chlorethylclonidine has been researched along with wb 4101 in 109 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (1.83) | 18.7374 |
1990's | 95 (87.16) | 18.2507 |
2000's | 10 (9.17) | 29.6817 |
2010's | 2 (1.83) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bondinell, WE; Hieble, JP; Ruffolo, RR | 1 |
Etgen, AM; Karkanias, GB; Petitti, N | 1 |
Aniukhovskiĭ, EP; Rozen, MP; Staĭnberg, SF | 1 |
Kowatch, MA; Miyamoto, A; Roth, GS; Villalobos-Molina, R | 1 |
Chiba, S; Skrbic, R | 1 |
Bevan, JA; Bevan, RD; Oriowo, MA | 1 |
Hayakawa, H; Shimizu, M; Yamawaki, S | 1 |
Kigoshi, S; Muramatsu, I; Ohmura, T; Oshita, M | 1 |
Kojima, C; Satoh, M; Takayanagi, I | 1 |
Harada, M; Koike, K; Satoh, M; Takayanagi, I | 1 |
Anyukhovsky, EP; Rosen, MR | 1 |
Abel, PW; Feng, F; Jeffries, WB; Pettinger, WA | 1 |
García-Sáinz, JA; Torres-Márquez, ME; Villalobos-Molina, R | 1 |
Anyukhovsky, EP; Molina-Viamonte, V; Rosen, MR | 1 |
Piascik, MT; Pruitt, TA; Soltis, EE; Sparks, MS | 1 |
Han, CD; Minneman, KP | 1 |
Moriya, M; Takayanagi, I | 1 |
Han, C; Li, J; Minneman, KP | 1 |
Hashimoto, S; Kigoshi, S; Muramatsu, I; Ohmura, T; Oshita, M | 1 |
Deth, RC; Gupta, S; Tian, WN | 1 |
Butler, BT; Kusiak, JW; Piascik, MT; Pruitt, TA | 1 |
Terman, BI | 1 |
Hashimoto, K; Suzuki, E; Tamura, K; Tsujimoto, G | 1 |
Hashimoto, K; Suzuki, E; Tsujimoto, G | 1 |
Minneman, KP; Wilson, KM | 1 |
del Balzo, U; Kaplan, LM; Malfatto, G; Rosen, MR; Steinberg, SF | 1 |
Bevan, JA; Oriowo, MA | 1 |
Bowersox, S; Ciaranello, R; Dement, WC; Frusthofer, B; Guilleminault, C; Maddaluno, J; Mignot, E; Nishino, S | 1 |
Abel, PW; Han, C; Minneman, KP | 1 |
Kow, LM; Pfaff, DW | 1 |
Han, C; Yu, GS | 1 |
Iwanov, V; Jiang, GC; Moulds, RF | 2 |
Badia, A; Gascón, S; Ivorra, D; Vila, E | 1 |
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H | 1 |
Kennedy, RH; Lindemann, JP; Seifen, E; Williamson, AP | 4 |
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M | 1 |
Aston, N; Chess-Williams, R; Couldwell, C | 1 |
Bowdish, DM; Gaspar, V; Low, AM; Prashad, TR | 1 |
Kigoshi, S; Muramatsu, I; Muraoka, R; Noguchi, H | 1 |
Kokubu, N; Satoh, M; Takayanagi, I | 1 |
Edwards, FR; Hill, CE; Hirst, GD; Klemm, M | 1 |
Badia, A; Dierssen, M; Gascón, S; Màrmol, F; Vivas, NM | 1 |
Chess-Williams, R; Couldwell, C; Jackson, A; O'Brien, H | 1 |
Aniukhovskiĭ, EP; Rosen, MR | 1 |
Anyukhovsky, EP; Cohen, IS; Rosen, MR; Steinberg, SF | 1 |
Badia, A; Sallés, J | 1 |
Chen, MZ; Han, QD; Yu, GS | 1 |
Daniel, EE; Hoo, KH; Kwan, CY | 1 |
Cable, DG; Dreyer, ER; Martins, JB; Rath, TE | 1 |
Oriowo, MA | 1 |
Anversa, P; Capasso, JM; Cheng, W; Coupet, J; Hamby, CV; Li, P; Meggs, LG; Reiss, K | 1 |
Nagashima, M | 1 |
Lepor, H; Meretyk, S; Shapiro, E; Tang, R | 1 |
Kennedy, RH; Lindemann, JP; Seifen, E; Stimers, JR; Williamson, AP | 1 |
Lepor, H; Shapiro, E; Tang, R | 1 |
Lee, JH; Rosen, MR | 1 |
Hagino, Y; Hasegawa, S; Kondo, H; Nomura, H; Nomura, T; Sumi-Ichinose, C; Tachibana, M; Ukai, K; Watanabe, T; Yokoyama, R | 1 |
Mironneau, C; Mironneau, J; Neuilly, G; Rakotoarisoa, L; Sayet, I | 1 |
