Topics: Antimalarials; Child; Child, Preschool; Chloroquine; Doxycycline; Humans; Infant; Malaria, Falciparum; Mefloquine; Primaquine

2001
Malaria chemoprophylaxis in the age of drug resistance. I. Currently recommended drug regimens.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2001, Jul-15, Volume: 33, Issue:2

    Topics: Animals; Antimalarials; Atovaquone; Azithromycin; Chloroquine; Drug Resistance; Health Planning Guidelines; Humans; Malaria, Falciparum; Mefloquine; Naphthoquinones; Plasmodium falciparum; Primaquine; Proguanil

2001
[Recommendations for prevention of malaria in patients with epilepsy].
    Der Nervenarzt, 2001, Volume: 72, Issue:6

    Topics: Adolescent; Adult; Aged; Antimalarials; Chloroquine; Electroencephalography; Epilepsy; Female; Humans; Malaria; Male; Mefloquine; Middle Aged

2001
[Malaria--chemoprophylaxis 2001].
    Therapeutische Umschau. Revue therapeutique, 2001, Volume: 58, Issue:6

    Topics: Africa; Antimalarials; Asia; Atovaquone; Chloroquine; Contraindications; Doxycycline; Drug Combinations; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum; Mefloquine; Naphthoquinones; Practice Guidelines as Topic; Proguanil; South America; Switzerland; Travel

2001
The Italian army standpoint on malaria chemoprophylaxis.
    Medecine tropicale : revue du Corps de sante colonial, 2001, Volume: 61, Issue:1

    Topics: Antimalarials; Chloroquine; Doxycycline; Drug Resistance; Drug Therapy, Combination; Endemic Diseases; Humans; Italy; Malaria; Malaria, Falciparum; Mefloquine; Military Personnel; Proguanil; Tropical Climate

2001
The malaria threat.
    Medecine tropicale : revue du Corps de sante colonial, 2001, Volume: 61, Issue:1

    Topics: Antimalarials; Chloroquine; Doxycycline; Drug Resistance; Health Policy; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Military Personnel; Proguanil

2001
Current drugs for antimalarial chemoprophylaxis: a review of efficacy and safety.
    Journal of travel medicine, 2001, Volume: 8, Issue:Suppl 3

    Topics: Antimalarials; Atovaquone; Chloroquine; Doxycycline; Humans; Malaria; Mefloquine; Naphthoquinones; Primaquine; Proguanil

2001
Clinical practice: antimalarial prophylaxis in patients with epilepsy [corrected].
    Epilepsy research, 2002, Volume: 51, Issue:1-2

    Topics: Antimalarials; Chemoprevention; Chloroquine; Epilepsy; Humans; Malaria; Mefloquine; Risk Factors; Travel; United Kingdom

2002
Safety evaluation of the drugs available to prevent malaria.
    Expert opinion on drug safety, 2002, Volume: 1, Issue:1

    Topics: Adult; Animals; Antimalarials; Chemical and Drug Induced Liver Injury; Chloroquine; Humans; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Randomized Controlled Trials as Topic; Travel

2002
Military aviators, special operations forces, and causal malaria prophylaxis.
    Military medicine, 2003, Volume: 168, Issue:12

    Topics: Aminoquinolines; Antimalarials; Atovaquone; Aviation; Chloroquine; Doxycycline; Drug Combinations; Humans; Malaria; Mefloquine; Military Personnel; Naphthoquinones; Primaquine; Proguanil; United States

2003
Genetic and biochemical aspects of drug resistance in malaria parasites.
    Current drug targets. Infectious disorders, 2004, Volume: 4, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dihydropteroate Synthase; Drug Resistance; Drug Resistance, Multiple; Humans; Linkage Disequilibrium; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Mutation; Phenanthrenes; Plasmodium falciparum; Plasmodium vivax; Protozoan Proteins; Pyrimethamine; Sulfadoxine; Tetrahydrofolate Dehydrogenase

2004
[Combined antimalarial therapy using artemisinin].
    Parassitologia, 2004, Volume: 46, Issue:1-2

    Topics: Amodiaquine; Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Chloroquine; Doxycycline; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Plasmodium; Pyrimethamine; Quinine; Sesquiterpenes; Sulfadoxine

2004
[Malaria: prophylaxis, treatment, stand-by medication. A single mosquito bite suffices].
    MMW Fortschritte der Medizin, 2004, Jun-17, Volume: 146, Issue:25

    Topics: Adult; Antimalarials; Artemether; Artemisinins; Atovaquone; Chloroquine; Climate; Doxycycline; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria; Male; Mefloquine; Naphthoquinones; Pregnancy; Proguanil; Risk Factors; Self Medication; Sesquiterpenes; Time Factors; Travel

2004
Malaria: prevention in travellers.
    Clinical evidence, 2003, Issue:10

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Doxycycline; Female; Humans; Insect Repellents; Insecticides; Malaria; Mefloquine; Mosquito Control; Naphthoquinones; Pregnancy; Proguanil; Travel

2003
Malaria: prevention in travellers.
    Clinical evidence, 2004, Issue:11

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Clothing; Doxycycline; Female; Humans; Insect Repellents; Insecticides; Malaria; Mefloquine; Mosquito Control; Naphthoquinones; Pregnancy; Proguanil; Travel

2004
Effectiveness of antimalarial drugs.
    The New England journal of medicine, 2005, Apr-14, Volume: 352, Issue:15

    Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Life Cycle Stages; Malaria; Mefloquine; Patient Compliance; Plasmodium; Primaquine; Pyrimethamine; Quinine; Secondary Prevention; Sulfadoxine; Treatment Failure

2005
Malaria: prevention in travellers.
    Clinical evidence, 2004, Issue:12

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Clothing; Doxycycline; Female; Humans; Insect Repellents; Insecticides; Malaria; Mefloquine; Mosquito Control; Naphthoquinones; Pregnancy; Travel

2004
Malaria: uncomplicated, caused by Plasmodium falciparum.
    Clinical evidence, 2005, Issue:13

    Topics: Amodiaquine; Antimalarials; Artemether; Artemisinins; Artesunate; Chloroquine; Dapsone; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Mefloquine; Proguanil; Pyrimethamine; Sesquiterpenes; Sulfadoxine

2005
[Malaria chemoprophylaxis].
    Ugeskrift for laeger, 2005, Oct-17, Volume: 167, Issue:42

    Topics: Antimalarials; Atovaquone; Chloroquine; Contraindications; Doxycycline; Drug Combinations; Female; Humans; Infant; Malaria, Falciparum; Mefloquine; Naphthoquinones; Practice Guidelines as Topic; Pregnancy; Proguanil; Risk Assessment; Travel

2005
Antimalarial multi-drug resistance in Asia: mechanisms and assessment.
    Current topics in microbiology and immunology, 2005, Volume: 295

    Topics: Animals; Antimalarials; Asia; ATP-Binding Cassette Transporters; Chloroquine; Dihydropteroate Synthase; DNA, Protozoan; Drug Resistance, Multiple; Folic Acid Antagonists; Genes, Protozoan; Humans; Malaria, Falciparum; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Plasmodium falciparum; Protozoan Proteins; Tetrahydrofolate Dehydrogenase

2005
[Cytochrome P-450 and the response to antimalarial drugs].
    Revista panamericana de salud publica = Pan American journal of public health, 2006, Volume: 19, Issue:1

    Topics: Administration, Oral; Adult; Amodiaquine; Animals; Antimalarials; Biotransformation; Child; Chloroquine; Cytochrome P-450 Enzyme System; Databases as Topic; Disease Models, Animal; Genotype; Humans; Malaria; Malaria, Falciparum; Mefloquine; Mice; Murinae; Mutation; Nutritional Status; Phenotype; Plasmodium berghei; Polymorphism, Genetic; Proguanil; Rats

2006
Antimalarial drugs: recent advances in molecular determinants of resistance and their clinical significance.
    Cellular and molecular life sciences : CMLS, 2006, Volume: 63, Issue:14

    Topics: Africa; Amino Alcohols; Animals; Antimalarials; Artemisinins; Asia, Southeastern; Biological Transport; Calcium-Transporting ATPases; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Drug Therapy, Combination; Gene Amplification; Humans; Malaria, Falciparum; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Models, Biological; Multidrug Resistance-Associated Proteins; Mutation; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Quinine; Sesquiterpenes

2006
Current malaria status and distribution of drug resistance in East and Southeast Asia with special focus to Thailand.
    The Tohoku journal of experimental medicine, 2007, Volume: 211, Issue:2

    Topics: Age Factors; Animals; Antimalarials; Artemisinins; Asia, Southeastern; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Plasmodium; Quinine; Sesquiterpenes; Sex Factors; Sulfadoxine

2007
Assessment of the relative advantage of various artesunate-based combination therapies by a multi-treatment Bayesian random-effects meta-analysis.
    The American journal of tropical medicine and hygiene, 2007, Volume: 77, Issue:6

    Topics: Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Bayes Theorem; Chloroquine; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Malaria; Mefloquine; Pyrimethamine; Randomized Controlled Trials as Topic; Sesquiterpenes; Sulfadoxine; Treatment Outcome

2007
Clinical inquiries. What is the most effective and safe malaria prophylaxis during pregnancy?
    The Journal of family practice, 2008, Volume: 57, Issue:1

    Topics: Abnormalities, Drug-Induced; Antimalarials; Chemoprevention; Chloroquine; Doxycycline; Female; Humans; Malaria; Mefloquine; Practice Guidelines as Topic; Pregnancy; Pregnancy Complications, Infectious

2008
Drugs for preventing malaria in travellers.
    The Cochrane database of systematic reviews, 2009, Oct-07, Issue:4

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Doxycycline; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Primaquine; Proguanil; Randomized Controlled Trials as Topic; Travel

2009
Azithromycin for treating uncomplicated malaria.
    The Cochrane database of systematic reviews, 2011, Feb-16, Issue:2

    Topics: Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Atovaquone; Azithromycin; Chloroquine; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Proguanil; Pyrimethamine; Randomized Controlled Trials as Topic; Sulfadoxine; Treatment Failure

2011
Malaria: prevention in travellers.
    BMJ clinical evidence, 2010, Jul-12, Volume: 2010

    Topics: Antimalarials; Bedding and Linens; Chloroquine; Humans; Malaria; Mefloquine; Primaquine; Travel

2010
Pharmacokinetics of antimalarials in pregnancy: a systematic review.
    Clinical pharmacokinetics, 2011, Nov-01, Volume: 50, Issue:11

    Topics: Anti-Bacterial Agents; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Proguanil; Pyrimethamine; Quinine; Sulfadoxine

2011
Primaquine for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2012, Sep-12, Issue:9

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2012
Malaria.
    Lancet (London, England), 2014, Feb-22, Volume: 383, Issue:9918

    Topics: Africa South of the Sahara; Amodiaquine; Animals; Anopheles; Antimalarials; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Drug Administration Schedule; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Female; Humans; Insecticide-Treated Bednets; Insecticides; Malaria; Malaria Vaccines; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Pregnancy; Pregnancy Complications, Infectious; Primary Prevention; Pyrimethamine; Quinine; Quinolines; Seasons; Sulfadoxine

2014
Monitoring antimalarial drug efficacy in the Greater Mekong Subregion: an overview of in vivo results from 2008 to 2010.
    The Southeast Asian journal of tropical medicine and public health, 2013, Volume: 44 Suppl 1

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Directly Observed Therapy; Drug Resistance; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Parasitemia; Quinolines

2013
Primaquine or other 8-aminoquinoline for reducing P. falciparum transmission.
    The Cochrane database of systematic reviews, 2014, Jun-30, Issue:6

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2014
Primaquine or other 8-aminoquinoline for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2015, Feb-19, Issue:2

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2015
WITHDRAWN: Drugs for preventing malaria in travellers.
    The Cochrane database of systematic reviews, 2015, Oct-05, Issue:10

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Doxycycline; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Primaquine; Proguanil; Randomized Controlled Trials as Topic; Travel

2015
Risk of drug resistance in Plasmodium falciparum malaria therapy-a systematic review and meta-analysis.
    Parasitology research, 2017, Volume: 116, Issue:2

    Topics: Amodiaquine; Antimalarials; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Risk; Sulfadoxine

2017
Mefloquine for preventing malaria during travel to endemic areas.
    The Cochrane database of systematic reviews, 2017, 10-30, Volume: 10

    Topics: Adult; Antimalarials; Atovaquone; Child; Chloroquine; Doxycycline; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Primaquine; Proguanil; Randomized Controlled Trials as Topic; Travel-Related Illness

2017
Primaquine or other 8-aminoquinolines for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2018, 02-02, Volume: 2

    Topics: Adult; Antimalarials; Artemisinins; Child; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Non-Randomized Controlled Trials as Topic; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine; Time Factors

2018
Mefloquine as a prophylaxis for malaria needs to be revisited.
    International journal for parasitology. Drugs and drug resistance, 2021, Volume: 17

    Topics: Antimalarials; Chloroquine; Humans; Malaria; Mefloquine; Military Personnel

2021
Transition Metal Complexes as Antimalarial Agents: A Review.
    ChemMedChem, 2023, 10-04, Volume: 18, Issue:19

    Topics: Antimalarials; Chloroquine; Coordination Complexes; Drug Resistance; Humans; Malaria; Malaria, Falciparum; Mefloquine; Plasmodium falciparum

2023

Trials

47 trial(s) available for chloroquine and mefloquine

ArticleYear
Fansimef for prophylaxis of malaria: a double-blind randomized placebo controlled trial.
    The Southeast Asian journal of tropical medicine and public health, 1992, Volume: 23, Issue:4

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Double-Blind Method; Drug Combinations; Humans; Incidence; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Pyrimethamine; Sulfadoxine; Treatment Outcome

1992
Mefloquine-sulphadoxine-pyrimethamine (Fansimef, Roche) in the prophylaxis of Plasmodium falciparum malaria: a double-blind, comparative, placebo-controlled study.
    Annals of tropical medicine and parasitology, 1992, Volume: 86, Issue:6

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Double-Blind Method; Drug Combinations; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Pyrimethamine; Sulfadoxine

1992
Clinical trials of mefloquine with tetracycline.
    The Southeast Asian journal of tropical medicine and public health, 1992, Volume: 23, Issue:3

    Topics: Acute Disease; Adolescent; Adult; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Prospective Studies; Pyrimethamine; Sulfadoxine; Tetracycline

1992
Evaluation of the relative efficacy of various antimalarial drugs in Nigerian children under five years of age suffering from acute uncomplicated falciparum malaria.
    Annals of tropical medicine and parasitology, 1992, Volume: 86, Issue:1

    Topics: Acute Disease; Amodiaquine; Antimalarials; Child, Preschool; Chloroquine; Drug Administration Schedule; Drug Combinations; Female; Humans; Infant; Infant, Newborn; Malaria, Falciparum; Male; Mefloquine; Nigeria; Pyrimethamine; Quinine; Sulfadoxine

1992
Comparison of mefloquine, chloroquine plus pyrimethamine-sulfadoxine (Fansidar), and chloroquine as malarial prophylaxis in eastern Thailand.
    The Southeast Asian journal of tropical medicine and public health, 1991, Volume: 22, Issue:2

    Topics: Adolescent; Adult; Aged; Analysis of Variance; Animals; Antimalarials; Cambodia; Chloroquine; Confidence Intervals; Double-Blind Method; Drug Combinations; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Middle Aged; Pyrimethamine; Sulfadoxine; Survival Analysis; Thailand

1991
Sensitivity of Plasmodium falciparum to chloroquine, amodiaquine and mefloquine in Ibadan, Nigeria.
    African journal of medicine and medical sciences, 1988, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; In Vitro Techniques; Infant; Malaria; Male; Mefloquine; Nigeria; Plasmodium falciparum; Quinolines

1988
Comparison of the susceptibility of falciparum malaria to mefloquine-sulphadoxine-pyrimethamine and chloroquine in Nigeria.
    African journal of medicine and medical sciences, 1988, Volume: 17, Issue:4

    Topics: Animals; Antimalarials; Child; Chloroquine; Clinical Trials as Topic; Drug Administration Schedule; Drug Combinations; Drug Resistance; Female; Humans; Malaria; Male; Mefloquine; Nigeria; Plasmodium falciparum; Pyrimethamine; Quinolines; Random Allocation; Sulfadoxine; Sulfanilamides

1988
Trials of mefloquine in vivax and of mefloquine plus 'fansidar' in falciparum malaria.
    Lancet (London, England), 1985, Apr-20, Volume: 1, Issue:8434

    Topics: Adolescent; Adult; Chloroquine; Clinical Trials as Topic; Double-Blind Method; Drug Combinations; Drug Therapy, Combination; Follow-Up Studies; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Plasmodium vivax; Pyrimethamine; Quinolines; Random Allocation; Sulfadoxine; Sulfanilamides

1985
Tolerability of long-term malaria prophylaxis with the combination mefloquine + sulfadoxine + pyrimethamine (Fansimef): results of a double blind field trial versus chloroquine in Nigeria.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:4

    Topics: Adolescent; Adult; Animals; Antimalarials; Aspartate Aminotransferases; Blood Cell Count; Child; Chloroquine; Clinical Trials as Topic; Double-Blind Method; Drug Combinations; Drug Therapy, Combination; Female; gamma-Glutamyltransferase; Humans; Malaria; Male; Mefloquine; Middle Aged; Nigeria; Plasmodium falciparum; Pyrimethamine; Quinolines; Random Allocation; Sulfadoxine; Sulfanilamides

1988
Sensitivity of Plasmodium falciparum to mefloquine-sulphadoxine-pyrimethamine (Fansimef) in vivo and to mefloquine alone in vitro in Nigeria.
    Annals of tropical medicine and parasitology, 1988, Volume: 82, Issue:4

    Topics: Animals; Antimalarials; Child; Chloroquine; Drug Combinations; Drug Evaluation; Drug Resistance; Female; Humans; Malaria; Male; Mefloquine; Nigeria; Plasmodium falciparum; Pyrimethamine; Quinolines; Random Allocation; Sulfadoxine; Sulfanilamides

1988
Parasitologic and clinical efficacy of 25 and 50 mg/kg of chloroquine for treatment of Plasmodium falciparum malaria in Rwandan children.
    The American journal of tropical medicine and hygiene, 1988, Volume: 38, Issue:2

    Topics: Animals; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; Infant; Malaria; Male; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Rwanda

1988
A phase-III clinical trial of mefloquine in children with chloroquine-resistant falciparum malaria in Thailand.
    Bulletin of the World Health Organization, 1987, Volume: 65, Issue:2

    Topics: Child; Child, Preschool; Chloroquine; Clinical Trials as Topic; Drug Resistance, Microbial; Female; Humans; Malaria; Male; Mefloquine; Plasmodium falciparum; Quinolines; Thailand

1987
A clinical trial of mefloquine in the treatment of Plasmodium vivax malaria.
    The American journal of tropical medicine and hygiene, 1985, Volume: 34, Issue:3

    Topics: Adult; Chloroquine; Clinical Trials as Topic; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Plasmodium vivax; Primaquine; Quinolines; Random Allocation

1985
The problem of drug resistance in malaria.
    Parasitology, 1985, Volume: 90 ( Pt 4)

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dapsone; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance, Microbial; Humans; India; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
A comparative clinical study of mefloquine and chloroquine in the treatment of vivax malaria.
    The Southeast Asian journal of tropical medicine and public health, 1985, Volume: 16, Issue:4

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium vivax; Quinolines

1985
A phase II clinical trial of mefloquine in patients with chloroquine-resistant falciparum malaria in Thailand.
    Bulletin of the World Health Organization, 1983, Volume: 61, Issue:2

    Topics: Adolescent; Adult; Aged; Antimalarials; Chloroquine; Clinical Trials as Topic; Double-Blind Method; Drug Resistance, Microbial; Humans; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines; Random Allocation

1983
A double-blind comparative clinical trial of mefloquine and chloroquine in symptomatic falciparum malaria.
    Bulletin of the World Health Organization, 1983, Volume: 61, Issue:4

    Topics: Adolescent; Adult; Animals; Antimalarials; Chloroquine; Clinical Trials as Topic; Double-Blind Method; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines

1983
The present status of malaria chemotherapy: mefloquine, a novel antimalarial.
    Medicinal research reviews, 1981,Fall, Volume: 1, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Aotus trivirgatus; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dogs; Drug Therapy, Combination; Erythrocytes; Female; Humans; Lethal Dose 50; Macaca mulatta; Malaria; Male; Mefloquine; Mice; Plasmodium berghei; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Protein Conformation; Pyrimethamine; Quinolines; Rats; Stereoisomerism; Swine

1981
Malaria prophylaxis. Toxicity of mefloquine is similar to that of other chemoprophylaxis.
    BMJ (Clinical research ed.), 1995, Jul-15, Volume: 311, Issue:6998

    Topics: Chloroquine; Double-Blind Method; Humans; Malaria; Mefloquine; Proguanil

1995
Daily primaquine is effective for prophylaxis against falciparum malaria in Kenya: comparison with mefloquine, doxycycline, and chloroquine plus proguanil.
    The Journal of infectious diseases, 1995, Volume: 171, Issue:6

    Topics: Adolescent; Child; Chloroquine; Doxycycline; Drug Administration Schedule; Humans; Kenya; Malaria, Falciparum; Mefloquine; Primaquine; Proguanil

1995
Prevention of Plasmodium falciparum malaria by Fansimef and Lariam in the northeastern part of Thailand.
    The Southeast Asian journal of tropical medicine and public health, 1993, Volume: 24, Issue:4

    Topics: Adult; Animals; Antibodies, Protozoan; Blood; Chloroquine; Drug Combinations; Humans; Malaria, Falciparum; Male; Mefloquine; Military Personnel; Plasmodium falciparum; Pyrimethamine; Sulfadoxine; Thailand

1993
Long-term malaria prophylaxis with weekly mefloquine.
    Lancet (London, England), 1993, Apr-03, Volume: 341, Issue:8849

    Topics: Africa, Western; Chloroquine; Cohort Studies; Drug Administration Schedule; Drug Therapy, Combination; Humans; Long-Term Care; Malaria, Falciparum; Mefloquine; Proguanil

1993
Mefloquine or doxycycline prophylaxis in US troops in Somalia.
    Lancet (London, England), 1993, Apr-17, Volume: 341, Issue:8851

    Topics: Animals; Chloroquine; Doxycycline; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Military Personnel; Patient Compliance; Plasmodium falciparum; Premedication; Somalia; United States

1993
Tolerability of prophylactic Lariam regimens.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1993, Volume: 44, Issue:3

    Topics: Adult; Anorexia; Chloroquine; Depression; Dizziness; Double-Blind Method; Dreams; Drug Tolerance; Eye; Humans; Irritable Mood; Malaria, Falciparum; Male; Mefloquine; Military Personnel; Nausea; Psychomotor Performance; Sleep; Sleep Initiation and Maintenance Disorders; Travel; United States

1993
Recent military experience with malaria chemoprophylaxis.
    The Medical journal of Australia, 1993, Apr-05, Volume: 158, Issue:7

    Topics: Antimalarials; Australia; Chloroquine; Dapsone; Doxycycline; Drug Administration Schedule; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Military Personnel; Primaquine; Pyrimethamine

1993
Efficacy of oral and intravenous artesunate in male Tanzanian adults with Plasmodium falciparum malaria and in vitro susceptibility to artemisinin, chloroquine, and mefloquine.
    The American journal of tropical medicine and hygiene, 1995, Volume: 53, Issue:6

    Topics: Administration, Oral; Adolescent; Adult; Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drugs, Chinese Herbal; Erythrocytes; Humans; Injections, Intravenous; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Parasitemia; Plasmodium falciparum; Recurrence; Sesquiterpenes; Tanzania

1995
Comparability of treatment groups and risk factors for parasitemia at the first antenatal clinic visit in a study of malaria treatment and prevention in pregnancy in rural Malawi.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:1 Suppl

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Humans; Malaria, Falciparum; Malawi; Mefloquine; Parasitemia; Pregnancy; Pregnancy Complications, Parasitic; Prenatal Care; Prospective Studies; Risk Factors; Rural Population; Seasons

1996
Malaria parasite infection during pregnancy and at delivery in mother, placenta, and newborn: efficacy of chloroquine and mefloquine in rural Malawi.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:1 Suppl

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Fetal Blood; Humans; Malaria, Falciparum; Malawi; Mefloquine; Obstetric Labor Complications; Parasitemia; Placenta Diseases; Pregnancy; Pregnancy Complications, Parasitic; Prospective Studies; Rural Population; Treatment Outcome

1996
Objectives and methodology in a study of malaria treatment and prevention in pregnancy in rural Malawi: The Mangochi Malaria Research Project.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:1 Suppl

    Topics: Antimalarials; Chloroquine; Female; Fetal Death; Follow-Up Studies; Humans; Infant, Low Birth Weight; Infant, Newborn; Infectious Disease Transmission, Vertical; Longitudinal Studies; Malaria, Falciparum; Malawi; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Prospective Studies; Research Design; Rural Population; Surveys and Questionnaires; Treatment Outcome

1996
[Malaria chemoprophylaxis: tolerance and compliance with mefloquine and proguanil/chloroquine combination in French tourists].
    Bulletin de la Societe de pathologie exotique (1990), 1997, Volume: 90, Issue:4

    Topics: Adult; Antimalarials; Chloroquine; Drug Combinations; Female; France; Humans; Kenya; Malaria; Male; Mefloquine; Patient Compliance; Proguanil; Senegal; Surveys and Questionnaires; Travel

1997
Response of falciparum malaria to different antimalarials in Myanmar.
    Bulletin of the World Health Organization, 1999, Volume: 77, Issue:3

    Topics: Adolescent; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Therapy, Combination; Humans; Infant; Malaria, Falciparum; Mefloquine; Myanmar; Pyrimethamine; Sulfadoxine

