chlorethylclonidine has been researched along with 5-methylurapidil in 76 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 52 (68.42) | 18.2507 |
2000's | 22 (28.95) | 29.6817 |
2010's | 2 (2.63) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bondinell, WE; Hieble, JP; Ruffolo, RR | 1 |
Etgen, AM; Karkanias, GB; Petitti, N | 1 |
Kowatch, MA; Miyamoto, A; Roth, GS; Villalobos-Molina, R | 1 |
Esbenshade, TA; Han, C; Minneman, KP | 1 |
Blue, DR; Clarke, DE; Vimont, RL | 1 |
Boer, R; Eltze, M | 1 |
Kojima, C; Satoh, M; Takayanagi, I | 1 |
García-Sáinz, JA; Torres-Márquez, ME; Villalobos-Molina, R | 1 |
Han, CD; Minneman, KP | 1 |
Gross, G; Ravens, U; Wang, XL; Wettwer, E | 1 |
Moriya, M; Takayanagi, I | 1 |
Bell, K; Insel, PA; Klijn, K; Slivka, SR | 1 |
Hashimoto, K; Suzuki, E; Tamura, K; Tsujimoto, G | 1 |
Kow, LM; Pfaff, DW | 1 |
Johns, EJ; Sattar, MA | 2 |
Abdul Sattar, M; Johns, EJ | 1 |
Han, C; Yu, GS | 1 |
Chueh, SC; Guh, JH; Ko, FN; Teng, CM | 1 |
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H | 1 |
Guarneri, L; Leonardi, A; Poggesi, E; Simonazzi, I; Taddei, C; Testa, R | 1 |
Aston, N; Chess-Williams, R; Couldwell, C | 1 |
Guh, JH; Ko, FN; Teng, CM | 1 |
Fleming, WW; Kong, JQ; Taylor, DA | 1 |
Gross, G; Hanft, G; Michel, MC | 1 |
Chen, MZ; Han, QD; Yu, GS | 1 |
Gorman, AJ; Vargas, HM; Zhou, L | 1 |
Lepor, H; Meretyk, S; Shapiro, E; Tang, R | 1 |
Lepor, H; Shapiro, E; Tang, R | 1 |
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T | 1 |
Ballejo, G; Queiroz-Neto, A | 1 |
García-Sáinz, JA; Romero-Avila, MT | 1 |
Chen, L; Eckhart, AD; Faber, JE; Xin, X; Yang, N | 1 |
Docherty, JR; Kearns, S; O'Rourke, M | 1 |
Benoit, JN; Gao, H; Korthuis, RJ | 1 |
Ibarra, M; López-Guerrero, JJ; Terrón, JA; Villalobos-Molina, R | 1 |
Ibarra, M; López-Guerrero, JJ; Villalobos-Molina, R | 2 |
Dougall, IG; Fagura, MS; Lydford, SJ | 1 |
Osnes, JB; Sandnes, D; Skomedal, T; Viko, H | 1 |
Andersen, GO; Enger, M; Osnes, JB; Skomedal, T | 1 |
Arai, M; Fujiwara, H; Fujiwara, T; Kariya, T; Koshiji, M; Minatoguchi, S; Ohno, T; Uno, Y; Yamashita, K | 1 |
Daniel, EE; Gaspar, V; Kwan, CY; Low, AM; Lu-Chao, H | 1 |
Hasegawa, Y; Ono, H; Wada, T | 1 |
Avkiran, M; Yasutake, M; Yokoyama, H | 1 |
Hattori, K; Makara, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Suzuki, M; Tsuchiya, M; Watanabe, K | 1 |
Demenge, P; Godin-Ribuot, D; Joyeux, M; Patel, A; Ribuot, C; Yellon, DM | 1 |
García-Sáinz, JA; Torres-Padilla, ME | 1 |
Li, W; Wang, XL; Zhang, Y | 1 |
Errasti, AE; Rothlin, RP; Sardi, SP; Torres, RM; Velo, MP | 1 |
Amobi, N; Coker, C; Guillebaud, J; Mulvin, D; Smith, IC | 1 |
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM | 1 |
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K | 1 |
Becker, K; Brodde, OE; Dhein, S; Giessler, C; Pönicke, K | 1 |
Coats, P; Hillier, C; Jarajapu, YP; MacDonald, A; McGrath, JC | 1 |
Hillier, C; Jarajapu, YP; MacDonald, A | 1 |
Koike, K; Yamamoto, Y | 1 |
D'Ocon, P; Gisbert, R; Ivorra, MD; Noguera, MA; Ziani, K | 1 |
Brodde, OE; Dhein, S; Giessler, C; Heinroth-Hoffmann, I; Leineweber, K; Seyfarth, T | 1 |
Han, Q; Peng, M; Xue, Z; Zhang, Y | 1 |
Brodde, OE; Dhein, S; Giessler, C; Silber, RE; Wangemann, T | 1 |
Arévalo-León, LE; Gallardo-Ortíz, IA; Urquiza-Marín, H; Villalobos-Molina, R | 1 |
Hillier, C; MacDonald, A; Zacharia, J | 2 |
Eltze, M; Jähnichen, S; Pertz, HH | 1 |
Abdullah, NA; Armenia, A; Helmi, A; Johns, EJ; Munavvar, AS | 1 |
