Page last updated: 2024-09-05

cgp 54626 and 3-aminopropylphosphinic acid

cgp 54626 has been researched along with 3-aminopropylphosphinic acid in 3 studies

Compound Research Comparison

Studies
(cgp 54626)
Trials
(cgp 54626)
Recent Studies (post-2010)
(cgp 54626)
Studies
(3-aminopropylphosphinic acid)
Trials
(3-aminopropylphosphinic acid)
Recent Studies (post-2010) (3-aminopropylphosphinic acid)
570163002

Protein Interaction Comparison

ProteinTaxonomycgp 54626 (IC50)3-aminopropylphosphinic acid (IC50)
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0052
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0051

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Angst, C; Bettler, B; Bischoff, S; Bittiger, H; Flor, PJ; Froestl, W; Heid, J; Huggel, K; Kaupmann, K; McMaster, G; Mickel, SJ1
Bernasconi, R; Bittiger, H; De Barry, J; Marescaux, C; Mathivet, P1
Farb, DH; Gravielle, MC; Lyons, HR; Martin, SC; Russek, SJ; Steiger, JL1

Other Studies

3 other study(ies) available for cgp 54626 and 3-aminopropylphosphinic acid

ArticleYear
Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors.
    Nature, 1997, Mar-20, Volume: 386, Issue:6622

    Topics: Adenylyl Cyclases; Affinity Labels; Amino Acid Sequence; Animals; Azides; Benzoates; Cell Line; Central Nervous System; Cloning, Molecular; COS Cells; DNA, Complementary; Escherichia coli; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Situ Hybridization; Ligands; Molecular Sequence Data; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Recombinant Proteins; RNA, Messenger; Sequence Alignment

1997
Binding characteristics of gamma-hydroxybutyric acid as a weak but selective GABAB receptor agonist.
    European journal of pharmacology, 1997, Feb-19, Volume: 321, Issue:1

    Topics: Animals; Anticonvulsants; Baclofen; Binding, Competitive; Brain Chemistry; Ethosuximide; GABA Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Organophosphorus Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-B; Sodium Oxybate; Valproic Acid

1997
Differential expression of gamma-aminobutyric acid type B receptor subunit mRNAs in the developing nervous system and receptor coupling to adenylyl cyclase in embryonic neurons.
    The Journal of comparative neurology, 2004, May-17, Volume: 473, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Binding Sites; Blotting, Western; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; In Situ Hybridization; Inhibitory Concentration 50; Male; Nervous System; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium

2004