Page last updated: 2024-08-17

chloramphenicol and fluconazole

chloramphenicol has been researched along with fluconazole in 59 studies

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's19 (32.20)29.6817
2010's39 (66.10)24.3611
2020's1 (1.69)2.80

Authors

AuthorsStudies
Duffy, EM; Jorgensen, WL1
Topliss, JG; Yoshida, F1
Abraham, MH; Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Chang, TK; Ensom, MH; Kiang, TK1
Bhadauria, D; Dubey, R; Halve, AK1
Liu, T; Lv, J; Wang, Y; Yin, L1
Bondock, S; Fadda, AA; Khalifa, W1
Carle, AO; Curti, C; Gellis, A; Laget, M; Vanelle, P1
Liu, T; Lv, J; Wang, Y1
Bondock, S; Etman, HA; Fadda, AA; Rabie, R1
Lombardo, F; Obach, RS; Waters, NJ1
Alimuddin, M; Bulloch, D; Dahl, R; Grant, D; Lee, N; Peacock, M1
Bhatia, RK; Gupta, V; Ishar, MP; Raj, T; Sharma, D; Sharma, RK1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Bondock, S; Fadaly, W; Metwally, MA1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Ahmad, A; Banday, MR; Farshori, NN; Khan, AU; Rauf, A1
Gan, LL; Zhang, FF; Zhou, CH1
Fang, B; Rao, XC; Zhou, CH1
Wan, K; Wang, XL; Zhou, CH1
Ghosh, I; Manoharlal, R; Prakash, O; Prasad, R; Puri, N; Sharma, M1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Shi, Y; Zhou, CH1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Zhang, YY; Zhou, CH1
Camps, I; Coelho, LF; D' Dego, JL; Dias, AL; Dias, KS; dos Santos, MH; Januário, JP; Viegas, C1
Barad, HA; Gupta, VK; Kant, R; Pansuriya, BR; Parmar, NJ; Teraiya, SB1
Barad, HA; Gupta, VK; Kant, R; Pansuriya, BR; Parmar, NJ1
Damu, GL; Geng, RX; Zhang, L; Zhang, SL; Zhou, CH1
Damu, GL; Geng, RX; Lv, JS; Wang, Y; Yang, DC; Zhou, CH1
Cui, SF; Damu, GL; Geng, RX; Peng, XM; Ren, Y; Zhang, SL; Zhou, CH1
Cai, GX; Damu, GL; Zhang, HZ; Zhou, CH1
Bhadraiah, UK; Javarasetty, C; Keshavamurthy, S; Ningaiah, S1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Geng, RX; Peng, XM; Rasheed, S; Yan, CY; Yin, BT; Zhang, SL; Zhou, CH1
Kishore, B; Lv, JS; Peng, XM; Zhou, CH1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Avula, SR; Jeyakkumar, P; Zhang, L; Zhou, CH1
Addla, D; Avula, SR; Cheng, Y; Gao, WW; Lin, JM; Tangadanchu, VKR; Zhang, L; Zhou, CH1
Cheng, Y; Geng, RX; Gopala, L; Jeyakkumar, P; Liu, HB; Peng, XM; Zhou, CH1
Gan, LL; Gopala, L; He, SC; Peng, YJ; Tangadanchu, VKR; Zhang, HJ; Zhang, HZ; Zhou, CH1
Bheemanaboina, RRY; Kannekanti, VK; Li, ZZ; Maddili, SK; Tangadanchu, VKR; Tuniki, B; Zhou, CH1
Zhang, B1
Blanchet, M; Bourguet-Kondracki, ML; Brunel, JM; Cadelis, MM; Copp, BR; Li, SA; Sue, K; Vidal, N1
Ba, Y; Hou, X; Wang, S; Xu, Z; Yang, H; Zhang, J1
Blanchet, M; Bourguet-Kondracki, ML; Brunel, JM; Cadelis, MM; Copp, BR; Kang, W; Pike, EIW; Vidal, N; Wu, Z1
Gao, F; Huang, G; Xiao, J1
Beteck, RM; Jesumoroti, OJ; Legoabe, LJ; Patel, OPS1
Goel, SL; Kumar, A; Saxena, KK; Singh, T; Srivastava, VK1
Geng, RX; Ji, QG; Shi, Y; Zhou, CH; Zhou, XD1
Devi, LS; Joshi, SR1
Al-Hakami, AM; Assiry, AM; Assiry, MM; Hamid, ME; Jamil, AS; Joseph, MR; Shaker, MA1
Baptista, P; de Pinho, PG; Malhadas, C; Malheiro, R; Pereira, JA1
Aboubakar, T; Bellet, V; Bertout, S; Delaporte, E; Doumbia, A; Drakulovski, P; Kassi, FK; Kouakou, GA; Krasteva, D; Menan, HIE; Reynes, J; Roger, F; Valérie, BA; Yavo, W1

