cgp 54626 has been researched along with baclofen in 19 studies
Studies (cgp 54626) | Trials (cgp 54626) | Recent Studies (post-2010) (cgp 54626) | Studies (baclofen) | Trials (baclofen) | Recent Studies (post-2010) (baclofen) |
---|---|---|---|---|---|
57 | 0 | 16 | 6,017 | 372 | 1,535 |
Protein | Taxonomy | cgp 54626 (IC50) | baclofen (IC50) |
---|---|---|---|
Gamma-aminobutyric acid type B receptor subunit 2 | Homo sapiens (human) | 0.05 | |
Gamma-aminobutyric acid type B receptor subunit 2 | Rattus norvegicus (Norway rat) | 0.2762 | |
Gamma-aminobutyric acid type B receptor subunit 1 | Homo sapiens (human) | 0.05 | |
Gamma-aminobutyric acid type B receptor subunit 1 | Rattus norvegicus (Norway rat) | 0.2762 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (5.26) | 18.2507 |
2000's | 11 (57.89) | 29.6817 |
2010's | 7 (36.84) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bernasconi, R; Bittiger, H; De Barry, J; Marescaux, C; Mathivet, P | 1 |
Ferguson, SC; McFarlane, S | 1 |
Medda, BK; Sengupta, JN; Shaker, R | 1 |
Bettler, B; Bräuner-Osborne, H; Cryan, JF; Froestl, W; Kaupmann, K; Klebs, K; Mombereau, C; Mosbacher, J; Sansig, G; Schmutz, M; van der Putten, H; Waldmeier, P; Wellendorph, P | 1 |
Farb, DH; Gravielle, MC; Lyons, HR; Martin, SC; Russek, SJ; Steiger, JL | 1 |
Bourova, L; Hejnova, L; Ihnatovych, I; Novotny, J; Stöhr, J; Svoboda, P | 1 |
Kerr, DI; Marino, V; Ong, J; Parker, DA | 1 |
Priest, CA; Puche, AC | 1 |
Carai, MA; Carboni, G; Castelli, MP; Gessa, GL; Pibiri, F | 1 |
Colón, J; Luján, R; Marker, CL; Wickman, K | 1 |
Friedrich, RW; Tabor, R; Yaksi, E | 1 |
Baumann, O; Blenau, W; Rotte, C; Walz, B; Witte, J | 1 |
Balana, B; Dolev, I; Laviv, T; Riven, I; Slesinger, PA; Slutsky, I; Vertkin, I | 1 |
Bernier, BE; Clements, MA; Morikawa, H; Perra, S | 1 |
Chen, CC; Cheng, SJ; Lin, CC; Lu, HC; Min, MY; Wang, HY; Wu, Y; Yang, HW | 1 |
Berdichevsky, Y; Bettler, B; Fogel, H; Laviv, T; Riven, I; Slesinger, PA; Slutsky, I; Vertkin, I | 1 |
Lalive, AL; Luján, R; Lüscher, C; Martínez-Hernández, J; Moss, SJ; Munoz, MB; Padgett, CL; Pangalos, MN; Slesinger, PA; Tan, KR; Terunuma, M; Watanabe, M | 1 |
Martire, M; Samengo, IA; Scotti, V | 1 |
Borst, JG; Hruskova, B; Rusu, SI; Turecek, R; Wang, T | 1 |
19 other study(ies) available for cgp 54626 and baclofen
Article | Year |
---|---|
Binding characteristics of gamma-hydroxybutyric acid as a weak but selective GABAB receptor agonist.
Topics: Animals; Anticonvulsants; Baclofen; Binding, Competitive; Brain Chemistry; Ethosuximide; GABA Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Organophosphorus Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-B; Sodium Oxybate; Valproic Acid | 1997 |
GABA and development of the Xenopus optic projection.