1999
In vivo-in vitro model for the assessment of clinically relevant antimalarial cross-resistance.
    The American journal of tropical medicine and hygiene, 2001, Volume: 65, Issue:6

    Topics: Adult; Animals; Antimalarials; Artemisinins; Chloroquine; Cross Reactions; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Models, Biological; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Recurrence; Sesquiterpenes

2001
Efficacy of chloroquine, sulfadoxine-pyrimethamine, and mefloquine for the treatment of uncomplicated Plasmodium falciparum malaria on the north coast of Peru.
    The American journal of tropical medicine and hygiene, 2003, Volume: 68, Issue:1

    Topics: Adolescent; Adult; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Peru; Plasmodium falciparum; Pyrimethamine; Sulfadoxine; Treatment Outcome

2003
Malaria in a cohort of Javanese migrants to Indonesian Papua.
    Annals of tropical medicine and parasitology, 2003, Volume: 97, Issue:6

    Topics: Adolescent; Adult; Antimalarials; Child; Chloroquine; Cross-Sectional Studies; Female; Follow-Up Studies; Humans; Incidence; Indonesia; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Papua New Guinea; Parasitemia; Prevalence; Transients and Migrants

2003
Randomized comparison of chloroquine plus sulfadoxine-pyrimethamine versus artesunate plus mefloquine versus artemether-lumefantrine in the treatment of uncomplicated falciparum malaria in the Lao People's Democratic Republic.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2004, Oct-15, Volume: 39, Issue:8

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Infant; Laos; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Pyrimethamine; Sesquiterpenes; Sulfadoxine

2004
Comparison of chloroquine, sulfadoxine/pyrimethamine, mefloquine and mefloquine-artesunate for the treatment of falciparum malaria in Kachin State, North Myanmar.
    Tropical medicine & international health : TM & IH, 2004, Volume: 9, Issue:11

    Topics: Adolescent; Adult; Age Distribution; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Therapy, Combination; Female; Hemoglobins; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Myanmar; Pyrimethamine; Recurrence; Sesquiterpenes; Sulfadoxine; Treatment Failure

2004
Efficacy of chloroquine + sulfadoxine--pyrimethamine, mefloquine + artesunate and artemether + lumefantrine combination therapies to treat Plasmodium falciparum malaria in the Chittagong Hill Tracts, Bangladesh.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 2005, Volume: 99, Issue:10

    Topics: Adolescent; Antimalarials; Artemether; Artemisinins; Artesunate; Bangladesh; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Treatment Outcome

2005
A randomized trial comparing the efficacy of four treatment regimens for uncomplicated falciparum malaria in Assam state, India.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 2006, Volume: 100, Issue:2

    Topics: Adolescent; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Therapy, Combination; Female; Humans; India; Infant; Malaria, Falciparum; Male; Mefloquine; Prospective Studies; Pyrimethamine; Quinolines; Sesquiterpenes; Sulfadoxine; Treatment Outcome

2006
Mefloquine is highly efficacious against chloroquine-resistant Plasmodium vivax malaria and Plasmodium falciparum malaria in Papua, Indonesia.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2006, Apr-15, Volume: 42, Issue:8

    Topics: Adult; Antimalarials; Child; Chloroquine; Drug Resistance; Humans; Indonesia; Japan; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Treatment Outcome

2006
Dramatically decreased therapeutic efficacy of chloroquine and sulfadoxine-pyrimethamine, but not mefloquine, in southern Benin.
    Tropical medicine & international health : TM & IH, 2007, Volume: 12, Issue:7

    Topics: Administration, Oral; Animals; Antigens, Protozoan; Antimalarials; Benin; Child, Preschool; Chloroquine; DNA, Protozoan; Drug Combinations; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Merozoite Surface Protein 1; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Pyrimethamine; Sulfadoxine; Treatment Failure; Treatment Outcome

2007
Prevention of malaria during pregnancy: assessing the effect of the distribution of IPTp through the national policy in Benin.
    The American journal of tropical medicine and hygiene, 2011, Volume: 84, Issue:2

    Topics: Adult; Antimalarials; Benin; Chloroquine; Drug Combinations; Female; Health Policy; HIV Infections; Humans; Infant, Low Birth Weight; Infant, Newborn; Malaria; Maternal Age; Mefloquine; Multivariate Analysis; Placenta; Pregnancy; Pregnancy Complications, Parasitic; Pyrimethamine; Risk Factors; Sulfadoxine; Young Adult

2011
A study protocol for a randomised open-label clinical trial of artesunate-mefloquine versus chloroquine in patients with non-severe Plasmodium knowlesi malaria in Sabah, Malaysia (ACT KNOW trial).
    BMJ open, 2014, Aug-19, Volume: 4, Issue:8

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Female; Humans; Malaria; Malaysia; Male; Mefloquine; Plasmodium knowlesi; Research Design; Severity of Illness Index

2014
Sporozoite immunization of human volunteers under mefloquine prophylaxis is safe, immunogenic and protective: a double-blind randomized controlled clinical trial.
    PloS one, 2014, Volume: 9, Issue:11

    Topics: Adolescent; Adult; Antibodies; Antimalarials; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Chloroquine; DNA, Protozoan; Double-Blind Method; Erythrocytes; Granzymes; Healthy Volunteers; Humans; Immunity, Cellular; Lysosomal-Associated Membrane Protein 1; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Sporozoites; Young Adult

2014
Efficacy and safety of a combination of azithromycin and chloroquine for the treatment of uncomplicated Plasmodium falciparum malaria in two multi-country randomised clinical trials in African adults.
    Malaria journal, 2014, Nov-25, Volume: 13

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Azithromycin; Chloroquine; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Parasitemia; Plasmodium falciparum; Polymerase Chain Reaction; Treatment Outcome; Uganda; Young Adult; Zambia

2014
Artesunate-mefloquine versus chloroquine for treatment of uncomplicated Plasmodium knowlesi malaria in Malaysia (ACT KNOW): an open-label, randomised controlled trial.
    The Lancet. Infectious diseases, 2016, Volume: 16, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Therapy, Combination; Female; Humans; Malaria; Malaysia; Male; Mefloquine; Middle Aged; Plasmodium knowlesi; Young Adult

2016
Efficacy of Artesunate-mefloquine for Chloroquine-resistant Plasmodium vivax Malaria in Malaysia: An Open-label, Randomized, Controlled Trial.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2016, 06-01, Volume: 62, Issue:11

    Topics: Adolescent; Adult; Aged; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; Infant; Malaria, Vivax; Male; Mefloquine; Middle Aged; Plasmodium vivax; Treatment Outcome; Young Adult

2016
Changing Antimalarial Drug Sensitivities in Uganda.
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:12

    Topics: Adolescent; Amodiaquine; Antimalarials; Artemisinins; Aspartic Acid Endopeptidases; Child; Child, Preschool; Chloroquine; Drug Resistance; Ethanolamines; Female; Fluorenes; Gene Expression; Humans; Infant; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Mutation; Parasitic Sensitivity Tests; Plasmodium falciparum; Protozoan Proteins; Quinolines; Uganda; Young Adult

2017

Other Studies

457 other study(ies) available for chloroquine and mefloquine

ArticleYear
From a cytotoxic agent to the discovery of a novel antimalarial agent.
    Bioorganic & medicinal chemistry letters, 2013, Jan-15, Volume: 23, Issue:2

    Topics: Antimalarials; Caco-2 Cells; Drug Discovery; Drug Resistance; Humans; Inhibitory Concentration 50; Morpholines; Piperidones; Plasmodium falciparum

2013
Comparative antimalarial activities and ADME profiles of ozonides (1,2,4-trioxolanes) OZ277, OZ439, and their 1,2-dioxolane, 1,2,4-trioxane, and 1,2,4,5-tetraoxane isosteres.
    Journal of medicinal chemistry, 2013, Mar-28, Volume: 56, Issue:6

    Topics: Absorption; Adamantane; Animals; Antimalarials; Dioxolanes; Heterocyclic Compounds; Heterocyclic Compounds, 1-Ring; Male; Mice; Peroxides; Plasmodium berghei; Plasmodium falciparum; Spiro Compounds; Structure-Activity Relationship; Tetraoxanes

2013
3,5-bis(benzylidene)-4-piperidones and related N-acyl analogs: a novel cluster of antimalarials targeting the liver stage of Plasmodium falciparum.
    Bioorganic & medicinal chemistry, 2013, Dec-01, Volume: 21, Issue:23

    Topics: Animals; Antimalarials; Drug Resistance; Hep G2 Cells; Humans; Liver; Malaria; Malaria, Falciparum; Mice; Piperidones; Plasmodium berghei; Plasmodium falciparum

2013
Design, synthesis and biological evaluation of 3-[4-(7-chloro-quinolin-4-yl)-piperazin-1-yl]-propionic acid hydrazones as antiprotozoal agents.
    European journal of medicinal chemistry, 2014, Mar-21, Volume: 75

    Topics: Antiprotozoal Agents; Drug Design; Entamoeba histolytica; Entamoebiasis; Humans; Hydrazones; Malaria, Falciparum; Plasmodium falciparum; Propionates

2014
Medicinal chemistry optimization of antiplasmodial imidazopyridazine hits from high throughput screening of a SoftFocus kinase library: part 1.
    Journal of medicinal chemistry, 2014, Mar-27, Volume: 57, Issue:6

    Topics: Animals; Antimalarials; Biological Availability; Drug Design; Drug Resistance; Drug Stability; Gene Library; Half-Life; High-Throughput Screening Assays; Imidazoles; Malaria; Malaria, Falciparum; Mice; Mice, SCID; Parasitic Sensitivity Tests; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Protein Kinase Inhibitors; Protein Kinases; Pyridazines; Rats; Structure-Activity Relationship

2014
Second generation steroidal 4-aminoquinolines are potent, dual-target inhibitors of the botulinum neurotoxin serotype A metalloprotease and P. falciparum malaria.
    Journal of medicinal chemistry, 2014, May-22, Volume: 57, Issue:10

    Topics: Aminoquinolines; Animals; Antimalarials; Botulinum Toxins, Type A; Chick Embryo; Chloroquine; Drug Resistance; Hep G2 Cells; Humans; Metalloproteases; Molecular Docking Simulation; Plasmodium falciparum; Protease Inhibitors; Structure-Activity Relationship

2014
Design, synthesis and biological evaluation of novel 4-alkapolyenylpyrrolo[1,2-a]quinoxalines as antileishmanial agents--part III.
    European journal of medicinal chemistry, 2014, Jun-23, Volume: 81

    Topics: Animals; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Female; Hep G2 Cells; Humans; Leishmania; Macrophages; Mice; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinoxalines; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2014
Sphingolipid analogues inhibit development of malaria parasites.
    ACS medicinal chemistry letters, 2012, Jan-12, Volume: 3, Issue:1

    Topics:

2012
Identification and optimization of an aminoalcohol-carbazole series with antimalarial properties.
    ACS medicinal chemistry letters, 2013, Nov-14, Volume: 4, Issue:11

    Topics:

2013
Blood schizontocidal and gametocytocidal activity of 3-hydroxy-N'-arylidenepropanehydrazonamides: a new class of antiplasmodial compounds.
    Journal of medicinal chemistry, 2014, Oct-09, Volume: 57, Issue:19

    Topics: Animals; Antimalarials; Chloroquine; Malaria; Mice; Parasitemia; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium berghei; Plasmodium falciparum; Rats; Structure-Activity Relationship

2014
Synthesis of novel triazole-linked mefloquine derivatives: biological evaluation against Plasmodium falciparum.
    Bioorganic & medicinal chemistry letters, 2014, Dec-01, Volume: 24, Issue:23

    Topics: Antimalarials; Humans; Malaria; Mefloquine; Molecular Structure; Plasmodium falciparum; Structure-Activity Relationship; Triazoles

2014
The synthesis, antimalarial activity and CoMFA analysis of novel aminoalkylated quercetin analogs.
    Bioorganic & medicinal chemistry letters, 2015, Jan-15, Volume: 25, Issue:2

    Topics: Antimalarials; Humans; Malaria; Models, Molecular; Molecular Structure; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quercetin; Stereoisomerism

2015
Prodrugs of reverse fosmidomycin analogues.
    Journal of medicinal chemistry, 2015, Feb-26, Volume: 58, Issue:4

    Topics: Animals; Antimalarials; Cell Survival; Disease Models, Animal; Dose-Response Relationship, Drug; Fosfomycin; HeLa Cells; Humans; Malaria; Mice; Mice, SCID; Molecular Structure; Plasmodium berghei; Plasmodium falciparum; Prodrugs; Structure-Activity Relationship

2015
Synthesis of 3-azabicyclo[3.2.2]nonanes and their antiprotozoal activities.
    Bioorganic & medicinal chemistry letters, 2015, Apr-01, Volume: 25, Issue:7

    Topics: Administration, Oral; Animals; Antiprotozoal Agents; Azabicyclo Compounds; Disease Models, Animal; Dose-Response Relationship, Drug; Injections, Intravenous; Male; Mice; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Rats; Structure-Activity Relationship; Tissue Distribution; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2015
Synthesis and antimalarial evaluation of prodrugs of novel fosmidomycin analogues.
    Bioorganic & medicinal chemistry letters, 2015, Volume: 25, Issue:10

    Topics: Antimalarials; Drug Evaluation, Preclinical; Fosfomycin; Humans; Prodrugs

2015
A Novel Pyrazolopyridine with in Vivo Activity in Plasmodium berghei- and Plasmodium falciparum-Infected Mouse Models from Structure-Activity Relationship Studies around the Core of Recently Identified Antimalarial Imidazopyridazines.
    Journal of medicinal chemistry, 2015, Nov-12, Volume: 58, Issue:21

    Topics: Animals; Antimalarials; Ether-A-Go-Go Potassium Channels; Humans; Liver; Malaria; Malaria, Falciparum; Mice; Plasmodium berghei; Plasmodium falciparum; Pyrazoles; Pyridines; Rats; Structure-Activity Relationship

2015
Reinvestigating Old Pharmacophores: Are 4-Aminoquinolines and Tetraoxanes Potential Two-Stage Antimalarials?
    Journal of medicinal chemistry, 2016, Jan-14, Volume: 59, Issue:1

    Topics: Aminoquinolines; Animals; Antimalarials; Drug Evaluation, Preclinical; Ether-A-Go-Go Potassium Channels; Hemin; Hepatocytes; Humans; In Vitro Techniques; Liver; Mice; Microsomes, Liver; Parasite Load; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship; Tetraoxanes

2016
Conjugation of N-acylhydrazone and 1,2,4-oxadiazole leads to the identification of active antimalarial agents.
    Bioorganic & medicinal chemistry, 2016, 11-15, Volume: 24, Issue:22

    Topics: Animals; Antimalarials; Cell Survival; Dose-Response Relationship, Drug; Hep G2 Cells; Humans; Hydrazones; Malaria; Mice; Molecular Structure; Oxadiazoles; Plasmodium falciparum; Structure-Activity Relationship

2016
Evaluation of the anti-malarial activity and cytotoxicity of 2,4-diamino-pyrimidine-based kinase inhibitors.
    European journal of medicinal chemistry, 2016, Nov-29, Volume: 124

    Topics: Animals; Antimalarials; Cell Line, Tumor; Chlorocebus aethiops; Drug Design; Humans; Molecular Docking Simulation; Plasmodium falciparum; Protein Conformation; Protein Kinase Inhibitors; Protein Kinases; Protozoan Proteins; Pyrimidines; Vero Cells

2016
Identification of a Potential Antimalarial Drug Candidate from a Series of 2-Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle.
    Journal of medicinal chemistry, 2016, 11-10, Volume: 59, Issue:21

    Topics: Animals; Antimalarials; Disease Models, Animal; Dose-Response Relationship, Drug; Ether-A-Go-Go Potassium Channels; Hep G2 Cells; Humans; Life Cycle Stages; Malaria; Mice; Mice, SCID; Microsomes, Liver; Molecular Structure; Parasitic Diseases, Animal; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Pyrazines; Solubility; Structure-Activity Relationship; Water

2016
2,8-bis(trifluoromethyl)quinoline analogs show improved anti-Zika virus activity, compared to mefloquine.
    European journal of medicinal chemistry, 2017, Feb-15, Volume: 127

    Topics: Animals; Antiviral Agents; Chlorocebus aethiops; Drug Design; Mefloquine; Quinolines; Structure-Activity Relationship; Vero Cells; Virus Replication; Zika Virus

2017
3-Hydroxy-N'-arylidenepropanehydrazonamides with Halo-Substituted Phenanthrene Scaffolds Cure P. berghei Infected Mice When Administered Perorally.
    Journal of medicinal chemistry, 2017, 07-27, Volume: 60, Issue:14

    Topics: Amides; Animals; Antimalarials; Hep G2 Cells; Humans; Hydrazones; Malaria; Mice; Phenanthrenes; Plasmodium berghei; Stereoisomerism; Structure-Activity Relationship

2017
Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P
    European journal of medicinal chemistry, 2018, Jun-25, Volume: 154

    Topics: Amino Acids; Antimalarials; Aspartic Acid Endopeptidases; Dose-Response Relationship, Drug; Molecular Structure; Parasitic Sensitivity Tests; Peptidomimetics; Plasmodium falciparum; Protease Inhibitors; Structure-Activity Relationship

2018
3,3'-Disubstituted 5,5'-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity.
    Journal of medicinal chemistry, 2019, 03-14, Volume: 62, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Mice; Molecular Structure; Plasmodium; Species Specificity; Structure-Activity Relationship; Triazines

2019
New hybrid trifluoromethylquinolines as antiplasmodium agents.
    Bioorganic & medicinal chemistry, 2019, 03-15, Volume: 27, Issue:6

    Topics: Animals; Antimalarials; Cell Line; Drug Discovery; Erythrocytes; Halogenation; Haplorhini; Humans; Malaria; Methylation; Mice; Plasmodium berghei; Plasmodium falciparum; Quinolines

2019
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
    Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7

    Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship

2019
Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in
    Journal of medicinal chemistry, 2021, 03-11, Volume: 64, Issue:5

    Topics: Amides; Antimalarials; Drug Resistance, Microbial; Hemeproteins; Hemoglobins; Hep G2 Cells; Humans; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Small Molecule Libraries; Structure-Activity Relationship; Tetrazoles

2021
Novel molecule combinations and corresponding hybrids targeting artemisinin-resistant Plasmodium falciparum parasites.
    Bioorganic & medicinal chemistry letters, 2021, 05-01, Volume: 39

    Topics: Antimalarials; Artemisinins; Atovaquone; Dose-Response Relationship, Drug; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Triclosan

2021
Discovery and development of 2-aminobenzimidazoles as potent antimalarials.
    European journal of medicinal chemistry, 2021, Oct-05, Volume: 221

    Topics: Antimalarials; Benzimidazoles; Dose-Response Relationship, Drug; Drug Discovery; HEK293 Cells; Humans; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship

2021
Design, synthesis, and characterization of novel aminoalcohol quinolines with strong in vitro antimalarial activity.
    European journal of medicinal chemistry, 2022, Jan-15, Volume: 228

    Topics: Amino Alcohols; Animals; Antimalarials; Cell Line; Cricetulus; Dose-Response Relationship, Drug; Drug Design; Ether-A-Go-Go Potassium Channels; Female; Humans; Malaria; Mice; Mice, Inbred BALB C; Microsomes, Liver; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2022
Sensitivity status of Plasmodium falciparum to chloroquine, amodiaquine, quinine, mefloquine and sulfadoxine/pyrimethamine in a tribal population of District Sundargarh, Orissa.
    Indian journal of malariology, 1992, Volume: 29, Issue:4

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; India; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1992
[Current health information for Spanish travellers to tropical areas].
    Enfermedades infecciosas y microbiologia clinica, 1992, Volume: 10, Issue:5

    Topics: Centers for Disease Control and Prevention, U.S.; Chloroquine; Health Education; Humans; Information Services; Malaria; Mefloquine; Proguanil; Spain; Travel; United States; World Health Organization

1992
[Treatment of malaria in children in France].
    Pediatrie, 1992, Volume: 47, Issue:5

    Topics: Antimalarials; Child; Chloroquine; France; Humans; Malaria, Cerebral; Malaria, Falciparum; Mefloquine; Phenanthrenes; Quinine

1992
Selection for high-level chloroquine resistance results in deamplification of the pfmdr1 gene and increased sensitivity to mefloquine in Plasmodium falciparum.
    The EMBO journal, 1992, Volume: 11, Issue:8

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chloroquine; Chromosome Deletion; Chromosome Mapping; Dose-Response Relationship, Drug; Drug Resistance; Gene Amplification; Mefloquine; Membrane Glycoproteins; Plasmodium falciparum; Restriction Mapping; Verapamil

1992
Inhibition of the Salmonella typhi oral vaccine strain, Ty21a, by mefloquine and chloroquine.
    The Journal of infectious diseases, 1992, Volume: 166, Issue:6

    Topics: Chloroquine; Humans; Mefloquine; Salmonella typhi; Typhoid-Paratyphoid Vaccines; Vaccines, Attenuated

1992
Chloroquine-resistant Plasmodium vivax: it may be a common problem.
    The Medical journal of Australia, 1992, Sep-21, Volume: 157, Issue:6

    Topics: Animals; Chloroquine; Drug Resistance; Female; Humans; Malaria, Vivax; Male; Mefloquine; Plasmodium vivax; Primaquine

1992
Effects of antimalarial chemoprophylactic agents on the viability of the Ty21a typhoid vaccine strain.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1992, Volume: 15, Issue:6

    Topics: Chloroquine; Mefloquine; Microbial Sensitivity Tests; Salmonella typhi; Typhoid-Paratyphoid Vaccines

1992
Proposals for a new therapeutic strategy for simple Plasmodium falciparum malaria attacks in Cameroon.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1992, Volume: 43, Issue:2

    Topics: Administration, Oral; Aminoquinolines; Amodiaquine; Animals; Antimalarials; Cameroon; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine

1992
Use of antiprotozoan and anthelmintic drugs during pregnancy: side-effects and contra-indications.
    The Journal of infection, 1992, Volume: 25, Issue:1

    Topics: Abnormalities, Drug-Induced; Anthelmintics; Antimalarials; Antiprotozoal Agents; Chloroquine; Contraindications; Female; Helminthiasis; Humans; Infant, Newborn; Mefloquine; Pregnancy; Pregnancy Complications, Infectious; Protozoan Infections

1992
Mefloquine-halofantrine cross-resistance in Plasmodium falciparum induced by intermittent mefloquine pressure.
    The American journal of tropical medicine and hygiene, 1992, Volume: 47, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine

1992
Susceptibility of Plasmodium falciparum strains to mefloquine in an urban area in Senegal.
    Bulletin of the World Health Organization, 1992, Volume: 70, Issue:3

    Topics: Adolescent; Adult; Aminoquinolines; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Humans; In Vitro Techniques; Infant; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum

1992
Type RI resistance to halofantrine in West Africa.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1991, Volume: 42, Issue:4

    Topics: Animals; Antimalarials; Biological Availability; Chloroquine; Cote d'Ivoire; Drug Resistance; Follow-Up Studies; France; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Phenanthrenes; Plasmodium falciparum; Quinine; Recurrence; Travel

1991
Effect on sodium sulphate on the adsorption of chloroquine and mefloquine to activated charcoal.
    East African medical journal, 1991, Volume: 68, Issue:6

    Topics: Adsorption; Charcoal; Chloroquine; Humans; Mefloquine; Sulfates

1991
[Malaria in the republic of São Tomé and Principe. Epidemiologic evaluation and chemoresistance of P. falciparum].
    Bulletin de la Societe de pathologie exotique (1990), 1991, Volume: 84, Issue:3

    Topics: Age Factors; Animals; Antimalarials; Atlantic Islands; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Seasons; Sex Factors; Splenomegaly

1991
Severe falciparum malaria (21 cases).
    Intensive care medicine, 1991, Volume: 17, Issue:8

    Topics: Adolescent; Adult; Child, Preschool; Chloroquine; Exchange Transfusion, Whole Blood; Female; Humans; Infusions, Intravenous; Intensive Care Units; Malaria, Cerebral; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Quinine; Respiration, Artificial; Retrospective Studies

1991
Malaria prophylaxis.
    The Central African journal of medicine, 1991, Volume: 37, Issue:10

    Topics: Chloroquine; Drug Resistance; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Travel; Zimbabwe

1991
Drug use and design in the nineties.
    Acta Leidensia, 1991, Volume: 60, Issue:1

    Topics: Aminoquinolines; Amodiaquine; Antimalarials; Artemisinins; Calcium Channel Blockers; Chloroquine; Humans; Malaria; Mefloquine; Naphthoquinones; Phenanthrenes; Primaquine; Quinine; Sesquiterpenes; Sulfadoxine

1991
[Prophylaxis of malaria].
    Presse medicale (Paris, France : 1983), 1991, Feb-16, Volume: 20, Issue:6

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Mefloquine

1991
[Prevention and treatment of malaria in expatriates living in Black Africa. Influence of chemoresistance. Investigations conducted in Brazzaville (Congo)].
    Presse medicale (Paris, France : 1983), 1991, Jun-22, Volume: 20, Issue:24

    Topics: Adolescent; Adult; Aged; Amodiaquine; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Congo; Drug Combinations; Drug Resistance, Microbial; Europe; Humans; Infant; Infant, Newborn; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1991
Resistance to antimalarials by Plasmodium falciparum in Arso PIR, Irian Jaya, Indonesia.
    The American journal of tropical medicine and hygiene, 1991, Volume: 44, Issue:6

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Indonesia; Malaria; Male; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1991
Infection of Aotus vociferans monkeys with different strains of Plasmodium falciparum.
    The Journal of parasitology, 1991, Volume: 77, Issue:4