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T | 1 |
Docherty, JR; Kearns, S; O'Rourke, M | 1 |
Cua, M; Danilo, P; Geller, JC; Guo, SD; Prieto, L; Rosen, MR | 1 |
Anwar, N; Klein, DC; Sugden, D | 1 |
Akaishi, Y; Hattori, Y; Kanno, M; Nagashima, M | 1 |
Akaishi, Y; Hattori, Y; Kanno, M; Kitabatake, A; Nagashima, M; Sakuma, I; Tohse, N | 1 |
Benoit, JN; Gao, H; Korthuis, RJ | 1 |
Choe, EU; Ferrara, JJ; Flint, LM; Hoang, TV; Hyman, AL; Lippton, HL | 1 |
Arias-Montaño, JA; De la Vega, MT; Trejo, F | 1 |
Aceves, J; Arias-Montaño, JA; Nuñez, A | 1 |
Homuth, V; Luther, HP; Wallukat, G | 1 |
Moulds, RF; Tognarini, DP | 1 |
Osnes, JB; Sandnes, D; Skomedal, T; Viko, H | 1 |
Dyer, DC; Hu, XQ | 1 |
Hattori, Y; Kanno, M; Nagashima, M; Tohse, N | 1 |
Cheng, JT; Tong, YC | 1 |
Han, C; Zhang, Y; Zhu, W | 1 |
Hattori, Y; Kanno, M | 1 |
Benoit de Coignac, A; Coudouel, N; Legrand, C; Limon-Boulez, I; Maltier, JP; Mhaouty-Kodja, S | 1 |
Macmillan, JB; McGrath, JC; Smith, KM | 1 |
Asakura, Y; Ebihara, Y; Hasegawa, H; Nakamura, Y; Shinmura, K; Suganuma, Y; Tani, M | 1 |
Chevalier, P; Danilo, P; Rosen, MR; Ruffy, F | 1 |
Hasegawa, Y; Ono, H; Wada, T | 1 |
Han, C; Lu, Z; Wei, H; Xu, K; Zhang, Y | 1 |
Capogrossi, MC; Gambassi, G; Lakatta, EG; Spurgeon, HA; Ziman, BD | 1 |
Brown, RD; Daniel, EE; Kwan, CY; Low, AM; Lu-Chao, H; Wang, YF | 1 |
Avkiran, M; Yasutake, M; Yokoyama, H | 1 |
Pupo, AS | 1 |
Hattori, K; Makara, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Suzuki, M; Tsuchiya, M; Watanabe, K | 1 |
Campos-Mello, C; Correa, FM; de Oliveira, AM; Leitão, MC | 1 |
García-Sáinz, JA; Torres-Padilla, ME | 1 |
Kocić, I | 1 |
Avellar, MC; Megale, A; Porto, CS; Silva, MA | 1 |
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM | 1 |
Antzelevitch, C; Burashnikov, A | 1 |
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K | 1 |
Chen, PC; Cheng, JT; Liu, IM; Yen, ST | 1 |
Hillier, C; Jarajapu, YP; MacDonald, A | 1 |
Koike, K; Yamamoto, Y | 1 |
Chiba, S; Taguchi, Y; Yang, XP | 1 |
Chiba, S; Tsukada, M | 1 |
Katus, HA; Kemken, D; Kurz, T; Mier, K; Richardt, G | 1 |
Campos, M; Morais, Pde L; Pupo, AS | 1 |
Avellar, MC; Hamamura, M; Mendes, FR; Porto, CS; Queiróz, DB | 1 |
Avellar, MC; Caricati-Neto, A; Jurkiewicz, A; Jurkiewicz, NH; Reuter, HR; Verde, LF | 1 |
Bockman, CS; Dang, HK; Gruber, DD; Scofield, MA; Wangemann, P; Witt, KM | 1 |
Dementieva, RE; Fashutdinov, LI; Zefirov, TL; Ziyatdinova, NI | 1 |
1 review(s) available for chlorethylclonidine and wb 4101
Article | Year |
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Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1995 |
108 other study(ies) available for chlorethylclonidine and wb 4101
Article | Year |
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Estradiol selectively regulates alpha 1B-noradrenergic receptors in the hypothalamus and preoptic area.
Topics: Animals; Clonidine; Cyclic AMP; Dioxanes; Estradiol; Female; Hypothalamus; Ovariectomy; Piperazines; Prazosin; Preoptic Area; Rats; Receptors, Adrenergic | 1992 |
[Modulation of heart rhythm by alpha-1 adrenoreceptors].
