chlorine and indazoles

chlorine has been researched along with indazoles in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19904 (30.77)18.7374
1990's1 (7.69)18.2507
2000's4 (30.77)29.6817
2010's3 (23.08)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Felińska, W; Linkowska, E; Wrzeciono, U1
Mörsdorf, K; Wolf, G1
Bruce, J; Bueding, E; Fisher, J1
Kim, TY; Ko, JH; Park, RE; Ryu, CK; Ryu, JS; Song, EH; Yeon, SW; You, HJ1
Balogh, G; Rákóczi, J; Vedres, A1
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ1
Cheng, CY; Gong, XD; Leung, GP; Silvestrini, B; Wong, PY; Wong, YL1
Gong, XD; Wong, PY1
Liu, X; Miller, MJ; Niu, X; Powell, A; Reddix, RA1
Bokonjić, D; Colić, M; Jelenković, A; Jovanović, MD; Ninković, M; Stevanović, ID1
Chen, WY; Cheng, CY; Ge, RS; He, Y; Li, K; Lu, JX; Ni, Y; Shi, QX1
Alessio, E; Arcangeli, A; Balducci, G; Battistin, F; Messori, L; Pillozzi, S; Scaletti, F1
Boccuto, A; Cirri, D; Dragoni, F; Marrone, A; Marzo, T; Messori, L; Saladini, F; Tolbatov, I; Vicenti, I1

Other Studies

13 other study(ies) available for chlorine and indazoles

ArticleYear
[Azoles. 3. Nitro derivatives of 3-chlorindazoles and the influence of C-5, C-6 and N-nitrogroups on the reaction capability of C-3 chlorine atoms].
    Die Pharmazie, 1978, Volume: 33, Issue:7

    Topics: Acetylation; Chemical Phenomena; Chemistry; Chlorine; Hydrolysis; Indazoles; Isomerism; Morpholines; Nitro Compounds; Piperidines; Pyrazoles; Pyrrolidines; Temperature

1978
[Comparative study on the efficiency of new antiphlogistics].
    Arzneimittel-Forschung, 1972, Volume: 22, Issue:12

    Topics: Acetates; Aniline Compounds; Animals; Anti-Inflammatory Agents; Autolysis; Chlorine; Edema; Evaluation Studies as Topic; Hydroxamic Acids; Indazoles; Indoles; Malonates; Nicotinic Acids; ortho-Aminobenzoates; Phenothiazines; Phenylacetates; Propionates; Proteins; Pyridazines; Rats; Thiazoles; Toluene; Triazines

1972
The antischistosomal activity of a chloroindazole analog of hycanthone in mice infected with Schistosoma mansoni.
    The Journal of pharmacology and experimental therapeutics, 1973, Volume: 186, Issue:3

    Topics: Animals; Anthelmintics; Chlorine; Ethylenediamines; Female; Glycogen; Indazoles; Lethal Dose 50; Methanol; Mice; Phosphorylases; Pyrazoles; Schistosoma mansoni; Schistosomiasis; Schistosomicides; Xanthenes

1973
Synthesis and biological evaluation of 5-arylamino-6-chloro-1H-indazole-4,7-diones as inhibitors of protein kinase B/Akt.
    Bioorganic & medicinal chemistry letters, 2006, Dec-01, Volume: 16, Issue:23

    Topics: Amination; Animals; Antineoplastic Agents; Catalysis; Cell Line, Tumor; Chlorine; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Indazoles; Mice; Mice, Nude; Molecular Structure; Neoplasms; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Structure-Activity Relationship; Xenograft Model Antitumor Assays

2006
[Synthesis of oxinazin (1-benzyl-3-3'-dimethyl aminopropoxy(-1H-indazole HC1), a new antiphlogistic].
    Acta pharmaceutica Hungarica, 1974, Volume: 44, Issue:1

    Topics: Alkylating Agents; Anti-Inflammatory Agents; Benzyl Compounds; Chlorides; Dimethylamines; Indazoles; Pyrazoles; Sulfonic Acids

1974
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
    European journal of pharmacology, 1994, Jul-15, Volume: 268, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis

