Compounds > chloroquine

chloroquine and bix 01294

chloroquine has been researched along with bix 01294 in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (83.33)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Biamonte, MA; Le Roch, KG; Wanner, J1
Chen, PB; Fuchter, MJ; Li, F; Lubin, AS; Lueg, GA; Malmquist, NA; Scherf, A; Sundriyal, S; Vedadi, M; White, AJP1
Andrews, KT; Arimondo, PB; Bouchut, A; Chua, MJ; Fabrizi, G; Hoglund, U; Khalife, J; Lafitte, S; Lucidi, A; Mai, A; Mazzone, R; Pechalrieu, D; Pierrot, C; Rotili, D; Schultz, J; Skinner-Adams, TS; Valente, S1
Chng, WJ; Dymock, BW; Fang Nee, AH; Haider, S; Mustafa, N; Ramanujulu, PM; Soumyanarayanan, U; Tan, KSW; Tong, JX1
Chen, Q; Deitsch, KW; Heinberg, AR; Ukaegbu, UE; Wele, M; Zhang, X1
Bao, X; Deng, A; Li, Q; Wang, L; Wang, M; Xiang, Y; Yu, W; Zhang, B; Zhang, Y1

Reviews

1 review(s) available for chloroquine and bix 01294

ArticleYear
Recent advances in malaria drug discovery.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure

2013

Other Studies

5 other study(ies) available for chloroquine and bix 01294

ArticleYear
Histone lysine methyltransferase structure activity relationships that allow for segregation of G9a inhibition and anti-
    MedChemComm, 2017, May-01, Volume: 8, Issue:5

    Topics:

2017
Identification of novel quinazoline derivatives as potent antiplasmodial agents.
    European journal of medicinal chemistry, 2019, Jan-01, Volume: 161

    Topics: Animals; Antimalarials; Dose-Response Relationship, Drug; Fibroblasts; Humans; Mice; Mice, Inbred BALB C; Molecular Conformation; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinazolines; Structure-Activity Relationship

2019
Discovery of a potent histone deacetylase (HDAC) 3/6 selective dual inhibitor.
    European journal of medicinal chemistry, 2019, Dec-15, Volume: 184

    Topics: Animals; Antimalarials; Apoptosis; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Drug Discovery; Histone Deacetylase 6; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Mice; Microsomes, Liver; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship

2019
A Unique Virulence Gene Occupies a Principal Position in Immune Evasion by the Malaria Parasite Plasmodium falciparum.
    PLoS genetics, 2015, Volume: 11, Issue:5

    Topics: Antigenic Variation; Antigens, Protozoan; Azepines; Chloroquine; Gene Expression Regulation; Genetic Loci; Histone Methyltransferases; Histone-Lysine N-Methyltransferase; Humans; Hydroxamic Acids; Immune Evasion; Inhibitory Concentration 50; Malaria, Falciparum; Models, Theoretical; Piperazines; Plasmodium falciparum; Promoter Regions, Genetic; Protozoan Proteins; Quinazolines; RNA Polymerase II; Terpenes; Transcriptional Activation; Transcriptome

2015
BIX-01294-enhanced chemosensitivity in nasopharyngeal carcinoma depends on autophagy-induced pyroptosis.
    Acta biochimica et biophysica Sinica, 2020, Oct-19, Volume: 52, Issue:10

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Autophagy; Autophagy-Related Protein 5; Azepines; bcl-2-Associated X Protein; Caspase 3; Cell Line, Tumor; Cell Survival; Chloroquine; Cisplatin; CRISPR-Cas Systems; Gene Knockout Techniques; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Microtubule-Associated Proteins; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Pyroptosis; Quinazolines; Receptors, Estrogen; Signal Transduction

2020