Page last updated: 2024-09-03

cgp 42112a and saralasin

cgp 42112a has been researched along with saralasin in 9 studies

Compound Research Comparison

Studies
(cgp 42112a)
Trials
(cgp 42112a)
Recent Studies (post-2010)
(cgp 42112a)
Studies
(saralasin)
Trials
(saralasin)
Recent Studies (post-2010) (saralasin)
2330351,4971316

Protein Interaction Comparison

ProteinTaxonomycgp 42112a (IC50)saralasin (IC50)
Type-1A angiotensin II receptor Rattus norvegicus (Norway rat)0.0017
Type-1B angiotensin II receptorRattus norvegicus (Norway rat)0.0017
Type-1 angiotensin II receptorHomo sapiens (human)0.0006
Type-2 angiotensin II receptorHomo sapiens (human)0.0008

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bogdal, Y; Bottari, SP; Deschepper, CF; Obermüller, N; Zahs, KR1
Bühlmayer, P; Criscione, L; de Gasparo, M; Herold, P; Kamber, B; Ostermayer, F; Thomann, H; Whitebread, S1
Bottari, SP; Culman, J; de Gasparo, M; Gohlke, P; Obermüller, N; Unger, T1
Heemskerk, FM; Saavedra, JM1
Bihoreau, C; Clauser, E; Conchon, S; Corvol, P; Monnot, C; Sirieix, ME1
Bensoussan, M; Mitchell, T; Reilly, T; Ronco, PM; Timmermans, PB; Verroust, PJ1
Betteridge, LJ; Hughes, AD; Patel, MK; Schachter, M1
Cooper, S; Pulakat, L; Turner, CA1
de Arruda Camargo, LA; Saad, WA1

Other Studies

9 other study(ies) available for cgp 42112a and saralasin

ArticleYear
Characterization and distribution of angiotensin II binding sites in fetal and neonatal astrocytes from different rat brain regions.
    Brain research, 1992, Jul-10, Volume: 585, Issue:1-2

    Topics: Angiotensin II; Animals; Animals, Newborn; Astrocytes; Binding Sites; Binding, Competitive; Biphenyl Compounds; Brain; Cells, Cultured; Fetus; Imidazoles; Losartan; Oligopeptides; Rats; Saralasin; Tetrazoles; Tissue Distribution

1992
Binding characteristics and vascular effects of various angiotensin II antagonists.
    Journal of cardiovascular pharmacology, 1990, Volume: 16 Suppl 4

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Angiotensins; Animals; Aorta; Biphenyl Compounds; Dose-Response Relationship, Drug; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Losartan; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Rats; Receptors, Angiotensin; Saralasin; Uterus

1990
Distribution of angiotensin II receptor subtypes in rat brain nuclei.
    Neuroscience letters, 1991, Oct-28, Volume: 132, Issue:1

    Topics: Angiotensin II; Animals; Binding, Competitive; Biphenyl Compounds; Brain; Brain Stem; Hypothalamus; Imidazoles; Iodine Radioisotopes; Losartan; Male; Mesencephalon; Oligopeptides; Organ Specificity; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Saralasin; Tetrazoles

1991
Quantitative autoradiography of angiotensin II AT2 receptors with [125I]CGP 42112.
    Brain research, 1995, Apr-17, Volume: 677, Issue:1

    Topics: Adrenal Medulla; Angiotensin II; Animals; Autoradiography; Binding, Competitive; Densitometry; Geniculate Bodies; Image Processing, Computer-Assisted; Iodine Radioisotopes; Male; Oligopeptides; Olivary Nucleus; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Saralasin

1995
Synthetic cDNA encoding the rat AT1a receptor: a useful tool for structure-function relationship analysis.
    Biochemical and biophysical research communications, 1994, Mar-30, Volume: 199, Issue:3

    Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Base Sequence; Biphenyl Compounds; CHO Cells; Codon; Cricetinae; DNA, Complementary; Imidazoles; Kinetics; Losartan; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligodeoxyribonucleotides; Oligopeptides; Open Reading Frames; Pyridines; Rats; Receptors, Angiotensin; Restriction Mapping; Saralasin; Signal Transduction; Structure-Activity Relationship; Tetrazoles; Transfection

1994
Immunological reactivity of angiotensin II receptor antagonists: possible implications for receptor binding sites.
    European journal of pharmacology, 1993, Oct-15, Volume: 247, Issue:2

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antihypertensive Agents; Biphenyl Compounds; Imidazoles; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Losartan; Molecular Conformation; Oligopeptides; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles

1993
Angiotensin II receptors are exclusively of the AT1 subtype in cultured human vascular smooth muscle cells.
    Biochemical Society transactions, 1995, Volume: 23, Issue:3

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Binding, Competitive; Biphenyl Compounds; Cells, Cultured; Humans; Imidazoles; Kinetics; Losartan; Muscle, Smooth, Vascular; Oligopeptides; Receptors, Angiotensin; Saralasin; Tetrazoles

1995
Role of the His273 located in the sixth transmembrane domain of the angiotensin II receptor subtype AT2 in ligand-receptor interaction.
    Biochemical and biophysical research communications, 1999, Apr-21, Volume: 257, Issue:3

    Topics: Amino Acid Substitution; Angiotensin II; Animals; Binding Sites; Cell Membrane; Histidine; Ligands; Lysine; Oligopeptides; Oocytes; Rats; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; RNA, Messenger; Saralasin; Structure-Activity Relationship; Xenopus laevis

1999
Renal effects of angiotensin II receptor subtype 1 and 2-selective ligands injected into the paraventricular nucleus of conscious rats.
    Regulatory peptides, 1999, Oct-22, Volume: 84, Issue:1-3

    Topics: Angiotensin II; Animals; Injections, Intraventricular; Kidney; Ligands; Losartan; Male; Oligopeptides; Paraventricular Hypothalamic Nucleus; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Saralasin; Sodium

1999