chloroquine and harmine

chloroquine has been researched along with harmine in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (28.57)29.6817
2010's2 (28.57)24.3611
2020's3 (42.86)2.80

Authors

AuthorsStudies
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Datti, A; Liang, M; Pillai, DR; Shahinas, D1
Fontinha, D; Held, J; Perković, I; Pessanha de Carvalho, L; Prudêncio, M; Raić-Malić, S; Rajić, Z; Tandarić, T; Vianello, R; Zorc, B1
Fontinha, D; Held, J; Marinović, M; Perković, I; Pessanha de Carvalho, L; Poje, G; Prudêncio, M; Rajić, Z; Tandarić, T; Vianello, R1
Held, J; Moita, D; Perković, I; Pessanha de Carvalho, L; Poje, G; Prudêncio, M; Rajić, Z; Tandarić, T; Vianello, R1
Azas, N; Delmas, F; Di, GC; Gasquet, M; Laget, M; Laurencin, N; Timon-David, P1
Benedict, C; Crandall, I; Macmullin, G; Pillai, DR; Shahinas, D1

Other Studies

7 other study(ies) available for chloroquine and harmine

ArticleYear
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
A repurposing strategy identifies novel synergistic inhibitors of Plasmodium falciparum heat shock protein 90.
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Adenosine Triphosphate; Antimalarials; Binding Sites; Binding, Competitive; Drug Evaluation, Preclinical; Drug Synergism; HSP90 Heat-Shock Proteins; Humans; Parasitic Sensitivity Tests; Plasmodium falciparum; Small Molecule Libraries; Substrate Specificity

2010
Harmicines - harmine and cinnamic acid hybrids as novel antiplasmodial hits.
    European journal of medicinal chemistry, 2020, Feb-01, Volume: 187

    Topics: Antimalarials; Cinnamates; Dose-Response Relationship, Drug; Harmine; Indole Alkaloids; Molecular Dynamics Simulation; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2020
Further investigation of harmicines as novel antiplasmodial agents: Synthesis, structure-activity relationship and insight into the mechanism of action.
    European journal of medicinal chemistry, 2021, Nov-15, Volume: 224

    Topics: Amides; Antimalarials; Binding Sites; Erythrocytes; HSP90 Heat-Shock Proteins; Humans; Indole Alkaloids; Life Cycle Stages; Molecular Dynamics Simulation; Plasmodium berghei; Plasmodium falciparum; Protozoan Proteins; Structure-Activity Relationship; Triazoles

2021
Design and synthesis of harmiquins, harmine and chloroquine hybrids as potent antiplasmodial agents.
    European journal of medicinal chemistry, 2022, Aug-05, Volume: 238

    Topics: Antimalarials; Chloroquine; Harmine; Heme; Humans; Malaria, Falciparum; Plasmodium falciparum

2022
Synergistic in vitro antimalarial activity of plant extracts used as traditional herbal remedies in Mali.
    Parasitology research, 2002, Volume: 88, Issue:2

    Topics: Animals; Antimalarials; Cell Culture Techniques; Chloroquine; Cytotoxins; Drug Synergism; Fluorescent Dyes; Harmine; Humans; Life Cycle Stages; Mali; Medicine, African Traditional; Mutagenesis; Plant Extracts; Plants, Medicinal; Plasmodium falciparum

2002
Harmine is a potent antimalarial targeting Hsp90 and synergizes with chloroquine and artemisinin.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:8

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Synergism; Harmaline; Harmine; HSP90 Heat-Shock Proteins; Malaria; Mice; Mice, Inbred BALB C; Mutagenesis, Site-Directed; Plasmodium berghei; Plasmodium falciparum; Protein Structure, Quaternary; Protein Structure, Tertiary; Surface Plasmon Resonance

2012