Reviews

6 review(s) available for chloramphenicol and fluconazole

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Comprehensive review on the anti-bacterial activity of 1,2,3-triazole hybrids.
    European journal of medicinal chemistry, 2019, Apr-15, Volume: 168

    Topics: Anti-Bacterial Agents; Bacteria; Bacterial Infections; Dose-Response Relationship, Drug; Humans; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Triazoles

2019
Nitroimidazole-containing compounds and their antibacterial and antitubercular activities.
    European journal of medicinal chemistry, 2019, Oct-01, Volume: 179

    Topics: Anti-Bacterial Agents; Bacterial Infections; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Molecular Structure; Nitroimidazoles

2019
Current scenario of tetrazole hybrids for antibacterial activity.
    European journal of medicinal chemistry, 2019, Dec-15, Volume: 184

    Topics: Anti-Bacterial Agents; Bacteria; Dose-Response Relationship, Drug; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Tetrazoles

2019
Metronidazole-conjugates: A comprehensive review of recent developments towards synthesis and medicinal perspective.
    European journal of medicinal chemistry, 2021, Jan-15, Volume: 210

    Topics: Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Antiprotozoal Agents; Drug Development; Humans; Hypoglycemic Agents; Metronidazole

2021

Other Studies

53 other study(ies) available for chloramphenicol and fluconazole

ArticleYear
Prediction of drug solubility from Monte Carlo simulations.
    Bioorganic & medicinal chemistry letters, 2000, Jun-05, Volume: 10, Issue:11

    Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogPoct: a tool for lipophilicity determination in drug discovery.
    Journal of medicinal chemistry, 2000, Jul-27, Volume: 43, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Solvents

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
N/C-4 substituted azetidin-2-ones: synthesis and preliminary evaluation as new class of antimicrobial agents.
    Bioorganic & medicinal chemistry letters, 2007, Jan-15, Volume: 17, Issue:2

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Azetidines; Bacteria; Cyclization; Drug Design; Drug Evaluation, Preclinical; Fungi; Indicators and Reagents; Microbial Sensitivity Tests; Structure-Activity Relationship

2007
Synthesis of pseudopeptides based L-tryptophan as a potential antimicrobial agent.
    Bioorganic & medicinal chemistry letters, 2007, Mar-15, Volume: 17, Issue:6

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Bacteria; Fungi; Hemolysis; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Peptides; Spectrometry, Mass, Electrospray Ionization; Spectrophotometry, Infrared; Tryptophan

2007
Synthesis and antimicrobial evaluation of some new thiazole, thiazolidinone and thiazoline derivatives starting from 1-chloro-3,4-dihydronaphthalene-2-carboxaldehyde.
    European journal of medicinal chemistry, 2007, Volume: 42, Issue:7

    Topics: Aldehydes; Anti-Bacterial Agents; Antifungal Agents; Bacteria; Dose-Response Relationship, Drug; Fungi; Molecular Structure; Naphthalenes; Thiazoles

2007
Rapid synthesis of sulfone derivatives as potential anti-infectious agents.
    European journal of medicinal chemistry, 2007, Volume: 42, Issue:6

    Topics: Anti-Infective Agents; Bacteria; Fungi; Microbial Sensitivity Tests; Molecular Structure; Sulfones

2007
Synthesis, structure and biological activity of pseudopeptidic macrolides based on an amino alcohol.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:1

    Topics: Amino Alcohols; Anti-Infective Agents; Crystallography, X-Ray; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Hemolysis; Macrolides; Microbial Sensitivity Tests; Structure-Activity Relationship

2008
Synthesis and antimicrobial activity of some new heterocycles incorporating antipyrine moiety.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:10

    Topics: Anti-Infective Agents; Antipyrine; Bacteria; Drug Design; Fungi; Heterocyclic Compounds; Nitriles

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Determination of log D via automated microfluidic liquid-liquid extraction.
    Journal of medicinal chemistry, 2008, Aug-28, Volume: 51, Issue:16

    Topics: Automation; Biopharmaceutics; Microfluidic Analytical Techniques; Pharmacokinetics

2008
Mechanism of unusual formation of 3-(5-phenyl-3H-[1,2,4]dithiazol-3-yl)chromen-4-ones and 4-oxo-4H-chromene-3-carbothioic acid N-phenylamides and their antimicrobial evaluation.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:8