    Topics: Amodiaquine; Animals; Anopheles; Cebidae; Chloroquine; Malaria; Mefloquine; Plasmodium falciparum; Time Factors

1991
Standard and reduced doses of mefloquine for treatment of Plasmodium falciparum in Tanzania: whole blood concentrations in relation to adverse reactions, in vivo response, and in vitro susceptibility.
    The American journal of tropical medicine and hygiene, 1991, Volume: 45, Issue:2

    Topics: Adolescent; Animals; Child; Chloroquine; Drug Administration Schedule; Humans; Malaria; Mefloquine; Plasmodium falciparum; Tanzania

1991
[Malaria of importation in the child: epidemiological, clinical and therapeutic analysis. Apropos of 70 cases observed in a pediatric hospital in Paris].
    Bulletin de la Societe de pathologie exotique (1990), 1991, Volume: 84, Issue:2

    Topics: Africa; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Infant; Malaria; Malaria, Falciparum; Mefloquine

1991
Imported Plasmodium falciparum malaria in American travelers to Africa. Implications for prevention strategies.
    JAMA, 1991, Jan-16, Volume: 265, Issue:3

    Topics: Africa, Eastern; Africa, Western; Animals; Chloroquine; Drug Resistance; Malaria; Mefloquine; Plasmodium falciparum; Population Surveillance; Travel; United States

1991
Chloroquine-resistant Plasmodium falciparum with reduced sensitivity in vitro to mefloquine and quinine in Zaria, northern Nigeria.
    The Journal of tropical medicine and hygiene, 1991, Volume: 94, Issue:2

    Topics: Animals; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Infant; Malaria; Mefloquine; Nigeria; Plasmodium falciparum; Quinine

1991
The chemical basis for the ferriprotoporphyrin IX-chloroquine complex induced lipid peroxidation.
    Biochimica et biophysica acta, 1991, May-24, Volume: 1074, Issue:1

    Topics: Animals; Antimalarials; Apoproteins; Benzoates; Benzoic Acid; Catalase; Chloroquine; Hemin; Hydrogen-Ion Concentration; Iron; Kinetics; Lipid Peroxidation; Liposomes; Mefloquine; Oxygen; Primaquine; Quinine; Rats; Spectrum Analysis; Superoxide Dismutase; Transferrin

1991
Widespread in vitro resistance to chloroquine of Plasmodium falciparum in the Congo, 1987.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1991, Volume: 42, Issue:1

    Topics: Adolescent; Animals; Child; Child, Preschool; Chloroquine; Congo; Drug Resistance; Humans; Infant; Malaria; Mefloquine; Plasmodium falciparum; Quinine; Regression Analysis

1991
In vitro and clinical correlates of mefloquine resistance of Plasmodium falciparum in eastern Thailand.
    The American journal of tropical medicine and hygiene, 1991, Volume: 44, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Butylated Hydroxytoluene; Chloroquine; Drug Resistance; Drugs, Chinese Herbal; Mefloquine; Molecular Structure; Phenanthrenes; Plasmodium falciparum; Pyridines; Pyrimethamine; Quinine; Sesquiterpenes; Thailand

1991
[Imported malaria in Bordeaux in 1989. Epidemiologic, clinical and therapeutic study of 71 cases].
    Bulletin de la Societe de pathologie exotique (1990), 1990, Volume: 83, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Female; France; Humans; Malaria; Male; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Travel

1990
An in-vitro profile of the action of four antimalarials on indigenous cases of Plasmodium falciparum malaria in Karnataka.
    The Journal of communicable diseases, 1990, Volume: 22, Issue:4

    Topics: Amodiaquine; Animals; Chloroquine; Drug Resistance, Microbial; Malaria; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine

1990
[A case of Plasmodium falciparum malaria contracted in Guinea-Bissau during chemoprophylaxis with chloroquine].
    Presse medicale (Paris, France : 1983), 1990, Nov-03, Volume: 19, Issue:36

    Topics: Animals; Chloroquine; Drug Resistance; Female; Humans; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Quinine

1990
Recommendations for the prevention of malaria among travelers.
    MMWR. Recommendations and reports : Morbidity and mortality weekly report. Recommendations and reports, 1990, Mar-09, Volume: 39, Issue:RR-3

    Topics: Adult; Animals; Antimalarials; Breast Feeding; Centers for Disease Control and Prevention, U.S.; Child; Chloroquine; Doxycycline; Drug Resistance; Female; Humans; Malaria; Mefloquine; Plasmodium falciparum; Pregnancy; Pregnancy Complications, Infectious; Primaquine; Proguanil; Risk Factors; Travel; United States

1990
Malaria prophylaxis in travellers to tropical Africa.
    Klinische Wochenschrift, 1990, Mar-05, Volume: 68, Issue:5

    Topics: Africa; Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Plasmodium falciparum; Proguanil; Pyrimethamine; Sulfadoxine; Travel

1990
[Cross resistance to mefloquine and halofantrine in a case of P. falciparum malaria contracted in Sierra Leone].
    Bulletin de la Societe de pathologie exotique (1990), 1990, Volume: 83, Issue:1

    Topics: Adult; Animals; Antimalarials; Chloroquine; Cross Reactions; Drug Resistance; Humans; Malaria; Male; Mefloquine; Phenanthrenes; Plasmodium falciparum

1990
[Uncomplicated malaria attack in an area with high resistance to chloroquine. 3. The use of second-choice oral drug treatment].
    Bulletin de la Societe de pathologie exotique (1990), 1990, Volume: 83, Issue:1

    Topics: Adolescent; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Infant; Malaria; Male; Mefloquine; Plasmodium falciparum; Pyrimethamine; Sulfadoxine; Sulfanilamides

1990
Micro in vitro assessment of Plasmodium falciparum sensitivity to chloroquine and mefloquine in Gujarat.
    Indian journal of malariology, 1990, Volume: 27, Issue:1

    Topics: Animals; Chloroquine; Drug Resistance; Humans; India; Mefloquine; Plasmodium falciparum

1990
Structure-activity relationships of analogs of pentamidine against Plasmodium falciparum and Leishmania mexicana amazonensis.
    Antimicrobial agents and chemotherapy, 1990, Volume: 34, Issue:7

    Topics: Animals; Chloroquine; Drug Resistance, Microbial; Leishmania mexicana; Mefloquine; Pentamidine; Plasmodium falciparum; Structure-Activity Relationship

1990
[Plasmodium falciparum drug resistance in the Congo. Evaluation of surveys carried out from 1985 to 1989].
    Bulletin de la Societe de pathologie exotique (1990), 1990, Volume: 83, Issue:2

    Topics: Adolescent; Aminoquinolines; Amodiaquine; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Congo; Drug Combinations; Drug Resistance; Humans; Infant; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1990
[Development of chemoresistance of Plasmodium falciparum to chloroquine and mefloquine in Benin between 1980 and 1989].
    Bulletin de la Societe de pathologie exotique (1990), 1990, Volume: 83, Issue:3

    Topics: Animals; Benin; Child; Chloroquine; Drug Resistance; Humans; Mefloquine; Plasmodium falciparum

1990
The Peruvian III strain of Plasmodium brasilianum in Saimiri sciureus boliviensis monkeys.
    The Journal of parasitology, 1990, Volume: 76, Issue:5

    Topics: Animals; Anopheles; Chloroquine; Malaria; Mefloquine; Monkey Diseases; Recurrence; Saimiri

1990
Potentiation of chloroquine activity against Plasmodium falciparum by the peroxidase-hydrogen peroxide system.
    Antimicrobial agents and chemotherapy, 1990, Volume: 34, Issue:10

    Topics: Animals; Cells, Cultured; Chloroquine; Drug Synergism; Hydrogen Peroxide; Hypoxanthine; Hypoxanthines; Mefloquine; Peroxidases; Plasmodium falciparum; Quinine

1990
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with lipids extracted from normal human erythrocytes.
    Molecular and biochemical parasitology, 1990, Jan-01, Volume: 38, Issue:1

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Deuterium; Erythrocytes; Humans; Magnetic Resonance Spectroscopy; Mefloquine; Membrane Lipids; Phosphatidylethanolamines; Phosphorus Isotopes; Quinacrine; Quinine

1990
Effects of mefloquine on the release of marker enzymes from the rat liver crude lysosomal fraction.
    Japanese journal of pharmacology, 1990, Volume: 53, Issue:2

    Topics: Acid Phosphatase; Animals; Biomarkers; Chloroquine; Glucuronidase; In Vitro Techniques; Liver; Lysosomes; Mefloquine; Proteins; Rats

1990
Effects of chloroquine, mefloquine and quinine on natural killer cell activity in vitro. An analysis of the inhibitory mechanism.
    Allergy, 1986, Volume: 41, Issue:7

    Topics: Cell Adhesion; Chloroquine; Cytotoxicity, Immunologic; Humans; Immunity, Cellular; Immunity, Innate; In Vitro Techniques; Interferons; Interleukin-2; Killer Cells, Natural; Mefloquine; Quinine; Quinolines

1986
[The role of mefloquine in the prevention of malaria].
    Bulletin de l'Academie nationale de medecine, 1989, Volume: 173, Issue:9

    Topics: Africa; Chloroquine; Drug Resistance, Microbial; Drug Tolerance; France; Humans; Malaria; Mefloquine

1989
A comparison of the in vitro activities of amodiaquine and desethylamodiaquine against isolates of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1989, Volume: 40, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinolines; Thailand

1989
The response of Plasmodium falciparum to chloroquine and mefloquine in Bandar-Abbas and Minab areas, Hormozgan Province, southern Iran.
    The Journal of tropical medicine and hygiene, 1989, Volume: 92, Issue:2

    Topics: Adolescent; Adult; Animals; Child; Chloroquine; Drug Resistance; Humans; Iran; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines

1989
Ultrastructure of Plasmodium falciparum "in vitro". II. Morphological patterns of different quinolines effects.
    Microbiologica, 1989, Volume: 12, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Indoles; Mefloquine; Microscopy, Electron; Molecular Structure; Plasmodium falciparum; Quinolines

1989
[Surveillance of Plasmodium falciparum drug sensitivity in Yaounde and its surroundings (Cameroon). In vivo and in vitro study].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1989, Volume: 82, Issue:2

    Topics: Adolescent; Adult; Amodiaquine; Animals; Antimalarials; Cameroon; Child; Child, Preschool; Chloroquine; Humans; In Vitro Techniques; Infant; Malaria; Mefloquine; Microbial Sensitivity Tests; Middle Aged; Plasmodium falciparum; Quinine; Quinolines; Rural Population

1989
Antimalarial drug susceptibility of Plasmodium falciparum isolates from forest fringe dwelling aborigines (Orang Asli) of Peninsular Malaysia.
    The American journal of tropical medicine and hygiene, 1989, Volume: 41, Issue:1

    Topics: Animals; Antimalarials; Child; Chloroquine; Drug Resistance; Humans; Malaria; Malaysia; Mefloquine; Plasmodium falciparum; Quinolines

1989
Drug resistant P. falciparum in Madras (Tamil Nadu) and district Jabalpur (Madhya Pradesh).
    Indian journal of malariology, 1989, Volume: 26, Issue:2

    Topics: Adolescent; Adult; Animals; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; India; Malaria; Male; Mefloquine; Plasmodium falciparum

1989
[A handy medium for in vitro assessment of sensitivity of Plasmodium falciparum to chloroquine and mefloquine in the field].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1989, Volume: 7, Issue:2

    Topics: Animals; Chloroquine; Culture Media; Drug Resistance; Mefloquine; Plasmodium falciparum

1989
[Sensitivity of Plasmodium falciparum to different antimalarials. A study in 1988 in a village in the Hauts-Plateaux of Madagascar].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1989, Volume: 82, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Madagascar; Mefloquine; Plasmodium falciparum; Quinine

1989
Status of the response of Plasmodium falciparum to chloroquine and mefloquine in Iran.
    Tropical and geographical medicine, 1989, Volume: 41, Issue:4

    Topics: Afghanistan; Animals; Chloroquine; Drug Resistance; Female; Humans; India; Iran; Malaria; Male; Mefloquine; Pakistan; Plasmodium falciparum

1989
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with dipalmitoylphosphatidylcholine bilayers.
    Molecular and biochemical parasitology, 1989, Volume: 35, Issue:3

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Mefloquine; Quinacrine; Quinine; Quinolines; Temperature

1989
Is plasmodium falciparum resistance to chloroquine reversible in absence of drug pressure?
    Lancet (London, England), 1985, Aug-03, Volume: 2, Issue:8449

    Topics: Adolescent; Child; Child, Preschool; Chloroquine; Drug Interactions; Drug Resistance, Microbial; Humans; Malaria; Mefloquine; Plasmodium falciparum; Quinolines; Vietnam

1985
In-vitro chloroquine and mefloquine-resistant Plasmodium falciparum in Nigeria.
    Lancet (London, England), 1987, Mar-07, Volume: 1, Issue:8532

    Topics: Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Infant; Mefloquine; Nigeria; Plasmodium falciparum; Quinolines

1987
High rate of Plasmodium vivax relapse following treatment of falciparum malaria in Thailand.
    Lancet (London, England), 1987, Nov-07, Volume: 2, Issue:8567

    Topics: Acute Disease; Adolescent; Adult; Animals; Antimalarials; Chloroquine; Female; Follow-Up Studies; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Plasmodium vivax; Quinidine; Quinine; Quinolines; Recurrence; Thailand

1987
In vitro sensitivity of Plasmodium falciparum isolates from Burma to chloroquine quinine and mefloquine.
    The Southeast Asian journal of tropical medicine and public health, 1985, Volume: 16, Issue:3

    Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Mefloquine; Myanmar; Plasmodium falciparum; Quinine; Quinolines

1985
Plasmodium falciparum: inhibition of dolichol kinase by mefloquine.
    Experimental parasitology, 1986, Volume: 62, Issue:3

    Topics: Animals; Artemisinins; Cations, Divalent; Chloroquine; Cytidine Triphosphate; Detergents; Dolichols; Egtazic Acid; Erythrocytes; Hydrogen-Ion Concentration; Kinetics; Mefloquine; Microsomes; Nucleotides; Phosphotransferases; Phosphotransferases (Alcohol Group Acceptor); Plasmodium falciparum; Quinolines; Sesquiterpenes; Trifluoperazine

1986
[In vitro activity of various antimalarials (chloroquine, amodiaquine, quinine and mefloquine) against 32 isolates of Plasmodium falciparum in French Guiana].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1988, Volume: 81, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Drug Resistance; French Guiana; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1988
Response of Kampuchean strains of Plasmodium falciparum to antimalarials: in-vivo assessment of quinine and quinine plus tetracycline; multiple drug resistance in vitro.
    The Journal of tropical medicine and hygiene, 1988, Volume: 91, Issue:4

    Topics: Adolescent; Adult; Animals; Cambodia; Chloroquine; Drug Administration Schedule; Drug Resistance; Drug Therapy, Combination; Humans; In Vitro Techniques; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinine; Quinolines; Tetracycline

1988
Patterns of in vitro resistance to chloroquine, quinine, and mefloquine of Plasmodium falciparum in Cameroon, 1985-1986.
    The American journal of tropical medicine and hygiene, 1988, Volume: 39, Issue:2

    Topics: Adolescent; Animals; Antimalarials; Cameroon; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Infant; Mefloquine; Plasmodium falciparum; Quinine; Quinolines; Time Factors

1988
[The chloroquine resistance of Plasmodium falciparum in Vanuatu (1980-1984): appearance, evolution, distribution].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1988, Volume: 81, Issue:2

    Topics: Adolescent; Adult; Animals; Child; Child, Preschool; Chloroquine; Culture Media; Drug Resistance; Humans; Infant; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines; Vanuatu

1988
Response of Plasmodium falciparum to antimalarial drugs in vitro at Wad Medani, Sudan.
    APMIS. Supplementum, 1988, Volume: 3

    Topics: Animals; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinolines; Sudan

1988
Serial studies on the evolution of drug resistance in malaria in an area of east Africa: findings from 1979 up to 1986.
    The Journal of tropical medicine and hygiene, 1988, Volume: 91, Issue:5

    Topics: Age Factors; Amodiaquine; Animals; Antibodies, Protozoan; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Drug Therapy, Combination; Humans; Infant; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinidine; Quinine; Quinolines; Sulfadoxine; Tanzania

1988
Susceptibility of Plasmodium falciparum to chloroquine and mefloquine in Somalia.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:2

    Topics: Adolescent; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Humans; Infant; Malaria; Mefloquine; Plasmodium falciparum; Quinolines; Somalia

1988
Antagonism of chloroquine with other antimalarials.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Combinations; Drug Interactions; Drug Resistance; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1988
In vitro response of Plasmodium falciparum to chloroquine and mefloquine in southeast Madagascar.
    Archives de l'Institut Pasteur de Madagascar, 1988, Volume: 54, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; In Vitro Techniques; Madagascar; Mefloquine; Plasmodium falciparum; Quinolines

1988
In-vivo susceptibility of Plasmodium falciparum to cholorquine in pregnant and non-pregnant women and in-vitro response of P. falciparum to chloroquine and mefloquine in Madang Province, Papua New Guinea.
    Acta Leidensia, 1988, Volume: 57, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Female; Humans; In Vitro Techniques; Malaria; Mefloquine; Papua New Guinea; Plasmodium falciparum; Pregnancy; Pregnancy Complications, Infectious; Quinolines

1988
Chloroquine-resistant Plasmodium falciparum in Mali revealed by congenital malaria.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:4

    Topics: Adult; Animals; Antimalarials; Chloroquine; Drug Resistance; Female; Humans; Infant, Newborn; Malaria; Mali; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1988
Multiple drug resistant Plasmodium falciparum malaria in a pregnant indigenous Zambian woman.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:4

    Topics: Adult; Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Erythromycin; Female; Humans; Malaria; Mefloquine; Plasmodium falciparum; Pregnancy; Pregnancy Complications, Infectious; Pyrimethamine; Quinine; Quinolines; Sulfadoxine

1988
[Characterization of 15 strains of Plasmodium falciparum in 8 areas of the Brazilian Amazon region].
    Revista brasileira de malariologia e doencas tropicais. Publicacoes avulsas, 1986, Volume: 38

    Topics: Animals; Antigens, Protozoan; Antimalarials; Brazil; Chloroquine; Mefloquine; Plasmodium falciparum

1986
Hypoglycaemia and antimalarial drugs: quinidine and release of insulin.
    British medical journal (Clinical research ed.), 1986, May-17, Volume: 292, Issue:6531

    Topics: Amodiaquine; Antimalarials; Blood Glucose; Chloroquine; Humans; Hypoglycemia; Insulin; Mefloquine; Phenanthrenes; Quinidine; Quinolines; Thailand

1986
Inhibition of human placental aromatase by mefloquine.
    Journal of steroid biochemistry, 1988, Volume: 29, Issue:1

    Topics: Antimalarials; Aromatase Inhibitors; Chloroquine; Female; Humans; Mefloquine; Microsomes; Placenta; Pregnancy; Quinolines; Structure-Activity Relationship

1988
Evidence for electrogenic accumulation of mefloquine by malarial parasites.
    Biochemical pharmacology, 1988, Oct-01, Volume: 37, Issue:19

    Topics: Animals; Antimalarials; Biological Transport; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Chloroquine; Dose-Response Relationship, Drug; Electrochemistry; Erythrocyte Membrane; Hydrogen-Ion Concentration; Ionophores; Mefloquine; Methylamines; Mice; Plasmodium; Quinolines; Temperature; Valinomycin

1988
Effects of amodiaquine, chloroquine, and mefloquine on human polymorphonuclear neutrophil function in vitro.
    Antimicrobial agents and chemotherapy, 1988, Volume: 32, Issue:8

    Topics: Amodiaquine; Antimalarials; Cell Survival; Cell-Free System; Chemotaxis, Leukocyte; Chloroquine; Humans; Mefloquine; Neutrophils; Oxidation-Reduction; Phagocytosis; Quinolines

1988
Simultaneous determination of mefloquine and chloroquine in biological fluids using high-performance liquid chromatography.
    Annales de biologie clinique, 1988, Volume: 46, Issue:9

    Topics: Antimalarials; Chloroquine; Chromatography, High Pressure Liquid; Humans; Mefloquine; Methaqualone; Quinolines

1988
Evaluation of an in vitro assay system for drug susceptibility of field isolates of Plasmodium falciparum from southern Thailand.
    The American journal of tropical medicine and hygiene, 1988, Volume: 38, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Butylated Hydroxytoluene; Chloroquine; Humans; Mefloquine; Parasitology; Phenanthrenes; Plasmodium falciparum; Pyridines; Pyrimethamine; Quinine; Quinolines; Thailand; Triazines

1988
In vitro activity of pyronaridine against field isolates and reference clones of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1988, Volume: 38, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Drug Resistance; Humans; Mefloquine; Naphthyridines; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Thailand

1988
Effects of quinoline-containing antimalarials on the erythrocyte membrane and their significance to drug action on Plasmodium falciparum.
    Biochemical pharmacology, 1988, May-15, Volume: 37, Issue:10

    Topics: Animals; Antimalarials; Chloroquine; Erythrocyte Membrane; Hemolysis; Humans; Hydrogen-Ion Concentration; Mefloquine; Phospholipids; Plasmodium falciparum; Potassium; Proteins; Quinine; Quinolines

1988
Concurrent chloroquine and Fansidar resistance of Plasmodium falciparum: an imported case from Gabon.
    Tropical and geographical medicine, 1988, Volume: 40, Issue:1

    Topics: Animals; Chloroquine; Drug Combinations; Drug Resistance; Gabon; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Sulfadoxine; Sulfanilamides

1988
In vitro susceptibility of Plasmodium falciparum to amodiaquine, mefloquine, quinine and chloroquine in Liberia, West Africa.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1986, Volume: 80, Issue:5

    Topics: Amodiaquine; Animals; Chloroquine; Drug Resistance; Liberia; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1986
A study of the sensitivity of Plasmodium falciparum to chloroquine and mefloquine using the in vitro microtechnique in Peninsular Malaysia.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1987, Volume: 81, Issue:2

    Topics: Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria; Malaysia; Mefloquine; Parasitology; Plasmodium falciparum; Quinolines

1987
Comparison of washed and unwashed specimens in the Plasmodium falciparum in vitro microculture drug assay.
    The Southeast Asian journal of tropical medicine and public health, 1987, Volume: 18, Issue:2

    Topics: Animals; Chloroquine; Drug Resistance; Humans; Mefloquine; Parasitology; Plasmodium falciparum; Quinolines; Specimen Handling

1987
In vitro drug response of Plasmodium falciparum in the Philippines: increased resistance to amodiaquine.
    The Southeast Asian journal of tropical medicine and public health, 1987, Volume: 18, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Philippines; Plasmodium falciparum; Quinine; Quinolines

1987
Flunarizine and verapamil inhibit chloroquine-resistant Plasmodium falciparum growth in vitro.
    The Southeast Asian journal of tropical medicine and public health, 1987, Volume: 18, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Chlorpromazine; Drug Resistance; Flunarizine; Mefloquine; Plasmodium falciparum; Quinine; Quinolines; Regression Analysis; Verapamil

1987
[2 cases of multiresistant Plasmodium falciparum malaria contracted in Douala with atypical clinical presentation].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1987, Volume: 80, Issue:3 Pt 2

    Topics: Adolescent; Adult; Amodiaquine; Animals; Antimalarials; Cameroon; Chloroquine; Drug Combinations; Drug Resistance; Humans; Malaria; Male; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Sulfadoxine

1987
[Sensitivity of Plasmodium falciparum to quinolines and therapeutic strategies: comparison of the situation in Africa and Madagascar between 1983 and 1986].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1987, Volume: 80, Issue:3 Pt 2

    Topics: Amodiaquine; Angola; Animals; Antimalarials; Burkina Faso; Cameroon; Chloroquine; Drug Resistance; Humans; Madagascar; Malaria; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1987
Amodiaquine fails to cure chloroquine resistant Plasmodium falciparum in the Punjab.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1987, Volume: 81, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Pakistan; Plasmodium falciparum; Quinolines

1987
[Susceptibility of Plasmodium falciparum to chloroquine, piperaquine, amodiaquine, mefloquine and quinine with in vitro microtechnique in Hainan Island].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1987, Volume: 5, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Synergism; Mefloquine; Plasmodium falciparum; Quinolines

1987
Filaricidal effect of mefloquine on adults and microfilariae of Brugia patei and Brugia malayi.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1987, Volume: 38, Issue:1

    Topics: Animals; Anthelmintics; Blood Proteins; Brugia; Chloroquine; Filaricides; Mefloquine; Microfilariae; Quinolines

1987
Effect of antimalarial drugs on stimulation and interleukin 2 production of human lymphocytes.
    International journal of immunopharmacology, 1987, Volume: 9, Issue:4

    Topics: Antimalarials; Candida; Cells, Cultured; Chloroquine; Drug Administration Schedule; Humans; In Vitro Techniques; Interleukin-2; Lymphocyte Activation; Mefloquine; Protein Biosynthesis; Pyrimethamine; Quinine; Quinolines; Tuberculin

1987
Adaptation of the Indochina I/CDC strain of Plasmodium falciparum to the squirrel monkey (Saimiri sciureus).
    The American journal of tropical medicine and hygiene, 1986, Volume: 35, Issue:3

    Topics: Animals; Aotus trivirgatus; Cebidae; Chloroquine; Disease Models, Animal; Drug Resistance; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Saimiri; Splenectomy; Sulfadoxine

1986
High level of sensitivity to chloroquine of 72 Plasmodium falciparum isolates from southern Cameroon in January 1985.
    The American journal of tropical medicine and hygiene, 1986, Volume: 35, Issue:4

