chloroquine and alpha-aminopyridine

chloroquine has been researched along with alpha-aminopyridine in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Avery, V; Bashyam, S; Bhamidipati, R; Charman, SA; Chibale, K; Douelle, F; Duffy, S; Feng, TS; González Cabrera, D; Hardick, D; Joseph, JT; Katneni, K; Le Manach, C; Mannila, J; Morizzi, J; Nchinda, AT; Shackleford, DM; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, KM1
Chen, M; Chen, T; Feng, J; Gao, L; Guo, H; Liang, Y; Liu, F; Liu, JJ; Ren, H; Shang, D; Shi, P; Thakur, A; Wang, T; Xu, F; Yang, T; Zhang, S1
Chibale, K; Egan, TJ; Hunter, R; Joshi, MC; Ndove, J; Nsumiwa, S; Okombo, J; Taylor, D; Wiesner, L1
Blanco-Aparicio, C; Hernández-Encinas, E; Llanos, S; Megias, D; Pietrocola, F; Rovira, M; Serrano, M1

Other Studies

4 other study(ies) available for chloroquine and alpha-aminopyridine

ArticleYear
3,5-Diaryl-2-aminopyridines as a novel class of orally active antimalarials demonstrating single dose cure in mice and clinical candidate potential.
    Journal of medicinal chemistry, 2012, Apr-12, Volume: 55, Issue:7

    Topics: Administration, Oral; Aminopyridines; Animals; Antimalarials; Biological Availability; Cell Line; Chloroquine; Cytochrome P-450 Enzyme Inhibitors; Drug Resistance; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Female; Humans; Isoenzymes; Malaria; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Rabbits; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

2012
Blockade efficacy of MEK/ERK-dependent autophagy enhances PI3K/Akt inhibitor NVP-BKM120's therapeutic effectiveness in lung cancer cells.
    Oncotarget, 2016, Oct-11, Volume: 7, Issue:41

    Topics: Aminopyridines; Animals; Antineoplastic Agents; Autophagy; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Chloroquine; Enzyme Inhibitors; Humans; Lung Neoplasms; MAP Kinase Signaling System; Mice; Morpholines; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Xenograft Model Antitumor Assays

2016
4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice.
    Journal of medicinal chemistry, 2017, 12-28, Volume: 60, Issue:24

    Topics: Administration, Oral; Aminopyridines; Aminoquinolines; Animals; Antimalarials; Cell Membrane Permeability; Chloroquine; CHO Cells; Cricetulus; Drug Evaluation, Preclinical; Drug Resistance, Microbial; ERG1 Potassium Channel; Hemeproteins; Humans; Malaria; Male; Mice, Inbred BALB C; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship

2017
Lysosomal trapping of palbociclib and its functional implications.
    Oncogene, 2019, Volume: 38, Issue:20

    Topics: Acridine Orange; Aminopyridines; Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Cellular Senescence; Chloroquine; Cyclin-Dependent Kinase 4; Cytokines; Fluorescent Dyes; Humans; Lysosomal Membrane Proteins; Lysosomes; Piperazines; Protein Kinase Inhibitors; Purines; Pyridines

2019