    Topics: Amides; Anti-Infective Agents; Bacteria; Chromones; Crystallography, X-Ray; Fungi; Microbial Sensitivity Tests; Spectrum Analysis; Structure-Activity Relationship

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Enaminonitrile in heterocyclic synthesis: synthesis and antimicrobial evaluation of some new pyrazole, isoxazole and pyrimidine derivatives incorporating a benzothiazole moiety.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:12

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzothiazoles; Botrytis; Drug Design; Fusarium; Heterocyclic Compounds; Heterocyclic Compounds, 2-Ring; Isoxazoles; Microbial Sensitivity Tests; Molecular Structure; Nitriles; Pyrazoles; Pyrimidines

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Synthesis and characterization of novel fatty acid analogs of cholesterol: in vitro antimicrobial activity.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:4

    Topics: Cholesterol; Fatty Acids; Gram-Negative Bacteria; Gram-Positive Bacteria; Magnetic Resonance Spectroscopy; Mass Spectrometry; Microbial Sensitivity Tests

2010
Synthesis, antibacterial and antifungal activities of some carbazole derivatives.
    Bioorganic & medicinal chemistry letters, 2010, Mar-15, Volume: 20, Issue:6

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aspergillus fumigatus; Bacteria; Candida albicans; Carbazoles; Microbial Sensitivity Tests

2010
Synthesis and biological activities of novel amine-derived bis-azoles as potential antibacterial and antifungal agents.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:9

    Topics: Amines; Anti-Bacterial Agents; Antifungal Agents; Azoles; Bacteria; Fungi; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Structure-Activity Relationship

2010
Synthesis of novel sulfanilamide-derived 1,2,3-triazoles and their evaluation for antibacterial and antifungal activities.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:10

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Bacteria; Bacterial Infections; Fungi; Humans; Magnetic Resonance Spectroscopy; Mycoses; Spectrophotometry, Infrared; Sulfanilamide; Sulfanilamides; Triazoles

2010
Analysis of physico-chemical properties of substrates of ABC and MFS multidrug transporters of pathogenic Candida albicans.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Candida albicans; Membrane Transport Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Substrate Specificity

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Synthesis and evaluation of a class of new coumarin triazole derivatives as potential antimicrobial agents.
    Bioorganic & medicinal chemistry letters, 2011, Feb-01, Volume: 21, Issue:3

    Topics: Anti-Infective Agents; Coumarins; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Triazoles

2011
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Synthesis and activities of naphthalimide azoles as a new type of antibacterial and antifungal agents.
    Bioorganic & medicinal chemistry letters, 2011, Jul-15, Volume: 21, Issue:14

    Topics: Anti-Bacterial Agents; Antifungal Agents; Azoles; Microbial Sensitivity Tests; Naphthalimides

2011
Semisynthesis and antimicrobial activity of novel guttiferone-A derivatives.
    Bioorganic & medicinal chemistry, 2012, Apr-15, Volume: 20, Issue:8

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzophenones; Cell Survival; Dose-Response Relationship, Drug; Fungi; Humans; Leukocytes, Mononuclear; Microbial Sensitivity Tests; Molecular Conformation; Stereoisomerism; Structure-Activity Relationship

2012
An efficient one-pot synthesis, structure, antimicrobial and antioxidant investigations of some novel quinolyldibenzo[b,e][1,4]diazepinones.
    Bioorganic & medicinal chemistry letters, 2012, Jun-01, Volume: 22, Issue:11

    Topics: Anti-Infective Agents; Antioxidants; Azepines; Crystallography, X-Ray; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Conformation; Quinolines

2012
An improved microwave assisted one-pot synthesis, and biological investigations of some novel aryldiazenyl chromeno fused pyrrolidines.
    Bioorganic & medicinal chemistry letters, 2012, Jun-15, Volume: 22, Issue:12

    Topics: Antifungal Agents; Antitubercular Agents; Aspergillus fumigatus; Azo Compounds; Benzopyrans; Candida albicans; Crystallography, X-Ray; Gram-Negative Bacteria; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Microwaves; Molecular Structure; Mycobacterium tuberculosis; Pyrrolidines; Stereoisomerism; Thiosemicarbazones

2012
Synthesis and biological evaluation of novel benzimidazole derivatives and their binding behavior with bovine serum albumin.
    European journal of medicinal chemistry, 2012, Volume: 55

