chelerythrine and y 27632

chelerythrine has been researched along with y 27632 in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's9 (52.94)29.6817
2010's8 (47.06)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
Fujita, A; Hata, F; Hirayama, N; Kitayama, M; Kushida, M; Takeuchi, T1
Molenaar, P; Russell, FD1
Kashihara, T; Nakayama, K; Nonogaki, A; Obara, K; Okamoto, Y1
Jarajapu, YP; Knot, HJ1
Ray, PE; Short, BL; Xie, H1
Azuma, YT; Hata, F; Nakajima, H; Takeuchi, T1
Chrones, T; Preiksaitis, HG; Sims, SM1
Díaz, M; Gómez, T; González-Montelongo, MC; Marín, R; Marrero-Alonso, J1
Bailey, SR; Berhane, Y; Elliott, J; Woodcock, H; Zerpa, H1
Enouri, S; Johnson, R; Monteith, G1
Lai, J; Leung, T; Li, SF; Tan, I; Yong, J1
Baik, J; Han, JY; Hong, JM; Kwon, SC; Oh, J; Ok, SH; Sohn, JT1
Khin, PP; Sohn, UD; Zaw, TS1

Other Studies

17 other study(ies) available for chelerythrine and y 27632

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Mechanisms involved in carbachol-induced Ca(2+) sensitization of contractile elements in rat proximal and distal colon.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: ADP Ribose Transferases; Alkaloids; Amides; Animals; Bacterial Toxins; Benzophenanthridines; Botulinum Toxins; Calcium; Carbachol; Cell Membrane Permeability; Colon, Ascending; Colon, Descending; Escin; Guanosine Triphosphate; Hemolysin Proteins; Intracellular Signaling Peptides and Proteins; Japan; Male; Muscle Contraction; Myocytes, Smooth Muscle; Peptide Fragments; Phenanthridines; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Wistar; Receptors, Muscarinic; rho-Associated Kinases; Tritium; Type C Phospholipases

2004
Investigation of signaling pathways that mediate the inotropic effect of urotensin-II in human heart.
    Cardiovascular research, 2004, Sep-01, Volume: 63, Issue:4

    Topics: Alkaloids; Amides; Androstadienes; Benzophenanthridines; Endothelin-1; Humans; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Myocardial Contraction; Myocardium; Myosin-Light-Chain Kinase; Phenanthridines; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Signal Transduction; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Urotensins; Wortmannin

2004
Differential interplay between protein kinase C and Rho-kinase in the endothelin-1-induced and pressure-induced contractions of rat posterior cerebral artery.
    Journal of cardiovascular pharmacology, 2004, Volume: 44 Suppl 1

    Topics: Amides; Animals; Benzophenanthridines; Blood Pressure; Calcium Signaling; Cytosol; Endothelin-1; In Vitro Techniques; Mechanotransduction, Cellular; Posterior Cerebral Artery; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; Rats; rho-Associated Kinases; Vasoconstriction

2004
Relative contribution of Rho kinase and protein kinase C to myogenic tone in rat cerebral arteries in hypertension.
    American journal of physiology. Heart and circulatory physiology, 2005, Volume: 289, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amides; Animals; Benzophenanthridines; Blood Pressure; Calcium; Calcium Signaling; Cerebral Arteries; Enzyme Inhibitors; Hypertension; Indoles; Intracellular Signaling Peptides and Proteins; Maleimides; Muscle Tonus; Muscle, Smooth, Vascular; Phenanthridines; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; rho-Associated Kinases

2005
Rho-kinase contributes to hypoxia/reoxygenation-induced cerebral endothelial dysfunction.
    Journal of cardiovascular pharmacology, 2006, Volume: 48, Issue:1

    Topics: Acetylcholine; Alkaloids; Amides; Animals; Benzophenanthridines; Cerebral Arteries; Endothelium, Vascular; Enzyme Inhibitors; Hypoxia; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxygen; Phenanthridines; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; Superoxides; Triazenes; Vasodilation; Vasodilator Agents

2006
A minor role for Ca2+ sensitization in sustained contraction through activation of muscarinic receptor in circular muscle of rat distal colon.
    Pflugers Archiv : European journal of physiology, 2007, Volume: 454, Issue:4

