Page last updated: 2024-09-03

changrolin and mexiletine

changrolin has been researched along with mexiletine in 2 studies

Compound Research Comparison

Studies
(changrolin)
Trials
(changrolin)
Recent Studies (post-2010)
(changrolin)
Studies
(mexiletine)
Trials
(mexiletine)
Recent Studies (post-2010) (mexiletine)
38001,488210227

Protein Interaction Comparison

ProteinTaxonomychangrolin (IC50)mexiletine (IC50)
5-hydroxytryptamine receptor 2BHomo sapiens (human)1.138
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)10
Sodium channel protein type 5 subunit alphaHomo sapiens (human)3
Sodium channel protein type 2 subunit alphaHomo sapiens (human)2.9

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, YH; Cheng, JH; Dai, DZ; Huang, J; Huang, WL; Liu, J; Peng, SX; Qiu, YT; Rong, P1
Kuang, Y; Liu, TP1

Other Studies

2 other study(ies) available for changrolin and mexiletine

ArticleYear
Anti-arrhythmic activities of six indole derivatives of changrolin.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1991, Volume: 12, Issue:5

    Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Guinea Pigs; Indoles; Mexiletine; Myocardial Reperfusion Injury; Quinazolines; Tachycardia; Ventricular Fibrillation

1991
Rate-dependent depression of maximal rate of depolarization in guinea pig papillary muscle action potentials by changrolin.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1990, Volume: 11, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Benzeneacetamides; Female; Guinea Pigs; In Vitro Techniques; Male; Mexiletine; Papillary Muscles; Piperidines; Quinazolines; Quinidine

1990