Baber, SR; Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD | 1 |
Ding, X; McCune, DF; Murray, PA; Perez, DM; Sohn, JT | 1 |
Farias-Rodríguez, VM; Gallardo-Ortíz, IA; Gómez-Zamudio, JH; Lázaro-Suárez, ML; Tanoue, A; Tsujimoto, G; Villalobos-Molina, R | 1 |
Abdullah, NA; Johns, EJ; Khan, AH; Sattar, MA | 1 |
Abdullah, NA; Armenia, A; Johns, EJ; Khan, MA; Sattar, MA | 1 |
Abdullah, NA; Johns, EJ; Kazi, RN; Khan, AH; Munavvar, AS | 1 |
Chu, CC; Lin, MT; Shieh, JP; Wang, JJ | 1 |
Bockman, CS; Dang, HK; Gruber, DD; Scofield, MA; Wangemann, P; Witt, KM | 1 |
Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD | 1 |
Abdulla, MH; Abdullah, NA; Ahmad, A; Azam, M; Hashmi, F; Johns, EJ; Khan, SA; Sattar, MA | 1 |
1 review(s) available for chlorethylclonidine and 5-methylurapidil
Article | Year |
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Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1995 |
75 other study(ies) available for chlorethylclonidine and 5-methylurapidil
Article | Year |
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Estradiol selectively regulates alpha 1B-noradrenergic receptors in the hypothalamus and preoptic area.
Topics: Animals; Clonidine; Cyclic AMP; Dioxanes; Estradiol; Female; Hypothalamus; Ovariectomy; Piperazines; Prazosin; Preoptic Area; Rats; Receptors, Adrenergic | 1992 |
Alpha 1-adrenoceptors in parotid cells: age does not alter the ratio of alpha 1A and alpha 1B subtypes.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Calcium; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Inosine Triphosphate; Male; Parotid Gland; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1992 |
Subtypes of alpha 1-adrenoceptors in DDT1 MF-2 and BC3H-1 clonal cell lines.
Topics: Adrenergic alpha-Antagonists; Binding, Competitive; Calcium; Cell Line; Clonidine; Inositol Phosphates; Muscle, Smooth; Norepinephrine; Phenethylamines; Piperazines; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones | 1992 |
Evidence for a noradrenergic innervation to alpha 1A-adrenoceptors in rat kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Calcium Channels; Clonidine; In Vitro Techniques; Kidney; Male; Nitrendipine; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Vasoconstriction | 1992 |
The adrenoceptor agonist, SDZ NVI 085, discriminates between alpha 1A- and alpha 1B-adrenoceptor subtypes in vas deferens, kidney and aorta of the rat.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Clonidine; In Vitro Techniques; Isradipine; Kidney; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Oxazines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Vas Deferens; Vasoconstriction | 1992 |
Pharmacological characterization of contractile responses induced by alpha 1-agonists, norepinephrine and clonidine, by selective antagonists of their subtypes in rabbit thoracic aorta.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rabbits | 1992 |
Alpha 1-adrenoceptor subtypes in aorta (alpha 1A) and liver (alpha 1B).
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Liver; Membranes; Muscle, Smooth, Vascular; Phosphatidylinositols; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha | 1991 |
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor binding sites in rat tissues.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dioxanes; Kinetics; Male; Membranes; Phentolamine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Time Factors | 1991 |
Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect?