Topics: Analysis of Variance; Animals; Baclofen; Blotting, Western; Culture Techniques; Dose-Response Relationship, Drug; Embryo, Nonmammalian; Embryonic Development; Epithelial Cells; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; Muscimol; Neurites; Neurons; Organophosphorus Compounds; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Retinal Ganglion Cells; Visual Pathways; Xenopus laevis | 2002 |
Effect of GABA(B) receptor agonist on distension-sensitive pelvic nerve afferent fibers innervating rat colon.
Topics: Afferent Pathways; Animals; Baclofen; Biomechanical Phenomena; Colon; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Male; Nerve Fibers; Organophosphorus Compounds; Pelvis; Physical Stimulation; Pressure; Rats; Rats, Long-Evans; Receptors, GABA-B; Spinal Nerve Roots | 2002 |
Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA(B)(1)-deficient mice.
Topics: 4-Butyrolactone; Adjuvants, Anesthesia; Animals; Anticonvulsants; Autoradiography; Baclofen; Behavior, Animal; Benzocycloheptenes; Binding, Competitive; Body Weight; Brain; Cell Membrane; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; Electroencephalography; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Guanosine 5'-O-(3-Thiotriphosphate); Mice; Mice, Inbred BALB C; Mice, Knockout; Motor Activity; Organophosphorus Compounds; Phenols; Radioligand Assay; Receptors, GABA-B; Sodium Oxybate; Time Factors | 2003 |
Differential expression of gamma-aminobutyric acid type B receptor subunit mRNAs in the developing nervous system and receptor coupling to adenylyl cyclase in embryonic neurons.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Binding Sites; Blotting, Western; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; In Situ Hybridization; Inhibitory Concentration 50; Male; Nervous System; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium | 2004 |
Increased baclofen-stimulated G protein coupling and deactivation in rat brain cortex during development.
Topics: Aging; Analysis of Variance; Animals; Animals, Newborn; Baclofen; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Male; Organophosphorus Compounds; Protein Binding; Proteins; Radioligand Assay; Rats; RGS Proteins; Tritium | 2004 |
Gabapentin activates presynaptic GABAB heteroreceptors in rat cortical slices.
Topics: Amines; Animals; Baclofen; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Gabapentin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Morpholines; Neocortex; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Presynaptic; Tritium | 2004 |
GABAB receptor expression and function in olfactory receptor neuron axon growth.
Topics: Analysis of Variance; Animals; Animals, Newborn; Axons; Baclofen; Cells, Cultured; Drug Interactions; Embryo, Mammalian; Female; GABA Agonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gene Expression Regulation; Glutamate Decarboxylase; Growth Cones; Immunohistochemistry; In Vitro Techniques; Male; Mice; Olfactory Bulb; Olfactory Mucosa; Olfactory Receptor Neurons; Organophosphorus Compounds; Pregnancy; Receptors, GABA-B; Time Factors | 2004 |
Up-regulation of GABA(B) receptors by chronic administration of the GABA(B) receptor antagonist SCH 50,911.
Topics: Animals; Baclofen; Binding, Competitive; Brain; Dose-Response Relationship, Drug; GABA Agonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Male; Mice; Mice, Inbred DBA; Morpholines; Organophosphorus Compounds; Receptors, GABA-B; Sulfur Radioisotopes; Tritium; Up-Regulation | 2005 |
Distinct populations of spinal cord lamina II interneurons expressing G-protein-gated potassium channels.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Baclofen; Blotting, Western; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; Immunohistochemistry; Immunoprecipitation; In Vitro Techniques; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Immunoelectron; Organophosphorus Compounds; Receptors, GABA; Receptors, Opioid, mu; Spinal Cord; Synapses | 2006 |
Multiple functions of GABA A and GABA B receptors during pattern processing in the zebrafish olfactory bulb.
Topics: Animals; Baclofen; Calcium; Food; GABA Agonists; GABA Antagonists; Neural Pathways; Neurons; Odorants; Olfactory Bulb; Organophosphorus Compounds; Patch-Clamp Techniques; Pyridazines; Receptors, GABA-A; Receptors, GABA-B; Smell; Zebrafish | 2008 |
Source, topography and excitatory effects of GABAergic innervation in cockroach salivary glands.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Electrophysiology; Fluorescent Antibody Technique; GABA Agonists; gamma-Aminobutyric Acid; Neurons; Organophosphorus Compounds; Periplaneta; Phosphinic Acids; Salivary Glands | 2009 |
Basal GABA regulates GABA(B)R conformation and release probability at single hippocampal synapses.