    Topics: Animals; Anti-Infective Agents; Bacteria; Benzimidazoles; Cattle; Chemistry Techniques, Synthetic; Fungi; Microbial Sensitivity Tests; Serum Albumin, Bovine; Thermodynamics

2012
Design, synthesis and evaluation of clinafloxacin triazole hybrids as a new type of antibacterial and antifungal agents.
    Bioorganic & medicinal chemistry letters, 2012, Sep-01, Volume: 22, Issue:17

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacterial Infections; Drug Design; Fluoroquinolones; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Mycoses; Staphylococcal Infections; Triazoles

2012
Synthesis and biological evaluation of a class of quinolone triazoles as potential antimicrobial agents and their interactions with calf thymus DNA.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Anti-Infective Agents; Bacteria; Cattle; DNA; DNA Replication; Drug Evaluation, Preclinical; Fungi; Intercalating Agents; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Quinolones; Spectrophotometry, Ultraviolet; Triazoles

2013
Design, synthesis and antimicrobial evaluation of novel benzimidazole type of Fluconazole analogues and their synergistic effects with Chloromycin, Norfloxacin and Fluconazole.
    European journal of medicinal chemistry, 2013, Volume: 64

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzimidazoles; Dose-Response Relationship, Drug; Drug Design; Drug Synergism; Fluconazole; Fungi; Microbial Sensitivity Tests; Norfloxacin; Structure-Activity Relationship

2013
Novel pyrazoline amidoxime and their 1,2,4-oxadiazole analogues: synthesis and pharmacological screening.
    Bioorganic & medicinal chemistry letters, 2013, Aug-15, Volume: 23, Issue:16

    Topics: Amides; Anti-Infective Agents; Anti-Inflammatory Agents; Antioxidants; Bacteria; Biological Assay; Drug Evaluation, Preclinical; Fatty Acids; Fungi; Molecular Structure; Oxadiazoles; Oximes; Pyrazoles

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Synthesis and biological evaluation of α-triazolyl chalcones as a new type of potential antimicrobial agents and their interaction with calf thymus DNA and human serum albumin.
    European journal of medicinal chemistry, 2014, Volume: 71

    Topics: Animals; Anti-Infective Agents; Bacteria; Bacterial Infections; Cattle; Chalcones; DNA; Fungi; Humans; Microbial Sensitivity Tests; Mycoses; Serum Albumin; Triazoles

2014
1,2,3-Triazole-derived naphthalimides as a novel type of potential antimicrobial agents: synthesis, antimicrobial activity, interaction with calf thymus DNA and human serum albumin.
    Bioorganic & medicinal chemistry letters, 2014, Jan-01, Volume: 24, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Bacteria; Cattle; DNA; DNA Replication; Dose-Response Relationship, Drug; Humans; Microbial Sensitivity Tests; Molecular Structure; Naphthalimides; Serum Albumin; Static Electricity; Structure-Activity Relationship; Triazoles

2014
Design, synthesis and biological evaluation of berberine-benzimidazole hybrids as new type of potentially DNA-targeting antimicrobial agents.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: Animals; Anti-Infective Agents; Bacteria; Benzimidazoles; Berberine; Cattle; Cell Membrane Permeability; Chemistry Techniques, Synthetic; DNA; Drug Design; Fungi; Humans; Microbial Sensitivity Tests; Molecular Docking Simulation; Protein Conformation; Serum Albumin; Water

2016
Multi-targeting exploration of new 2-aminothiazolyl quinolones: Synthesis, antimicrobial evaluation, interaction with DNA, combination with topoisomerase IV and penetrability into cells.
    European journal of medicinal chemistry, 2016, Nov-29, Volume: 124

    Topics: Animals; Anti-Infective Agents; Biological Transport; Cattle; Cell Line; Cell Membrane Permeability; Chemistry Techniques, Synthetic; DNA; DNA Replication; DNA Topoisomerase IV; Drug Design; Kinetics; Mice; Microbial Sensitivity Tests; Molecular Docking Simulation; Permeability; Quinolones

2016
Novel benzimidazolyl tetrahydroprotoberberines: Design, synthesis, antimicrobial evaluation and multi-targeting exploration.
    Bioorganic & medicinal chemistry letters, 2017, 04-15, Volume: 27, Issue:8

    Topics: Animals; Anti-Infective Agents; Bacteria; Bacterial Infections; Benzimidazoles; Berberine Alkaloids; Cattle; DNA; Fungi; Humans; Microbial Sensitivity Tests; Molecular Docking Simulation; Mycoses

2017
Design, synthesis and antimicrobial evaluation of novel benzimidazole-incorporated sulfonamide analogues.
    European journal of medicinal chemistry, 2017, Aug-18, Volume: 136