Topics: Animals; Arrhythmias, Cardiac; Clonidine; Dioxanes; Dogs; Electrocardiography; Heart Rate; Myocardial Ischemia; Phentolamine; Rats; Receptors, Adrenergic, alpha | 1992 |
Alpha 1-adrenoceptors in parotid cells: age does not alter the ratio of alpha 1A and alpha 1B subtypes.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Calcium; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Inosine Triphosphate; Male; Parotid Gland; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1992 |
Pharmacological properties of alpha 1-adrenoceptor-mediated vasoconstrictions in dog and monkey lingual arteries: evidence for subtypes of alpha 1-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channels; Clonidine; Diltiazem; Dioxanes; Dogs; Dose-Response Relationship, Drug; Macaca; Muscle, Smooth, Vascular; Norepinephrine; Receptors, Adrenergic; Signal Transduction; Species Specificity; Tongue; Vasoconstriction | 1992 |
Vascular alpha-adrenoceptor affinity variation is not due to varying populations of subtypes distinguished by WB 4101 and chlorethylclonidine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Clonidine; Dioxanes; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rabbits; Receptors, Adrenergic, alpha | 1992 |
The effects of electroconvulsive shock or imipramine on subtypes of alpha 1-adrenoceptors in the frontal cortex of the rat.
Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Clonidine; Dioxanes; Electroshock; Hippocampus; Imipramine; In Vitro Techniques; Kinetics; Male; Prazosin; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Adrenergic, alpha | 1992 |
Identification of alpha 1-adrenoceptor subtypes in the rat vas deferens: binding and functional studies.
Topics: Acetonitriles; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Electric Stimulation; Epididymis; In Vitro Techniques; Kinetics; Male; Muscle, Smooth; Nifedipine; Norepinephrine; Oxathiins; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Vas Deferens | 1992 |
Pharmacological characterization of contractile responses induced by alpha 1-agonists, norepinephrine and clonidine, by selective antagonists of their subtypes in rabbit thoracic aorta.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rabbits | 1992 |
Differences in alpha 1-adrenoceptor mechanisms for phenylephrine and tizanidine in rabbit thoracic aorta and common iliac artery.
Topics: Animals; Aorta, Thoracic; Clonidine; Dioxanes; Iliac Artery; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Receptors, Adrenergic, alpha; Tissue Distribution; Vasoconstriction | 1991 |
Abnormal automatic rhythms in ischemic Purkinje fibers are modulated by a specific alpha 1-adrenergic receptor subtype.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Clonidine; Coronary Disease; Dioxanes; Dogs; Extracellular Space; Heart Rate; Phenylephrine; Propranolol; Purkinje Fibers; Receptors, Adrenergic, alpha | 1991 |
Regional distribution of alpha 1-adrenoceptor subtypes in rat kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Cell Membrane; Clonidine; Dioxanes; Kidney; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1991 |
Alpha 1-adrenoceptor subtypes in aorta (alpha 1A) and liver (alpha 1B).
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Liver; Membranes; Muscle, Smooth, Vascular; Phosphatidylinositols; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha | 1991 |
An alpha-1-adrenergic receptor subtype is responsible for delayed afterdepolarizations and triggered activity during simulated ischemia and reperfusion of isolated canine Purkinje fibers.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Clonidine; Dioxanes; Dogs; Myocardial Reperfusion Injury; Phenylephrine; Purkinje Fibers; Receptors, Adrenergic, alpha | 1991 |
Evidence for a complex interaction between the subtypes of the alpha 1-adrenoceptor.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Kinetics; Male; Methoxamine; Muscle, Smooth, Vascular; Phenoxybenzamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1991 |
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor binding sites in rat tissues.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dioxanes; Kinetics; Male; Membranes; Phentolamine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Time Factors | 1991 |
Alpha 1A-adrenoceptors in rabbit bronchus.
Topics: Adrenergic alpha-Antagonists; Animals; Bronchi; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha | 1991 |
Subtypes of alpha 1-adrenoceptors in rat blood vessels.
Topics: Animals; Aorta, Thoracic; Blood Vessels; Clonidine; Dioxanes; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Renal Artery | 1990 |
Pharmacological subclassification of alpha 1-adrenoceptors in vascular smooth muscle.
Topics: Acetonitriles; Adrenergic alpha-Antagonists; Animals; Blood Vessels; Clonidine; Dioxanes; Dogs; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Phentolamine; Prazosin; Rabbits; Rats; Receptors, Adrenergic, alpha; Species Specificity; Yohimbine | 1990 |
Species differences in chlorethylclonidine antagonism at vascular alpha-1 adrenergic receptors.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Male; Muscle, Smooth, Vascular; Norepinephrine; Rabbits; Rats; Receptors, Adrenergic, alpha; Species Specificity; Vasoconstriction | 1990 |
Agonist interaction with alkylation-sensitive and -resistant alpha-1 adrenoceptor subtypes.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Clonidine; Diltiazem; Dioxanes; Drug Interactions; Heart; Inositol Phosphates; Male; Muscle, Smooth, Vascular; Myocardium; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1990 |
[The identification and characteristics of subpopulations of alpha 1-adrenergic receptors].