Topics: Analysis of Variance; Anesthetics, Local; Animals; Animals, Newborn; Baclofen; CA1 Region, Hippocampal; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Egtazic Acid; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agents; gamma-Aminobutyric Acid; In Vitro Techniques; Microscopy, Confocal; Neurons; Nipecotic Acids; Organophosphorus Compounds; Potassium Chloride; Presynaptic Terminals; Probability; Protein Conformation; Pyridinium Compounds; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Synapses; Tetrodotoxin | 2010 |
In vivo ethanol experience increases D(2) autoinhibition in the ventral tegmental area.
Topics: Action Potentials; Analysis of Variance; Animals; Baclofen; Central Nervous System Depressants; Chelating Agents; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Stimulation; Enzyme Inhibitors; Estrenes; Ethanol; GABA Antagonists; GABA-B Receptor Agonists; In Vitro Techniques; Indoles; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Pyrrolidinones; Receptors, Dopamine D2; Time Factors; Ventral Tegmental Area | 2011 |
GABAB receptor-mediated tonic inhibition of noradrenergic A7 neurons in the rat.
Topics: Analysis of Variance; Animals; Anisoles; Baclofen; Barium; Bee Venoms; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation; In Vitro Techniques; Lysine; Male; Morpholines; Neural Inhibition; Neurons; Nipecotic Acids; Norepinephrine; Organophosphorus Compounds; Oximes; Patch-Clamp Techniques; Pons; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; RNA, Messenger | 2011 |
Compartmentalization of the GABAB receptor signaling complex is required for presynaptic inhibition at hippocampal synapses.
Topics: Analysis of Variance; Animals; Baclofen; Calcium; Calcium Channels, N-Type; Cyclic AMP; Electric Stimulation; GABA Antagonists; GABA-B Receptor Agonists; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; Hippocampus; Luminescent Proteins; Mice; Mice, Inbred BALB C; Mice, Knockout; Microscopy, Confocal; Mutation; Neural Inhibition; Organophosphorus Compounds; Pertussis Toxin; Picrotoxin; Presynaptic Terminals; Rats; Rats, Wistar; Receptors, GABA-B; Signal Transduction; Spectroscopy, Fourier Transform Infrared; Synapses; Synaptic Vesicles | 2011 |
Methamphetamine-evoked depression of GABA(B) receptor signaling in GABA neurons of the VTA.
Topics: Action Potentials; Animals; Animals, Newborn; Baclofen; Bacterial Proteins; Central Nervous System Stimulants; Channelrhodopsins; Dopamine; Dopamine Agents; Down-Regulation; Drug Interactions; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Green Fluorescent Proteins; Homeodomain Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Luminescent Proteins; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Mice, Transgenic; Microscopy, Immunoelectron; Neurons; Organophosphorus Compounds; Phosphorylation; Receptors, GABA-A; Transcription Factors; Ventral Tegmental Area | 2012 |
Co-application of the GABAB receptor agonist, baclofen, and the mGlu receptor agonist, L-CCG-I, facilitates [(3)H]GABA release from rat cortical nerve endings.
Topics: Amino Acids, Dicarboxylic; Animals; Baclofen; Cerebral Cortex; Chelating Agents; Estrenes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; gamma-Aminobutyric Acid; Male; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Wistar; Synaptosomes; Time Factors | 2013 |
Modulation of synaptic depression of the calyx of Held synapse by GABA(B) receptors and spontaneous activity.
Topics: Acoustic Stimulation; Action Potentials; Age Factors; Animals; Baclofen; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Long-Term Synaptic Depression; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Receptors, GABA-B; Synapses; Synaptic Potentials; Tegmentum Mesencephali | 2013 |