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Benzimidazoles; Cattle; DNA; Dose-Response Relationship, Drug; Drug Design; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Molecular Structure; Serum Albumin; Structure-Activity Relationship; Sulfonamides

2017
Azoalkyl ether imidazo[2,1-b]benzothiazoles as potentially antimicrobial agents with novel structural skeleton.
    Bioorganic & medicinal chemistry letters, 2018, 08-01, Volume: 28, Issue:14

    Topics: Anti-Bacterial Agents; Antifungal Agents; Benzothiazoles; Dose-Response Relationship, Drug; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Quantum Theory; Structure-Activity Relationship

2018
6-Bromoindolglyoxylamido derivatives as antimicrobial agents and antibiotic enhancers.
    Bioorganic & medicinal chemistry, 2019, 05-15, Volume: 27, Issue:10

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cell Line; Cell Survival; Drug Resistance, Bacterial; Erythrocytes; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Hemolysis; Humans; Indoles; Microbial Sensitivity Tests; Polyamines

2019
Exploration of the antibiotic potentiating activity of indolglyoxylpolyamines.
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Anti-Bacterial Agents; Cell Line; Cell Membrane Permeability; Cell Survival; Cephalosporins; Gram-Negative Bacteria; Hemolysis; Humans; Hydrolysis; Indoles; Microbial Sensitivity Tests; Signal Transduction; Spermine

2019
Synthesis of new thiazolylthiazolidinylbenzothiazoles and thiazolylazetidinylbenzothiazoles as potential insecticidal, antifungal, and antibacterial agents.
    Archiv der Pharmazie, 2006, Volume: 339, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Azetidines; Benzothiazoles; Candida; Chloramphenicol; Escherichia coli; Fluconazole; Insecticides; Molecular Structure; Parathion; Periplaneta; Staphylococcus aureus

2006
[Synthesis and antimicrobial evaluation of coumarin-based benzotriazoles and their synergistic effects with chloromycin and fluconazole].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2011, Volume: 46, Issue:7

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aspergillus fumigatus; Chloramphenicol; Coumarins; Drug Synergism; Fluconazole; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Methicillin-Resistant Staphylococcus aureus; Staphylococcus aureus; Triazoles

2011
Evaluation of the antimicrobial potency of silver nanoparticles biosynthesized by using an endophytic fungus, Cryptosporiopsis ericae PS4.
    Journal of microbiology (Seoul, Korea), 2014, Volume: 52, Issue:8

    Topics: Anti-Bacterial Agents; Antifungal Agents; Candida albicans; Chloramphenicol; Enterococcus faecalis; Escherichia coli; Fluconazole; Fungi; Metal Nanoparticles; Microbial Sensitivity Tests; Microscopy, Electron, Scanning; Microscopy, Electron, Transmission; Salmonella enterica; Silver; Spectrometry, X-Ray Emission; Spectrophotometry; Staphylococcus aureus

2014
In vitro anti-yeast activity of chloramphenicol: A preliminary report.
    Journal de mycologie medicale, 2015, Volume: 25, Issue:1

    Topics: Antifungal Agents; Candida; Caspofungin; Chloramphenicol; Cryptococcus neoformans; Echinocandins; Fluconazole; Humans; Ketoconazole; Lipopeptides; Microbial Sensitivity Tests; Pilot Projects; Saccharomyces cerevisiae

2015
Antimicrobial activity of endophytic fungi from olive tree leaves.
    World journal of microbiology & biotechnology, 2017, Volume: 33, Issue:3

    Topics: Acetates; Alternaria; Chloramphenicol; Endophytes; Fluconazole; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Olea; Penicillium; Pentanols; Phenylethyl Alcohol; Plant Extracts; Plant Leaves; Volatile Organic Compounds; Yeasts

2017
Comparative typing analyses of clinical and environmental strains of the Cryptococcus neoformans/Cryptococcus gattii species complex from Ivory Coast.
    Journal of medical microbiology, 2018, Volume: 67, Issue:1

    Topics: Adult; Amphotericin B; Antifungal Agents; Chloramphenicol; Cote d'Ivoire; Cryptococcosis; Cryptococcus gattii; Cryptococcus neoformans; DNA, Fungal; Environmental Microbiology; Female; Fluconazole; Flucytosine; Genotype; HIV Infections; Humans; Male; Microbial Sensitivity Tests; Middle Aged; Molecular Typing; Mycological Typing Techniques; Prospective Studies; Serotyping; Young Adult

2018