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain Chemistry; Calcium; Clonidine; Dioxanes; GTP-Binding Proteins; Liver; Microsomes; Phentolamine; Prazosin; Rats; Receptors, Adrenergic, alpha | 1990 |
Two pharmacologically distinct alpha 1-adrenoceptor subtypes in the contraction of rabbit aorta: each subtype couples with a different Ca2+ signalling mechanism and plays a different physiological role.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Binding Sites; Calcium; Clonidine; Dioxanes; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenethylamines; Phenoxybenzamine; Piperazines; Rabbits; Receptors, Adrenergic, alpha; Signal Transduction; Tetralones; Vasoconstriction | 1990 |
Different desensitization mechanisms of two alpha 1-adrenoceptor subtypes in the contraction of rabbit aorta.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenethylamines; Rabbits; Receptors, Adrenergic, alpha; Tetralones | 1990 |
Pertussis toxin inhibits norepinephrine-stimulated inositol phosphate formation in primary brain cell cultures.
Topics: Animals; Brain; Calcium; Carbachol; Cells, Cultured; Clonidine; Cyclic AMP; Dioxanes; GTP-Binding Proteins; Inositol Phosphates; Norepinephrine; Pertussis Toxin; Phenethylamines; Prazosin; Rats; Receptors, Adrenergic, alpha; Tetralones; Virulence Factors, Bordetella; Yohimbine | 1990 |
Specific alpha 1-adrenergic receptor subtypes modulate catecholamine-induced increases and decreases in ventricular automaticity.
Topics: Age Factors; Animals; Binding Sites; Cells, Cultured; Clonidine; Dioxanes; Dogs; Electrophysiology; Heart Ventricles; Inositol Phosphates; Norepinephrine; Purkinje Fibers; Receptors, Adrenergic, alpha; Stimulation, Chemical; Ventricular Function | 1990 |
Chloroethylclonidine unmasks a non-alpha-adrenoceptor noradrenaline binding site in the rat aorta.
Topics: Animals; Aorta, Thoracic; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Rats; Receptors, Adrenergic; Yohimbine | 1990 |
Central alpha 1 adrenoceptor subtypes in narcolepsy-cataplexy: a disorder of REM sleep.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Cataplexy; Clonidine; Dioxanes; Dogs; Narcolepsy; Phenoxybenzamine; Prazosin; Receptors, Adrenergic, alpha; Sleep, REM | 1989 |
Comparison of alpha 1-adrenergic receptor subtypes distinguished by chlorethylclonidine and WB 4101.
Topics: Animals; Clonidine; Dioxanes; Dioxins; Hippocampus; In Vitro Techniques; Inositol Phosphates; Male; Norepinephrine; Osmolar Concentration; Rats; Receptors, Adrenergic, alpha; Solubility; Spleen; Tissue Distribution; Vas Deferens | 1988 |
Functional analyses of alpha 1-adrenoceptor subtypes in rat hypothalamic ventromedial nucleus neurons.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Hypothalamus, Middle; In Vitro Techniques; Neurons; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1995 |
Role of alpha 1A- and alpha 1B-adrenoceptors in phenylephrine-induced positive inotropic response in isolated rat left atrium.
Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Inositol Phosphates; Male; Myocardial Contraction; Phenethylamines; Phenylephrine; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Tetralones | 1994 |
Increased sensitivity to inhibition by nifedipine of responses of the mesenteric artery bed of the SHRSP to noradrenaline is not dependent on alpha 1-adrenoceptor subtypes.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Clonidine; Dioxanes; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Hypertension; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Vascular Resistance | 1995 |
Alpha 1-adrenoceptor subtypes and inositol phosphates production in heart ventricles of spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Heart Ventricles; Hypertension; Inositol Phosphates; Male; Myocardium; Norepinephrine; Prazosin; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha | 1993 |
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine | 1995 |
Alpha 1a-adrenergic receptor mediated positive chronotropic effect in right atria isolated from rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Atrial Function; Clonidine; Dioxanes; Heart Atria; Heart Rate; In Vitro Techniques; Male; Phenoxybenzamine; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1994 |
The difference in nifedipine sensitivity between hypertensive and normotensive rat aortae is dependent on age.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Aorta, Thoracic; Clonidine; Dioxanes; Hypertension; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred WKY | 1995 |
Pharmacological evidence of distinct alpha 1-adrenoceptor subtypes mediating the contraction of human prostatic urethra and peripheral artery.
Topics: Aged; Aged, 80 and over; Arteries; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Phenylephrine; Receptors, Adrenergic, alpha-1; Urethra; Vasoconstriction | 1994 |
Alpha 1A-adrenoceptor subtype mediates contraction of the rat urethra.
Topics: Aminoquinolines; Animals; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetrahydroisoquinolines; Urethra | 1994 |
Interactions of chloroethylclonidine with rauwolscine- and prazosin-sensitive adrenoceptors in dog saphenous vein.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Calcium; Calcium Channel Blockers; Clonidine; Dioxanes; Dogs; Extracellular Space; In Vitro Techniques; Membranes; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Saphenous Vein; Yohimbine | 1994 |
Alpha 1-adrenoceptor subtype involved in the positive inotropic response to phenylephrine in rat atria.