    Topics: Animals; Antimalarials; Cameroon; Child; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1986
Digestion of the host erythrocyte by malaria parasites is the primary target for quinoline-containing antimalarials.
    Biochemical pharmacology, 1986, Jul-15, Volume: 35, Issue:14

    Topics: Amino Acids; Ammonium Chloride; Animals; Antimalarials; Chloroquine; Erythrocytes; Host-Parasite Interactions; Humans; Mefloquine; Methylamines; Plasmodium falciparum; Quinine; Quinolines; Vacuoles

1986
[Preliminary study, in vitro, of the sensitivity of P. falciparum to chloroquine, mefloquine and quinine during 1985, in Kampuchea].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1986, Volume: 79, Issue:3

    Topics: Adult; Antimalarials; Cambodia; Chloroquine; Humans; Malaria; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine; Quinolines

1986
In vitro effect of chloroquine, mefloquine and quinine on human lymphocyte proliferative responses to malaria antigens and other antigens/mitogens.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1986, Volume: 37, Issue:3

    Topics: Adult; Antigens, Fungal; Antigens, Protozoan; Candida albicans; Chloroquine; Humans; Lymphocyte Activation; Mefloquine; Mitogens; Plasmodium falciparum; Quinine; Quinolines; Tuberculin

1986
Effects of combinations of quinoline-containing antimalarials on Plasmodium falciparum in culture.
    Annals of tropical medicine and parasitology, 1986, Volume: 80, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Interactions; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1986
Chloroquine-resistant falciparum malaria from East Africa.
    The Journal of tropical medicine and hygiene, 1986, Volume: 89, Issue:6

    Topics: Adult; Africa, Eastern; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Drug Therapy, Combination; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sulfadoxine

1986
Plasmodium falciparum drug resistance in West Africa.
    Annales de la Societe belge de medecine tropicale, 1986, Volume: 66, Issue:4

    Topics: Africa, Western; Animals; Antimalarials; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1986
[Development of P. falciparum sensitivity to chloroquine, to quinine and to mefloquine between 1983 and 1985 in Zaire].
    Annales de la Societe belge de medecine tropicale, 1986, Volume: 66, Issue:4

    Topics: Animals; Antimalarials; Chloroquine; Democratic Republic of the Congo; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1986
[Comparison of the effectiveness of two kinds of media for in vitro microtest of sensitivity of Plasmodium falciparum to chloroquine and mefloquine].
    Ji sheng chong xue yu ji sheng chong bing za zhi = Journal of parasitology & parasitic diseases, 1986, Volume: 4, Issue:4

    Topics: Animals; Chloroquine; Culture Media; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinolines

1986
Plasmodium falciparum: S-adenosyl-L-methionine decarboxylase.
    Experimental parasitology, 1987, Volume: 63, Issue:2

    Topics: Adenosylmethionine Decarboxylase; Animals; Carboxy-Lyases; Chloroquine; Erythrocytes; Humans; Hydrogen-Ion Concentration; Kinetics; Mefloquine; Mitoguazone; Plasmodium falciparum; Polyamines; Putrescine; Quinolines

1987
In vitro susceptibility of chloroquine resistant Plasmodium falciparum to mefloquine in Delhi.
    Indian journal of malariology, 1986, Volume: 23, Issue:2

    Topics: Adolescent; Adult; Animals; Antimalarials; Child; Chloroquine; Drug Resistance; Humans; India; Malaria; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines

1986
Plasma and whole blood mefloquine concentrations during treatment of chloroquine-resistant falciparum malaria with the combination mefloquine-sulphadoxine-pyrimethamine.
    British journal of clinical pharmacology, 1987, Volume: 23, Issue:4

    Topics: Adolescent; Adult; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Female; Humans; Intestinal Absorption; Kinetics; Malaria; Male; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Sulfadoxine; Sulfanilamides

1987
[A case of malaria tropicameningoencephalitis (neuromalaria) with chloroquine and pyrimethamine/sulfadoxine resistance].
    Der Nervenarzt, 1985, Volume: 56, Issue:2

    Topics: Adult; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Male; Mefloquine; Meningoencephalitis; Plasmodium falciparum; Pyrimethamine; Quinolines; Sulfadoxine; Sulfanilamides

1985
Use of non-human plasma for in vitro cultivation and antimalarial drug susceptibility testing of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1985, Volume: 34, Issue:2

    Topics: Animals; Antimalarials; Cattle; Chloroquine; Culture Media; Goats; Horses; Humans; Mefloquine; Plasma; Plasmodium falciparum; Quinolines; Sheep; Swine

1985
Antimalarial drug susceptibility testing of Plasmodium falciparum in Thailand using a microdilution radioisotope method.
    The American journal of tropical medicine and hygiene, 1985, Volume: 34, Issue:2

    Topics: Adult; Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Lethal Dose 50; Malaria; Male; Mefloquine; Microbial Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Quinine; Quinolines; Thailand

1985
Studies of resistance to chloroquine, quinine, amodiaquine and mefloquine among Philippine strains of Plasmodium falciparum.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1985, Volume: 79, Issue:1

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Mefloquine; Philippines; Plasmodium falciparum; Quinine; Quinolines

1985
Sensitivity of Plasmodium falciparum to antimalarial drugs in Colombia.
    The American journal of tropical medicine and hygiene, 1985, Volume: 34, Issue:4

    Topics: Amodiaquine; Antimalarials; Chloroquine; Colombia; Drug Combinations; Drug Resistance, Microbial; Geography; Humans; Malaria; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Pyrimethamine; Quinolines; Sulfadoxine

1985
Mefloquine failure in a case of falciparum malaria induced with a multidrug-resistant isolate in a non-immune subject.
    The American journal of tropical medicine and hygiene, 1985, Volume: 34, Issue:4

    Topics: Adult; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Male; Mefloquine; Phenanthrenes; Plasmodium falciparum; Pyridines; Quinine; Quinolines

1985
Antimalarials increase vesicle pH in Plasmodium falciparum.
    The Journal of cell biology, 1985, Volume: 101, Issue:6

    Topics: Ammonia; Animals; Antimalarials; Biological Transport; Chloroquine; Erythrocytes; Hydrogen-Ion Concentration; Lysosomes; Mefloquine; Organoids; Plasmodium falciparum; Quinine; Quinolines

1985
[Studies on the chemoresistance of Plasmodium falciparum in Africa: current data].
    Annales de la Societe belge de medecine tropicale, 1985, Volume: 65 Suppl 2

    Topics: Africa; Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Mefloquine; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinolines

1985
[Sensitivity of strains of Plasmodium falciparum to chloroquine, mefloquine and quinine in 1983 in Zaire].
    Annales de la Societe belge de medecine tropicale, 1985, Volume: 65 Suppl 2

    Topics: Animals; Antimalarials; Chloroquine; Democratic Republic of the Congo; Drug Resistance, Microbial; In Vitro Techniques; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1985
In vitro response of Plasmodium falciparum to mefloquine. Studies conducted in West and East Africa.
    Annales de la Societe belge de medecine tropicale, 1985, Volume: 65 Suppl 2

    Topics: Africa, Eastern; Africa, Western; Animals; Chloroquine; Drug Resistance, Microbial; In Vitro Techniques; Mefloquine; Plasmodium falciparum; Quinolines

1985
Plasmodium falciparum in Madagascar: in vivo and in vitro sensitivity to seven drugs.
    Annals of tropical medicine and parasitology, 1985, Volume: 79, Issue:4

    Topics: Adolescent; Adult; Aged; Amodiaquine; Antimalarials; Child; Child, Preschool; Chloroquine; Humans; Infant; Madagascar; Malaria; Mefloquine; Microbial Sensitivity Tests; Middle Aged; Phenanthrenes; Piperazines; Plasmodium falciparum; Quinine; Quinolines

1985
[8 cases of drug-resistant Plasmodium falciparum malaria contracted in Mozambique].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1985, Volume: 78, Issue:4

    Topics: Adult; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria; Male; Mefloquine; Mozambique; Plasmodium falciparum; Quinolines

1985
[Development of a piperaquine-resistant line of Plasmodium berghei K 173 strain].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1985, Volume: 20, Issue:6

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance; Malaria; Male; Mefloquine; Mice; Plasmodium berghei; Quinolines; Sesquiterpenes

1985
In vitro assessment of sensitivity of Plasmodium falciparum to chloroquine and mefloquine in Ghana.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1985, Volume: 79, Issue:6

    Topics: Adolescent; Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Female; Ghana; Humans; Malaria; Male; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinolines

1985
[Malaria chemoprophylaxis. Resistance problems].
    Archives francaises de pediatrie, 1985, Volume: 42 Suppl 2

    Topics: Antimalarials; Child; Child, Preschool; Chloroquine; Dapsone; Drug Combinations; Drug Resistance, Microbial; Humans; Infant; Malaria; Mefloquine; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Quinolines; Sulfadoxine

1985
Recent trends of chemotherapy and vaccination against malaria: new lamps for old.
    British medical journal (Clinical research ed.), 1985, Oct-19, Volume: 291, Issue:6502

    Topics: Antibodies, Monoclonal; Chloroquine; Drug Resistance, Microbial; Global Health; Humans; Immunotherapy; Malaria; Mefloquine; Plasmodium falciparum; Quinolines; Vaccines

1985
A rabbit--in vitro system to evaluate drug action against Plasmodium falciparum.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:1

    Topics: Acedapsone; Animals; Antimalarials; Chloroquine; Drug Evaluation, Preclinical; Male; Mefloquine; Microbial Sensitivity Tests; Models, Biological; Plasmodium falciparum; Pyrimethamine; Quinolines; Rabbits; Time Factors; Triazines

1983
Interactions of hemin, antimalarial drugs and hemin-antimalarial complexes with phospholipid monolayers.
    Chemistry and physics of lipids, 1984, Volume: 35, Issue:4

    Topics: Animals; Antimalarials; Cattle; Chloroquine; Heme; Hemin; Mathematics; Mefloquine; Membranes, Artificial; Phospholipids; Quinine; Quinolines; Surface Properties

1984
The effect of anti-malarial drugs on human natural killer cells in vitro.
    Parasite immunology, 1984, Volume: 6, Issue:6

    Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines

1984
In vitro study of drug sensitivity of Plasmodium falciparum: evaluation of a new semi-micro test.
    The American journal of tropical medicine and hygiene, 1983, Volume: 32, Issue:3

    Topics: Antimalarials; Chloroquine; Evaluation Studies as Topic; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine; Quinolines

1983
Susceptibility of Plasmodium falciparum to five drugs: an in vitro study of isolates mainly from Thailand.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:2

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; In Vitro Techniques; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Thailand

1983
Plasmodium falciparum: drug sensitivity in vitro of isolates before and after adaptation to continuous culture.
    Experimental parasitology, 1983, Volume: 56, Issue:1

    Topics: Adaptation, Physiological; Animals; Antimalarials; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1983
Plasmodium falciparum-malaria: resistance to chloroquine, but sensitivity to mefloquine in the Gabon. A prospective in-vitro study.
    Tropenmedizin und Parasitologie, 1984, Volume: 35, Issue:1

    Topics: Adolescent; Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Gabon; Humans; Infant; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Prospective Studies; Quinolines

1984
The treatment of falciparum malaria.
    The Journal of antimicrobial chemotherapy, 1984, Volume: 13, Issue:4

    Topics: Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Plasmodium falciparum; Quinidine; Quinine; Quinolines; Sesquiterpenes

1984
The relationship between the in vitro response of Plasmodium falciparum to chloroquine, quinine and mefloquine.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1984, Volume: 78, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1984
Application of an in vitro semi-microtest to the study of drug sensitivity of 66 Plasmodium falciparum isolates from 15 countries.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1984, Volume: 78, Issue:4

    Topics: Animals; Chloroquine; Drug Resistance, Microbial; Mefloquine; Microbial Sensitivity Tests; Piperazines; Plasmodium falciparum; Quinine; Quinolines

1984
A comparative micro in-vitro test of P. falciparum to mefloquine and chloroquine in Gadchiroli District, Maharashtra State.
    The Journal of communicable diseases, 1984, Volume: 16, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Humans; India; Malaria; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinolines

1984
[In vitro sensitivity tests of Plasmodium falciparum samples of the Amazonian Basin (Brazil)].
    Revista brasileira de malariologia e doencas tropicais. Publicacoes avulsas, 1983, Volume: 35

    Topics: Amodiaquine; Animals; Antimalarials; Brazil; Chloroquine; In Vitro Techniques; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines

1983
African serum interference in the determination of chloroquine sensitivity in Plasmodium falciparum.
    Zeitschrift fur Parasitenkunde (Berlin, Germany), 1984, Volume: 70, Issue:5

    Topics: Adult; Animals; Antimalarials; Child; Chloroquine; Drug Resistance, Microbial; Humans; Immune Sera; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines; Sudan

1984
[Drug sensitivity of Plasmodium falciparum in Madagascar. V. Study of the in vitro activity of quinine, mefloquine and halofantrine].
    Archives de l'Institut Pasteur de Madagascar, 1984, Volume: 51, Issue:1

    Topics: Antimalarials; Chloroquine; Humans; Mefloquine; Microbial Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Quinine; Quinolines

1984
Inhibition of ornithine decarboxylase of in vitro cultured Plasmodium falciparum by chloroquine.
    Tropenmedizin und Parasitologie, 1983, Volume: 34, Issue:1

    Topics: Carboxy-Lyases; Chloroquine; Culture; DNA; Eflornithine; Humans; Mefloquine; Ornithine; Ornithine Decarboxylase; Ornithine Decarboxylase Inhibitors; Plasmodium falciparum; Quinolines

1983
Diverse membrane-active agents modify the hemolytic response to ferriprotoporphyrin IX.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:3

    Topics: Adult; Antimalarials; Calcium; Chloroquine; Drug Synergism; Erythrocytes; Female; Heme; Hemin; Hemolysis; Humans; Male; Mefloquine; Osmotic Fragility; Quinine; Quinolines; Sodium Chloride

1983
[Standardisation of the in vitro chemosensitivity test for Plasmodium falciparum ].
    Pathologie-biologie, 1982, Volume: 30, Issue:6 Pt 2

    Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Erythrocytes; Humans; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine; Quinolines

1982
In vitro assessment of 2-acetylpyridine thiosemicarbazones against chloroquine-resistant Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 1982, Volume: 22, Issue:6

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Malaria; Mefloquine; Mice; Plasmodium falciparum; Pyrimethamine; Quinolines; Structure-Activity Relationship; Thiosemicarbazones

1982
Plasmodium chabaudi-infection of mice: effects of chloroquine and mefloquine. Inhibition of ornithine decarboxylase activity.
    Tropenmedizin und Parasitologie, 1981, Volume: 32, Issue:2

    Topics: Acridines; Animals; Antimalarials; Carboxy-Lyases; Chloroquine; Enzyme Repression; Erythrocyte Membrane; Malaria; Mefloquine; Mice; Ornithine Decarboxylase Inhibitors; Piperidines; Plasmodium; Primaquine; Quinolines

1981
Antimalarial activity of mefloquine and chloroquine against blood induced Plasmodium knowlesi infection in rhesus monkeys.
    The Indian journal of medical research, 1981, Volume: 73 Suppl

    Topics: Animals; Antimalarials; Chloroquine; Female; Macaca mulatta; Malaria; Male; Mefloquine; Piperidines; Quinolines

1981
The inhibitory effect of a drug combination on the development of mefloquine resistance in Plasmodium berghei.
    Annals of tropical medicine and parasitology, 1980, Volume: 74, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Drug Therapy, Combination; Erythrocytes; Male; Mefloquine; Mice; Piperidines; Plasmodium berghei; Pyrimethamine; Quinolines; Sulfadoxine

1980
Binding of antimalarial drugs to hemozoin from Plasmodium berghei.
    Experientia, 1980, Sep-15, Volume: 36, Issue:9

    Topics: Animals; Antimalarials; Chloroquine; Heme; Hemeproteins; Mefloquine; Methemoglobin; Pigments, Biological; Piperidines; Plasmodium berghei; Protein Binding; Protoporphyrins; Quinacrine; Quinolines; Spectrophotometry

1980
Decrease in susceptibility of Plasmodium falciparum to mefloquine in continuous culture.
    Bulletin of the World Health Organization, 1981, Volume: 59, Issue:2

    Topics: Animals; Chloroquine; Culture Media; Drug Resistance, Microbial; Humans; In Vitro Techniques; Malaria; Mefloquine; Piperidines; Plasmodium falciparum; Quinolines

1981
Use of the in vitro microtechnique for the assessment of drug sensitivity of Plasmodium falciparum in Sennar, Sudan.
    Bulletin of the World Health Organization, 1980, Volume: 58, Issue:5

    Topics: Adolescent; Adult; Aged; Aminoquinolines; Child; Child, Preschool; Chloroquine; Humans; In Vitro Techniques; Malaria; Mefloquine; Microbiological Techniques; Middle Aged; Piperidines; Plasmodium falciparum; Quinolines; Sudan

1980
Sustained-release implants in the chemotherapy of experimental rodent malaria I. A comparison of the effects of some antimalarials in polydimethylsiloxane matrices.
    Annals of tropical medicine and parasitology, 1981, Volume: 75, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Dimethylpolysiloxanes; Drug Implants; Malaria; Male; Mefloquine; Mice; Mice, Inbred Strains; Naphthoquinones; Piperidines; Plasmodium berghei; Primaquine; Proguanil; Pyrimethamine; Quinolines; Silicone Elastomers; Sulfadiazine; Triazines

1981
In vitro susceptibility of Plasmodium falciparum to chloroquine, amodiaquine, quinine, mefloquine, and sulfadoxine/pyrimethamine in Equatorial Guinea.
    The American journal of tropical medicine and hygiene, 1995, Volume: 53, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Child; Chloroquine; Drug Combinations; Equatorial Guinea; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Regression Analysis; Sulfadoxine

1995
The chemotherapy of rodent malaria. LII. Response of Plasmodium yoelii ssp. NS to mefloquine and its enantiomers.
    Annals of tropical medicine and parasitology, 1995, Volume: 89, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Malaria; Mefloquine; Mice; Plasmodium yoelii; Stereoisomerism

1995
Assessment of interactions of the antimalarial drugs chloroquine and mefloquine with NaNO2 and HgCl2 in rodents.
    Mutation research, 1994, Mar-01, Volume: 305, Issue:2

    Topics: Animals; Bone Marrow; Bone Marrow Cells; Chloroquine; Chromosome Aberrations; Dose-Response Relationship, Drug; Drug Interactions; Mefloquine; Mercuric Chloride; Mice; Mice, Inbred BALB C; Micronucleus Tests; Mitotic Index; Mutagenicity Tests; Mutagens; Rats; Rats, Wistar; Sodium Nitrite

1994
Antimalarials for Africa.
    Communicable disease report. CDR weekly, 1994, Jul-29, Volume: 4, Issue:30

    Topics: Africa; Chloroquine; Humans; Malaria; Mefloquine; Travel; United Kingdom

1994
Malaria prophylaxis. Mefloquine toxicity should limit its use to treatment alone.
    BMJ (Clinical research ed.), 1995, Jul-15, Volume: 311, Issue:6998

    Topics: Africa; Antimalarials; Chloroquine; Humans; Malaria; Malaria, Falciparum; Mefloquine; Proguanil; Travel

1995
Malaria prophylaxis. Psychological problems after mefloquine and chloroquine.
    BMJ (Clinical research ed.), 1995, Jul-15, Volume: 311, Issue:6998

    Topics: Chloroquine; Humans; Malaria; Mefloquine; Mental Disorders

1995
Quinine resistant falciparum malaria acquired in east Africa.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1995, Volume: 46, Issue:1

    Topics: Adult; Africa, Eastern; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Male; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Tetracycline

1995
Sensitivity to antimalarial drugs by Plasmodium falciparum in Goundry, Oubritenga province, Burkina Faso.
    Parassitologia, 1994, Volume: 36, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Burkina Faso; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; National Health Programs; Parasitemia; Plasmodium falciparum; Pyrimethamine; Sulfadoxine; Treatment Outcome

1994
[Malaria prevention with mefloquine].
    Deutsche medizinische Wochenschrift (1946), 1995, Aug-18, Volume: 120, Issue:33

    Topics: Altitude Sickness; Calcium Channel Blockers; Chloroquine; Drug Interactions; Humans; Malaria; Mefloquine; Nifedipine

1995
Drug-resistant Plasmodium falciparum malaria in the eastern Transvaal.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1994, Volume: 84, Issue:7

    Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1994
[Development and trends from 1986 to 1993 of the attitude of intercontinental travellers on departure from France, with respect to malaria prophylaxis].
    Bulletin de la Societe de pathologie exotique (1990), 1993, Volume: 86, Issue:5 Pt 2

    Topics: Africa South of the Sahara; Attitude to Health; Chloroquine; France; Humans; Malaria; Mefloquine; Mosquito Control; Proguanil; Risk Factors; Travel

1993
Plasmodium falciparum and Plasmodium vivax: lactate dehydrogenase activity and its application for in vitro drug susceptibility assay.
    Experimental parasitology, 1995, Volume: 80, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Colorimetry; Erythrocytes; Humans; L-Lactate Dehydrogenase; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Parasitemia; Phenanthrenes; Plasmodium falciparum; Plasmodium vivax; Quinine

1995
Confused malaria chemoprophylaxis.
    Lancet (London, England), 1994, Feb-26, Volume: 343, Issue:8896

    Topics: Chloroquine; Clinical Protocols; Drug Resistance; Humans; Malaria; Mefloquine; Proguanil; Risk Factors; Travel; United Kingdom

1994
[In vitro sensitivity of Plasmodium falciparum to mefloquine, quinine, amodiaquine, chloroquine, pyronaridine and sulfadoxine/pyrimethamine in south Yunnan].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1994, Volume: 12, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Mefloquine; Naphthyridines; Plasmodium falciparum; Pyrimethamine; Quinine; Sulfadoxine

1994
A strong association between mefloquine and halofantrine resistance and amplification, overexpression, and mutation in the P-glycoprotein gene homolog (pfmdr) of Plasmodium falciparum in vitro.
    The American journal of tropical medicine and hygiene, 1994, Volume: 51, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Sequence; Blotting, Northern; Blotting, Southern; Chloroquine; DNA Primers; DNA, Protozoan; Drug Resistance; Gene Amplification; Gene Expression; Genes, Protozoan; Mefloquine; Molecular Sequence Data; Phenanthrenes; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Quinine; RNA, Messenger; Selection, Genetic; Sequence Homology, Nucleic Acid; Sesquiterpenes

1994
Ten-year surveillance of drug-resistant malaria in Burkina Faso (1982-1991).
    The American journal of tropical medicine and hygiene, 1994, Volume: 50, Issue:6

    Topics: Adolescent; Animals; Antimalarials; Burkina Faso; Child; Chloroquine; Drug Resistance; Humans; Longitudinal Studies; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Prevalence; Pyrimethamine; Quinine; Retrospective Studies; Sulfadoxine

1994
[Cytokines and malaria. A study of TNF-alpha, IL1-beta, IL6 and IL2R in 28 patients].
    Bulletin de la Societe de pathologie exotique (1990), 1994, Volume: 87, Issue:2

    Topics: Adolescent; Adult; Amodiaquine; C-Reactive Protein; Chloroquine; Humans; Interleukin-1; Interleukin-6; Leukocyte Count; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Middle Aged; Neutrophils; Platelet Count; Prognosis; Receptors, Interleukin-2; Retrospective Studies; Tumor Necrosis Factor-alpha

1994
Susceptibility of Plasmodium falciparum to chloroquine and mefloquine in Ouagadougou area (Burkina Faso).
    Parassitologia, 1993, Volume: 35, Issue:1-3

    Topics: Animals; Burkina Faso; Child; Child, Preschool; Chloroquine; Drug Evaluation; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Treatment Outcome

1993
In vitro susceptibility of Cambodian isolates of Plasmodium falciparum to halofantrine, pyronaridine and artemisinin derivatives.
    Annals of tropical medicine and parasitology, 1994, Volume: 88, Issue:2

    Topics: Adult; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; Mefloquine; Naphthyridines; Phenanthrenes; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Sesquiterpenes; Triazines

1994
Travellers' malaria risks.
    BMJ (Clinical research ed.), 1994, Jul-30, Volume: 309, Issue:6950

    Topics: Africa, Western; Chloroquine; Humans; Malaria; Mefloquine; Proguanil; Travel; United Kingdom

1994
[Subacute Plasmodium falciparum malaria in 43 patients returning from areas with chloroquine in Africa].
    Annales de medecine interne, 1994, Volume: 145, Issue:3

    Topics: Adult; Africa; Aged; Antibodies, Protozoan; Blood Cell Count; Chloroquine; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Risk Factors; Time Factors; Travel

1994
Sensitivity of Plasmodium falciparum field-isolates from Tanzania to chloroquine, mefloquine and pyrimethamine during in vitro cultivation.
    Acta tropica, 1993, Volume: 52, Issue:4

    Topics: Animals; Chloroquine; Drug Resistance; Mefloquine; Parasitology; Plasmodium falciparum; Pyrimethamine; Tanzania

1993
Antimalarial chemoprophylaxis for west Africa.
    Lancet (London, England), 1993, Apr-03, Volume: 341, Issue:8849

    Topics: Africa, Western; Antimalarials; Chloroquine; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Patient Compliance; Proguanil

1993
Mefloquine compared with other malaria chemoprophylactic regimens in tourists visiting east Africa.
    Lancet (London, England), 1993, May-22, Volume: 341, Issue:8856

    Topics: Adult; Antimalarials; Chloroquine; Female; Humans; Kenya; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Proguanil; Pyrimethamine; Sulfadoxine; Travel