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dihydropyridines; Electrophysiology; Heart; Membrane Potentials; Myocardium; Phenylephrine; Piperazines; Propranolol; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1991 |
Alpha 1A-adrenoceptors in rabbit bronchus.
Topics: Adrenergic alpha-Antagonists; Animals; Bronchi; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha | 1991 |
Renal alpha 1-adrenergic receptor subtypes: MDCK-D1 cells, but not rat cortical membranes possess a single population of receptors.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Binding, Competitive; Cell Membrane; Clonidine; Dogs; In Vitro Techniques; Kidney; Kidney Cortex; Kidney Tubules; Phosphatidylcholines; Phosphatidylinositols; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Signal Transduction; Tissue Distribution | 1991 |
Two pharmacologically distinct alpha 1-adrenoceptor subtypes in the contraction of rabbit aorta: each subtype couples with a different Ca2+ signalling mechanism and plays a different physiological role.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Binding Sites; Calcium; Clonidine; Dioxanes; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenethylamines; Phenoxybenzamine; Piperazines; Rabbits; Receptors, Adrenergic, alpha; Signal Transduction; Tetralones; Vasoconstriction | 1990 |
Functional analyses of alpha 1-adrenoceptor subtypes in rat hypothalamic ventromedial nucleus neurons.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Hypothalamus, Middle; In Vitro Techniques; Neurons; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1995 |
Evidence for an alpha 1-adrenoceptor subtype mediating adrenergic vasoconstriction in Wistar normotensive and stroke-prone spontaneously hypertensive rat kidney.
Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Cerebrovascular Disorders; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Renal Circulation; Sympathetic Nervous System; Vasoconstriction | 1994 |
Alpha 1-adrenoceptor subtypes mediating adrenergic vasoconstriction in kidney, one-clip Goldblatt and deoxycorticosterone acetate-salt hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Clonidine; Desoxycorticosterone; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Hypertension, Renovascular; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Vasoconstriction | 1994 |
Role of alpha 1A- and alpha 1B-adrenoceptors in phenylephrine-induced positive inotropic response in isolated rat left atrium.
Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Inositol Phosphates; Male; Myocardial Contraction; Phenethylamines; Phenylephrine; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Tetralones | 1994 |
Characterization of alpha 1-adrenoceptor subtypes in tension response of human prostate to electrical field stimulation.
Topics: Adrenergic Antagonists; Animals; Clonidine; Electric Stimulation; Humans; Hyperplasia; In Vitro Techniques; Isometric Contraction; Male; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens; Yohimbine | 1995 |
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine | 1995 |
Mediation of noradrenaline-induced contractions of rat aorta by the alpha 1B-adrenoceptor subtype.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Computer Simulation; Hippocampus; In Vitro Techniques; Liver; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Regression Analysis; Spiperone; Stereoisomerism; Sulfonamides | 1995 |
Alpha 1A-adrenoceptor subtype mediates contraction of the rat urethra.
Topics: Aminoquinolines; Animals; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetrahydroisoquinolines; Urethra | 1994 |
Functional identification of alpha 1-adrenoceptor subtypes in human prostate: comparison with those in rat vas deferens and spleen.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Animals; Clonidine; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens | 1994 |
Functional distribution and role of alpha-1 adrenoceptor subtypes in the mesenteric vasculature of the rat.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Clonidine; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1994 |
Radioligand binding studies of alpha 1-adrenoceptor subtypes in rat heart.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cadmium; Cadmium Chloride; Calcium; Chlorides; Clonidine; Epinephrine; Heart Ventricles; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1994 |
A new alpha 1-adrenergic receptor subtype with low affinity for 5-methyl-urapidil but insensitive to chlorethylclonidine.
Topics: Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Clonidine; Dioxanes; Male; Myocardium; Phenethylamines; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetralones | 1993 |
Role of vascular alpha-1 adrenoceptor subtypes in the pressor response to sympathetic nerve stimulation in the pithed rat.
Topics: Animals; Blood Pressure; Blood Vessels; Clonidine; Decerebrate State; Dioxanes; Electric Stimulation; Idazoxan; Male; Nifedipine; Piperazines; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Sympathetic Nervous System | 1994 |
Alpha 1 adrenoceptor subtypes in the human prostate.