Topics: Acetonitriles; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Heart Atria; In Vitro Techniques; Male; Myocardial Contraction; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha | 1993 |
Chloroethylclonidine discriminates between alpha 1A- and alpha 1B-adrenoceptors in the presence of guanosine 5'-triphosphate in rabbit thoracic aorta.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding Sites; Clonidine; Dioxanes; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Phenylephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha | 1993 |
Sympathetic transmission to the dilator muscle of the rat iris.
Topics: Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Clonidine; Dioxanes; Iris; Membrane Potentials; Neuroeffector Junction; Norepinephrine; Parasympathetic Nervous System; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sympathetic Nervous System; Synaptic Transmission; Synaptic Vesicles; Yohimbine | 1993 |
Effects of age on alpha 1-adrenoceptor subtypes in the heart ventricular muscle of the rat.
Topics: Adrenergic alpha-Antagonists; Aging; Alkylating Agents; Animals; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Myocardium; Norepinephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1993 |
Characterization of the alpha 1-adrenoceptors of the rat prostate gland.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Clonidine; Dioxanes; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Phenylephrine; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens | 1993 |
Effects of WB4101 and chloroethylclonidine on the positive and negative inotropic actions of phenylephrine in rat cardiac muscle.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Drug Antagonism; In Vitro Techniques; Male; Myocardial Contraction; Phenylephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1994 |
[The modulation of anomalous automatism in ischemic Purkinje fibers by a specific subclass of alpha 1-adrenoblockers].
Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Arrhythmias, Cardiac; Clonidine; Dioxanes; Dogs; Heart Rate; In Vitro Techniques; Myocardial Ischemia; Myocardial Reperfusion; Perfusion; Purkinje Fibers; Receptors, Adrenergic, alpha-1 | 1993 |
Receptor-effector coupling pathway for alpha 1-adrenergic modulation of abnormal automaticity in 'ischemic' canine Purkinje fibers.
Topics: Adrenergic alpha-Antagonists; Animals; Barium; Clonidine; Dioxanes; Dogs; Membrane Potentials; Myocardial Ischemia; Pertussis Toxin; Phenylephrine; Purkinje Fibers; Receptors, Adrenergic, alpha-1; Virulence Factors, Bordetella | 1994 |
Selective enrichment with alpha 1A- and alpha 1B-adrenoceptor subtypes in rat brain cortical membranes.
Topics: Adrenergic alpha-Antagonists; Alkylating Agents; Alkylation; Animals; Binding Sites; Cerebral Cortex; Clonidine; Cystamine; Dihydropyridines; Dioxanes; Phenoxybenzamine; Phentolamine; Prazosin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha | 1994 |
A new alpha 1-adrenergic receptor subtype with low affinity for 5-methyl-urapidil but insensitive to chlorethylclonidine.
Topics: Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Clonidine; Dioxanes; Male; Myocardium; Phenethylamines; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetralones | 1993 |
Investigation of alpha 1-adrenoceptor subtypes in canine aorta, using alkylating agents.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Aorta; Binding, Competitive; Clonidine; Dioxanes; Dogs; Female; In Vitro Techniques; Male; Mesenteric Veins; Muscle, Smooth, Vascular; Oxymetazoline; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1 | 1994 |
WB4101- and CEC-sensitive positive inotropic actions of phenylephrine in rat cardiac muscle.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; Heart Atria; In Vitro Techniques; Male; Myocardial Contraction; Osmolar Concentration; Papillary Muscles; Phenylephrine; Rats; Rats, Sprague-Dawley | 1994 |
Refractory period response of cardiac Purkinje tissue to alpha 1- and alpha 2-adrenergic influences.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Dioxanes; Dogs; Female; Male; Norepinephrine; Phenylephrine; Purkinje Fibers; Receptors, Adrenergic, alpha; Refractory Period, Electrophysiological | 1994 |
Alpha 1-adrenoceptor subtype(s) mediating noradrenaline-induced contractions of the guinea-pig aorta.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Clonidine; Dioxanes; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Oxazines; Prazosin; Receptors, Adrenergic, alpha-1 | 1994 |
Coronary artery constriction in rats affects the activation of alpha 1 adrenergic receptors in cardiac myocytes.
Topics: Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Base Sequence; Calcium; Cell Size; Cells, Cultured; Clonidine; Constriction; Coronary Vessels; Cytosol; Dioxanes; Inositol Phosphates; Male; Molecular Sequence Data; Myocardium; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1994 |
[Pharmacological study on functional significance of alpha 1-adrenoceptor subtypes in mammalian ventricular myocardium].
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Heart Ventricles; Hydrolysis; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Phenylephrine; Phosphatidylinositols; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Stimulation, Chemical | 1994 |
Alpha 1 adrenoceptor subtypes in the human prostate.
Topics: Adrenergic alpha-Antagonists; Aged; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Male; Middle Aged; Phenethylamines; Piperazines; Prostate; Receptors, Adrenergic, alpha; Tetralones | 1993 |
Alpha 1b-adrenoceptor-mediated stimulation of Na-K pump current in adult rat ventricular myocytes.
Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; Heart Ventricles; Male; Myocardium; Ouabain; Phenoxybenzamine; Phenylephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Sodium-Potassium-Exchanging ATPase; Ventricular Function, Left | 1993 |
The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylephrine; Piperazines; Prostate; Receptors, Adrenergic, alpha | 1993 |
Modulation of delayed afterdepolarisations by alpha 1 adrenergic receptor subtypes.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Clonidine; Culture Techniques; Dioxanes; Dogs; Heart; Ouabain; Phenylephrine; Purkinje Fibers; Receptors, Adrenergic, alpha | 1993 |
Alpha 1B-adrenoceptor-mediated stimulation of Ca2+ mobilization and cAMP accumulation in isolated rat hepatocytes.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Clonidine; Cyclic AMP; Dioxanes; In Vitro Techniques; Liver; Male; Methoxamine; Norepinephrine; Pertussis Toxin; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Signal Transduction; Tetradecanoylphorbol Acetate; Vasopressins; Virulence Factors, Bordetella | 1993 |
Relation between alpha 1-adrenoceptor subtypes and noradrenaline-induced contraction in rat portal vein smooth muscle.
Topics: Acetonitriles; Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Clonidine; Dioxanes; Horses; In Vitro Techniques; Isometric Contraction; Kinetics; Microsomes; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Portal Vein; Prazosin; Rats; Receptors, Adrenergic, alpha-1 | 1993 |
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine | 1993 |
Investigation of the actions of chloroethylclonidine in rat aorta.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine | 1995 |
Chloroethylclonidine increases the incidence of lethal arrhythmias during coronary occlusion in anesthetized dogs.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Clonidine; Dioxanes; Dogs; Female; Male; Myocardial Ischemia; Receptors, Adrenergic, alpha-1 | 1995 |
The positive inotropic effect of alpha 1A-adrenoceptor stimulation is inhibited by 4-aminopyridine.
Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Cardiotonic Agents; Clonidine; Dioxanes; Heart Atria; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Staurosporine | 1996 |
Rat pineal alpha 1-adrenoceptor subtypes: studies using radioligand binding and reverse transcription-polymerase chain reaction analysis.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dioxanes; Male; Phenethylamines; Pineal Gland; Polymerase Chain Reaction; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Tetralones; Transcription, Genetic | 1996 |
Alpha 1-adrenoceptor subtype distribution and the coupling to phosphoinositide hydrolysis in rat and rabbit ventricular myocardium.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Heart Ventricles; Hydrolysis; Kinetics; Lithium Chloride; Male; Myocardium; Phosphatidylinositols; Prazosin; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tritium | 1996 |
Alpha 1-adrenoceptor subtypes mediating inotropic and electrophysiological effects in mammalian myocardium.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Electric Conductivity; Electrophysiology; Female; Heart; Male; Myocardial Contraction; Papillary Muscles; Phenylephrine; Rabbits; Rats; Receptors, Adrenergic, alpha | 1996 |
Hypoxia/reoxygenation selectively impairs alpha 1b-adrenoceptor function in small mesenteric arteries.
Topics: Adrenergic alpha-Antagonists; Aerobiosis; Animals; Catalase; Clonidine; Dioxanes; Hypoxia; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Yohimbine | 1996 |
Characterization of alpha-adrenoceptor activity in term-newborn piglet mesentery.
Topics: Animals; Animals, Newborn; Benzazepines; Clonidine; Dioxanes; Female; Male; Mesenteric Arteries; Receptors, Adrenergic, alpha; Swine; Vasoconstriction | 1996 |
Functional characterisation of alpha 1-adrenoceptor subtypes mediating noradrenaline-induced inositol phosphate formation in rat thalamus slices.