1993
Malaria chemoprophylaxis.
    Lancet (London, England), 1993, Aug-21, Volume: 342, Issue:8869

    Topics: Chloroquine; Drug Combinations; Humans; Malaria; Mefloquine; Patient Compliance; Proguanil; Risk Factors; Travel

1993
Malaria chemoprophylaxis.
    Lancet (London, England), 1993, Aug-21, Volume: 342, Issue:8869

    Topics: Africa, Eastern; Africa, Western; Chloroquine; Drug Combinations; Humans; Malaria; Mefloquine; Patient Compliance; Proguanil; Risk Factors; Travel

1993
Mefloquine prophylaxis.
    Lancet (London, England), 1993, Aug-28, Volume: 342, Issue:8870

    Topics: Chloroquine; Humans; Malaria, Falciparum; Mefloquine

1993
In vitro activity of pyrimethamine, cycloguanil, and other antimalarial drugs against African isolates and clones of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1994, Volume: 50, Issue:2

    Topics: Africa; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Mefloquine; Phenanthrenes; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Triazines

1994
[A case of mefloquine-resistant Plasmodium falciparum malaria with convulsion after antimalarial treatment].
    Kansenshogaku zasshi. The Journal of the Japanese Association for Infectious Diseases, 1994, Volume: 68, Issue:1

    Topics: Adult; Animals; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Male; Mefloquine; Seizures; Travel; Uganda

1994
Malaria chemoprophylactic regimens for travellers.
    Bulletin of the World Health Organization, 1994, Volume: 72, Issue:2

    Topics: Chloroquine; Doxycycline; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Proguanil; Travel

1994
Efficacy of chloroquine on Plasmodium falciparum transmitted at Amani, eastern Usambara Mountains, north-east Tanzania: an area where malaria has recently become endemic.
    The Journal of tropical medicine and hygiene, 1993, Volume: 96, Issue:6

    Topics: Adolescent; Adult; Amodiaquine; Animals; Child; Child, Preschool; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Female; Follow-Up Studies; Hemoglobins; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinine; Regression Analysis; Sickle Cell Trait; Tanzania

1993
Malaria prophylaxis. Mefloquine should be first choice.
    BMJ (Clinical research ed.), 1993, Dec-11, Volume: 307, Issue:6918

    Topics: Chloroquine; Humans; Malaria; Mefloquine; Proguanil

1993
Warning--misleading malaria advice.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1993, Volume: 83, Issue:9

    Topics: Chloroquine; Health Education; Humans; Malaria; Mefloquine; Pamphlets; Proguanil; South Africa

1993
Enhancement of drug susceptibility in Plasmodium falciparum in vitro and Plasmodium berghei in vivo by mixed-function oxidase inhibitors.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:6

    Topics: Adolescent; Animals; Child; Child, Preschool; Chloroquine; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Desipramine; Drug Interactions; Drug Resistance, Microbial; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Mice; Mice, Inbred Strains; Microbial Sensitivity Tests; Mixed Function Oxygenases; Plasmodium berghei; Plasmodium falciparum

1993
In vitro activity of artemisinin derivatives against African isolates and clones of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1993, Volume: 49, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

1993
Comparison of beta-artemether and beta-arteether against malaria parasites in vitro and in vivo.
    The American journal of tropical medicine and hygiene, 1993, Volume: 48, Issue:3

    Topics: Animals; Antimalarials; Aotus trivirgatus; Artemether; Artemisinins; Chloroquine; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Malaria; Malaria, Falciparum; Male; Mefloquine; Mice; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes; Structure-Activity Relationship

1993
Derivation of highly mefloquine-resistant lines from Plasmodium falciparum in vitro.
    The American journal of tropical medicine and hygiene, 1993, Volume: 48, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Erythrocytes; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Serial Passage; Vacuoles

1993
Plasmodium falciparum: role of absolute stereochemistry in the antimalarial activity of synthetic amino alcohol antimalarial agents.
    Experimental parasitology, 1993, Volume: 76, Issue:4

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Pyridines; Quinolines; Stereoisomerism; Structure-Activity Relationship

1993
The antimalarial drug, Ro 42-1611 (arteflene), does not affect cytoadherence and cytokine-inducing properties of Plasmodium falciparum malaria parasites.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1995, Volume: 46, Issue:2

    Topics: Adult; Animals; Antigens, Protozoan; Antimalarials; Artemisinins; Bridged Bicyclo Compounds, Heterocyclic; Cell Adhesion; Cell Survival; Chloroquine; Cytokines; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Erythrocytes; Humans; Immunoglobulin G; Interleukin-1; Interleukin-6; Lipopolysaccharides; Lymphocytes; Malaria, Falciparum; Mefloquine; Melanoma; Plasmodium falciparum; Styrenes; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha

1995
Canadian recommendations for the prevention and treatment of malaria among international travellers. Committee to Advise on Tropical Medicine and Travel (CATMAT).
    Canada communicable disease report = Releve des maladies transmissibles au Canada, 1995, Volume: 21 Suppl 3

    Topics: Animals; Antimalarials; Canada; Child; Chloroquine; Culicidae; Drug Resistance; Female; Humans; Malaria; Malaria, Falciparum; Mefloquine; Pregnancy; Recurrence; Risk Factors; Travel

1995
Malaria among United States troops in Somalia.
    The American journal of medicine, 1996, Volume: 100, Issue:1

    Topics: Anti-Bacterial Agents; Antimalarials; Chemoprevention; Chloroquine; Clothing; Cohort Studies; Doxycycline; Drug Resistance; Humans; Malaria, Cerebral; Malaria, Falciparum; Male; Mefloquine; Military Personnel; Population Surveillance; Prospective Studies; Protective Devices; Pyrimethamine; Quinine; Risk Factors; Somalia; Sulfadoxine; Treatment Failure; Treatment Refusal; United States

1996
Effect of pH on in vitro potency of amantadine against Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1996, Volume: 54, Issue:3

    Topics: Adamantane; Amantadine; Ammonium Chloride; Animals; Antimalarials; Chloroquine; Culture Media; Dose-Response Relationship, Drug; Drug Resistance; Humans; Hydrogen-Ion Concentration; Mefloquine; Plasmodium falciparum; Quinine

1996
Plasmodium falciparum: molecular characterization of multidrug-resistant Cambodian isolates.
    Experimental parasitology, 1996, Volume: 82, Issue:2

    Topics: Alleles; Animals; Antimalarials; Blotting, Southern; Cambodia; Chloroquine; Codon; DNA Fingerprinting; DNA, Protozoan; Drug Resistance, Multiple; Folic Acid Antagonists; Genes, Protozoan; Genetic Variation; Humans; Mefloquine; Phenanthrenes; Plasmodium falciparum; Polymorphism, Genetic; Proguanil; Pyrimethamine; Triazines

1996
The effect of malaria and malaria prevention in pregnancy on offspring birthweight, prematurity, and intrauterine growth retardation in rural Malawi.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:1 Suppl

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Fetal Growth Retardation; Humans; Infant, Low Birth Weight; Infant, Newborn; Infant, Premature; Malaria, Falciparum; Malawi; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Risk Factors; Rural Population; Treatment Outcome

1996
Malaria treatment and prevention in pregnancy: indications for use and adverse events associated with use of chloroquine or mefloquine.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:1 Suppl

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Fetal Death; Fever; Humans; Malaria, Falciparum; Malawi; Mefloquine; Parasitemia; Pregnancy; Pregnancy Complications, Parasitic; Pregnancy Outcome; Rural Population

1996
Analysis of pfmdr1 and drug susceptibility in fresh isolates of Plasmodium falciparum from subsaharan Africa.
    Molecular and biochemical parasitology, 1995, Volume: 74, Issue:2

    Topics: Africa South of the Sahara; Alleles; Animals; Antimalarials; Base Sequence; Chloroquine; Codon; DNA Fingerprinting; DNA, Protozoan; Drug Resistance, Multiple; Genes, Protozoan; Genetic Variation; Humans; Malaria, Falciparum; Mefloquine; Phenotype; Plasmodium falciparum

1995
[Informal care of malaria: determinants of demand and supply inventory. A study conducted in Touba City (Senegal)].
    Bulletin de la Societe de pathologie exotique (1990), 1996, Volume: 89, Issue:1

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Female; Health Care Costs; Humans; Malaria; Male; Mefloquine; Middle Aged; Senegal; Surveys and Questionnaires

1996
Comparison of adverse events associated with use of mefloquine and combination of chloroquine and proguanil as antimalarial prophylaxis: postal and telephone survey of travellers.
    BMJ (Clinical research ed.), 1996, Aug-31, Volume: 313, Issue:7056

    Topics: Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Female; Health Surveys; Hospitalization; Humans; Malaria; Male; Mefloquine; Mental Disorders; Nervous System Diseases; Proguanil; Retrospective Studies; Travel; Treatment Refusal; United Kingdom

1996
In vitro drug sensitivity and clinical aspects of Plasmodium falciparum malaria in African children.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1995, Volume: 46, Issue:4

    Topics: Animals; Child; Child, Preschool; Chloroquine; Congo; Humans; Infant; Malaria, Falciparum; Mefloquine; Parasitemia; Plasmodium falciparum; Quinine

1995
Modulation of the function of human MDR1 P-glycoprotein by the antimalarial drug mefloquine.
    Biochemical pharmacology, 1996, Nov-22, Volume: 52, Issue:10

    Topics: Affinity Labels; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Binding, Competitive; Biological Transport, Active; Chloroquine; Drug Interactions; Drug Resistance, Multiple; Fluorescent Dyes; Humans; Kinetics; Mefloquine; Neoplasms; Prazosin; Tumor Cells, Cultured; Verapamil; Vinblastine

1996
Adverse events associated with mefloquine. Study in returned travellers confirms authors' findings.
    BMJ (Clinical research ed.), 1996, Dec-14, Volume: 313, Issue:7071

    Topics: Adult; Antimalarials; Chloroquine; Drug Combinations; Humans; Mefloquine; Mental Disorders; Proguanil; Travel

1996
Adverse events associated with mefloquine. Risk-benefit ratio must be taken into account.
    BMJ (Clinical research ed.), 1996, Dec-14, Volume: 313, Issue:7071

    Topics: Antimalarials; Chloroquine; Drug Combinations; Humans; Mefloquine; Mental Disorders; Proguanil; Risk Factors; Travel

1996
In vitro selection of halofantrine resistance in Plasmodium falciparum is not associated with increased expression of Pgh1.
    Molecular and biochemical parasitology, 1996, Dec-02, Volume: 83, Issue:1

    Topics: Animals; Antimalarials; ATP-Binding Cassette Transporters; Biological Transport; Chloroquine; DNA Fingerprinting; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Gene Dosage; Gene Expression; Immunoblotting; Mefloquine; Phenanthrenes; Plasmodium falciparum; Protozoan Proteins; Quinine; Selection, Genetic; Sequence Analysis, DNA; Verapamil

1996
High prevalence of chloroquine resistant Plasmodium falciparum infection in Rajasthan epidemic.
    Acta tropica, 1996, Dec-16, Volume: 62, Issue:3

    Topics: Animals; Antibodies, Protozoan; Antimalarials; Chloroquine; Disease Outbreaks; Drug Resistance, Microbial; Enzyme-Linked Immunosorbent Assay; Humans; Immunoglobulin G; Immunoglobulin M; India; Malaria, Falciparum; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Pyrimethamine; Quinine; Seroepidemiologic Studies; Sulfadoxine; Tumor Necrosis Factor-alpha

1996
In vitro susceptibility of Plasmodium falciparum isolates in Vietnam to artemisinin derivatives and other antimalarials.
    Acta tropica, 1997, Volume: 63, Issue:2-3

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine; Sesquiterpenes; Vietnam

1997
The chemotherapy of rodent malaria. LIV. Combinations of 'Fenozan B07' (Fenozan-50F), a difluorinated 3,3'-spirocyclopentane 1,2,4-trioxane, with other drugs against drug-sensitive and drug-resistant parasites.
    Annals of tropical medicine and parasitology, 1997, Volume: 91, Issue:1

    Topics: Aminoquinolines; Animals; Antimalarials; Chloroquine; Drug Antagonism; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Malaria; Mefloquine; Mice; Naphthyridines; Parasitemia; Phenanthrenes; Phenylpropionates; Plasmodium berghei; Plasmodium yoelii

1997
[Not more symptoms with mefloquine use than with other drugs in malaria prophylaxis].
    Nederlands tijdschrift voor geneeskunde, 1997, Feb-15, Volume: 141, Issue:7

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Patient Compliance; Proguanil; Retrospective Studies

1997
In vitro susceptibility of Tanzanian wild isolates of Plasmodium falciparum to artemisinin, chloroquine, sulfadoxine/pyrimethamine and mefloquine.
    Parasitology, 1997, Volume: 114 ( Pt 6)

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Humans; Mefloquine; Plasmodium falciparum; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Tanzania

1997
Activity of pyronaridine and mepacrine against twelve strains of Plasmodium falciparum in vitro.
    The Journal of antimicrobial chemotherapy, 1996, Volume: 37, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Mefloquine; Naphthyridines; Plasmodium falciparum; Quinacrine; Quinine

1996
[There is no evidence of more symptoms with mefloquine than with other drugs in malaria prophylaxis].
    Nederlands tijdschrift voor geneeskunde, 1997, Apr-19, Volume: 141, Issue:16

    Topics: Antimalarials; Chloroquine; Humans; Mefloquine; Proguanil

1997
[Adverse effects associated with antimalarial chemoprophylaxis].
    Medicina clinica, 1997, May-24, Volume: 108, Issue:20

    Topics: Adolescent; Adult; Aged; Antimalarials; Body Weight; Child; Child, Preschool; Chloroquine; Drug Therapy, Combination; Female; Humans; Male; Mefloquine; Middle Aged; Proguanil; Surveys and Questionnaires; Travel

1997
Compliance with and tolerance of mefloquine and chloroquine + proguanil malaria chemoprophylaxis in French short-term travellers to sub-Saharan Africa.
    Tropical medicine & international health : TM & IH, 1997, Volume: 2, Issue:10

    Topics: Adult; Antimalarials; Chloroquine; Drug Therapy, Combination; Female; Humans; Kenya; Malaria; Male; Mefloquine; Patient Compliance; Proguanil; Senegal; Surveys and Questionnaires; Travel

1997
Update on prevention of malaria for travelers.
    JAMA, 1997, Dec-03, Volume: 278, Issue:21

    Topics: Animals; Antimalarials; Chloroquine; Doxycycline; Drug Resistance; Global Health; Guidelines as Topic; Humans; Malaria; Mefloquine; Plasmodium; Primaquine; Proguanil; Travel

1997
A simplified in vivo drug sensitivity test for malaria in the field.
    The Southeast Asian journal of tropical medicine and public health, 1997, Volume: 28, Issue:2

    Topics: Adult; Animals; Antimalarials; Child; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Myanmar; Plasmodium falciparum; Pyrimethamine; Sulfadoxine; Time Factors

1997
Pfmdr1 Asn1042Asp and Asp1246Tyr polymorphisms, thought to be associated with chloroquine resistance, are present in chloroquine-resistant and -sensitive Brazilian field isolates of Plasmodium falciparum.
    Experimental parasitology, 1998, Volume: 88, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Mefloquine; Plasmodium falciparum; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Quinine

1998
On achieving consensus on the prevention of malaria.
    The Journal of antimicrobial chemotherapy, 1998, Volume: 41, Issue:1

    Topics: Antimalarials; Chemoprevention; Chloroquine; Guidelines as Topic; Humans; Malaria, Falciparum; Mefloquine; Travel

1998
In vitro activity of artemether against African isolates (Senegal) of Plasmodium falciparum in comparison with standard antimalarial drugs.
    The American journal of tropical medicine and hygiene, 1998, Volume: 58, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance; Erythrocytes; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Senegal; Sesquiterpenes

1998
A primary malarial infection is composed of a very wide range of genetically diverse but related parasites.
    The Journal of clinical investigation, 1998, May-01, Volume: 101, Issue:9

    Topics: Africa; Animals; Antimalarials; Biomarkers; Chloroquine; Clone Cells; Culicidae; Drug Resistance; Genetic Variation; Humans; Insect Bites and Stings; Malaria, Falciparum; Mefloquine; Parasitology; Phenotype; Plasmodium falciparum; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Quinine; Thailand

1998
New aspects of malaria imported from Ethiopia.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1998, Volume: 26, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Culicidae; Disease Reservoirs; Drug Therapy, Combination; Ethiopia; Humans; Incidence; Insect Vectors; Israel; Malaria, Vivax; Mefloquine; Primaquine; Travel

1998
Follow-up of the susceptibility of Plasmodium falciparum to antimalarials in Gabon.
    The American journal of tropical medicine and hygiene, 1998, Volume: 58, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Follow-Up Studies; Gabon; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes; Sulfadoxine

1998
The effect of chemoprophylaxis on the timing of onset of falciparum malaria.
    Tropical medicine & international health : TM & IH, 1998, Volume: 3, Issue:4

    Topics: Antimalarials; Chemoprevention; Chloroquine; Drug Combinations; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Proguanil; Retrospective Studies; Time Factors; Travel

1998
Effectiveness of chemoprophylaxis and other determinants of malaria in travellers to Kenya.
    Tropical medicine & international health : TM & IH, 1998, Volume: 3, Issue:5

    Topics: Adult; Animals; Antimalarials; Case-Control Studies; Chloroquine; Humans; Kenya; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Proguanil; Risk Factors; Travel

1998
In vitro sensitivity of Plasmodium falciparum to halofantrine compared with chloroquine, quinine and mefloquine in the region of Bobo-Dioulasso, Burkina Faso (West Africa).
    Tropical medicine & international health : TM & IH, 1998, Volume: 3, Issue:5

    Topics: Animals; Antimalarials; Burkina Faso; Chloroquine; Drug Resistance; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine

1998
Mefloquine to prevent malaria. Withdrawal rates are misleading measure of tolerability.
    BMJ (Clinical research ed.), 1998, Jun-27, Volume: 316, Issue:7149

    Topics: Anti-Bacterial Agents; Antimalarials; Chloroquine; Doxycycline; Humans; Malaria; Mefloquine; Proguanil; Travel; Treatment Refusal

1998
[Chemoprophylaxis of malaria in travelers to endemic zones].
    Revista clinica espanola, 1998, Volume: 198, Issue:6

    Topics: Antimalarials; Chloroquine; Dapsone; Doxycycline; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Proguanil; Pyrimethamine; Travel

1998
Functional analysis of pfmdr1 gene of Plasmodium falciparum.
    Methods in enzymology, 1998, Volume: 292

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chloroquine; CHO Cells; Cricetinae; Drug Resistance, Multiple; Genes, Protozoan; Mefloquine; Phenotype; Plasmodium falciparum; Recombinant Proteins; Transfection

1998
Safety of mefloquine and other antimalarial agents in the first trimester of pregnancy.
    Journal of travel medicine, 1998, Volume: 5, Issue:3

    Topics: Abnormalities, Drug-Induced; Abortion, Spontaneous; Adult; Adverse Drug Reaction Reporting Systems; Antimalarials; Chloroquine; Databases, Factual; Drug Combinations; Drug Industry; Female; Humans; Malaria; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Pregnancy Trimester, First; Proguanil; Prospective Studies; Pyrimethamine; Risk Factors; Safety; Sulfadoxine; Surveys and Questionnaires

1998
[Considering disparities in resistance of Plasmodium falciparum in Africa in chemoprevention decisions].
    Presse medicale (Paris, France : 1983), 1998, Sep-26, Volume: 27, Issue:28

    Topics: Africa; Animals; Antimalarials; Chloroquine; Cross-Cultural Comparison; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Folic Acid Antagonists; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Proguanil; Seasons; Travel; Triazines

1998
Adverse effects of antimalarial prophylactic drugs: an important consideration in the risk-benefit equation.
    The Annals of pharmacotherapy, 1998, Volume: 32, Issue:10

    Topics: Animals; Anti-Bacterial Agents; Antimalarials; Atovaquone; Azithromycin; Chloroquine; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Naphthoquinones; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Risk Assessment

1998
Central role of hemoglobin degradation in mechanisms of action of 4-aminoquinolines, quinoline methanols, and phenanthrene methanols.
    Antimicrobial agents and chemotherapy, 1998, Volume: 42, Issue:11

    Topics: Amodiaquine; Antimalarials; Chloroquine; Hemoglobins; Humans; Leucine; Mefloquine; Phenanthrenes; Primaquine; Protease Inhibitors

1998
In vitro susceptibility studies of Malaysian Plasmodium falciparum isolates and clones against schizontocidal drugs.
    Folia parasitologica, 1998, Volume: 45, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Malaysia; Mefloquine; Plasmodium falciparum; Quinine

1998
A common mechanism for blockade of heme polymerization by antimalarial quinolines.
    The Journal of biological chemistry, 1998, Nov-20, Volume: 273, Issue:47

    Topics: Animals; Antimalarials; Chloroquine; Erythrocytes; Heme; Hemeproteins; Mefloquine; Plasmodium falciparum; Polymers; Quinidine; Quinolines

1998
Malaria at Christmas: risks of prophylaxis versus risks of malaria.
    BMJ (Clinical research ed.), 1998, Nov-28, Volume: 317, Issue:7171

    Topics: Adult; Antimalarials; Chloroquine; Disease Outbreaks; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Proguanil; Risk Factors; Travel; United Kingdom

1998
Science commentary: protection against malaria.
    BMJ (Clinical research ed.), 1998, Nov-28, Volume: 317, Issue:7171

    Topics: Antimalarials; Chloroquine; Humans; Malaria; Mefloquine; Proguanil; Travel

1998
A severe adverse reaction to mefloquine and chloroquine prophylaxis.
    Australian family physician, 1998, Volume: 27, Issue:12

    Topics: Adult; Antimalarials; Chloroquine; Drug Hypersensitivity; Humans; Malaria; Male; Mefloquine; Severity of Illness Index

1998
8-Aminoquinolines active against blood stage Plasmodium falciparum in vitro inhibit hematin polymerization.
    Antimicrobial agents and chemotherapy, 1999, Volume: 43, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Hemin; Humans; Hydrogen-Ion Concentration; Mefloquine; Models, Molecular; Plasmodium falciparum; Quinolines

1999
[The proper use of antimalarial drugs currently available].
    Bulletin de la Societe de pathologie exotique (1990), 1998, Volume: 91, Issue:5 Pt 1-2

    Topics: Animals; Antimalarials; Chemoprevention; Chloroquine; Contraindications; Drug Combinations; Drug Resistance; Endemic Diseases; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Phenanthrenes; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Proguanil; Pyrimethamine; Quinine; Sulfadoxine; Travel

1998
[Pulmonary manifestations associated with malaria].
    Revue de pneumologie clinique, 1998, Volume: 54, Issue:6

    Topics: Adult; Anti-Bacterial Agents; Antimalarials; Bronchitis; Child; Chloroquine; Female; Humans; Infant, Newborn; Lung Diseases; Malaria, Falciparum; Male; Mefloquine; Oxygen Inhalation Therapy; Phenanthrenes; Pleurisy; Pregnancy; Pregnancy Complications, Parasitic; Pulmonary Edema; Quinidine; Quinine; Respiratory Distress Syndrome, Newborn; Travel

1998
Malaria prophylaxis for the 1990s and beyond.
    British journal of hospital medicine, 1997, Dec-10, Volume: 58, Issue:11

    Topics: Antimalarials; Atovaquone; Chloroquine; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum; Mefloquine; Naphthoquinones; Proguanil

1997
In vitro susceptibility of African Plasmodium falciparum isolates to dihydroartemisinin and the risk factors for resistance to qinghaosu.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chloroquine; Cross Reactions; Drug Evaluation, Preclinical; Drug Resistance; France; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes; Travel

1998
Antimalarial drug resistance and combination chemotherapy.
    Philosophical transactions of the Royal Society of London. Series B, Biological sciences, 1999, Apr-29, Volume: 354, Issue:1384

    Topics: Animals; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Naphthoquinones; Plasmodium falciparum; Sesquiterpenes

1999
Efficacy and tolerability of a low-dose mefloquine-sulfadoxine-pyrimethamine combination compared with chloroquine in the treatment of acute malaria infection in a population with multiple drug-resistant Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1999, Volume: 61, Issue:1

    Topics: Adolescent; Adult; Animals; Antimalarials; Blood; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance, Multiple; Female; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Nigeria; Plasmodium falciparum; Prospective Studies; Pyrimethamine; Random Allocation; Sulfadoxine

1999
Plasmodium chabaudi: effect of antimalarial drugs on gametocytogenesis.
    Experimental parasitology, 1999, Volume: 93, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Gametogenesis; Malaria; Male; Mefloquine; Mice; Mice, Inbred C57BL; Plasmodium chabaudi; Pyrimethamine; Quinine

1999
Phenotypic and genotypic characteristics of recently adapted isolates of Plasmodium falciparum from Thailand.
    The American journal of tropical medicine and hygiene, 1999, Volume: 60, Issue:3

    Topics: Animals; Antimalarials; Blotting, Western; Chloroquine; DNA Fingerprinting; DNA, Protozoan; Drug Resistance; Electrophoresis, Agar Gel; Gene Dosage; Genotype; Humans; Malaria, Falciparum; Mefloquine; Penfluridol; Phenanthrenes; Phenotype; Plasmodium falciparum; Polymerase Chain Reaction; Quinine; Thailand; Verapamil

1999
The microculture tetrazolium assay (MTA): another colorimetric method of testing Plasmodium falciparum chemosensitivity.
    Annals of tropical medicine and parasitology, 1999, Volume: 93, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Colorimetry; Dose-Response Relationship, Drug; Drug Resistance; L-Lactate Dehydrogenase; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Tetrazolium Salts

1999
[Prevention of malaria].
    Revista clinica espanola, 1999, Volume: 199, Issue:8