Topics: Adrenergic alpha-Antagonists; Aged; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Male; Middle Aged; Phenethylamines; Piperazines; Prostate; Receptors, Adrenergic, alpha; Tetralones | 1993 |
The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylephrine; Piperazines; Prostate; Receptors, Adrenergic, alpha | 1993 |
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine | 1993 |
Alpha 1-adrenoceptor subtypes mediating the norepinephrine-induced contractile response in the rat vas deferens.
Topics: Adrenergic alpha-1 Receptor Antagonists; Alkylating Agents; Animals; Clonidine; Epididymis; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperazines; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Ryanodine; Vas Deferens | 1993 |
Characterization of the alpha 1A-adrenoceptors of guinea pig liver membranes: studies using 5-[3H]methylurapidil.
Topics: Alkylating Agents; Animals; Binding, Competitive; Clonidine; Guinea Pigs; In Vitro Techniques; Liver; Male; Piperazines; Radioligand Assay; Receptors, Adrenergic, alpha | 1993 |
Regulation of vascular smooth muscle growth by alpha 1-adrenoreceptor subtypes in vitro and in situ.
Topics: Actins; Adrenergic alpha-Antagonists; Animals; Aorta; Cell Division; Cells, Cultured; Clonidine; In Vitro Techniques; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; RNA, Messenger; Venae Cavae | 1995 |
Investigation of the actions of chloroethylclonidine in rat aorta.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine | 1995 |
alpha1-Adrenoceptor subtypes mediating antinatriuresis in Wistar and stroke-prone spontaneously hypertensive rats.
Topics: Animals; Clonidine; Diuresis; Hypertension; Male; Natriuresis; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1995 |
Hypoxia/reoxygenation selectively impairs alpha 1b-adrenoceptor function in small mesenteric arteries.
Topics: Adrenergic alpha-Antagonists; Aerobiosis; Animals; Catalase; Clonidine; Dioxanes; Hypoxia; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Yohimbine | 1996 |
Evidence for an age-dependent functional expression of alpha 1D-adrenoceptors in the rat vasculature.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Blood Pressure; Blood Vessels; Clonidine; Male; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1997 |
Alpha 1D- and alpha 1A-adrenoceptors mediate contraction in rat renal artery.
Topics: Animals; Clonidine; Male; Muscle Contraction; Norepinephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Renal Artery | 1997 |
Pharmacological classification of alpha 1-adrenoceptors mediating contractions of rabbit isolated ear artery: comparison with rat isolated thoracic aorta.
Topics: Animals; Aorta, Thoracic; Clonidine; Dose-Response Relationship, Drug; Ear; In Vitro Techniques; Male; Piperazines; Rabbits; Rats; Receptors, Adrenergic, alpha-1; Vasoconstriction | 1997 |
Alpha 1-adrenoceptor subtypes involved in increased 86Rb+ influx rate and inositol 1,4,5-trisphosphate mass in adult rat cardiomyocytes.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Clonidine; Dioxanes; Heart Ventricles; Inositol 1,4,5-Trisphosphate; Myocardium; Piperazines; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Rubidium Radioisotopes | 1997 |
Alpha 1-adrenoceptor mediated activation of Na/K/2Cl cotransport and K+ channels in the rat heart involves different receptor subtypes.
Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Bumetanide; Carrier Proteins; Chlorides; Clonidine; Heart; In Vitro Techniques; Male; Myocardium; Phenylephrine; Piperazines; Potassium; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sodium; Sodium-Potassium-Chloride Symporters | 1997 |
Infarct size-reducing effect of ischemic preconditioning is related to alpha1b-adrenoceptors but not to alpha1a-adrenoceptors in rabbits.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Ischemic Preconditioning, Myocardial; Male; Phenoxybenzamine; Piperazines; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1 | 1997 |
Characterization of alpha-adrenoceptors in canine mesenteric vein.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dogs; Female; Male; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Yohimbine | 1997 |
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord | 1997 |
Alpha1-adrenergic stimulation of sarcolemmal Na+-H+ exchanger activity in rat ventricular myocytes: evidence for selective mediation by the alpha1A-adrenoceptor subtype.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cattle; Clonidine; Dioxanes; Heart Ventricles; Humans; Imidazoles; Kinetics; Myocardium; Phenylephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sarcolemma; Sodium-Hydrogen Exchangers; Tetrahydronaphthalenes | 1998 |
Discrimination of alpha1-adrenoceptor subtypes in rat aorta and prostate.
Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vasoconstriction; Vasodilator Agents | 1998 |
Infarct size-reducing effect of heat stress and alpha1 adrenoceptors in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Heat Stress Disorders; Heat-Shock Proteins; HSP72 Heat-Shock Proteins; Infarction; Male; Myocardial Ischemia; Organ Culture Techniques; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reperfusion Injury | 1998 |
Modulation of basal intracellular calcium by inverse agonists and phorbol myristate acetate in rat-1 fibroblasts stably expressing alpha1d-adrenoceptors.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cell Line; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Endothelin-1; Fibroblasts; Norepinephrine; Phentolamine; Piperazines; Protein Kinase C; Rats; Receptors, Adrenergic, alpha-1; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1999 |
Altered alpha 1-adrenoceptor subtypes mediated cardiac function after treatment of propranolol to rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Clonidine; Heart Rate; Male; Myocardial Contraction; Phenylephrine; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Stimulation, Chemical | 1997 |
Characterization of alpha1-adrenoceptor subtypes mediating vasoconstriction in human umbilical vein.
Topics: Adrenergic Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Humans; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Umbilical Veins; Vasoconstriction; Vasoconstrictor Agents | 1999 |
Functional characterization of alpha1-adrenoceptor subtypes in longitudinal and circular muscle of human vas deferens.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Alkylating Agents; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Piperazines; Prazosin; Receptors, Adrenergic; Spiperone; Vas Deferens | 1999 |
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured | 1999 |
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine | 2000 |
Inositolphosphate formation in thoracic and abdominal rat aorta following Gq/11-coupled receptor stimulation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Abdominal; Aorta, Thoracic; Clonidine; Endothelin Receptor Antagonists; Endothelin-1; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; In Vitro Techniques; Inositol Phosphates; Male; Muscle Contraction; Norepinephrine; Peptides, Cyclic; Piperazines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptors, Adrenergic, alpha; Receptors, Endothelin; Receptors, Thromboxane; Vasoconstrictor Agents | 2001 |
Functional characterization of alpha(1)-adrenoceptor subtypes in human skeletal muscle resistance arteries.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Arteries; Clonidine; Dose-Response Relationship, Drug; Humans; Imidazoles; In Vitro Techniques; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vasoconstriction | 2001 |
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction | 2001 |
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction | 2001 |
Modulatory role of a constitutively active population of alpha(1D)-adrenoceptors in conductance arteries.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Arteries; Calcium; Clonidine; Dose-Response Relationship, Drug; Female; Iliac Artery; Mesenteric Arteries; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance | 2002 |
Changes in alpha(1)-adrenergic vascular reactivity in monocrotaline-treated rats.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Hypertension, Pulmonary; Hypertrophy, Right Ventricular; In Vitro Techniques; Male; Mesenteric Arteries; Monocrotaline; Norepinephrine; Piperazines; Pulmonary Artery; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Thoracic Arteries; Vasoconstriction | 2002 |
[Alpha1-adrenoceptor subtypes in rabbit penile corpus cavernosum].
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Male; Norepinephrine; Penile Erection; Penis; Piperazines; Protein Isoforms; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha-1 | 1998 |
Noradrenaline-induced contraction of human saphenous vein and human internal mammary artery: involvement of different alpha-adrenoceptor subtypes.
Topics: Adrenergic alpha-Antagonists; Aged; Clonidine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Mammary Arteries; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Regression Analysis; Saphenous Vein; Yohimbine | 2002 |
Evidence for the role of alpha1D- and alpha1A-adrenoceptors in contraction of the rat mesenteric artery.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxymetazoline; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 2003 |
Alpha1-adrenoceptor subtypes involved in vasoconstrictor responses to exogenous and neurally released noradrenaline in rat femoral resistance arteries.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cocaine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents | 2004 |
Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Arteries; Clonidine; Dioxins; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Pyrimidinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tail | 2004 |
The contribution of adrenoceptor subtype(s) in the renal vasculature of diabetic spontaneously hypertensive rats.