    Topics: Alkaloids; Amides; Animals; Benzophenanthridines; Calcium; Carbachol; Carcinogens; Cholinergic Agonists; Colon; Dose-Response Relationship, Drug; Guanosine Triphosphate; Male; Muscle Contraction; Muscle Relaxants, Central; Muscle, Smooth; Phorbol 12,13-Dibutyrate; Pyridines; Rats; Rats, Wistar; Receptors, Muscarinic

2007
Calcium sensitization in human esophageal muscle: role for RhoA kinase in maintenance of lower esophageal sphincter tone.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Benzophenanthridines; Calcium; Electric Stimulation; Esophageal Sphincter, Lower; Humans; In Vitro Techniques; Muscle Contraction; Naphthalenes; Protein Kinase C; Pyridines; rhoA GTP-Binding Protein

2008
Androgens induce nongenomic stimulation of colonic contractile activity through induction of calcium sensitization and phosphorylation of LC20 and CPI-17.
    Molecular endocrinology (Baltimore, Md.), 2010, Volume: 24, Issue:5

    Topics: Amides; Androgens; Animals; Benzophenanthridines; Blotting, Western; Calcium; Colon; Cycloheximide; Dactinomycin; Dihydrotestosterone; Enzyme Inhibitors; Finasteride; Flutamide; In Vitro Techniques; Male; Mice; Models, Biological; Models, Theoretical; Muscle Contraction; Muscle, Smooth; Phosphorylation; Protein Kinase C; Pyridines; Receptors, Androgen; rho-Associated Kinases; Signal Transduction; Testosterone

2010
Rho kinase activation and ROS production contributes to the cooling enhanced contraction in cutaneous equine digital veins.
    Journal of applied physiology (Bethesda, Md. : 1985), 2010, Volume: 109, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Amides; Animals; Antioxidants; Benzophenanthridines; Body Temperature Regulation; Brimonidine Tartrate; Cold Temperature; Cyclic N-Oxides; Cytoskeletal Proteins; Female; Horses; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; Quinoxalines; Reactive Oxygen Species; rho-Associated Kinases; Rotenone; Spin Labels; Vasoconstriction; Vasodilator Agents; Veins

2010
Characteristics of myogenic reactivity in isolated rat mesenteric veins.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2011, Volume: 300, Issue:2

    Topics: Amides; Animals; Benzophenanthridines; Calcium; Calcium Channels, L-Type; Compliance; Endothelin-1; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitric Oxide Synthase Type III; Nitroarginine; Norepinephrine; Pressure; Protein Kinase C; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases

2011
Chelerythrine perturbs lamellar actomyosin filaments by selective inhibition of myotonic dystrophy kinase-related Cdc42-binding kinase.
    FEBS letters, 2011, May-06, Volume: 585, Issue:9

    Topics: Actomyosin; Amides; Animals; Antineoplastic Agents; Benzophenanthridines; Biocatalysis; Cell Line, Tumor; Cell Movement; Chlorocebus aethiops; COS Cells; Cytoskeleton; Dose-Response Relationship, Drug; Enzyme Inhibitors; HeLa Cells; Humans; Immunoblotting; Microscopy, Fluorescence; Molecular Structure; Myosins; Myotonin-Protein Kinase; Phosphorylation; Protein Serine-Threonine Kinases; Pyridines; Recombinant Proteins; rho-Associated Kinases; Serine

2011
Dexmedetomidine-Induced Contraction Involves CPI-17 Phosphorylation in Isolated Rat Aortas.
    International journal of molecular sciences, 2016, Sep-30, Volume: 17, Issue:10

    Topics: Adrenergic alpha-2 Receptor Agonists; Amides; Animals; Aorta; Benzophenanthridines; Calcium; Cells, Cultured; Dexmedetomidine; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Myosin Light Chains; Phosphoproteins; Phosphorylation; Protein Kinase C; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; Yohimbine

2016
Signal Transduction Underlying the Inhibitory Mechanism of Fluoxetine on Electrical Field Stimulation Response in Rat Ileal Smooth Muscle.
    Pharmacology, 2017, Volume: 99, Issue:5-6

    Topics: 4-Aminopyridine; Amides; Animals; Atropine; Azepines; Benzophenanthridines; Bicuculline; Calcimycin; Drug Interactions; Electric Stimulation; Estrenes; Fluoxetine; Glyburide; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Ondansetron; Pyridines; Pyrrolidinones; Rats; Signal Transduction; Sulfonamides; Tetraethylammonium

2017