Topics: Adrenergic alpha-Agonists; Animals; Calcium; Clonidine; Dioxanes; In Vitro Techniques; Inositol Phosphates; Male; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Thalamus | 1996 |
Noradrenaline-induced inositol phosphate formation in rat striatum is mediated by alpha 1A-adrenoceptors.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Calcium; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dioxanes; In Vitro Techniques; Inositol Phosphates; Male; Neostriatum; Norepinephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1996 |
Alpha 1-adrenergic receptor antibodies in patients with primary hypertension.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Amino Acid Sequence; Animals; Animals, Newborn; Autoantibodies; Blood Proteins; Cells, Cultured; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Heart; Humans; Hypertension; Male; Middle Aged; Molecular Sequence Data; Peptides; Phenylephrine; Prazosin; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance | 1997 |
Intracellular Ca2+ and contractile responses to alpha 1-adrenoceptor subtype activation in rat aortic vascular smooth muscle.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Calcium; Clonidine; Dioxanes; Female; Fluorescent Dyes; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Sprague-Dawley | 1997 |
Alpha 1-adrenoceptor subtypes involved in increased 86Rb+ influx rate and inositol 1,4,5-trisphosphate mass in adult rat cardiomyocytes.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Clonidine; Dioxanes; Heart Ventricles; Inositol 1,4,5-Trisphosphate; Myocardium; Piperazines; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Rubidium Radioisotopes | 1997 |
Heterogeneity and complexity of alpha 1-adrenoceptors in the ovine uterine artery and umbilical vein.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Binding, Competitive; Calcium Channel Blockers; Clonidine; Dioxanes; Drug Interactions; Drug Synergism; Female; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Prazosin; Pregnancy; Receptors, Adrenergic, alpha-1; Sheep; Umbilical Veins; Uterus; Vasoconstriction | 1997 |
Alpha 1-adrenoceptor subtype involved in the positive and negative inotropic responses to phenylephrine in rat papillary muscle.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Carcinogens; Cardiotonic Agents; Clonidine; Dioxanes; Electrophysiology; In Vitro Techniques; Myocardial Contraction; Nifedipine; Papillary Muscles; Phenylephrine; Phorbol 12,13-Dibutyrate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1997 |
Subtyping of alpha1-adrenoceptors responsible for the contractile response in the rat corpus cavernosum.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Penis; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1997 |
Characterization of subtype of alpha1-adrenoceptor mediating vasoconstriction in perfused rat hind limb.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Cell Line; Clonidine; Cloning, Molecular; Dioxanes; Dose-Response Relationship, Drug; Extremities; Humans; Indoles; Norepinephrine; Perfusion; Piperazines; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Vasoconstriction | 1997 |
Involvement of alpha1B-adrenoceptors in the positive inotropic effect of endogenous noradrenaline in rabbit myocardium.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Male; Myocardial Contraction; Norepinephrine; Papillary Muscles; Phenylephrine; Propranolol; Rabbits; Receptors, Adrenergic, alpha-1; Stimulation, Chemical; Tyramine | 1997 |
The alpha1B-adrenergic receptor subtype activates the phospholipase C signaling pathway in rat myometrium at parturition.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Membrane; Clonidine; Dioxanes; Female; Guanylyl Imidodiphosphate; Labor, Obstetric; Myometrium; Pregnancy; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Signal Transduction; Type C Phospholipases | 1997 |
Investigation of alpha1-adrenoceptor subtypes mediating vasoconstriction in rabbit cutaneous resistance arteries.
Topics: Acetonitriles; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1; Skin; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction | 1997 |
Effects of alpha 1-adrenoreceptor subtype blockade on ischemia-reperfusion injury.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Clonidine; Dioxanes; Energy Metabolism; In Vitro Techniques; Male; Myocardial Reperfusion Injury; Quinazolines; Rats; Rats, Sprague-Dawley | 1997 |
Interaction between alpha-1 adrenergic and vagal effects on cardiac rate and repolarization.
Topics: Animals; Clonidine; Dioxanes; Electrocardiography; GTP-Binding Proteins; Guinea Pigs; Heart; Heart Rate; Male; Membrane Potentials; Phenylephrine; Receptors, Adrenergic, alpha-1; Vagus Nerve | 1998 |
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord | 1997 |
Alteration of alpha1-adrenoceptor subtypes in aortas of 12-month-old spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; Hypertension; Indoles; Male; Muscle Contraction; Norepinephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Ribonucleases | 1998 |
Opposing effects of alpha 1-adrenergic receptor subtypes on Ca2+ and pH homeostasis in rat cardiac myocytes.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Clonidine; Dioxanes; Drug Combinations; Drug Synergism; Fluorescent Dyes; Homeostasis; Hydrogen; Hydrogen-Ion Concentration; Indoles; Male; Myocardial Contraction; Myocardium; Phenylephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1998 |
Pharmacological and immunocytochemical characterization of subtypes of alpha-1 adrenoceptors in dog aorta.
Topics: Animals; Aorta; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Immunohistochemistry; Indoles; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Spiro Compounds | 1998 |
Alpha1-adrenergic stimulation of sarcolemmal Na+-H+ exchanger activity in rat ventricular myocytes: evidence for selective mediation by the alpha1A-adrenoceptor subtype.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cattle; Clonidine; Dioxanes; Heart Ventricles; Humans; Imidazoles; Kinetics; Myocardium; Phenylephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sarcolemma; Sodium-Hydrogen Exchangers; Tetrahydronaphthalenes | 1998 |
Functional effects of castration on alpha1-adrenoceptors in rat vas deferens.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Castration; Clonidine; Dioxanes; Male; Muscle Contraction; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vas Deferens; Vasoconstrictor Agents | 1998 |
Discrimination of alpha1-adrenoceptor subtypes in rat aorta and prostate.
Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vasoconstriction; Vasodilator Agents | 1998 |
Maturation and aging-related differences in responsiveness of rat aorta and carotid arteries to alpha1-adrenoceptor stimulation.