Topics: Animals; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Electric Stimulation; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intravenous; Kidney; Kidney Cortex; Malaysia; Male; Methoxamine; Muscle, Smooth, Vascular; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-1; Streptozocin; Time Factors; Vasoconstriction | 2004 |
Pharmacological characterization of alpha1-adrenoceptors in mouse isolated femoral small arteries.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents | 2004 |
Effects of norepinephrine on alpha-subtype receptors in the feline pulmonary vascular bed.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Angiotensin II; Animals; Cats; Clonidine; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation, Preclinical; Ephedrine; Female; Injections, Intra-Arterial; Injections, Intravenous; Male; Norepinephrine; Phenylephrine; Piperazines; Pulmonary Artery; Pulmonary Circulation; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstrictor Agents | 2004 |
Postjunctional alpha1-adrenoceptors in the vasculature of the pithed mouse are of the alpha1A-subtype.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Carotid Arteries; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Drug Synergism; Heart Rate; Male; Mice; Models, Animal; Norepinephrine; Piperazines; Receptors, Adrenergic, alpha-1; Vagotomy; Vasoconstrictor Agents | 2005 |
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction.
Topics: Anesthetics, Intravenous; Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Fentanyl; Hydrogen-Ion Concentration; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Receptors, Adrenergic, alpha-1; Vasoconstriction | 2005 |
Chloroethylclonidine reveals that alpha (1 A)-adrenoceptors mediate contraction in aorta of alpha (1 D)-adrenoceptor knockout mice.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dose-Response Relationship, Drug; Imines; In Vitro Techniques; Mice; Mice, Knockout; Norepinephrine; Piperazines; Piperidines; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents | 2005 |
Influence of cisplatin-induced renal failure on the alpha(1)-adrenoceptor subtype causing vasoconstriction in the kidney of the rat.
Topics: Amlodipine; Animals; Cisplatin; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Injections, Intraperitoneal; Kidney; Male; Methoxamine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Renal Insufficiency; Vasoconstriction; Vasodilator Agents | 2007 |
Functional subtypes of renal alpha1-adrenoceptor in diabetic and non-diabetic 2K1C Goldblatt renovascular hypertension.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Clonidine; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension, Renovascular; Kidney; Male; Methoxamine; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Vasoconstriction | 2008 |
Influence of high dietary sodium intake on the functional subtypes of alpha-adrenoceptors in the renal cortical vasculature of Wistar-Kyoto rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Body Weight; Clonidine; Drinking; Hydroxylamines; Kidney Cortex; Male; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Sodium; Sodium, Dietary; Urine; Vasoconstriction; Vasoconstrictor Agents | 2009 |
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Anesthesia, Local; Anesthetics, Local; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Methoxamine; Nifedipine; Nitroglycerin; Pain Measurement; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 2009 |
Molecular and pharmacological characteristics of the gerbil α(1a)-adrenergic receptor.
Topics: Adrenergic alpha-1 Receptor Antagonists; Amino Acid Sequence; Animals; Arteries; Chlorocebus aethiops; Clonidine; Cloning, Molecular; Cochlea; Conserved Sequence; COS Cells; Dioxanes; Dose-Response Relationship, Drug; Gerbillinae; Humans; Mice; Molecular Sequence Data; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Sequence Analysis, Protein; Transfection; Vasoconstriction | 2012 |
Ma huang and alpha subtype adrenoceptors in the cat pulmonary vascular bed.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Ephedra sinica; Female; Lung; Male; Phentolamine; Piperazines; Prazosin; Prospective Studies; Pulmonary Circulation; Receptors, Adrenergic; Vasoconstrictor Agents | 2008 |
Cystathione gamma lyase/Hydrogen Sulphide Pathway Up Regulation Enhances the Responsiveness of α1A and α1B-Adrenoreceptors in the Kidney of Rats with Left Ventricular Hypertrophy.
Topics: Adrenergic beta-Antagonists; Animals; Clonidine; Cystathionine gamma-Lyase; Hydrogen Sulfide; Hypertrophy, Left Ventricular; Kidney; Male; Nitric Oxide; Nitric Oxide Synthase Type III; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Renal Circulation; Sulfurtransferases; Up-Regulation | 2016 |