Page last updated: 2024-09-05

cgp 54626 and n-(4,4-diphenyl-3-butenyl)nipecotic acid

cgp 54626 has been researched along with n-(4,4-diphenyl-3-butenyl)nipecotic acid in 1 studies

Compound Research Comparison

Studies
(cgp 54626)
Trials
(cgp 54626)
Recent Studies (post-2010)
(cgp 54626)
Studies
(n-(4,4-diphenyl-3-butenyl)nipecotic acid)
Trials
(n-(4,4-diphenyl-3-butenyl)nipecotic acid)
Recent Studies (post-2010) (n-(4,4-diphenyl-3-butenyl)nipecotic acid)
57016121022

Protein Interaction Comparison

ProteinTaxonomycgp 54626 (IC50)n-(4,4-diphenyl-3-butenyl)nipecotic acid (IC50)
Cytochrome P450 3A4Homo sapiens (human)0.6918
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)0.165
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)0.4099

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balana, B; Dolev, I; Laviv, T; Riven, I; Slesinger, PA; Slutsky, I; Vertkin, I1

Other Studies

1 other study(ies) available for cgp 54626 and n-(4,4-diphenyl-3-butenyl)nipecotic acid

ArticleYear
Basal GABA regulates GABA(B)R conformation and release probability at single hippocampal synapses.
    Neuron, 2010, Jul-29, Volume: 67, Issue:2

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Animals, Newborn; Baclofen; CA1 Region, Hippocampal; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Egtazic Acid; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agents; gamma-Aminobutyric Acid; In Vitro Techniques; Microscopy, Confocal; Neurons; Nipecotic Acids; Organophosphorus Compounds; Potassium Chloride; Presynaptic Terminals; Probability; Protein Conformation; Pyridinium Compounds; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Synapses; Tetrodotoxin

2010