Page last updated: 2024-09-05

cgs 20625 and diazepam

cgs 20625 has been researched along with diazepam in 4 studies

Compound Research Comparison

Studies
(cgs 20625)
Trials
(cgs 20625)
Recent Studies (post-2010)
(cgs 20625)
Studies
(diazepam)
Trials
(diazepam)
Recent Studies (post-2010) (diazepam)
90218,3772,3291,790

Protein Interaction Comparison

ProteinTaxonomycgs 20625 (IC50)diazepam (IC50)
Gamma-aminobutyric acid receptor subunit piHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit deltaHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-1Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0108
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0227
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0106
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-4Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit epsilonHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit gamma-1Homo sapiens (human)0.0101
GABA theta subunitRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit gamma-3Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit thetaHomo sapiens (human)0.0101

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's2 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Franklin, SR; Tang, AH1
Bennett, DA; Braunwalder, AF; Jarvis, MF; Loo, PA; Schmutz, M; Thompson, TN; Wasley, JW; Williams, M; Yokoyoma, N1
Amrick, CL; Bennett, DA; Braunwalder, AF; Loo, PS; Schmutz, M; Thompson, TN; Wasley, JW; Williams, M; Wilson, DE; Yokoyoma, N1
Bennett, DA1

Reviews

1 review(s) available for cgs 20625 and diazepam

ArticleYear
Pharmacology of the pyrazolo-type compounds: agonist, antagonist and inverse agonist actions.
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Hypnotics and Sedatives; Muscle Relaxants, Central; Pyrazoles; Rats; Receptors, GABA-A

1987

Other Studies

3 other study(ies) available for cgs 20625 and diazepam

ArticleYear
The discriminative stimulus effects of diazepam in rats at two training doses.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam

1991
CGS 20625, a novel pyrazolopyridine with selective anxiolytic activity.
    Progress in clinical and biological research, 1990, Volume: 361

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Biological Availability; Diazepam; Flunitrazepam; Learning; Male; Motor Activity; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter

1990
CGS 20625, a novel pyrazolopyridine anxiolytic.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Male; Motor Activity; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Receptors, GABA-A

1989