    Topics: Anti-Bacterial Agents; Antimalarials; Chloroquine; Doxycycline; Female; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Primaquine; Proguanil; Risk Assessment; Risk Factors; Time Factors; Travel

1999
Suboptimal prophylaxis for P. falciparum.
    Journal of travel medicine, 1999, Volume: 6, Issue:4

    Topics: Antimalarials; Chloroquine; Fatal Outcome; Humans; Kenya; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Multiple Organ Failure; Treatment Failure

1999
Analysis of mefloquine resistance and amplification of pfmdr1 in multidrug-resistant Plasmodium falciparum isolates from Thailand.
    The American journal of tropical medicine and hygiene, 1999, Volume: 61, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Chromosome Mapping; DNA Primers; DNA, Protozoan; Drug Resistance, Multiple; Electrophoresis, Agar Gel; Electrophoresis, Gel, Pulsed-Field; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Quinine; Scintillation Counting; Sequence Analysis, DNA; Thailand

1999
Inoculum effect leads to overestimation of in vitro resistance for artemisinin derivatives and standard antimalarials: a Gambian field study.
    Parasitology, 1999, Volume: 119 ( Pt 5)

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Gambia; Hematocrit; Humans; Malaria, Falciparum; Mefloquine; Parasitemia; Phenanthrenes; Plasmodium falciparum; Quinine; Scintillation Counting; Sensitivity and Specificity; Sesquiterpenes

1999
Potent antimalarial activity of clotrimazole in in vitro cultures of Plasmodium falciparum.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Jan-04, Volume: 97, Issue:1

    Topics: Animals; Antifungal Agents; Antimalarials; Cells, Cultured; Chloroquine; Clotrimazole; Growth Inhibitors; Histocytochemistry; Hypoxanthine; Mefloquine; Plasmodium falciparum

2000
Prevention of malaria.
    The Medical letter on drugs and therapeutics, 2000, Jan-24, Volume: 42, Issue:1070

    Topics: Antimalarials; Chloroquine; Doxycycline; Drug Resistance; Humans; Malaria; Mefloquine

2000
Pgh1 modulates sensitivity and resistance to multiple antimalarials in Plasmodium falciparum.
    Nature, 2000, Feb-24, Volume: 403, Issue:6772

    Topics: Amino Acid Substitution; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Chloroquine; Cloning, Molecular; Drug Resistance; Mefloquine; Mutation; Phenanthrenes; Plasmodium falciparum; Protozoan Proteins; Quinine; Sesquiterpenes; Verapamil

2000
Gametocytocidal activity of pyronaridine and DNA topoisomerase II inhibitors against multidrug-resistant Plasmodium falciparum in vitro.
    Parasitology international, 2000, Volume: 48, Issue:4

    Topics: Amsacrine; Animals; Antimalarials; Chloroquine; Drug Resistance, Multiple; Enzyme Inhibitors; Etoposide; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Naphthyridines; Norfloxacin; Nucleic Acid Synthesis Inhibitors; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Thailand; Topoisomerase II Inhibitors; Triazines

2000
Management of a case of chloroquine-resistant falciparum malaria in a pregnant woman with glucose-6-phosphate dehydrogenase (G6PD) deficiency.
    American journal of perinatology, 1999, Volume: 16, Issue:8

    Topics: Adult; Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Drug Therapy, Combination; Female; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Microbial Sensitivity Tests; Pregnancy; Pregnancy Complications; Pregnancy Outcome; Pyrimethamine

1999
Prevention and treatment of malaria in UK travellers.
    Hospital medicine (London, England : 1998), 2000, Volume: 61, Issue:3

    Topics: Age Factors; Antimalarials; Chloroquine; Contraindications; Doxycycline; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Proguanil; Quinine; Risk Factors; Travel

2000
An unusual case of multidrug-resistant Plasmodium vivax malaria in Mumbai (Bombay), India.
    Annals of tropical medicine and parasitology, 2000, Volume: 94, Issue:2

    Topics: Adolescent; Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance, Multiple; Humans; India; Malaria, Vivax; Male; Mefloquine; Plasmodium vivax; Primaquine; Pyrimethamine; Sesquiterpenes; Sulfadoxine

2000
[Malaria imported to Norway 1989-98].
    Tidsskrift for den Norske laegeforening : tidsskrift for praktisk medicin, ny raekke, 2000, May-30, Volume: 120, Issue:14

    Topics: Adolescent; Adult; Aged; Antimalarials; Child; Child, Preschool; Chloroquine; Disease Notification; Emigration and Immigration; Female; Humans; Infant; Insect Bites and Stings; Malaria; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Norway; Proguanil; Travel

2000
In vitro susceptibility of Plasmodium falciparum to four antimalarial drugs in the Central Province of Papua New Guinea.
    Papua and New Guinea medical journal, 1998, Volume: 41, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Mefloquine; Microbial Sensitivity Tests; Papua New Guinea; Phenanthrenes; Plasmodium falciparum; Quinine

1998
Interaction of chloroquine and its analogues with heme: An isothermal titration calorimetric study.
    Biochemical and biophysical research communications, 2000, Oct-05, Volume: 276, Issue:3

    Topics: Amodiaquine; Antimalarials; Binding Sites; Calorimetry; Chloroquine; Hemin; Hydrogen-Ion Concentration; Mefloquine; Octoxynol; Quinidine; Quinine; Solubility; Spectrophotometry, Ultraviolet; Temperature; Thermodynamics; Titrimetry

2000
Treatment of uncomplicated Plasmodium falciparum malaria in Myanmar: a clinical decision analysis.
    The Southeast Asian journal of tropical medicine and public health, 2000, Volume: 31, Issue:2

    Topics: Antimalarials; Chloroquine; Cost-Benefit Analysis; Decision Support Techniques; Decision Trees; Drug Combinations; Humans; Malaria, Falciparum; Mefloquine; Myanmar; Pyrimethamine; Sulfadoxine; Treatment Failure; Treatment Outcome

2000
Adaptation of a chloroquine-resistant strain of Plasmodium vivax from Indonesia to New World monkeys.
    The American journal of tropical medicine and hygiene, 2000, Volume: 62, Issue:4

    Topics: Adaptation, Physiological; Adult; Amodiaquine; Animals; Antimalarials; Aotidae; Child; Chloroquine; Disease Models, Animal; Drug Resistance; Female; Humans; Indonesia; Malaria, Vivax; Male; Mefloquine; Parasitemia; Plasmodium vivax; Saimiri; Splenectomy

2000
Coadministration of mefloquine and chloroqine: use of a pharmacokinetic-based approach to reduce toxicity.
    The Pediatric infectious disease journal, 2001, Volume: 20, Issue:2

    Topics: Antimalarials; Child; Chloroquine; Drug Overdose; Drug Synergism; Drug Therapy, Combination; Humans; Malaria; Male; Mefloquine

2001
Vivax malaria: also a challenge to biomedical sciences and services.
    The Journal of the Association of Physicians of India, 1999, Volume: 47, Issue:12

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria, Vivax; Mefloquine; Plasmodium vivax; Primaquine

1999
Declining chloroquine resistance of Plasmodium falciparum in Lambaréné, Gabon from 1992 to 1998.
    Wiener klinische Wochenschrift, 2001, Jan-15, Volume: 113, Issue:1-2

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Gabon; Humans; In Vitro Techniques; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Practice Guidelines as Topic; Prospective Studies; Quinine

2001
Madagascan isolates of Plasmodium falciparum showing low sensitivity to artemether in vitro.
    Annals of tropical medicine and parasitology, 2001, Volume: 95, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Confidence Intervals; Drug Resistance; Drug Therapy, Combination; Humans; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Sesquiterpenes; Statistics, Nonparametric

2001
Use of the DELI-microtest to determine the drug sensitivity of Plasmodium falciparum in Burkina Faso.
    Annals of tropical medicine and parasitology, 2001, Volume: 95, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Malaria, Falciparum; Mefloquine; Parasitemia; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Reagent Kits, Diagnostic; Sensitivity and Specificity; Statistics, Nonparametric

2001
Reversal of chloroquine and mefloquine resistance in Plasmodium falciparum by the two monoindole alkaloids, icajine and isoretuline.
    Planta medica, 2001, Volume: 67, Issue:6

    Topics: Alkaloids; Animals; Antimalarials; Chloroquine; Colon; Drug Resistance, Multiple; Drug Synergism; Humans; Indoles; Inhibitory Concentration 50; Mefloquine; Molecular Structure; Plasmodium falciparum; Strychnine; Tumor Cells, Cultured

2001
Death from malaria following inappropriate chemoprophylaxis.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2001, Sep-01, Volume: 33, Issue:5

    Topics: Africa; Animals; Antimalarials; Centers for Disease Control and Prevention, U.S.; Chemoprevention; Child; Chloroquine; Drug Resistance; Fatal Outcome; Humans; Malaria, Falciparum; Mefloquine; Middle Aged; Plasmodium falciparum; Proguanil; Travel; United States

2001
Antimalarial drugs clear resistant parasites from partially immune hosts.
    Antimicrobial agents and chemotherapy, 2001, Volume: 45, Issue:10

    Topics: Animals; Antimalarials; Chloroquine; Disease Models, Animal; Drug Resistance; Immunization; Malaria; Mefloquine; Mice; Plasmodium chabaudi

2001
In vitro susceptibility of Plasmodium falciparum isolates from Myanmar to antimalarial drugs.
    The American journal of tropical medicine and hygiene, 2001, Volume: 65, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Sesquiterpenes

2001
Malaria remains a military medical problem.
    Journal of the Royal Army Medical Corps, 2001, Volume: 147, Issue:3

    Topics: Adult; Animals; Antimalarials; Atovaquone; Chloroquine; Drug Combinations; Global Health; Humans; Kenya; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Military Medicine; Military Personnel; Naphthoquinones; Patient Compliance; Plasmodium falciparum; Plasmodium vivax; Proguanil; Sierra Leone; Treatment Failure; Treatment Outcome; United Kingdom

2001
Differential effects of 4-aminoquinoline-containing antimalarial drugs on hemoglobin digestion in Plasmodium falciparum-infected erythrocytes.
    Biochemical pharmacology, 2002, Feb-01, Volume: 63, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Erythrocytes; Hemoglobins; Mefloquine; Plasmodium falciparum

2002
Efficacy of scopadulcic acid A against Plasmodium falciparum in vitro.
    Journal of natural products, 2002, Volume: 65, Issue:4

    Topics: Animals; Antimalarials; Chloroquine; Diterpenes; Drug Resistance; Humans; In Vitro Techniques; Inhibitory Concentration 50; Mefloquine; Plants, Medicinal; Plasmodium falciparum; Scrophulariaceae

2002
Design, synthesis, and evaluation of new chemosensitizers in multi-drug-resistant Plasmodium falciparum.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Animals; Antimalarials; Cell Line; Chloroquine; Diphenylamine; Drug Resistance, Multiple; Imines; Mefloquine; Molecular Conformation; Phenothiazines; Plasmodium falciparum; Pyrrolidines; Stilbenes; Structure-Activity Relationship

2002
Resistant malaria in a neonate.
    Indian pediatrics, 2002, Volume: 39, Issue:6

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance, Multiple; Drug Therapy, Combination; Female; Follow-Up Studies; Humans; Infant, Newborn; Malaria, Falciparum; Mefloquine; Quinine; Risk Assessment; Sesquiterpenes; Severity of Illness Index; Treatment Outcome

2002
[Many travellers suffer of side-effects of malaria prophylaxis].
    Lakartidningen, 2002, Jun-27, Volume: 99, Issue:26-27

    Topics: Antimalarials; Chloroquine; Drug Eruptions; Gastrointestinal Diseases; Humans; Malaria; Mefloquine; Mental Disorders; Proguanil; Surveys and Questionnaires; Travel

2002
Ligands of the peripheral benzodiazepine receptor are potent inhibitors of Plasmodium falciparum and Toxoplasma gondii in vitro.
    Antimicrobial agents and chemotherapy, 2002, Volume: 46, Issue:10

    Topics: Animals; Antimalarials; Chloroquine; Erythrocytes; Fibroblasts; Flurazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hemeproteins; Humans; Isoquinolines; Ligands; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Toxoplasma

2002
Chloroquine resistance in Plasmodium falciparum malaria parasites conferred by pfcrt mutations.
    Science (New York, N.Y.), 2002, Oct-04, Volume: 298, Issue:5591

    Topics: Alleles; Amodiaquine; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Chloroquine; Cloning, Molecular; Drug Resistance; Genes, Protozoan; Haplotypes; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Parasitic Sensitivity Tests; Phenotype; Plasmodium falciparum; Point Mutation; Protozoan Proteins; Quinine; Sesquiterpenes; Transfection; Verapamil

2002
Haem polymerase as a novel target of antimalarial action of cyproheptadine.
    Biochemical pharmacology, 2002, Nov-01, Volume: 64, Issue:9

    Topics: Animals; Antimalarials; Chloroquine; Cyproheptadine; Disease Models, Animal; Drug Resistance; Enzyme Inhibitors; Hemeproteins; Mefloquine; Mice; Plasmodium yoelii; Quinine; Transferases; Treatment Outcome

2002
Molecular characterisation of drug-resistant Plasmodium falciparum from Thailand.
    Malaria journal, 2002, Oct-14, Volume: 1

    Topics: Amodiaquine; Animals; Antimalarials; ATP-Binding Cassette Transporters; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Gene Frequency; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine; Thailand

2002
Discovery of novel targets of quinoline drugs in the human purine binding proteome.
    Molecular pharmacology, 2002, Volume: 62, Issue:6

    Topics: Adenosine Triphosphate; Aldehyde Dehydrogenase; Aldehyde Dehydrogenase 1 Family; Animals; Antimalarials; Chloroquine; Chromatography, Agarose; Enzyme Inhibitors; Erythrocytes; Humans; Isoenzymes; Mefloquine; Mice; NAD(P)H Dehydrogenase (Quinone); Plasmodium falciparum; Primaquine; Proteome; Retinal Dehydrogenase; Sepharose

2002
Drug-resistant Plasmodium falciparum infection in immigrants and non-immune travellers.
    Clinical microbiology and infection : the official publication of the European Society of Clinical Microbiology and Infectious Diseases, 2002, Volume: 8, Issue:11

    Topics: Adult; Africa; Animals; Antimalarials; Asia, Southeastern; Chloroquine; Drug Resistance; Emigration and Immigration; Female; Humans; Inhibitory Concentration 50; Kuwait; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Travel

2002
In vitro activity of chloroquine, quinine, mefloquine and halofantrine against Gabonese isolates of Plasmodium falciparum.
    Tropical medicine & international health : TM & IH, 2003, Volume: 8, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Gabon; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Quinine

2003
[Assay of sensitivity of Plasmodium falciparum to chloroquine, amodiaquine, piperaquine, mefloquine and quinine in Yunnan province].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1999, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

1999
Profile and evolution of the chemosusceptibility of falciparum malaria imported into France in 2000.
    Euro surveillance : bulletin Europeen sur les maladies transmissibles = European communicable disease bulletin, 2002, Volume: 7, Issue:7

    Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; France; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Proguanil; Quinine; Triazines

2002
In-vitro sensitivity of Plasmodium falciparum to chloroquine, halofantrine, mefloquine and quinine in Madagascar.
    East African medical journal, 2002, Volume: 79, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Evaluation, Preclinical; Drug Resistance; Hospitals, Public; Hospitals, Urban; Humans; Madagascar; Malaria, Falciparum; Mefloquine; Microbial Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Quinine; Rural Health

2002
Drug-resistant malaria in Bangladesh: an in vitro assessment.
    The American journal of tropical medicine and hygiene, 2003, Volume: 68, Issue:2

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Bangladesh; Chloroquine; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Sesquiterpenes

2003
In vitro sensitivity of Plasmodium falciparum to amodiaquine compared with other major antimalarials in Madagascar.
    Parassitologia, 2002, Volume: 44, Issue:3-4

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Humans; Inhibitory Concentration 50; Madagascar; Malaria, Falciparum; Mefloquine; Parasitemia; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Triazines

2002
Malaria in Austria 1990-2000.
    Euro surveillance : bulletin Europeen sur les maladies transmissibles = European communicable disease bulletin, 2003, Volume: 8, Issue:4

    Topics: Adolescent; Adult; Age Distribution; Animals; Austria; Chemoprevention; Child; Child, Preschool; Chloroquine; Disease Notification; Drug Combinations; Female; Humans; Infant; Infant, Newborn; Malaria; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Patient Compliance; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Proguanil; Pyrimethamine; Sex Distribution; Sulfadoxine

2003
Failure of a chloroquine chemoprophylaxis program to adequately prevent malaria during pregnancy in Koupéla District, Burkina Faso.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2003, Jun-01, Volume: 36, Issue:11

    Topics: Adolescent; Adult; Animals; Antimalarials; Burkina Faso; Chemoprevention; Chloroquine; Cross-Sectional Studies; Culicidae; Disease Vectors; Female; Humans; Infant, Low Birth Weight; Infant, Newborn; Insecticides; Malaria, Falciparum; Mefloquine; Parasitemia; Pregnancy; Pregnancy Complications, Parasitic; Treatment Outcome

2003
[Malaria--case report].
    Deutsche medizinische Wochenschrift (1946), 2003, Jun-06, Volume: 128, Issue:23

    Topics: Adult; Anti-Infective Agents; Antidiarrheals; Antimalarials; Chloroquine; Ciprofloxacin; Diarrhea; Emergencies; Fluid Therapy; Glasgow Coma Scale; Humans; Loperamide; Malaria, Cerebral; Malaria, Falciparum; Male; Mefloquine; Nigeria; Parasitemia; Positive-Pressure Respiration; Proguanil; Quinine; Respiratory Distress Syndrome; Travel

2003
The chemotherapy of rodent malaria. LXI. Drug combinations to impede the selection of drug resistance, part 4: the potential role of 8-aminoquinolines.
    Annals of tropical medicine and parasitology, 2003, Volume: 97, Issue:3

    Topics: Aminoquinolines; Animals; Antimalarials; Chloroquine; Disease Models, Animal; Drug Resistance; Drug Therapy, Combination; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Mice; Plasmodium berghei; Plasmodium chabaudi; Plasmodium yoelii; Primaquine; Time Factors

2003
Mapping of the Plasmodium falciparum multidrug resistance gene 5'-upstream region, and evidence of induction of transcript levels by antimalarial drugs in chloroquine sensitive parasites.
    Molecular microbiology, 2003, Volume: 49, Issue:3

    Topics: 5' Untranslated Regions; Animals; Antimalarials; ATP-Binding Cassette Transporters; Base Sequence; Chloroquine; Chromosome Mapping; Drug Resistance, Multiple; Gene Expression Regulation; Genes, MDR; Genes, Protozoan; Genes, Reporter; Luciferases; Mefloquine; Molecular Sequence Data; Plasmodium falciparum; Polymerase Chain Reaction; Protozoan Proteins; Pyrimethamine; Quinine; Reverse Transcriptase Polymerase Chain Reaction; Sequence Alignment; Sequence Homology, Nucleic Acid; Transcription, Genetic

2003
Asymptomatic, recrudescent, chloroquine-resistant Plasmodium falciparum infections in Nigerian children: clinical and parasitological characteristics and implications for the transmission of drug-resistant parasites.
    Annals of tropical medicine and parasitology, 2003, Volume: 97, Issue:5

    Topics: Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Nigeria; Plasmodium falciparum; Prevalence; Pyrimethamine; Recurrence; Statistics as Topic; Sulfadoxine; Treatment Failure

2003
Delayed onset of malaria--implications for chemoprophylaxis in travelers.
    The New England journal of medicine, 2003, Oct-16, Volume: 349, Issue:16

    Topics: Antimalarials; Chloroquine; Drug Resistance; Endemic Diseases; Humans; Israel; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Population Surveillance; Time Factors; Travel; United States

2003
Diagnosis and treatment of malaria in children.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2003, Nov-15, Volume: 37, Issue:10

    Topics: Animals; Antimalarials; Atovaquone; Child; Chloroquine; Drug Combinations; Humans; Malaria; Malaria, Falciparum; Mefloquine; Naphthoquinones; Plasmodium falciparum; Proguanil; Pyrimethamine; Sulfadoxine

2003
A cost-effectiveness analysis of three antimalarial treatments for acute, uncomplicated Plasmodium falciparum malaria in Mumbai, India.
    The Journal of the Association of Physicians of India, 2003, Volume: 51

    Topics: Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Chloroquine; Clinical Trials as Topic; Cost-Benefit Analysis; Drug Combinations; Economics, Pharmaceutical; Ethanolamines; Female; Fluorenes; Hospitalization; Humans; India; Malaria, Falciparum; Male; Mefloquine; Sesquiterpenes

2003
Malaria during pregnancy in a reference centre from the Brazilian Amazon: unexpected increase in the frequency of Plasmodium falciparum infections.
    Memorias do Instituto Oswaldo Cruz, 2004, Volume: 99, Issue:1

    Topics: Adolescent; Adult; Antimalarials; Brazil; Child; Chloroquine; Cross-Sectional Studies; Female; Humans; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Prevalence; Quinine

2004
Defective DNA repair as a potential mechanism for the rapid development of drug resistance in Plasmodium falciparum.
    Biochemistry, 2004, May-04, Volume: 43, Issue:17

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; DNA Damage; DNA Repair; Drug Resistance; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Pyrimethamine; Quinine; Sesquiterpenes; Sulfanilamide; Sulfanilamides; Ultraviolet Rays

2004
In vitro susceptibility of Plasmodium falciparum isolates to chloroquine and mefloquine in southeastern Mindanao Island, the Philippines.
    The Southeast Asian journal of tropical medicine and public health, 2003, Volume: 34, Issue:3

    Topics: Adolescent; Adult; Animals; Antimalarials; Chloroquine; Drug Resistance, Multiple; Female; Humans; In Vitro Techniques; Malaria, Falciparum; Male; Mefloquine; Parasitic Sensitivity Tests; Philippines; Plasmodium falciparum; Residence Characteristics

2003
Polymorphism of the Plasmodium falciparum multidrug resistance and chloroquine resistance transporter genes and in vitro susceptibility to aminoquinolines in isolates from the Peruvian Amazon.
    The American journal of tropical medicine and hygiene, 2004, Volume: 70, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance, Multiple; Genes, MDR; Genotype; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Mutation; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine

2004
Antimalarial quinolines and artemisinin inhibit endocytosis in Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2004, Volume: 48, Issue:7

    Topics: Ammonium Chloride; Animals; Antimalarials; Artemisinins; Biotin; Blotting, Western; Chloroquine; Dextrans; Endocytosis; Fluorescein-5-isothiocyanate; Fluorescent Antibody Technique; Fluorescent Dyes; Hemoglobins; Mefloquine; Microscopy, Electron; Microscopy, Fluorescence; Monensin; Plasmodium falciparum; Quinolones; Sesquiterpenes; Transport Vesicles; Vacuoles

2004
Application of multi-component reactions to antimalarial drug discovery. Part 1: Parallel synthesis and antiplasmodial activity of new 4-aminoquinoline Ugi adducts.
    Bioorganic & medicinal chemistry letters, 2004, Aug-02, Volume: 14, Issue:15

    Topics: Animals; Antimalarials; Chloroquine; Mefloquine; Molecular Conformation; Molecular Structure; Plasmodium falciparum; Quinine; Structure-Activity Relationship

2004
The in-vitro antimalarial activity of ferrochloroquine, measured against Cambodian isolates of Plasmodium falciparum.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Cambodia; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Mutation; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Sesquiterpenes

2004
The sensitivities of yeast strains deficient in PDR ABC transporters, to quinoline-ring antimalarial drugs.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:6

    Topics: Antimalarials; ATP-Binding Cassette Transporters; Chloroquine; Cycloheximide; Drug Resistance, Multiple, Fungal; Gene Deletion; Genes, Fungal; Mefloquine; Mutation; Quinacrine; Quinidine; Quinine; Saccharomyces cerevisiae; Transcription, Genetic

2004
[Acute malaria in an Israeli tourist to Kenya].
    Harefuah, 1999, Apr-02, Volume: 136, Issue:7

    Topics: Acidosis; Adult; Chloroquine; Drug Therapy, Combination; Humans; Malaria, Falciparum; Male; Mefloquine; Treatment Outcome

1999
In vitro monitoring of Plasmodium falciparum susceptibility to artesunate, mefloquine, quinine and chloroquine in Cambodia: 2001-2002.
    Acta tropica, 2005, Volume: 93, Issue:1

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Cambodia; Chloroquine; Drug Resistance; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Quinine; Sesquiterpenes; Statistics, Nonparametric

2005
Efficacy of antimalarial chemoprophylaxis among French residents travelling to Africa.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 2005, Volume: 99, Issue:2

    Topics: Adult; Africa South of the Sahara; Africa, Western; Antimalarials; Case-Control Studies; Chloroquine; Drug Therapy, Combination; Female; France; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Patient Compliance; Proguanil; Travel; Treatment Outcome

2005
Absence of nucleotide polymorphism in a Plasmodium vivax multidrug resistance gene after failure of mefloquine prophylaxis in French Guyana.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 2005, Volume: 99, Issue:3

    Topics: Adult; Animals; Antimalarials; Chloroquine; Drug Resistance, Multiple; Humans; Malaria, Vivax; Male; Mefloquine; Military Personnel; Mutation; Plasmodium vivax; Polymorphism, Single Nucleotide

2005
Syndromic management of prolonged fever: a cost-effective approach.
    Tropical doctor, 2005, Volume: 35, Issue:1

    Topics: Anti-Infective Agents; Antimalarials; Chloramphenicol; Chloroquine; Cost-Benefit Analysis; Drug Therapy, Combination; Fever; Humans; Infant; Mefloquine; Time Factors; Trimethoprim, Sulfamethoxazole Drug Combination

