Page last updated: 2024-09-03

cgp 46381 and gamma-aminobutyric acid

cgp 46381 has been researched along with gamma-aminobutyric acid in 3 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Compound Research Comparison

Studies
(cgp 46381)
Trials
(cgp 46381)
Recent Studies (post-2010)
(cgp 46381)
Studies
(gamma-aminobutyric acid)
Trials
(gamma-aminobutyric acid)
Recent Studies (post-2010) (gamma-aminobutyric acid)
250540,2151,4239,631

Protein Interaction Comparison

ProteinTaxonomycgp 46381 (IC50)gamma-aminobutyric acid (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0292
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0332
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0323
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.152
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0333
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.2623
Sodium- and chloride-dependent taurine transporterHomo sapiens (human)354
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)2.51
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)6.349
Sodium- and chloride-dependent GABA transporter 2Mus musculus (house mouse)7.0795
Sodium- and chloride-dependent GABA transporter 3Mus musculus (house mouse)8.1283
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent betaine transporterHomo sapiens (human)6.4082
Sodium- and chloride-dependent GABA transporter 3Homo sapiens (human)3.9953
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0333
GABA theta subunitRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0292

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Curtis, DR; Lacey, G1
Bowery, NG; Da Silva, H; Malcangio, M1
Akiba, Y; Baker, H; Cave, JW; Estevez, AG; Huerta, PT; Sasaki, H1

Other Studies

3 other study(ies) available for cgp 46381 and gamma-aminobutyric acid

ArticleYear
GABA-B receptor-mediated spinal inhibition.
    Neuroreport, 1994, Jan-31, Volume: 5, Issue:5

    Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Cats; Decerebrate State; Depression, Chemical; GABA Antagonists; gamma-Aminobutyric Acid; Organophosphorus Compounds; Phosphinic Acids; Receptors, GABA; Reflex, Monosynaptic; Spinal Cord; Tetany

1994
Plasticity of GABAB receptor in rat spinal cord detected by autoradiography.
    European journal of pharmacology, 1993, Nov-30, Volume: 250, Issue:1

    Topics: Animals; Autoradiography; Baclofen; Binding Sites; gamma-Aminobutyric Acid; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B; Spinal Cord; Up-Regulation

1993
gamma-Aminobutyric acid-mediated regulation of the activity-dependent olfactory bulb dopaminergic phenotype.
    Journal of neuroscience research, 2009, Aug-01, Volume: 87, Issue:10

    Topics: Agatoxins; Amino Acids; Animals; Animals, Newborn; Bicuculline; Calcium Channel Blockers; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Green Fluorescent Proteins; Interneurons; Mice; Mice, Transgenic; Olfactory Bulb; Phosphinic Acids; Potassium Chloride; Prosencephalon; Spider Venoms; Tissue Culture Techniques; Tyrosine 3-Monooxygenase; Xanthenes

2009