1994
Lonidamine and analogue AF2785 block the cyclic adenosine 3', 5'-monophosphate-activated chloride current and chloride secretion in the rat epididymis.
    Biology of reproduction, 2000, Volume: 63, Issue:3

    Topics: Animals; Benzyl Compounds; Bicarbonates; Chloride Channels; Chlorides; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Epididymis; Epithelial Cells; Indazoles; Male; Rats; Rats, Sprague-Dawley

2000
Characterization of Lonidamine and AF2785 blockade of the cyclic AMP-activated chloride current in rat epididymal cells.
    The Journal of membrane biology, 2000, Dec-01, Volume: 178, Issue:3

    Topics: Animals; Antispermatogenic Agents; Benzyl Compounds; Chlorides; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Epididymis; Epithelial Cells; Indazoles; Ion Channel Gating; Ion Transport; Male; Molecular Structure; ortho-Aminobenzoates; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Second Messenger Systems

2000
Constitutive nitric oxide release modulates neurally-evoked chloride secretion in guinea pig colon.
    Autonomic neuroscience : basic & clinical, 2000, Dec-28, Volume: 86, Issue:1-2

    Topics: Animals; Chloride Channels; Chlorides; Colon; Electric Stimulation; Enteric Nervous System; Enzyme Inhibitors; Gastrointestinal Motility; Guinea Pigs; Hemoglobins; Indazoles; Intestinal Absorption; Male; Neural Inhibition; Neurons, Efferent; NG-Nitroarginine Methyl Ester; Nitric Oxide

2000
Nitric oxide synthase inhibitors protect cholinergic neurons against AlCl3 excitotoxicity in the rat brain.
    Brain research bulletin, 2010, Apr-05, Volume: 81, Issue:6

    Topics: Acetylcholinesterase; Aluminum Chloride; Aluminum Compounds; Animals; Avoidance Learning; Brain; Chlorides; Enzyme Activation; Enzyme Inhibitors; Guanidines; Hippocampus; Indazoles; Male; Memory; Neurons; Neuroprotective Agents; Neurotoxins; Nitric Oxide Synthase; Rats; Time Factors

2010
Inhibition of sperm capacitation and fertilizing capacity by adjudin is mediated by chloride and its channels in humans.
    Human reproduction (Oxford, England), 2013, Volume: 28, Issue:1

    Topics: Acrosome Reaction; Adenylyl Cyclase Inhibitors; Adult; Animals; Chloride Channels; Chlorides; Contraceptive Agents, Male; Cricetinae; Cyclic AMP; Egg Proteins; Enzyme Inhibitors; Female; Fertilization; Humans; Hydrazines; Indazoles; Male; Membrane Glycoproteins; Membrane Transport Modulators; Phosphodiesterase Inhibitors; Phosphorylation; Protein Processing, Post-Translational; Receptors, Cell Surface; Recombinant Proteins; Sperm Capacitation; Spermatozoa; Zona Pellucida Glycoproteins

2013
Water-soluble Ru(II)- and Ru(III)-halide-PTA complexes (PTA=1,3,5-triaza-7-phosphaadamantane): Chemical and biological properties.
    Journal of inorganic biochemistry, 2016, Volume: 160

    Topics: Adamantane; Antineoplastic Agents; Bromides; Cell Line, Tumor; Cell Survival; Chlorides; Coordination Complexes; Cytochromes c; Filaggrin Proteins; HCT116 Cells; Humans; Hydrogen-Ion Concentration; Imidazoles; Indazoles; Inhibitory Concentration 50; Ligands; Oligonucleotides; Organometallic Compounds; Organophosphorus Compounds; Protons; Ribonuclease, Pancreatic; Ruthenium; Solubility; Structure-Activity Relationship; Water

2016
In Vitro Anti-SARS-CoV-2 Activity of Selected Metal Compounds and Potential Molecular Basis for Their Actions Based on Computational Study.
    Biomolecules, 2021, 12-10, Volume: 11, Issue:12

    Topics: 2,2'-Dipyridyl; Animals; Antimony; Antiviral Agents; Cell Line; Chlorides; Chlorocebus aethiops; COVID-19 Drug Treatment; Drug Discovery; Humans; Indazoles; Organogold Compounds; Organometallic Compounds; Ruthenium Compounds; SARS-CoV-2; Vero Cells

2021