Topics: Adrenergic alpha-Antagonists; Aging; Analysis of Variance; Animals; Aorta, Thoracic; Carotid Arteries; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Male; Muscle, Smooth, Vascular; Phenylephrine; Potassium Chloride; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vasoconstrictor Agents | 1998 |
Modulation of basal intracellular calcium by inverse agonists and phorbol myristate acetate in rat-1 fibroblasts stably expressing alpha1d-adrenoceptors.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cell Line; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Endothelin-1; Fibroblasts; Norepinephrine; Phentolamine; Piperazines; Protein Kinase C; Rats; Receptors, Adrenergic, alpha-1; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1999 |
Preconditioning prevents the negative inotropic action of phenylephrine in rat isolated stunned papillary muscle.
Topics: Adrenergic alpha-Antagonists; Animals; Cardiotonic Agents; Clonidine; Dioxanes; Female; Ischemic Preconditioning, Myocardial; Isoproterenol; Male; Muscle Contraction; Papillary Muscles; Phenylephrine; Rats; Rats, Wistar; Reperfusion Injury; Yohimbine | 1999 |
Expression and pharmacological characterization of alpha1-adrenoceptors in rat seminal vesicle.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenoxybenzamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Seminal Vesicles | 1999 |
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured | 1999 |
Differences in the electrophysiologic response of four canine ventricular cell types to alpha 1-adrenergic agonists.
Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Endocardium; Heart Ventricles; In Vitro Techniques; Methoxamine; Microelectrodes; Pericardium; Phenylephrine; Prazosin; Propranolol; Purkinje Fibers | 1999 |
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine | 2000 |
Role of alpha1A-adrenoceptor in the regulation of glucose uptake into white adipocyte of rats in vitro.
Topics: Adipocytes; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkaloids; Animals; Benzophenanthridines; Biological Transport, Active; Chromones; Clonidine; Deoxyglucose; Dioxanes; Enzyme Inhibitors; Estrenes; Glucose; Glucose Transporter Type 4; Indoles; Male; Maleimides; Methoxamine; Monosaccharide Transport Proteins; Morpholines; Muscle Proteins; Phenanthridines; Phosphoinositide-3 Kinase Inhibitors; Prazosin; Protein Kinase C; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Type C Phospholipases | 2000 |
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction | 2001 |
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction | 2001 |
Existence of alpha(1A)- and alpha(1B)-adrenoceptor subtypes in canine mandibular alveolar arteries.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alveolar Process; Animals; Arteries; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Mandible; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction; Xylazine; Yohimbine | 2001 |
Existence of functional alpha1A- and alpha1D- but no alpha1B-adrenoceptor subtypes in rat common carotid arteries.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Methoxamine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vasoconstriction | 2002 |
Adrenergic activation of cardiac phospholipase D: role of alpha(1)-adrenoceptor subtypes.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cardiomegaly; Clonidine; Dioxanes; Male; Myocardium; Norepinephrine; Perfusion; Phospholipase D; Piperazines; Prazosin; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Signal Transduction; Stimulation, Chemical | 2002 |
Effects of castration and of testosterone replacement on alpha(1)-adrenoceptor subtypes in the rat vas deferens.
Topics: Animals; Castration; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Neuronal Plasticity; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Testosterone; Time Factors; Vas Deferens; Yohimbine | 2003 |
Effects of androgen manipulation on alpha1-adrenoceptor subtypes in the rat seminal vesicle.
Topics: Adrenergic alpha-1 Receptor Antagonists; Analysis of Variance; Androgens; Animals; Autoradiography; Barium Compounds; Chlorides; Clonidine; Cyproterone Acetate; Dioxanes; Gene Expression Regulation; Male; Orchiectomy; Organ Size; Phenylephrine; Piperazines; Quinazolines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; RNA, Messenger; Seminal Vesicles; Testosterone | 2004 |
Sympathetic neurotransmission in the rat testicular capsule: functional characterization and identification of mRNA encoding alpha1-adrenoceptor subtypes.
Topics: Acetyl-CoA C-Acyltransferase; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Calcium Channel Blockers; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Male; Muscle Contraction; Nifedipine; Norepinephrine; Prazosin; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Purinergic P2; Reserpine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spiperone; Suramin; Sympathetic Nervous System; Synaptic Transmission; Testis | 2006 |
Molecular and pharmacological characteristics of the gerbil α(1a)-adrenergic receptor.
Topics: Adrenergic alpha-1 Receptor Antagonists; Amino Acid Sequence; Animals; Arteries; Chlorocebus aethiops; Clonidine; Cloning, Molecular; Cochlea; Conserved Sequence; COS Cells; Dioxanes; Dose-Response Relationship, Drug; Gerbillinae; Humans; Mice; Molecular Sequence Data; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Sequence Analysis, Protein; Transfection; Vasoconstriction | 2012 |
Blockade of different subtypes of α(1)-adrenoceptors produces opposite effect on heart chronotropy in newborn rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Animals, Newborn; Clonidine; Dioxanes; Heart Rate; Piperazines; Rats; Receptors, Adrenergic, alpha-1 | 2012 |