chlordiazepoxide and cimetidine

chlordiazepoxide has been researched along with cimetidine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199012 (54.55)18.7374
1990's0 (0.00)18.2507
2000's4 (18.18)29.6817
2010's6 (27.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Barclay, AM1
Bergman, J; Spealman, RD1
Kurowski, M; Reim, HG1
D'Arcy, PF1
Bleger, G1
Chojnacki, J; Grzegorczyk, K; Klupińska, G; Michowicz, A; Tkaczewski, W1
Jenike, MA1
Johnson, RF; Patwardhan, RV; Schenker, S; Sinclair, AP; Speeg, KV1
File, SE; Pearce, JB1
Babb, RR1
Desmond, PV; Patwardhan, RV; Schenker, S; Speeg, KV1

Reviews

2 review(s) available for chlordiazepoxide and cimetidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Cimetidine in elderly patients: review of uses and risks.
    Journal of the American Geriatrics Society, 1982, Volume: 30, Issue:3

    Topics: Administration, Oral; Aged; Antacids; Chemical Phenomena; Chemistry; Chlordiazepoxide; Cimetidine; Diazepam; Drug Interactions; Duodenal Ulcer; Female; Gastric Acid; Guanidines; Humans; Mental Disorders; Middle Aged; Peptic Ulcer; Phenytoin; Zollinger-Ellison Syndrome

1982

Trials

1 trial(s) available for chlordiazepoxide and cimetidine

ArticleYear
[Metabolic interaction between cimetidine, ranitidine and amitriptyline/chlordiazepoxide].
    Zeitschrift fur Gastroenterologie, 1986, Volume: 24, Issue:10

    Topics: Adult; Amitriptyline; Biotransformation; Chlordiazepoxide; Cimetidine; Drug Combinations; Gastric Acidity Determination; Half-Life; Humans; Male; Metabolic Clearance Rate; Ranitidine

1986

Other Studies

19 other study(ies) available for chlordiazepoxide and cimetidine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Psychotropic drugs in the elderly. Selection of the appropriate agent.
    Postgraduate medicine, 1985, Volume: 77, Issue:8

    Topics: Age Factors; Aged; Antidepressive Agents; Antipsychotic Agents; Benzodiazepines; Chlordiazepoxide; Cimetidine; Diazepam; Flurazepam; Haloperidol; Humans; Kinetics; Lithium; Phenothiazines; Physostigmine; Psychotropic Drugs; Thiothixene; Trazodone

1985
Some behavioral effects of histamine H1 antagonists in squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:1

    Topics: Animals; Behavior, Animal; Chlordiazepoxide; Chlorpheniramine; Cimetidine; Clozapine; Cocaine; Conditioning, Operant; Dextroamphetamine; Diphenhydramine; Electroshock; Feeding Behavior; Histamine H1 Antagonists; Male; Promethazine; Saimiri; Self Administration; Tripelennamine

1986
Early reports on drug interactions.
    Drug intelligence & clinical pharmacy, 1983, Volume: 17, Issue:2

    Topics: Acetaminophen; Amiodarone; Apazone; Aspirin; Carbamazepine; Chlordiazepoxide; Cimetidine; Coumarins; Drug Interactions; Erythromycin; Ethanol; Furosemide; Gentamicins; Humans; Levodopa; Lidocaine; Phenytoin; Prenylamine; Quinidine

1983
[Long term medical treatment of ulcer excluding acute attacks].
    Medecine & chirurgie digestives, 1980, Volume: 9, Issue:5

    Topics: Chlordiazepoxide; Cimetidine; Drug Combinations; Duodenal Ulcer; Guanidines; Humans; Quinuclidines; Stomach Ulcer

1980
[Prevention of duodenal ulcer recurrences after treatment with cimetidine preparations].
    Wiadomosci lekarskie (Warsaw, Poland : 1960), 1982, Jun-01, Volume: 35, Issue:6

    Topics: Adolescent; Adult; Chlordiazepoxide; Cimetidine; Double-Blind Method; Doxepin; Drug Combinations; Duodenal Ulcer; Guanidines; Humans; Middle Aged; Quinuclidines; Recurrence

1982
Lack of tolerance and rapid recovery of cimetidine-inhibited chlordiazepoxide (Librium) elimination.
    Gastroenterology, 1981, Volume: 81, Issue:3

    Topics: Adult; Chlordiazepoxide; Cimetidine; Female; Guanidines; Humans; Kinetics; Male

1981
Benzodiazepines reduce gastric ulcers induced in rats by stress.
    British journal of pharmacology, 1981, Volume: 74, Issue:3

    Topics: Animals; Atropine; Benzodiazepines; Chlordiazepoxide; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Hypnotics and Sedatives; In Vitro Techniques; Lorazepam; Male; Rats; Rats, Inbred Strains; Stomach Ulcer; Stress, Physiological

1981
Drug interactions with cimetidine.
    Postgraduate medicine, 1981, Volume: 70, Issue:5

    Topics: Chlordiazepoxide; Cimetidine; Diazepam; Drug Interactions; Guanidines; Humans; Phenytoin; Propranolol; Theophylline; Warfarin

1981
Cimetidine impairs elimination of chlordiazepoxide (Librium) in man.
    Annals of internal medicine, 1980, Volume: 93, Issue:2

    Topics: Adult; Chlordiazepoxide; Cimetidine; Drug Interactions; Female; Guanidines; Half-Life; Humans; Liver; Male

1980