2005
ATPase activity of purified plasma membranes and digestive vacuoles from Plasmodium falciparum.
    Molecular and biochemical parasitology, 2005, Volume: 141, Issue:1

    Topics: Adenosine Triphosphatases; Animals; Antimalarials; Artemisinins; Cell Membrane; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinine; Sesquiterpenes; Subcellular Fractions; Vacuoles

2005
Molecular epidemiology of drug resistance markers of Plasmodium falciparum malaria in Thailand.
    Tropical medicine & international health : TM & IH, 2005, Volume: 10, Issue:8

    Topics: Animals; Antimalarials; ATP-Binding Cassette Transporters; Biomarkers; Chloroquine; Drug Resistance; Endemic Diseases; Genes, MDR; Genotype; Humans; Malaria, Falciparum; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Microbial Sensitivity Tests; Mutation; Plasmodium falciparum; Polymorphism, Restriction Fragment Length; Protozoan Proteins; Thailand

2005
In vitro antimalarial drug susceptibility in Thai border areas from 1998-2003.
    Malaria journal, 2005, Aug-02, Volume: 4

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Quinine; Sesquiterpenes; Thailand; Time Factors

2005
[Malaria prophylaxis for long-term travellers and expatriates].
    Ugeskrift for laeger, 2005, Oct-17, Volume: 167, Issue:42

    Topics: Antimalarials; Atovaquone; Chloroquine; Counseling; Doxycycline; Drug Combinations; Humans; Insect Bites and Stings; Malaria; Mefloquine; Mosquito Control; Naphthoquinones; Proguanil; Risk Assessment; Risk Factors; Travel

2005
In vitro susceptibility and genetic variations for chloroquine and mefloquine in Plasmodium falciparum isolates from Thai-Myanmar border.
    The Southeast Asian journal of tropical medicine and public health, 2005, Volume: 36 Suppl 4

    Topics: Animals; Chloroquine; Disease Susceptibility; Drug Resistance, Microbial; Genetic Variation; Humans; In Vitro Techniques; Malaria; Mefloquine; Mutation; Myanmar; Plasmodium falciparum; Polymorphism, Genetic; Risk Factors; Thailand

2005
Mefloquine-induced mania in a 22-year-old Chinese man.
    Singapore medical journal, 2006, Volume: 47, Issue:6

    Topics: Acute Disease; Adult; Animals; Antimalarials; Bipolar Disorder; Chloroquine; Contraindications; Humans; Malaria, Falciparum; Male; Mefloquine; Nonprescription Drugs; Risk Factors; Risperidone; Singapore

2006
In vitro study assessing the response of plasmodium falciparum malaria to chloroquine, sulfadoxine/pyrimethamine, quinine and mefloquine in Wad Medani District, Sudan.
    Saudi medical journal, 2006, Volume: 27, Issue:6

    Topics: Animals; Antimalarials; Chloroquine; In Vitro Techniques; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrimethamine; Quinine; Sudan; Sulfadoxine

2006
Carbenoxolone and mefloquine suppress tremor in the harmaline mouse model of essential tremor.
    Movement disorders : official journal of the Movement Disorder Society, 2006, Volume: 21, Issue:10

    Topics: 1-Octanol; Animals; Carbenoxolone; Central Nervous System Stimulants; Cerebellum; Chloroquine; Connexins; Disease Models, Animal; Dose-Response Relationship, Drug; Essential Tremor; Female; Gap Junction delta-2 Protein; Gap Junctions; Glycyrrhizic Acid; Harmaline; Heptanol; Injections, Subcutaneous; Mefloquine; Mice; Mice, Inbred ICR; Olivary Nucleus

2006
Drug interactions and pharmacogenetic reactions are the basis for chloroquine and mefloquine-induced psychosis.
    Medical hypotheses, 2006, Volume: 67, Issue:5

    Topics: Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chloroquine; Drug Interactions; Drug-Related Side Effects and Adverse Reactions; Humans; Loperamide; Mefloquine; Mental Disorders; Psychotic Disorders

2006
Fluoxetine potentiates chloroquine and mefloquine effect on multidrug-resistant Plasmodium falciparum in vitro.
    Japanese journal of infectious diseases, 2006, Volume: 59, Issue:5

    Topics: Animals; Antimalarials; Cells, Cultured; Chloroquine; Drug Resistance, Multiple; Drug Synergism; Erythrocytes; Fluoxetine; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Plasmodium falciparum

2006
Synergistic interactions of the antiretroviral protease inhibitors saquinavir and ritonavir with chloroquine and mefloquine against Plasmodium falciparum in vitro.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Drug Synergism; HIV Protease Inhibitors; Humans; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Ritonavir; Saquinavir

2007
Roxithromycin potentiates the effects of chloroquine and mefloquine on multidrug-resistant Plasmodium falciparum in vitro.
    Experimental parasitology, 2007, Volume: 115, Issue:4

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Synergism; Inhibitory Concentration 50; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Roxithromycin

2007
[A plasmodium alciparum malaria case originated from Mozambique: clues for the diagnosis and therapy].
    Mikrobiyoloji bulteni, 2006, Volume: 40, Issue:4

    Topics: Animals; Antimalarials; Canada; Chloroquine; Doxycycline; Drug Resistance; Erythrocytes; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Mozambique; Parasitemia; Plasmodium falciparum; Quinine; Secondary Prevention; Travel; Turkey

2006
Overestimating resistance in field testing of malaria parasites: simple methods for estimating high EC50 values using a Bayesian approach.
    Malaria journal, 2007, Jan-17, Volume: 6

    Topics: Algorithms; Animals; Antimalarials; Artemisinins; Artesunate; Bayes Theorem; Chloroquine; Computer Simulation; Dose-Response Relationship, Drug; Drug Resistance; False Positive Reactions; Inhibitory Concentration 50; Mefloquine; Models, Biological; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes

2007
In vitro antimalarial drug susceptibility and pfcrt mutation among fresh Plasmodium falciparum isolates from the Lao PDR (Laos).
    The American journal of tropical medicine and hygiene, 2007, Volume: 76, Issue:2

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; DNA, Protozoan; Drug Resistance; Ethanolamines; Female; Fluorenes; Humans; Inhibitory Concentration 50; Laos; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Protozoan Proteins; Sesquiterpenes

2007
A non-radiolabeled heme-GSH interaction test for the screening of antimalarial compounds.
    Experimental parasitology, 2007, Volume: 116, Issue:3

    Topics: Amodiaquine; Animals; Antimalarials; Artemether; Artemisinins; Atovaquone; Chloroquine; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; Glutathione; Heme; Indicators and Reagents; Mefloquine; Methylene Blue; o-Phthalaldehyde; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Spectrometry, Fluorescence

2007
The antimalarial drugs quinine, chloroquine and mefloquine are antagonists at 5-HT3 receptors.
    British journal of pharmacology, 2007, Volume: 151, Issue:5

    Topics: Algorithms; Animals; Antimalarials; Binding, Competitive; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Electrophysiology; Female; Granisetron; In Vitro Techniques; Kinetics; Mefloquine; Models, Molecular; Oocytes; Quinine; Radioligand Assay; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Xenopus laevis

2007
The in-vitro susceptibilities of Ghanaian Plasmodium falciparum to antimalarial drugs.
    Annals of tropical medicine and parasitology, 2007, Volume: 101, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Artesunate; Child, Preschool; Chloroquine; Drug Resistance; Ghana; Humans; Infant; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

2007
Prevalent pfmdr1 n86y mutant Plasmodium falciparum in Madagascar despite absence of pfcrt mutant strains.
    The American journal of tropical medicine and hygiene, 2007, Volume: 76, Issue:6

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; DNA, Protozoan; Drug Resistance; Humans; Inhibitory Concentration 50; Madagascar; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Prevalence; Protozoan Proteins; Quinine; Rural Population

2007
Adaptation of a multi-drug resistant strain of Plasmodium falciparum from Peru to Aotus lemurinus griseimembra, A. nancymaae, and A. vociferans monkeys.
    The American journal of tropical medicine and hygiene, 2007, Volume: 77, Issue:2

    Topics: Animals; Antimalarials; Aotidae; Chloroquine; Cytochromes b; Dihydropteroate Synthase; Disease Models, Animal; DNA, Protozoan; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Mefloquine; Monkey Diseases; Parasitemia; Peru; Plasmodium falciparum; Sequence Analysis, DNA; Tetrahydrofolate Dehydrogenase

2007
[Polymorphisms of the pfmdr1 gene in field samples of Plasmodium falciparum and their association with therapeutic response to antimalarial drugs and severe malaria in Colombia].
    Biomedica : revista del Instituto Nacional de Salud, 2007, Volume: 27, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Colombia; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Mefloquine; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins

2007
Pharmacologic advances in the global control and treatment of malaria: combination therapy and resistance.
    Clinical pharmacology and therapeutics, 2007, Volume: 82, Issue:5

    Topics: Amodiaquine; Antimalarials; Artemether; Artemisinins; Artesunate; Chloroquine; Dapsone; Drug Design; Drug Resistance; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Global Health; Half-Life; Humans; Lumefantrine; Malaria; Mefloquine; Pregnancy; Pregnancy Complications, Infectious; Proguanil; Pyrimethamine; Quinine; Sesquiterpenes; Sulfadoxine

2007
Clinical inquiries. When should travelers begin malaria prophylaxis?
    The Journal of family practice, 2007, Volume: 56, Issue:11

    Topics: Antimalarials; Chloroquine; Contraindications; Doxycycline; Humans; Insect Repellents; Insecticides; Internet; Malaria; Mefloquine; Occlusive Dressings; Permethrin; Practice Guidelines as Topic; Primaquine; Time Factors; Travel

2007
Susceptibility to chloroquine, mefloquine and artemisinin of Plasmodium vivax in northwestern Thailand.
    Wiener klinische Wochenschrift, 2007, Volume: 119, Issue:19-20 Supp

    Topics: Antimalarials; Artemisinins; Chloroquine; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Humans; Lethal Dose 50; Malaria, Vivax; Mefloquine; Plasmodium vivax; Survival Rate; Thailand; Treatment Outcome

2007
Pharmacokinetic determinants of the window of selection for antimalarial drug resistance.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:5

    Topics: Algorithms; Amodiaquine; Animals; Antimalarials; Artemisinins; Chloroquine; Computer Simulation; Drug Resistance; Malaria; Mefloquine; Models, Theoretical; Pyrimethamine; Quinine

2008
Antimalarial drugs inhibit human 5-HT(3) and GABA(A) but not GABA(C) receptors.
    British journal of pharmacology, 2008, Volume: 153, Issue:8

    Topics: Animals; Antimalarials; Binding, Competitive; Cells, Cultured; Chloroquine; Electrophysiology; Female; GABA-A Receptor Antagonists; Humans; Inhibitory Concentration 50; Mefloquine; Oocytes; Quinine; Receptors, GABA; Serotonin 5-HT3 Receptor Antagonists; Xenopus laevis

2008
Differential effects of quinoline antimalarials on endocytosis in Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Blotting, Western; Chloroquine; Endocytosis; Erythrocytes; Hemoglobins; Humans; Mefloquine; Peroxidase; Phenanthrenes; Plasmodium falciparum; Protein Binding; Protozoan Proteins; Quinolines

2008
Malaria in Egypt, Saudi Arabia and Yemen: a clinical pilot study.
    Journal of the Egyptian Society of Parasitology, 2007, Volume: 37, Issue:3

    Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Chloroquine; Egypt; Female; Humans; Infant; Malaria; Male; Mefloquine; Middle Aged; Pilot Projects; Quinine; Saudi Arabia; Severity of Illness Index; Yemen

2007
Studies on antimalarial drug susceptibility in Colombia, in relation to Pfmdr1 and Pfcrt.
    Parasitology, 2008, Volume: 135, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Colombia; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Polymorphism, Single Nucleotide; Protozoan Proteins

2008
In vitro activity of ferroquine is independent of polymorphisms in transport protein genes implicated in quinoline resistance in Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:8

    Topics: Aminoquinolines; Amodiaquine; Animals; Chloroquine; Drug Resistance, Bacterial; Ferrous Compounds; Mefloquine; Membrane Transport Proteins; Metallocenes; Microsatellite Repeats; Molecular Structure; Plasmodium falciparum; Polymorphism, Genetic; Polymorphism, Single Nucleotide; Protozoan Proteins; Quinolines

2008
In vitro and in vivo properties of ellagic acid in malaria treatment.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:3

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Atovaquone; Chloroquine; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ellagic Acid; Erythrocytes; Female; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Mice; Mice, Inbred Strains; Molecular Structure; Molecular Weight; Parasitemia; Parasitic Sensitivity Tests; Plasmodium; Plasmodium falciparum; Schizonts; Trophozoites

2009
Failure of artesunate-mefloquine combination therapy for uncomplicated Plasmodium falciparum malaria in southern Cambodia.
    Malaria journal, 2009, Jan-12, Volume: 8

    Topics: Adult; Animals; Antimalarials; Artemisinins; Artesunate; Cambodia; Child; Chloroquine; Drug Therapy, Combination; Female; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Multidrug Resistance-Associated Proteins; Parasitemia; Plasmodium falciparum; Polymerase Chain Reaction; Survival Analysis; Treatment Failure

2009
Assessment of malaria in vitro drug combination screening and mixed-strain infections using the malaria Sybr green I-based fluorescence assay.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:6

    Topics: Animals; Antimalarials; Artemisinins; Benzothiazoles; Chloroquine; Diamines; Drug Combinations; Drug Evaluation, Preclinical; Drug Interactions; Fluorescent Dyes; Hypoxanthine; Mefloquine; Organic Chemicals; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2009
Drug resistance and in vitro susceptibility of Plasmodium falciparum in Thailand during 1988-2003.
    The Korean journal of parasitology, 2009, Volume: 47, Issue:2

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Thailand

2009
Monitoring of in vitro susceptibilities and molecular markers of resistance of Plasmodium falciparum isolates from Thai-Myanmar border to chloroquine, quinine, mefloquine and artesunate.
    Acta tropica, 2010, Volume: 113, Issue:2

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance; Gene Dosage; Genetic Markers; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Myanmar; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine; Thailand

2010
Decreased in vitro susceptibility of Plasmodium falciparum isolates to artesunate, mefloquine, chloroquine, and quinine in Cambodia from 2001 to 2007.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:5

    Topics: Antimalarials; Artemisinins; Artesunate; Cambodia; Chloroquine; Drug Resistance, Bacterial; Geographic Information Systems; In Vitro Techniques; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Oligonucleotide Array Sequence Analysis; Plasmodium falciparum; Point Mutation; Polymorphism, Single Nucleotide; Quinine

2010
Chloroquine-induced autophagic vacuole accumulation and cell death in glioma cells is p53 independent.
    Neuro-oncology, 2010, Volume: 12, Issue:5

    Topics: Antineoplastic Agents; Autophagy; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Chloroquine; Glioma; Humans; Immunohistochemistry; Mefloquine; Quinacrine; Tumor Suppressor Protein p53; Vacuoles

2010
Synergy of mefloquine activity with atorvastatin, but not chloroquine and monodesethylamodiaquine, and association with the pfmdr1 gene.
    The Journal of antimicrobial chemotherapy, 2010, Volume: 65, Issue:7

    Topics: Amodiaquine; Antimalarials; Atorvastatin; Chloroquine; DNA, Protozoan; Drug Synergism; Gene Dosage; Genotype; Heptanoic Acids; Humans; Inhibitory Concentration 50; Mefloquine; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrroles

2010
Purified Plasmodium falciparum multi-drug resistance protein (PfMDR 1) binds a high affinity chloroquine analogue.
    Molecular and biochemical parasitology, 2010, Volume: 173, Issue:2

    Topics: Antimalarials; Binding Sites; Chloroquine; Drug Resistance, Multiple; Mefloquine; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Protein Binding; Quinine

2010
Residual antimalarial concentrations before treatment in patients with malaria from Cambodia: indication of drug pressure.
    The Journal of infectious diseases, 2010, Oct-01, Volume: 202, Issue:7

    Topics: Adolescent; Adult; Antimalarials; Cambodia; Child; Child, Preschool; Chloroquine; Chromatography, Liquid; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Quinine; Quinolines; Selection, Genetic; Serum; Tandem Mass Spectrometry; Young Adult

2010
In-vitro culture of Plasmodium falciparum: utility of modified (RPNI) medium for drug-sensitivity studies using SYBR Green I assay.
    Experimental parasitology, 2011, Volume: 127, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Benzothiazoles; Chloroquine; Culture Media; Diamines; Fluorescent Dyes; Mefloquine; Organic Chemicals; Plasmodium falciparum; Quinine; Quinolines

2011
Potentiation of the mutagenicity and recombinagenicity of bleomycin in yeast by unconventional intercalating agents.
    Environmental and molecular mutagenesis, 2011, Volume: 52, Issue:2

    Topics: Amines; Animals; Benzophenones; Bleomycin; Cell Line; Chloroquine; Chlorpromazine; Cricetinae; DNA Damage; Drug Synergism; Gene Conversion; Intercalating Agents; Mefloquine; Mutagenicity Tests; Mutagens; Recombination, Genetic; Saccharomyces cerevisiae; Tamoxifen

2011
Enantiomeric separation of antimalarial drugs by capillary electrophoresis using neutral and negatively charged cyclodextrins.
    Journal of pharmaceutical and biomedical analysis, 2011, Feb-20, Volume: 54, Issue:3

    Topics: Aminoquinolines; Anions; Antimalarials; beta-Cyclodextrins; Chloroquine; Cyclodextrins; Electrophoresis, Capillary; Humans; Magnetic Resonance Spectroscopy; Mass Spectrometry; Mefloquine; Primaquine; Stereoisomerism

2011
Suicide by skull stab wounds: a case of drug-induced psychosis.
    The American journal of forensic medicine and pathology, 2010, Volume: 31, Issue:4

    Topics: Adult; Antimalarials; Arm Injuries; Chloroquine; Forensic Toxicology; Gastrointestinal Contents; Head Injuries, Penetrating; Humans; Male; Mefloquine; Psychoses, Substance-Induced; Shoulder; Shoulder Injuries; Suicide; Temporal Lobe; Wounds, Stab

2010
Incorporation of basic side chains into cryptolepine scaffold: structure-antimalarial activity relationships and mechanistic studies.
    Journal of medicinal chemistry, 2011, Feb-10, Volume: 54, Issue:3

    Topics: Animals; Antimalarials; Cell Line, Tumor; Chlorocebus aethiops; Chloroquine; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; DNA; Drug Resistance; Erythrocytes; Hemin; Humans; Indole Alkaloids; Mefloquine; Oligonucleotides; Plasmodium falciparum; Pyrimethamine; Quinolines; Structure-Activity Relationship; Vero Cells

2011
Increased prevalence of the Plasmodium falciparum Pfmdr1 86N genotype among field isolates from Franceville, Gabon after replacement of chloroquine by artemether-lumefantrine and artesunate-mefloquine.
    Infection, genetics and evolution : journal of molecular epidemiology and evolutionary genetics in infectious diseases, 2011, Volume: 11, Issue:2

    Topics: Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Gabon; Genotype; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Parasitemia; Plasmodium falciparum; Polymorphism, Genetic; Prevalence; Protozoan Proteins

2011
Human p38 mitogen-activated protein kinase inhibitor drugs inhibit Plasmodium falciparum replication.
    Experimental parasitology, 2011, Volume: 128, Issue:2

    Topics: Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Erythrocytes; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Mefloquine; p38 Mitogen-Activated Protein Kinases; Plasmodium falciparum; Protein Kinase Inhibitors; Pyridines

2011
In vitro activity of Proveblue (methylene blue) on Plasmodium falciparum strains resistant to standard antimalarial drugs.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; Ethanolamines; Fluorenes; Inhibitory Concentration 50; Lumefantrine; Mefloquine; Methylene Blue; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine

2011
2,4-diarylthiazole antiprion compounds as a novel structural class of antimalarial leads.
    Bioorganic & medicinal chemistry letters, 2011, Jun-15, Volume: 21, Issue:12

    Topics: Antimalarials; Chloroquine; Mefloquine; Molecular Structure; Plasmodium falciparum; Prions; Quinacrine; Structure-Activity Relationship; Thiazoles

2011
Radical curative efficacy of tafenoquine combination regimens in Plasmodium cynomolgi-infected Rhesus monkeys (Macaca mulatta).
    Malaria journal, 2011, Jul-29, Volume: 10

    Topics: Aminoquinolines; Animals; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Chloroquine; Chromatography, Liquid; Disease Models, Animal; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Macaca mulatta; Malaria; Male; Mass Spectrometry; Mefloquine; Plasma; Plasmodium cynomolgi; Primate Diseases; Quinine; Treatment Outcome

2011
Sensitivity of Plasmodium vivax to chloroquine, mefloquine, artemisinin and atovaquone in north-western Thailand.
    Wiener klinische Wochenschrift, 2011, Volume: 123 Suppl 1

    Topics: Animals; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Dose-Response Relationship, Drug; Lethal Dose 50; Mefloquine; Plasmodium vivax; Thailand

2011
Quality of essential drugs in tropical countries: evaluation of antimalarial drugs in the Brazilian Health System.
    Revista da Sociedade Brasileira de Medicina Tropical, 2011, Volume: 44, Issue:5

    Topics: Antimalarials; Brazil; Chloroquine; Chromatography, High Pressure Liquid; Drug Storage; Drugs, Essential; Humans; Mefloquine; Primaquine; Quality Control; Quinine

2011
Eritrean and Sudanese migrants presenting with malaria in Israel.
    Travel medicine and infectious disease, 2011, Volume: 9, Issue:6

    Topics: Adult; Antigens, Protozoan; Antimalarials; Chloroquine; Eritrea; Female; Hospitalization; Humans; Israel; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Plasmodium falciparum; Plasmodium vivax; Population Surveillance; Retrospective Studies; Sudan; Transients and Migrants; Treatment Outcome; Young Adult

2011
Prophylactic use of antimalarials during pregnancy.
    Canadian family physician Medecin de famille canadien, 2011, Volume: 57, Issue:11

    Topics: Antimalarials; Atovaquone; Chemoprevention; Chloroquine; Doxycycline; Drug Combinations; Female; Humans; Hydroxychloroquine; Malaria; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Primaquine; Proguanil; Travel

2011
Extracellular heme enhances the antimalarial activity of artemisinin.
    Biological & pharmaceutical bulletin, 2012, Volume: 35, Issue:1

    Topics: Antimalarials; Antioxidants; Artemisia; Artemisinins; Chloroquine; Cholesterol, LDL; Fluorescence; Heme; Hemin; Humans; Lipid Peroxidation; Mefloquine; Oxidants; Oxidation-Reduction; Plasmodium falciparum; Quinine; Tryptophan; Vitamin E

2012
Discordant temporal evolution of Pfcrt and Pfmdr1 genotypes and Plasmodium falciparum in vitro drug susceptibility to 4-aminoquinolines after drug policy change in French Guiana.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:3

    Topics: Aminoquinolines; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance; Ethanolamines; Evolution, Molecular; Fluorenes; French Guiana; Gene Dosage; Haplotypes; Humans; Inhibitory Concentration 50; Longitudinal Studies; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Practice Guidelines as Topic; Protozoan Proteins; Quinine

2012
Anti-malarial chemoprophylaxis following evacuation from Afghanistan.
    Journal of the Royal Army Medical Corps, 2012, Volume: 158, Issue:1

    Topics: Afghan Campaign 2001-; Antimalarials; Atovaquone; Chemoprevention; Chloroquine; Clinical Audit; Doxycycline; Drug Combinations; Drug Prescriptions; Humans; Malaria; Mefloquine; Military Personnel; Proguanil

2012
Distribution of drug resistance genotypes in Plasmodium falciparum in an area of limited parasite diversity in Saudi Arabia.
    The American journal of tropical medicine and hygiene, 2012, Volume: 86, Issue:5

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Genotype; Humans; Infant; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Multidrug Resistance-Associated Proteins; Mutation; Phenanthrenes; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Pyrimethamine; Saudi Arabia; Sulfadoxine; Tetrahydrofolate Dehydrogenase; Young Adult

2012
In vitro assessment of drug resistance in Plasmodium falciparum in five States of India.
    The Indian journal of medical research, 2012, Volume: 135, Issue:4

    Topics: Amodiaquine; Artemisinins; Artesunate; Biomarkers, Pharmacological; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; India; Mefloquine; Membrane Transport Proteins; Mutation; Plasmodium falciparum; Protozoan Proteins

2012
Efficacy of dihydroartemisinin-piperaquine for treatment of uncomplicated Plasmodium falciparum and Plasmodium vivax in Cambodia, 2008 to 2010.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:2

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Cambodia; Child; Chloroquine; Drug Resistance; Drug Therapy, Combination; Female; Genotype; Humans; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Parasitic Sensitivity Tests; Plasmodium falciparum; Plasmodium vivax; Protozoan Proteins; Quinolines; Treatment Outcome; Young Adult

2013
Defining the timing of action of antimalarial drugs against Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:3

    Topics: Amodiaquine; Antimalarials; Artemisinins; Artesunate; Chloroquine; Erythrocytes; Flow Cytometry; High-Throughput Screening Assays; Hydroxamic Acids; Inhibitory Concentration 50; Mefloquine; Merozoites; Plasmodium falciparum; Quinine; Quinolines; Schizonts; Time Factors

2013
Ketoconazole, a cytochrome P(450) inhibitor can potentiate the antimalarial action of α/β arteether against MDR Plasmodium yoelii nigeriensis.
    Acta tropica, 2013, Volume: 126, Issue:2

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance, Multiple; Drug Synergism; Drug Therapy, Combination; Female; Humans; Ketoconazole; Liver; Malaria; Male; Mefloquine; Mice; Plasmodium falciparum; Plasmodium yoelii; Quinine

2013
An in vivo drug screening model using glucose-6-phosphate dehydrogenase deficient mice to predict the hemolytic toxicity of 8-aminoquinolines.
    The American journal of tropical medicine and hygiene, 2013, Volume: 88, Issue:6

    Topics: Acute Disease; Aminoquinolines; Anemia, Hemolytic; Animals; Antimalarials; Chloroquine; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Genotype; Glucosephosphate Dehydrogenase Deficiency; Glutathione; Haptoglobins; Hemolytic Agents; Male; Mefloquine; Mice; Phenotype; Primaquine; Reticulocyte Count

2013
Chemosensitization potential of P-glycoprotein inhibitors in malaria parasites.
    Experimental parasitology, 2013, Volume: 134, Issue:2

    Topics: Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Boron Compounds; Chloroquine; Chlorpheniramine; Dibenzocycloheptenes; Drug Interactions; Drug Resistance, Multiple; Erythrocytes; Fluorescent Dyes; Gefitinib; Humans; Imatinib Mesylate; Mefloquine; Piperazines; Plasmodium falciparum; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Quinolines

2013
High-throughput analysis of antimalarial susceptibility data by the WorldWide Antimalarial Resistance Network (WWARN) in vitro analysis and reporting tool.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:7

    Topics: Amodiaquine; Antimalarials; Artemisinins; Automation, Laboratory; Chloroquine; Drug Resistance; Drug Therapy, Combination; High-Throughput Screening Assays; Internet; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine

2013
The role of Pfmdr1 and Pfcrt in changing chloroquine, amodiaquine, mefloquine and lumefantrine susceptibility in western-Kenya P. falciparum samples during 2008-2011.
    PloS one, 2013, Volume: 8, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; DNA, Protozoan; Drug Resistance; Ethanolamines; Fluorenes; Haplotypes; Humans; Inhibitory Concentration 50; Kenya; Lumefantrine; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Retrospective Studies

2013
In vitro chloroquine resistance for Plasmodium vivax isolates from the Western Brazilian Amazon.
    Malaria journal, 2013, Jul-03, Volume: 12

    Topics: Adolescent; Adult; Antimalarials; Brazil; Cell Survival; Child; Chloroquine; Female; Humans; Inhibitory Concentration 50; L-Lactate Dehydrogenase; Malaria, Vivax; Male; Mefloquine; Middle Aged; Mutation, Missense; Parasitic Sensitivity Tests; Plasmodium vivax; Protozoan Proteins; Young Adult

2013
Nonlinear mixed-effects modelling of in vitro drug susceptibility and molecular correlates of multidrug resistant Plasmodium falciparum.
    PloS one, 2013, Volume: 8, Issue:7

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Ethanolamines; Fluorenes; Lumefantrine; Mefloquine; Models, Statistical; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Genetic; Polymorphism, Single Nucleotide; Protozoan Proteins

2013
Repeat polymorphisms in the low-complexity regions of Plasmodium falciparum ABC transporters and associations with in vitro antimalarial responses.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:12

    Topics: Amino Acid Motifs; Antimalarials; Artemisinins; Asparagine; Aspartic Acid; Chloroquine; Drug Resistance; Ethanolamines; Fluorenes; Gene Expression; Genome, Protozoan; Lumefantrine; Mefloquine; Molecular Sequence Data; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine

2013
Humanized mouse model of glucose 6-phosphate dehydrogenase deficiency for in vivo assessment of hemolytic toxicity.
    Proceedings of the National Academy of Sciences of the United States of America, 2013, Oct-22, Volume: 110, Issue:43

    Topics: Aminoquinolines; Anemia, Hemolytic; Animals; Antimalarials; Chloroquine; Combined Modality Therapy; Dapsone; Dose-Response Relationship, Drug; Doxycycline; Drug Evaluation, Preclinical; Erythrocyte Count; Erythrocyte Transfusion; Female; Glucosephosphate Dehydrogenase Deficiency; Humans; Mefloquine; Mice; Mice, Inbred NOD; Mice, SCID; Primaquine; Pyrimethamine; Reproducibility of Results; Sensitivity and Specificity; Transplantation, Heterologous

2013
Formulation and evaluation of Pheroid vesicles containing mefloquine for the treatment of malaria.
    The Journal of pharmacy and pharmacology, 2014, Volume: 66, Issue:1

    Topics: Animals; Biological Availability; Cell Line, Tumor; Chemistry, Pharmaceutical; Chloroquine; Coated Vesicles; Drug Delivery Systems; Half-Life; Humans; Malaria; Male; Mefloquine; Mice; Mice, Inbred C57BL; Neuroblastoma; Particle Size; Solubility

2014
Susceptibility of human Plasmodium knowlesi infections to anti-malarials.
    Malaria journal, 2013, Nov-19, Volume: 12

    Topics: Animals; Antimalarials; Artemisinins; Borneo; Chloroquine; Humans; Malaria; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Plasmodium knowlesi; Plasmodium vivax; Zoonoses

2013
Co-treatment with the anti-malarial drugs mefloquine and primaquine highly sensitizes drug-resistant cancer cells by increasing P-gp inhibition.
    Biochemical and biophysical research communications, 2013, Nov-22, Volume: 441, Issue:3

    Topics: Antimalarials; Antineoplastic Agents; Apoptosis; Artemisinins; Artesunate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Chloroquine; Doxycycline; Drug Resistance, Neoplasm; Humans; Mefloquine; Primaquine; Verapamil; Vinblastine

2013
Four years' monitoring of in vitro sensitivity and candidate molecular markers of resistance of Plasmodium falciparum to artesunate-mefloquine combination in the Thai-Myanmar border.
    Malaria journal, 2014, Jan-15, Volume: 13

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Drug Resistance; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinine; Seasons; Thailand; Time Factors

2014
Mefloquine and psychotomimetics share neurotransmitter receptor and transporter interactions in vitro.
    Psychopharmacology, 2014, Volume: 231, Issue:14

    Topics: Animals; Antimalarials; Central Nervous System Stimulants; Chloroquine; CHO Cells; Cricetinae; Cricetulus; Hallucinogens; HEK293 Cells; Humans; Mefloquine; Mice; Receptors, Dopamine; Receptors, Serotonin; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism

2014
Plasmodium vivax and Plasmodium falciparum ex vivo susceptibility to anti-malarials and gene characterization in Rondônia, West Amazon, Brazil.
    Malaria journal, 2014, Feb-28, Volume: 13

    Topics: Adult; Antimalarials; Artemisinins; Artesunate; Brazil; Chloroquine; DNA, Protozoan; Drug Resistance; Female; Genotype; Humans; Inhibitory Concentration 50; Malaria; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Multidrug Resistance-Associated Proteins; Mutation, Missense; Parasitic Sensitivity Tests; Plasmodium falciparum; Plasmodium vivax; Protozoan Proteins

2014
Imported malaria is stable from Africa but declining from Asia.
    Danish medical journal, 2014, Volume: 61, Issue:5

    Topics: Adolescent; Adult; Africa; Aged; Antimalarials; Asia; Atovaquone; Chemoprevention; Child; Child, Preschool; Chloroquine; Delayed Diagnosis; Denmark; Drug Combinations; Female; Humans; Incidence; Infant; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Middle Aged; Primaquine; Proguanil; Recurrence; Risk Factors; Severity of Illness Index; Travel; Young Adult

2014
Plasmodium falciparum multidrug resistance protein 1 (pfmrp1) gene and its association with in vitro drug susceptibility of parasite isolates from north-east Myanmar.
    The Journal of antimicrobial chemotherapy, 2014, Volume: 69, Issue:8

    Topics: Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Sequence; Chloroquine; Drug Resistance; Ethanolamines; Fluorenes; Geography; Humans; Lumefantrine; Malaria, Falciparum; Mefloquine; Multidrug Resistance-Associated Proteins; Mutation; Myanmar; Naphthyridines; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Single Nucleotide; Selection, Genetic; Sequence Analysis, DNA

2014
Treatment of murine cerebral malaria by artemisone in combination with conventional antimalarial drugs: antiplasmodial effects and immune responses.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:8

    Topics: Animals; Antimalarials; Artemisinins; Cell Line; Cell Survival; Cells, Cultured; Chloroquine; Doxycycline; Drug Synergism; Drug Therapy, Combination; Erythrocytes; Humans; Interleukin-10; Interleukin-4; Malaria, Cerebral; Mefloquine; Mice; Mice, Inbred C57BL; Monocytes; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium berghei; Plasmodium falciparum

2014
Imported malaria in a non-endemic area: the experience of the university of Campinas hospital in the Brazilian Southeast.
    Malaria journal, 2014, Jul-22, Volume: 13

    Topics: Acquired Immunodeficiency Syndrome; Adolescent; Adult; Anemia; Antimalarials; Artemether; Artemisinins; Brazil; Chloroquine; Comorbidity; Female; Follow-Up Studies; Humans; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Middle Aged; Parasitemia; Primaquine; Recurrence; Retrospective Studies; Tertiary Care Centers; Thrombocytopenia; Travel; Young Adult

2014
In vitro susceptibility of Plasmodium vivax to antimalarials in Colombia.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:11

    Topics: Amodiaquine; Antimalarials; Artemisinins; Artesunate; Chloroquine; Colombia; Drug Resistance; Malaria, Vivax; Mefloquine; Parasitic Sensitivity Tests; Plasmodium vivax; Quinine

2014
Role of Pfmdr1 in in vitro Plasmodium falciparum susceptibility to chloroquine, quinine, monodesethylamodiaquine, mefloquine, lumefantrine, and dihydroartemisinin.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:12

    Topics: Adult; Amodiaquine; Antimalarials; Artemisinins; Biological Transport; Child; Chloroquine; Drug Resistance; Erythrocytes; Ethanolamines; Female; Fluorenes; Gene Expression; Haplotypes; Humans; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Single Nucleotide; Quinine; Senegal

2014
Complex polymorphisms in the Plasmodium falciparum multidrug resistance protein 2 gene and its contribution to antimalarial response.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:12

    Topics: Amino Acid Sequence; Antimalarials; Artemisinins; Biological Transport; Chloroquine; Chromosomes; Drug Resistance, Multiple; Erythrocytes; Humans; INDEL Mutation; Malaria, Falciparum; Mefloquine; Molecular Sequence Data; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Single Nucleotide; Quinolines; Thailand

2014
Studying the effect of chloroquine on sporozoite-induced protection and immune responses in Plasmodium berghei malaria.
    Malaria journal, 2015, Mar-26, Volume: 14

    Topics: Animals; Antimalarials; CD8-Positive T-Lymphocytes; Chloroquine; Immunity, Cellular; Immunologic Memory; Interferon-gamma; Malaria; Mefloquine; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Plasmodium berghei; Sporozoites

2015
Ex Vivo Drug Susceptibility Testing and Molecular Profiling of Clinical Plasmodium falciparum Isolates from Cambodia from 2008 to 2013 Suggest Emerging Piperaquine Resistance.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:8

    Topics: Adolescent; Adult; Aged; Antimalarials; Artemisinins; Cambodia; Chloroquine; Drug Resistance; Female; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Young Adult

2015
In Vitro and Molecular Surveillance for Antimalarial Drug Resistance in Plasmodium falciparum Parasites in Western Kenya Reveals Sustained Artemisinin Sensitivity and Increased Chloroquine Sensitivity.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:12

    Topics: Alleles; Amodiaquine; Animals; Antimalarials; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Resistance; Epidemiological Monitoring; Ethanolamines; Fluorenes; Gene Dosage; Gene Expression; Genotype; Humans; Kenya; Lumefantrine; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins

2015
In Vitro Activities of Primaquine-Schizonticide Combinations on Asexual Blood Stages and Gametocytes of Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:12

    Topics: Antimalarials; Benzothiazoles; Chloroquine; Diamines; Drug Combinations; Drug Interactions; Erythrocytes; Ethanolamines; Flow Cytometry; Fluorenes; Humans; Lumefantrine; Mefloquine; Organic Chemicals; Parasitic Sensitivity Tests; Plasmodium falciparum; Primaquine; Quinolines; Sporozoites; Trophozoites

2015
Expression of Plasmodium vivax crt-o Is Related to Parasite Stage but Not Ex Vivo Chloroquine Susceptibility.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:1

    Topics: Amodiaquine; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance, Multiple; Erythrocytes; Fructose-Bisphosphate Aldolase; Gene Expression Regulation; Humans; Inhibitory Concentration 50; Life Cycle Stages; Malaria, Vivax; Mefloquine; Membrane Transport Proteins; Plasmodium vivax; Protozoan Proteins; Quinolines; Transcription, Genetic; Tubulin

2016
Characterizing Types of Human Mobility to Inform Differential and Targeted Malaria Elimination Strategies in Northeast Cambodia.
    Scientific reports, 2015, Nov-23, Volume: 5

    Topics: Animals; Anopheles; Antimalarials; Artemisinins; Artesunate; Cambodia; Chloroquine; Disease Eradication; Health Surveys; Humans; Insect Vectors; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Plasmodium falciparum; Plasmodium vivax; Transients and Migrants

2015
Artemisinin-based combination therapy for knowlesi malaria.
    The Lancet. Infectious diseases, 2016, Volume: 16, Issue:2

    Topics: Antimalarials; Artemisinins; Chloroquine; Female; Humans; Malaria; Male; Mefloquine; Plasmodium knowlesi

2016
An improved SYBR Green-1-based fluorescence method for the routine monitoring of Plasmodium falciparum resistance to anti-malarial drugs.
    Malaria journal, 2015, Dec-01, Volume: 14

    Topics: Antimalarials; Artemisinins; Artesunate; Benzothiazoles; Child; Child, Preschool; Chloroquine; Diamines; Drug Resistance; Fluorometry; Humans; Inhibitory Concentration 50; Mefloquine; Organic Chemicals; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Staining and Labeling

2015
Assessment of the Worldwide Antimalarial Resistance Network Standardized Procedure for In Vitro Malaria Drug Sensitivity Testing Using SYBR Green Assay for Field Samples with Various Initial Parasitemia Levels.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:4

    Topics: Antimalarials; Artemisinins; Atovaquone; Benzothiazoles; Biological Assay; Chloroquine; Diamines; DNA, Protozoan; Drug Resistance; Erythrocytes; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Organic Chemicals; Parasitemia; Plasmodium falciparum; Public Health Surveillance; Quinolines; Reproducibility of Results; Sensitivity and Specificity

2016
Repetitive live sporozoites inoculation under arteether chemoprophylaxis confers protection against subsequent sporozoite challenge in rodent malaria model.
    Acta tropica, 2016, Volume: 158

    Topics: Animals; Antimalarials; Artemisinins; Chemoprevention; Chloroquine; Female; Immunization; Malaria; Mefloquine; Mice; Parasite Load; Plasmodium yoelii; Primaquine; Sporozoites; Vaccination

2016
Effect of mild medical hypothermia on in vitro growth of Plasmodium falciparum and the activity of anti-malarial drugs.
    Malaria journal, 2016, Mar-15, Volume: 15

    Topics: Antimalarials; Artemisinins; Chloroquine; Cold Temperature; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum

2016
Absence of Association between Polymorphisms in the RING E3 Ubiquitin Protein Ligase Gene and Ex Vivo Susceptibility to Conventional Antimalarial Drugs in Plasmodium falciparum Isolates from Dakar, Senegal.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:8

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Doxycycline; Ethanolamines; Fluorenes; Lumefantrine; Mefloquine; Naphthyridines; Plasmodium falciparum; Polymorphism, Genetic; Quinine; Quinolines; Senegal; Ubiquitin-Protein Ligases

2016
Highly active ozonides selected against drug resistant malaria.
    Memorias do Instituto Oswaldo Cruz, 2016, Jun-07, Volume: 0

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Disease Models, Animal; Female; Humans; Malaria, Falciparum; Mefloquine; Mice; Parasitemia; Plasmodium falciparum

2016
In vitro sensitivity of antimalarial drugs and correlation with clinico-parasitological response following treatment with a 3-day artesunate-mefloquine combination in patients with falciparum malaria along the Thai-Myanmar border.
    Acta tropica, 2017, Volume: 166

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Myanmar; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Thailand; Young Adult

2017
Association between Polymorphisms in the Pf
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:3

    Topics: Amodiaquine; Antimalarials; Artemisinins; Artesunate; Asparagine; ATP-Binding Cassette Transporters; Chloroquine; Doxycycline; Drug Resistance; Ethanolamines; Fluorenes; Gene Expression; Humans; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mefloquine; Naphthyridines; Plasmodium falciparum; Polymorphism, Genetic; Protein Isoforms; Protozoan Proteins; Quinine; Quinolines; Repetitive Sequences, Amino Acid; Senegal

2017
Antibody Responses to
    The American journal of tropical medicine and hygiene, 2017, Volume: 96, Issue:5

    Topics: Adaptive Immunity; Antibodies, Protozoan; Antimalarials; Artemisinins; Artesunate; Chloroquine; Cohort Studies; Disease Resistance; Disease Susceptibility; Female; Humans; Immunoglobulin G; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Merozoite Surface Protein 1; Parasitemia; Parturition; Plasmodium falciparum; Plasmodium vivax; Pregnancy; Proportional Hazards Models; Risk; Time Factors

2017
Synthesis and Antimalarial Activity of New Enantiopure Aminoalcoholpyrrolo[ 1,2-a]quinoxalines.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2018, Volume: 14, Issue:3

    Topics: Amino Alcohols; Animals; Antimalarials; Cell Line, Tumor; Chloroquine; CHO Cells; Cricetulus; Humans; Mefloquine; Plasmodium falciparum; Pyrroles; Quinoxalines; Stereoisomerism

2018
In vitro anti-malarial interaction and gametocytocidal activity of cryptolepine.
    Malaria journal, 2017, 12-28, Volume: 16, Issue:1

    Topics: Alkaloids; Antimalarials; Chloroquine; Ethanolamines; Fluorenes; Gametogenesis; Ghana; Humans; Indole Alkaloids; Life Cycle Stages; Lumefantrine; Malaria; Malaria, Falciparum; Mefloquine; Plant Extracts; Plasmodium falciparum; Quinolines

2017
Heterologous Expression of a Novel Drug Transporter from the Malaria Parasite Alters Resistance to Quinoline Antimalarials.
    Scientific reports, 2018, 02-06, Volume: 8, Issue:1

    Topics: Amino Acid Transport Systems; Amodiaquine; Animals; Antimalarials; Biological Transport; Chloroquine; Conserved Sequence; Drug Resistance; Gene Expression; Humans; Mefloquine; Mutation; Plasmodium chabaudi; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Quinine; Recombinant Proteins; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Transgenes

2018
Prediction Model for Antimalarial Activities of Hemozoin Inhibitors by Using Physicochemical Properties.
    Antimicrobial agents and chemotherapy, 2018, Volume: 62, Issue:5

    Topics: Animals; Antimalarials; Bayes Theorem; Chloroquine; Hemeproteins; Humans; Malaria; Mefloquine; Plasmodium falciparum

2018
    The Indian journal of medical research, 2017, Volume: 146, Issue:5

    Topics: Anti-Bacterial Agents; Antimalarials; Artemether; Artemisinins; Atovaquone; Azithromycin; Chloroquine; Doxycycline; Ethanolamines; Fluorenes; Humans; India; Lumefantrine; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

2017
A survey on outcomes of accidental atovaquone-proguanil exposure in pregnancy.
    Malaria journal, 2018, May-15, Volume: 17, Issue:1

    Topics: Abnormalities, Drug-Induced; Abortion, Spontaneous; Adult; Antimalarials; Atovaquone; Chemoprevention; Chloroquine; Drug Combinations; Female; Humans; Live Birth; Mefloquine; Middle Aged; Pregnancy; Pregnancy Outcome; Premature Birth; Proguanil; Stillbirth; United States; Young Adult

2018
Nanomolar binding affinity of quinine-based antimalarial compounds by the cocaine-binding aptamer.
    Bioorganic & medicinal chemistry, 2018, 11-01, Volume: 26, Issue:20

    Topics: Amodiaquine; Antimalarials; Aptamers, Nucleotide; Binding Sites; Chloroquine; Cocaine; Ligands; Mefloquine; Primaquine; Quinine; Thermodynamics

2018
Application of the automated haematology analyzer XN-30 for discovery and development of anti-malarial drugs.
    Malaria journal, 2019, Jan-14, Volume: 18, Issue:1

    Topics: Antimalarials; Atovaquone; Automation, Laboratory; Chloroquine; Drug Discovery; Hematology; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Schizonts; Trophozoites

2019
Chloroquine and mefloquine resistance profiles are not related to the circumsporozoite protein (CSP) VK210 subtypes in field isolates of Plasmodium vivax from Manaus, Brazilian Amazon.
    Memorias do Instituto Oswaldo Cruz, 2019, Volume: 114

    Topics: Antimalarials; Chloroquine; Genotype; Humans; Malaria, Vivax; Mefloquine; Parasitic Sensitivity Tests; Plasmodium vivax; Polymerase Chain Reaction; Protozoan Proteins

2019
Deployment and Travel Medicine Knowledge, Attitudes, Practices, and Outcomes Study (KAPOS): Malaria Chemoprophylaxis Prescription Patterns in the Military Health System.
    The American journal of tropical medicine and hygiene, 2020, Volume: 103, Issue:1

    Topics: Adolescent; Adult; Aged; Antimalarials; Atovaquone; Chemoprevention; Chloroquine; Doxycycline; Drug Combinations; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Military Medicine; Military Personnel; Practice Patterns, Physicians'; Primaquine; Proguanil; United States; Young Adult

2020
Malaria in the pregnant traveler.
    Journal of travel medicine, 2020, Jul-14, Volume: 27, Issue:4

    Topics: Antimalarials; Chemoprevention; Chloroquine; Drug Resistance; Female; Humans; Malaria; Mefloquine; Pregnancy; Proguanil; Travel

2020
Ex-vivo Sensitivity of Plasmodium falciparum to Common Anti-malarial Drugs: The Case of Kéniéroba, a Malaria Endemic Village in Mali.
    Drugs in R&D, 2020, Volume: 20, Issue:3

    Topics: Adolescent; Amodiaquine; Antimalarials; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Resistance; Endemic Diseases; Humans; Infant; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mali; Mefloquine; Plasmodium falciparum; Quinine; Quinolines

2020
Genetic analysis of the orthologous crt and mdr1 genes in Plasmodium malariae from Thailand and Myanmar.
    Malaria journal, 2020, Aug-31, Volume: 19, Issue:1

    Topics: Chloroquine; Drug Resistance; Insecticides; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Myanmar; Plasmodium malariae; Polymorphism, Genetic; Protozoan Proteins; Thailand

2020
Comparison of chloroquine-like molecules for lysosomal inhibition and measurement of autophagic flux in the brain.
    Biochemical and biophysical research communications, 2021, 01-01, Volume: 534

    Topics: Animals; Autophagy; Brain; Chloroquine; Drug Evaluation, Preclinical; Female; HeLa Cells; Humans; Lysosomes; Macrolides; Male; Mefloquine; Mice, Inbred C57BL; Mice, Transgenic; Microtubule-Associated Proteins; Promazine; Quinacrine; Trifluoperazine

2021
Ex vivo susceptibility of Plasmodium falciparum to antimalarial drugs in Northern Uganda.
    Parasitology international, 2021, Volume: 81

    Topics: Amodiaquine; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Lumefantrine; Mefloquine; Plasmodium falciparum; Quinine; Uganda

2021
Cryptic Plasmodium inui and Plasmodium fieldi Infections Among Symptomatic Malaria Patients in Thailand.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2022, 09-14, Volume: 75, Issue:5

    Topics: Animals; Artemisinins; Chloroquine; Electron Transport Complex IV; Humans; Macaca; Malaria; Mefloquine; Phylogeny; Plasmodium; Plasmodium knowlesi; Retrospective Studies; Thailand

2022
Unlike Chloroquine, Mefloquine Inhibits SARS-CoV-2 Infection in Physiologically Relevant Cells.
    Viruses, 2022, 02-11, Volume: 14, Issue:2

    Topics: Adenosine Monophosphate; Alanine; Alveolar Epithelial Cells; Antiviral Agents; Cell Line; Chloroquine; COVID-19 Drug Treatment; Drug Repositioning; Humans; Mefloquine; SARS-CoV-2; Serine Endopeptidases; Virus Internalization

2022
Mechanistic basis for multidrug resistance and collateral drug sensitivity conferred to the malaria parasite by polymorphisms in PfMDR1 and PfCRT.
    PLoS biology, 2022, Volume: 20, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Lumefantrine; Malaria, Falciparum; Mefloquine; Multidrug Resistance-Associated Proteins; Parasites; Plasmodium falciparum; Protein Isoforms; Protozoan Proteins

2022
Opioidergic and nitrergic systems mediate the anticonvulsant effect of mefloquine and chloroquine on seizures induced by pentylenetetrazol and maximal electroshock in mice.
    Acta neurobiologiae experimentalis, 2022, Volume: 82, Issue:2

    Topics: Animals; Anticonvulsants; Chloroquine; Disease Models, Animal; Electroshock; Mefloquine; Mice; Naltrexone; Nitrites; Pentylenetetrazole; Seizures

2022
Genome-wide functional screening of drug-resistance genes in Plasmodium falciparum.
    Nature communications, 2022, 10-18, Volume: 13, Issue:1

    Topics: Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Protozoan Proteins

2022
Integrative Genetic Manipulation of Plasmodium cynomolgi Reveals Multidrug Resistance-1 Y976F Associated With Increased In Vitro Susceptibility to Mefloquine.
    The Journal of infectious diseases, 2023, 05-12, Volume: 227, Issue:10

    Topics: Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Mefloquine; Plasmodium cynomolgi; Plasmodium falciparum; Plasmodium vivax

2023